Patent number: 4087422
Abstract: Dihydrotetrazolo [1,5-a] quinazolines having the formula: ##STR1## wherein (a) n is 0, X is oxygen, and R is optionally unsubstituted alkyl, alkenyl of at least 4 carbon atoms, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, amino or substituted aryl; or (b) n is 1 or 2, X is oxygen, R is hydrogen, or optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy or (c) n is 0, 1 or 2, X is sulphur, R is hydrogen, or optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy; or (d) n is 0, 1 or 2, X is NR.sub.2 where R.sub.2 is hydrogen, alkyl having 1 to 10 carbon atoms, benzyl or hydroxyalkyl, R is optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy; and salts thereof. These compounds demonstrate pesticidal activity.
Type:
Grant
Filed:
June 13, 1977
Date of Patent:
May 2, 1978
Assignee:
Imperial Chemical Industries Limited
Inventors:
Raymond Alexander Bowie, John Michael Cox, Gordon Michael Farrell, Margaret Claire Shephard
Patent number: 4056384
Abstract: Dihydrotetrazolo [1,5-a] quinazolines having the formula ##STR1## wherein (a) n is zero, X is oxygen, and R is optionally unsubstituted alkyl, alkenyl of at least 4 carbon atoms, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, amino or substituted aryl; or (b) n is 1 or 2, X is oxygen, R is hydrogen, or optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy or (c) n is zero, 1 or 2, X is sulphur, R is hydrogen, or optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy; or (d) n is 0, 1 or 2, X is NR.sub.2 where R.sub.2 is hydrogen, alkyl having 1 to 10 carbon atoms, benzyl or hydroxyalkyl, R is optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy; and salts thereof. These compounds demonstrate pesticidal activity.
Type:
Grant
Filed:
August 25, 1975
Date of Patent:
November 1, 1977
Assignee:
Imperial Chemical Industries Limited
Inventors:
Raymond Alexander Bowie, John Michael Cox, Gordon Michael Farrell, Margaret Claire Shephard