Patents by Inventor Michael Pieper

Michael Pieper has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20080063608
    Abstract: A pharmaceutical composition comprising: (a) an anticholinergic of formula 1 wherein X? is an anion with a single negative charge; (b) a corticosteroid; and (c) a betamimetic, wherein each component (a), (b), and (c) are optionally in the form of the solvates or hydrates thereof, processes for preparing them, and their use in the treatment of respiratory diseases.
    Type: Application
    Filed: June 7, 2007
    Publication date: March 13, 2008
    Applicant: Boehringer Ingelheim Pharma GmbH & Co. KG
    Inventors: Michael Pieper, Christopher Meade, Michel Pairet
  • Publication number: 20080051444
    Abstract: The invention relates to the use of dopamine receptor agonists for preparing a pharmaceutical composition for the reduction of excessive food intake.
    Type: Application
    Filed: September 18, 2007
    Publication date: February 28, 2008
    Inventors: Michael Pieper, Joachim Mierau
  • Publication number: 20080051443
    Abstract: The invention relates to the use of dopamine receptor agonists for preparing a pharmaceutical composition for the reduction of excessive food intake.
    Type: Application
    Filed: September 18, 2007
    Publication date: February 28, 2008
    Inventors: Michael Pieper, Joachim Mierau
  • Publication number: 20070259855
    Abstract: Disclosed are compounds of general formula (I), wherein the groups R1, R2, Ra and Rb have the meanings given in the claims and specification, the tautomers, racemates, enantiomers, diastereomers and the mixtures thereof, and optionally the pharmacologically acceptable acid addition salts, solvates and hydrates thereof, and processes for preparing these thiazolyl-dihydro-indazoles and the use thereof as pharmaceutical compositions.
    Type: Application
    Filed: March 23, 2007
    Publication date: November 8, 2007
    Inventors: Udo Maier, Matthias Grauert, Matthias Hoffmann, Christoph Hoenke, Anne Joergensen, Alexander Pautsch, Trixi Brandl, Steffen Breitfelder, Stefan Scheuerer, Klaus Erb, Michael Pieper, Ingo Pragst
  • Publication number: 20070244104
    Abstract: Disclosed are thiazolyl-dihydro-quinazolines of general formula (I) wherein the groups R1 to R4 have the meanings given in the claims and specification, the isomers thereof, and processes for preparing these compounds and their use as pharmaceutical compositions.
    Type: Application
    Filed: March 23, 2007
    Publication date: October 18, 2007
    Inventors: Trixi Brandl, Udo Maier, Matthias Hoffmann, Stefan Scheuerer, Anne Joergensen, Alexander Pautsch, Steffen Breitfelder, Matthias Grauert, Christoph Hoenke, Klaus Erb, Michael Pieper, Ingo Pragst
  • Publication number: 20070238718
    Abstract: The present invention relates to new thiazolyl-dihydro-indazoles of general formula (I) wherein the groups R1, R2 and R3 have the meanings given in the claims and specification, the tautomers, racemates, enantiomers, diastereomers and the mixtures thereof, and optionally the pharmacologically acceptable acid addition salts, solvates and hydrates thereof, and processes for preparing these thiazolyl-dihydro-indazoles and the use thereof as pharmaceutical compositions.
    Type: Application
    Filed: March 23, 2007
    Publication date: October 11, 2007
    Inventors: Matthias GRAUERT, Udo Maier, Matthias Hoffmann, Stefan Scheuerer, Anne Joergensen, Alexander Pautsch, Trixi Brandl, Christoph Hoenke, Steffen Breitfelder, Klaus Erb, Michael Pieper, Ingo Pragst
  • Publication number: 20070238746
    Abstract: Disclosed are compounds of general formula (I), wherein the groups A, R1, R2, Ra and Rb have the meanings given in the claims and specification, the tautomers, racemates, enantiomers, diastereomers and the mixtures thereof, and optionally the pharmacologically acceptable acid addition salts, solvates and hydrates thereof, and processes for preparing these thiazolyl-dihydro-quinazolines and the use thereof as pharmaceutical compositions.
    Type: Application
    Filed: March 23, 2007
    Publication date: October 11, 2007
    Inventors: Trixi Brandl, Udo Maier, Christoph Hoenke, Anne Joergensen, Alexander Pautsch, Steffen Breitfelder, Matthias Grauert, Matthias Hoffmann, Stefan Scheuerer, Klaus Erb, Michael Pieper, Ingo Pragst
  • Publication number: 20070238730
    Abstract: Disclosed are compounds of general formula (I), wherein the groups R1, R2, Ra and Rb have the meanings given in the claims and specification, the tautomers, racemates, enantiomers, diastereomers and the mixtures thereof, and optionally the pharmacologically acceptable acid addition salts, solvates and hydrates thereof, and processes for preparing these thiazolyl-dihydro-cyclopentapyrazoles and the use thereof as pharmaceutical compositions.
    Type: Application
    Filed: March 23, 2007
    Publication date: October 11, 2007
    Inventors: Steffen Breitfelder, Udo Maier, Christoph Hoenke, Anne Joergensen, Alexander Pautsch, Trixi Brandl, Matthias Grauert, Matthias Hoffmann, Stefan Scheuerer, Klaus Erb, Michael Pieper, Ingo Pragst
  • Publication number: 20070086951
    Abstract: Fluorenecarboxylic acid esters of general formula 1 wherein X? and the groups A, R, R1, R2, R3, R3?, R4, and R4? have the meanings given in the claims and in the specification, processes for the manufacture thereof and the use thereof a medicaments.
    Type: Application
    Filed: November 10, 2006
    Publication date: April 19, 2007
    Inventors: Sabine Germeyer, Helmut Meissner, Gerd Morschhauser, Sabine Pestel, Michael Pieper, Gerald Pohl, Richard Reichl, Georg Speck
  • Publication number: 20070086957
    Abstract: A pharmaceutical composition comprising: (a) a compound of formula 1 wherein: n is 1 or 2; R1 is hydrogen, halogen, C1-4-alkyl, or O—C1-4-alkyl; R2 is hydrogen, halogen, C1-4-alkyl, or O—C1-4-alkyl; and R3 is hydrogen, C1-4-alkyl, OH, halogen, O—C1-4-alkyl, O—C1-4-alkylene-COOH, or O—C1-4-alkylene-COO—C1-4-alkyl, or an enantiomer, mixture of enantiomers, or racemate thereof, or an acid addition salt with pharmacologically acceptable acids thereof, or a solvate or hydrate thereof; and (b) another active substance 2, wherein the molar ratio of the compound of formula 1 to the active substance 2 is 1:10 to 12:1.
    Type: Application
    Filed: October 5, 2006
    Publication date: April 19, 2007
    Inventors: Thierry Bouyssou, Michael Pieper, Andreas Schnapp
  • Publication number: 20070021333
    Abstract: The present invention relates to novel pharmaceutical compositions based on anticholinergics and soluble TNF receptor fusion proteins, processes for preparing them and their use in the treatment of respiratory diseases.
    Type: Application
    Filed: February 7, 2004
    Publication date: January 25, 2007
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Christopher Meade, Michael Pieper, Michel Pairet
  • Publication number: 20060286040
    Abstract: The present invention relates to novel pharmaceutical compositions based on anticholinergics of the formula 1; wherein X?, R1 ? and Ar are defined as in claim 1, and a heterocyclic compound of the formula 2. Furthermore, the invention relates to processes for preparing them and their use in the treatment of respiratory complaints.
    Type: Application
    Filed: August 5, 2004
    Publication date: December 21, 2006
    Applicant: Kyowa Hakko Kogyo Co., Ltd.
    Inventors: Christopher Meade, Michel Pairet, Michael Pieper, Yuzuru Abe, Ichiro Miki
  • Publication number: 20060287530
    Abstract: The invention relates to a process for preparing new tiotropium salts, these new tiotropium salts as such, pharmaceutical formulations containing them and their use for preparing a medicament.
    Type: Application
    Filed: June 15, 2006
    Publication date: December 21, 2006
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Mihaela Pop, Stephanie Mulder Houdayer, Peter Sieger, Michael Pieper
  • Publication number: 20060276441
    Abstract: A pharmaceutical composition comprising: (a) a salt of formula 1 wherein: X? is an anion with a single negative charge; and (b) a steroid 2, processes for preparing such pharmaceutical composition, and their use in the treatment of respiratory complaints.
    Type: Application
    Filed: April 20, 2006
    Publication date: December 7, 2006
    Applicant: Boehringer Ingelheim Pharma GmbH & Co. KG
    Inventors: Rolf Banholzer, Helmut Meissner, Gerd Morschhaeuser, Michael Pieper, Gerald Pohl, Richard Reichl, Georg Speck, Christopher Meade, Michel Pairet
  • Publication number: 20060270667
    Abstract: The present invention relates to new medicament combinations which contain in addition to one or more, preferably one, betamimetic 1, at least one anticholinergic 2 and at least one PDEIV-inhibitor 3, processes for preparing them and their use as pharmaceutical compositions.
    Type: Application
    Filed: May 30, 2006
    Publication date: November 30, 2006
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Michael PIEPER, Andreas Schnapp, Peter Nickolaus
  • Publication number: 20060251656
    Abstract: The present invention relates to novel pharmaceutical compositions based on anticholinergies and anti-TNF antibodies, processes for preparing them and their use in the treatment of respiratory diseases.
    Type: Application
    Filed: February 7, 2004
    Publication date: November 9, 2006
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Christopher Meade, Michael Pieper, Michel Pairet
  • Publication number: 20060239935
    Abstract: The present invention relates to new pharmaceutical compositions for inhalation containing one or more, preferably one anticholinergic 1 in combination with one or more pharmacologically acceptable acid addition salts of a compound of formula 2?, wherein the groups R1, R2, R3 and R4 may have the meanings given in the specification and in the claims, processes for preparing them and their use in the treatment of respiratory complaints.
    Type: Application
    Filed: April 21, 2006
    Publication date: October 26, 2006
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Thierry Bouyssou, Ingo Konetzki, Michael Pieper, Andreas Schnapp
  • Publication number: 20060239908
    Abstract: The present invention relates to new pharmaceutical compositions for inhalation containing one or more, preferably one anticholinergic 1 in combination with one or more betamimetics 2 and one or more steroids 3, processes for preparing them and their use in the treatment of respiratory complaints.
    Type: Application
    Filed: April 21, 2006
    Publication date: October 26, 2006
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Thierry Bouyssou, Ingo Konetzki, Michael Pieper, Andreas Schnapp
  • Publication number: 20060228305
    Abstract: The present invention relates to novel pharmaceutical compositions based on anticholinergics and TNF-alpha-antagonists, processes for preparing them and their use in the treatment of respiratory diseases.
    Type: Application
    Filed: February 7, 2004
    Publication date: October 12, 2006
    Applicant: Boehringer Ingelheim International GmbH
    Inventors: Christopher Meade, Michael Pieper, Michel Pairet
  • Publication number: 20060223869
    Abstract: The invention relates to the use of dopamine receptor agonists for preparing a pharmaceutical composition for the reduction of excessive food intake.
    Type: Application
    Filed: June 26, 2006
    Publication date: October 5, 2006
    Applicant: Boehringer Ingelheim Pharma GmbH & Co. KG
    Inventors: Michael PIEPER, Joachim Mierau