Patents by Inventor Nicholas Paschalides

Nicholas Paschalides has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Processes for making a solid-state form of relugolix
    Patent number: 11655256
    Abstract: The present invention is directed to processes for making an anhydrous form of relugolix, designated herein as Form T of anhydrous relugolix. The processes of making Form T of anhydrous relugolix are from the following: (i) Form A of the DMF solvate of relugolix; (ii) Form B of anhydrous relugolix; or (iii) amorphous relugolix.
    Type: Grant
    Filed: November 6, 2021
    Date of Patent: May 23, 2023
    Assignee: Macfarlan Smith Limited
    Inventor: Nicholas Paschalides
  • SOLID SALT FORM OF ALPHA-6-MPEG6-O-HYDROXYCODONE AS OPIOID AGONISTS AND USES THEREOF
    Publication number: 20170226119
    Abstract: Solid forms of certain opioid agonists are provided herein. Methods of preparing the solid forms, methods of using the solid forms, and pharmaceutical compositions comprising the solid forms are also provided herein.
    Type: Application
    Filed: April 26, 2017
    Publication date: August 10, 2017
    Inventors: Patricia Andres, Yogesh Datar, Ramakrishna Gadiraju, Bruce Andrew Kowalczyk, Gabriel Christian Kuklis, Mahmoud Mirmehrabi, Nicholas Paschalides
  • Solid salt form of ?-6-mPEG-O-hydroxycodone as opioid agonists and uses thereof
    Patent number: 9682988
    Abstract: Solid forms of certain opioid agonists are provided herein. Methods of preparing the solid forms, methods of using the solid forms, and pharmaceutical compositions comprising the solid forms are also provided herein.
    Type: Grant
    Filed: October 29, 2013
    Date of Patent: June 20, 2017
    Assignee: Nektar Therapeutics
    Inventors: Patricia Andres, Yogesh Datar, Ramakrishna Gadiraju, Bruce Andrew Kowalczyk, Gabriel Christian Kuklis, Mahmoud Mirmehrabi, Nicholas Paschalides
  • Solid Salt Form of Alpha-6-MPEG6-O-Hydroxycodone as Opioid Agonists and Uses Thereof
    Publication number: 20150284402
    Abstract: Solid forms of certain opioid agonists are provided herein. Methods of preparing the solid forms, methods of using the solid forms, and pharmaceutical compositions comprising the solid forms are also provided herein.
    Type: Application
    Filed: October 29, 2013
    Publication date: October 8, 2015
    Applicant: Nektar Therapeutics
    Inventors: Patricia Andres, Yogesh Datar, Ramakrishna Gadiraju, Bruce Andrew Kowalczyk, Gabriel Christian Kuklis, Mahmoud Mirmehrabi, Nicholas Paschalides