Patents by Inventor Patrick G. Guerret

Patrick G. Guerret has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4808582
    Abstract: Compounds of formula: ##STR1## wherein: Ar is an aromatic group; R and R.sub.1 are H or CH.sub.3 ; A represents a nitrogenized heterocyclic radical; B is OH or forms with the adjacent CO group, either an amido group, or a carbonyloxy group; R.sub.2 and R.sub.3 are H or alkyl; m=0 or 1; and n=0, 1, 2 or 3.These compounds are useful as drugs having stimulating, protecting and/or correcting activities of the cerebral functions.
    Type: Grant
    Filed: March 19, 1987
    Date of Patent: February 28, 1989
    Assignee: Delalande S.A.
    Inventors: Alain Y. Platel, Guy R. Bourgery, Patrick G. Guerret
  • Patent number: 4598084
    Abstract: N-arylated oxazolidine-2-one derivatives corresponding to the formula: ##STR1## and of S(+) configuration, A representing in this case the hydroxyl radical or of R (+) configuration, A designating then the N-methylamino group, as well as the acid addition salts thereof.Application in therapeutics more particularly as monoamine oxidase inhibitors.
    Type: Grant
    Filed: June 3, 1983
    Date of Patent: July 1, 1986
    Assignee: Delalande S.A.
    Inventors: Margherita Strolin-Benedetti, Patrick G. Guerret, Michel Langlois, Philippe L. Dostert
  • Patent number: 4526786
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 16, 1982
    Date of Patent: July 2, 1985
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Phillippe L. Dostert
  • Patent number: 4517197
    Abstract: A compound of the formula ##STR1## where R is selected from the group consisting of CH.sub.3 --CO--(CH.sub.2).sub.2 --O--, ##STR2## The compounds are useful in treating depression.
    Type: Grant
    Filed: July 29, 1983
    Date of Patent: May 14, 1985
    Assignee: Delalande S.A.
    Inventors: Jean-Francois R. Ancher, Guy R. Bourgery, Philippe L. Dostert, Colette A. Douzon, Patrick G. Guerret, Alain P. Lacour, Michel Langlois
  • Patent number: 4470993
    Abstract: Method of treating the central nervous system troubles such as the Parkinson's disease and the senescence troubles, generally treated by the B type monoamine oxidase inhibitors, which comprises administering internally to a human being requiring such treatment a therapeutically effective amount of N-aryl 5-aminomethyl oxazolidine-2-one derivatives.
    Type: Grant
    Filed: March 3, 1983
    Date of Patent: September 11, 1984
    Assignee: Delalande S.A.
    Inventors: Jean-Francois R. Ancher, Guy R. Bourgery, Philippe L. Dostert, Colette A. Douzon, Patrick G. Guerret, Alain P. Lacour, Michel Langlois, Margherita Strolin-Benedetti
  • Patent number: 4463004
    Abstract: Compounds having analgesic activity are disclosed which have the general formula: ##STR1## wherein R.sub.1 is hydrogen, alkyl having 1 to 4 carbon atoms, cyclohexyl or benzyl; R is selected from the group consisting of alkyl having at least 4 carbon atoms; cyclohexyl; unsubstituted phenyl or phenyl substituted with one or more halogen atoms, methyl, methoxy, hydroxy, cyano, nitro, trifluoromethyl, carboxyl, ethoxycarbonyl, acetamido, methylsulfonyl, phenoxy, benzoyl, phenyl, .alpha.-hydroxybenzyl, cyclohexyl or carbamoyl; thienyl; pyridyl; naphthyl; naphthyl substituted with methoxy; adamantyl; and benzyl; and n is 1, 2 or 3, with the provisos that (1) when R is carboxyphenyl, benzoylphenyl, or (.alpha.-hydroxybenzyl) phenyl, n is not 3, and (2) when R is (.alpha.-hydroxy benzyl) phenyl, R.sub.1 is not benzyl, and acid addition salts thereof.
    Type: Grant
    Filed: April 16, 1982
    Date of Patent: July 31, 1984
    Assignee: Delalande S.A.
    Inventors: Patrick G. Guerret, Bernard P. Bucher, Philippe L. Dostert, Gisele C. Mocquet, Alain L. Nedelec
  • Patent number: 4459296
    Abstract: There are disclosed piperidinio, piperazino and homopiperazino derivatives wherein there is N-substitution by a heterocyclic compound taken from the group benzimidazole, indole, purine or benzotriazole and to the organic or mineral acid addition salts of these derivatives. The process for preparation of such compounds and their use is also disclosed.
    Type: Grant
    Filed: April 20, 1982
    Date of Patent: July 10, 1984
    Assignee: Delalande S.A.
    Inventors: Jean-Francois R. Ancher, Patrick G. Guerret, Michel Langlois, Jacky A. Tisne-Versailles
  • Patent number: 4435415
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 16, 1982
    Date of Patent: March 6, 1984
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Philippe L. Dostert
  • Patent number: 4413001
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 16, 1982
    Date of Patent: November 1, 1983
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Philippe L. Dostert
  • Patent number: 4348393
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: June 4, 1979
    Date of Patent: September 7, 1982
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Phillippe L. Dostert
  • Patent number: 4287351
    Abstract: N-aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones are disclosed. These compounds possess antidepressant activity.
    Type: Grant
    Filed: February 6, 1980
    Date of Patent: September 1, 1981
    Assignee: Delalande S.A.
    Inventors: Guy R. Bourgery, Colette A. Douzon, Jean-Francois R. Ancher, Alain P. Lacour, Patrick G. Guerret, Michel Langlois, Phillippe L. Dostert
  • Patent number: 4016154
    Abstract: A compound having the formula ##STR1## and its pharmacologically acceptable acid addition salts. The compound is prepared by condensing N-(3,4,5-trimethoxy cinnamoyl) piperazine with N-(2-pyrrolidinone) chloroacetamide. The compounds possess peripheral and coronary vasodilatatory properties and hypotensive and antihypertensive properties.
    Type: Grant
    Filed: July 15, 1975
    Date of Patent: April 5, 1977
    Assignee: Delalande S.A.
    Inventors: Michel J. Turin, Guy M. Raynaud, Bernard M. Pourrias, Patrick G. Guerret