Patents by Inventor Klaus Hasspacher

Klaus Hasspacher has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4980359
    Abstract: Compounds of formula I ##STR1## wherein R.sub.1 is hydrogen or C.sub.1-4 alkyl; R.sub.2 is hydrogen and R.sub.3 is hydrogen or C.sub.1-4 alkyl, or R.sub.2 and R.sub.3 together represent an additional bond as indicated by the dotted line; R.sub.4 is hydrogen, C.sub.1-4 alkyl or phenyl; R.sub.5 is methoxy or ethoxy; R.sub.6 is hydrogen, hydroxy, C.sub.1-4 alkoxy, hydroxy-(C.sub.2-4 alkoxy) or (C.sub.1-4 alkoxy)-(C.sub.2-4 alkoxy); R.sub.7 and R.sub.8 are each independently C.sub.1-4 alkoxy or (C.sub.1-4 alkoxy)-(C.sub.2-4 alkoxy); and R.sub.9 is hydrogen or halogen,in free form or pharmaceutically acceptable salt form, have pharmaceutical utility, in particular as bronchodilators, eosinophil accumulation and/or activation inhibiting agents and in the treatment of prophylactic treatment of obstructive or inflammatory airways diseases.
    Type: Grant
    Filed: April 10, 1990
    Date of Patent: December 25, 1990
    Assignee: Sandoz Ltd.
    Inventors: Klaus Hasspacher, Reto Naef
  • Patent number: 4609664
    Abstract: Piperidylidene derivatives of formula ##STR1## wherein n is 2 or 3, R.sub.1 comprises a tricyclic nucleus and R.sub.2 is hydrogen or an acid residue, useful in the treatment and prophylaxis of asthmatic conditions.
    Type: Grant
    Filed: July 16, 1984
    Date of Patent: September 2, 1986
    Assignee: Sandoz Ltd.
    Inventor: Klaus Hasspacher
  • Patent number: 4351838
    Abstract: The invention provides compounds of formula ##STR1## wherein R.sub.1 and R.sub.2 are alkyl, R.sub.3 is hydrogen, alkyl, alkenyl, phenylalkyl or a group --(CH.sub.2 --CH.sub.2 --O).sub.n --R.sub.4 in which n is 1 to 3 and R.sub.4 is hydrogen or an acid residue, and the ring A is unsubstituted or substituted, with the proviso that when R.sub.3 is methyl the ring A is substituted. The compounds are useful in the treatment and prophylaxis of allergic conditions.
    Type: Grant
    Filed: February 12, 1981
    Date of Patent: September 28, 1982
    Assignee: Sandoz Ltd.
    Inventor: Klaus Hasspacher
  • Patent number: 4123545
    Abstract: The present invention provides a compound of the formula ##STR1## which possesses pharmacological activity, for example anti-psychotic activity.
    Type: Grant
    Filed: June 30, 1977
    Date of Patent: October 31, 1978
    Assignee: Sandoz Ltd.
    Inventors: Klaus Hasspacher, Michael Strasser
  • Patent number: 4094987
    Abstract: This invention provides compounds of formula I, ##STR1## wherein R.sub.1 is alkyl of 4 to 8 carbon atoms; cycloalkyl of 4 to 6 carbon atoms; phenethyl or phenethyl monosubstituted in the phenyl residue with fluorine, chlorine, bromine, methoxy or alkyl of 1 to 4 carbon atoms; 2-tetrahydrofurylmethyl or 2-furylmethyl,Useful as analgesic agents.
    Type: Grant
    Filed: January 24, 1977
    Date of Patent: June 13, 1978
    Assignee: Sandoz Ltd.
    Inventors: Klaus Hasspacher, Michael Strasser
  • Patent number: 3958003
    Abstract: The present invention concerns new heterocyclic compounds of the formula: ##SPC1##WhereinR.sub.1 and R.sub.2 are inter alia alkyl, chlorine or methoxy,R.sub.3 is hydroxy, alkylcarboxy or monoalkylcarbamoyloxy, andA is protected or unprotected carbonyl.The compounds possess analgesic and central nervous system depressant properties.
    Type: Grant
    Filed: May 2, 1975
    Date of Patent: May 18, 1976
    Assignee: Sandoz Ltd.
    Inventors: Jean-Michel Bastian, Klaus Hasspacher, Michael Strasser