Patent number: 6696607
Abstract: Use of phenethylacrylamides of the formula I:
in which the substituents have the following meanings:
X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and —O—C(Ra,Rb)—C≡C—R6;
Ra,Rb and Rc have the meanings given in the description;
m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1;
Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl;
R1,R2 independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3;
R3,R4,R5,R6 independently of one another are hydrogen, halogen, alkyl, alkoxy, or
R3 and R4 together form a cyclopropyl ring, it being possible for the C—R5— and C—R6 bonds can be in the E- or Z-position relative to each other;
for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.
Type:
Grant
Filed:
December 4, 2002
Date of Patent:
February 24, 2004
Assignee:
BASF Aktiengesellschaft
Inventors:
Wassilios Grammenos, Hubert Sauter, Oliver Cullmann, Markus Gewehr, Bernd Müller, Jordi Tormo i Blasco, Norbert Götz, Thorsten Volk, Gisela Lorenz, Eberhard Ammermann, Reinhard Stierl, Siegfried Strathmann
Publication number: 20030191190
Abstract: The invention relates to the use of phenethyl acrylamides of formula I for controlling phytopathogenic fungi, wherein the substituents of said phenethyl acrylamides have the following significations: X signifies halogen, alkyl, halogenalkyl, alkoxy halogenalkoxy and —O—C(Ra, Rb)—C≡C—R6; Ra, Rb and Rc have the signification given in the description; m, n independently signify 1 to 4, the radicals X or Y being potentially different if m or n is higher than 1; Y signifies halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl; R1, R2 independently signify hydrogen, halogen, alkyl, alkoxy, halogenalkoxy and CF3; R3, R4, R5, and R6 independently signify hydrogen, alkyl and alkoxy, or R3 and R4 together form a cyclopropyl ring, whereby the C—R5 and C—R6 bonds can be in position E or Z in relation to each other. The invention also relates to novel phenethyl acrylamides, a method for the productio thereof, and agents containing the same.
Type:
Application
Filed:
December 4, 2002
Publication date:
October 9, 2003
Inventors:
Wassilios Grammenos, Hubert Sauter, Oliver Cullmann, Markus Gewehr, Bernd Muller, Jordi Tormo i Blasco, Norbert Gotz, Thorsten Volk, Gisela Lorenz, Eberhard Ammermann, Reinhard Stierl, Siegfried Strathman
Patent number: 6593315
Abstract: Salicylic acid derivatives of the formula I,
where the index and the substituents have the following meanings:
X is halogen, NO2, cyano, alkyl or alkoxy;
m is 0, 1, 2 or 3, it being possible for the substituents X to be different from each other if n is greater than 1;
A is OH, alkoxy, NH2, NHCH3 or N(CH3)2;
R1 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, comprising one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted;
R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio,
processes for the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.
Type:
Grant
Filed:
July 2, 2001
Date of Patent:
July 15, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Andreas Gypser, Thomas Grote, Joachim Rheinheimer, Ingo Rose, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Jordi Tormo i Blasco, Bernd Müller, Hubert Sauter, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl
Patent number: 6562833
Abstract: 2-(N-phenylamino)pyrimidines of the formula I,
where:
R1, R3 independently of one another are cyano, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or are C3-C8-cycloalkyl or a group C(═NORx)Ry
R2 is halogen, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or
R1 and R2 together with the two linking carbon atoms form a fused-on partially unsaturated 4- to 8-membered ring which may be up to trisubstituted by identical or different substituents selected from the group consisting of C1-C4-alkyl, halogen and C1-C4-alkoxy-carbonyl, which may contain a carbonyl group and/or, in addition to the multiple bond of the pyrimidine ring, a double bond and/or which may be interrupted by O, S or N—(C1-C4-alkyl);
the substituents R4 to R8, Rx, Ry, Ra and Rb are
Type:
Grant
Filed:
December 5, 2000
Date of Patent:
May 13, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Bernd Müller, Hubert Sauter, Herbert Bayer, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Andreas Gypser, Arne Ptock, Norbert Götz, Thomas Grote, Michael Rack, Eberhard Ammermann, Gisela Lorenz, Siegfried Strathmann, John-Bryan Speakman
Patent number: 6537989
Abstract: The present invention relates to azadioxacycloalkenes of the formula I
in which the substituents R1 to R5 and X, the index n and the bridge member W have the following meanings:
R1 is C1-C4-alkyl, halogen, C1-C4-haloalkyl, C3-C6-cycloalkyl;
R2 is C1-C4-alkyl, C1-C4-haloalkyl, C3-C4-alkenyl, C3-C4-haloalkenyl, C3-C4-alkynyl or C3-C4-haloalkynyl;
R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl or unsubstituted or substituted phenyl;
R4 is ═CRaRb, —CRd═CRaRb or ═N—ORc, where Ra, Rb, Rc and Rd are each as defined in claim 1;
R5 is nitro, cyano, halogen, C1-C6-alkyl or, in the case that n is 2, additionally a bridge which is attached to two adjacent ring atoms;
n is 0, 1, 2, 3 or 4, where the substituents R1 may be different if n is greater than 1;
X is C1-C4-alkoxy-N═, C1-C4-alkoxy-CH═ or R6—CH═, where R6 is as defined in claim 1
W is unsubstituted or substituted C1-C3-alkylene.
Type:
Grant
Filed:
April 2, 2001
Date of Patent:
March 25, 2003
Assignee:
BASF Aktiengesellschaft
Inventors:
Markus Gewehr, Wassilios Grammenos, Hubert Sauter, Herbert Bayer, Andreas Gypser, Bernd Müller, Arne Ptock, Oliver Cullmann, Thomas Grote, Eberhard Ammermann, Gisela Lorenz, Siegfried Strathmann, Volker Harries
Patent number: 6455515
Abstract: Salicylohydrazide derivatives of the formula I
in which the index and the substituents have the following meanings:
X is halogen, NO2, cyano, alkyl or alkoxy;
m is 0, 1, 2 or 3, it being possible for the substituents X to differ from each other if n is greater than 1;
R1 is NO2, NH2 or NH—CO—A;
A is hydrogen, alkyl, alkoxy, NH2, NHCH3 or N(CH3)2;
R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio;
it being possible for the hydrocarbon radicals to be unsubstituted or substituted,
R3 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl containing one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted;
the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.
Type:
Grant
Filed:
June 14, 2001
Date of Patent:
September 24, 2002
Assignee:
BASF Aktiengesellschaft
Inventors:
Andreas Gypser, Thomas Grote, Joachim Rheinheimer, Ingo Rose, Peter Schäfer, Oliver Cullmann, Markus Gewehr, Wassilios Grammenos, Jordi Tormo i Blasco, Bernd Müller, Hubert Sauter, Eberhard Ammermann, Siegfried Strathmann, Gisela Lorenz, Reinhard Stierl