Patents by Inventor Julius Diamond

Julius Diamond has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Amidinoureas for treating diarrhea
    Patent number: 4060635
    Abstract: A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-diarrheal agents.
    Type: Grant
    Filed: March 31, 1975
    Date of Patent: November 29, 1977
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, George H. Douglas
  • Amidinoureas
    Patent number: 4025652
    Abstract: A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-diarrheal agents.
    Type: Grant
    Filed: March 31, 1975
    Date of Patent: May 24, 1977
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, George H. Douglas
  • Carbamylguanidine antimicrobial compounds
    Patent number: 4022962
    Abstract: Antimicrobial compounds are disclosed having the formula:Z--B--Y--B'--Z .nHAwherein B is carbamylguaidino, or thiocarbamylguanidino and B' is B or biguanidino provided that B' is biguanidino only when B is carbamylguanidino bonded to Y through the guanidino portion of the group, Y is a bivalent organic radical selected from the group consisting of C.sub.2 -C.sub.12 alkylene, C.sub.5 -C.sub.12 cycloalkylene, C.sub.5 -C.sub.12 cycloalkylenebis(loweralkyl), C.sub.6 -C.sub.12 arylene and loweralkylarylene, C.sub.7 -C.sub.12 aryleneloweralkyl, and C.sub.8 -C.sub.12 arylenebis(loweralkyl) and Z is selected from the group consisting of C.sub.1 -C.sub.12 alkyl; C.sub.4 -C.sub.12 dialkylaminoalkyl; C.sub.3 -C.sub.12 alkenyl; C.sub.3 -C.sub.12 alkynyl; C.sub.3 -C.sub.12 cycloalkyl, C.sub.4 -C.sub.12 cycloalkylalkyl; C.sub.1 -C.sub.10 alkoxy C.sub.10 -C.sub.2 alkyl having a total carbon content of C.sub.3 -C.sub.14 ; C.sub.1 -C.sub.10 alkylthio C.sub.10 -C.sub.2 alkyl having a total carbon content of C.sub.3 -C.sub.
    Type: Grant
    Filed: February 3, 1975
    Date of Patent: May 10, 1977
    Assignee: Cooper Laboratories, Inc.
    Inventor: Julius Diamond
  • Phenylacetic acids
    Patent number: 4008269
    Abstract: Novel .alpha.-halo-p-cycloalkylphenylacetic acids and their derivatives have been prepared. Compounds of this invention possess useful anti-inflammatory, analgesic and antipyretic properties.
    Type: Grant
    Filed: December 10, 1973
    Date of Patent: February 15, 1977
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, Norman Julian Santora
  • Process for making a methenamine salt of an optically active acid
    Patent number: 4001231
    Abstract: Novel salts of hexamethylenetetramine formed from d- or l- enantiamorph of a selected acid are disclosed, and a process for the preparation is described. A new method for the treatment of urinary tract infections is also described.
    Type: Grant
    Filed: March 29, 1973
    Date of Patent: January 4, 1977
    Assignee: William H. Rorer, Inc.
    Inventor: Julius Diamond
  • 1,5-Disubstituted biguanides
    Patent number: 3996232
    Abstract: Novel 1-aryl and aralkyl 5-substituted biguanide compounds have been prepared. The compounds of this invention possess useful antiulcerogenic properties.
    Type: Grant
    Filed: October 3, 1973
    Date of Patent: December 7, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, Bernard J. Burns
  • Ethynylaryl compounds and derivatives thereof
    Patent number: 3987116
    Abstract: Novel ethynylaryl compounds and derivatives are described. Their use in the treatment of inflammation is also disclosed.
    Type: Grant
    Filed: August 1, 1974
    Date of Patent: October 19, 1976
    Assignee: William H. Rorer, Inc.
    Inventor: Julius Diamond
  • Phenyl propionic acids and derivatives thereof
    Patent number: 3985788
    Abstract: Novel .alpha.-halo-.beta.-(4-cyclohexylphenyl)propionic acids and their salts and esters are described. Therapeutic compositions containing same and a method of treating inflammation by their administration are also disclosed.
    Type: Grant
    Filed: October 4, 1973
    Date of Patent: October 12, 1976
    Assignee: William H. Rorer, Inc.
    Inventor: Julius Diamond
  • Ethynylindenyl compounds and derivatives thereof used in the treatment of pain, fever and inflammation
    Patent number: 3983253
    Abstract: Novel ethynylindenyl compounds and derivatives are described. Their use in the treatment of inflammation is also disclosed.
    Type: Grant
    Filed: January 16, 1974
    Date of Patent: September 28, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, George H. Douglas
  • Ethynylbenzene compounds and derivatives thereof
    Patent number: 3981932
    Abstract: Novel ethynylbenzene compounds and derivatives are described. Their use in the treatment of inflammation is also disclosed.
    Type: Grant
    Filed: May 14, 1975
    Date of Patent: September 21, 1976
    Assignee: William H. Rorer, Inc.
    Inventor: Julius Diamond
  • Phenylacetic acids
    Patent number: 3979428
    Abstract: Novel p-cycloalkylphenylacetic acids which are substituted in .alpha.-position by a carbamylthio, loweralkylcarbamylthio, or diloweralkylcarbamylthio group, and their salts have been prepared. They possess useful antiinflammatory, analgesic, and antipyretic properties.
    Type: Grant
    Filed: June 24, 1975
    Date of Patent: September 7, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, Norman Julian Santora
  • Guanidines
    Patent number: 3976643
    Abstract: Novel substituted phenylquanidine compounds and processes for their preparation are disclosed. Their use as anti-hypertensive agents is also revealed.
    Type: Grant
    Filed: February 20, 1975
    Date of Patent: August 24, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, George H. Douglas
  • D-aminophenylacetic acid compounds and derivatives
    Patent number: 3969401
    Abstract: Certain substituted .alpha.-halo and .alpha.-mercaptophenylacetic acids and substituted phenylacetic acids having in .alpha.-position a sulfur-containing group, a cyano group, or an amino group, their substantially non-toxic esters, salts, and acid amides as well as 5-phenyl substituted 2-imino-4-oxothiazolidines and 5-phenyl substituted 2,4-dioxothiazolidines have a high anti-inflammatory, analgesic, and antipyretic activity, low toxicity, and/or a favorable therapeutic index with minor or no side-effects. Preferred compounds of this invention are .alpha.,m-dichloro-p-cyclohexylphenylacetic acids and its esters and salts.
    Type: Grant
    Filed: August 14, 1973
    Date of Patent: July 13, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, Norman J. Santora
  • Phenyl butyric acids and derivatives thereof
    Patent number: 3966801
    Abstract: Novel substituted phenyl butyric acids and their derivatives are described. Therapeutic compositions and method of treatment of inflammation is also disclosed.
    Type: Grant
    Filed: December 13, 1973
    Date of Patent: June 29, 1976
    Assignee: William H. Rorer, Inc.
    Inventor: Julius Diamond
  • 1-Substituted biguanides for treating hyperacidity or ulceration
    Patent number: 3959488
    Abstract: The 1-substituted biguanides of this invention possess useful gastric anti-secretory and spasmolytic properties. Compounds of this type which also display anti-hypertensive and CNS depressant properties are also disclosed.
    Type: Grant
    Filed: December 6, 1973
    Date of Patent: May 25, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, George H. Douglas, Bernard J. Burns
  • 2-Thiosulfo biphenylylacetic acids
    Patent number: 3941821
    Abstract: Novel .alpha.-mercapto-p-biphenylylacetic acids and their derivatives have been prepared. Compounds of this invention possess useful anti-inflammatory, analgesic and antipyretic properties.
    Type: Grant
    Filed: March 8, 1974
    Date of Patent: March 2, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, Norman Julian Santora
  • Alpha-acyl substituted naphthylacetic acids
    Patent number: 3931269
    Abstract: Novel naphthylalkanoic acids and their derivatives are described. Therapeutic compositions and method of treatment of inflammation is also disclosed.
    Type: Grant
    Filed: February 28, 1975
    Date of Patent: January 6, 1976
    Assignee: William H. Rorer, Inc.
    Inventors: Julius Diamond, Ching Tan Tsuei