Patents by Inventor Patrick Saur

Patrick Saur has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 5322846
    Abstract: The present invention relates to novel 4-methylthiazole derivatives, to tr methods of preparation and to the pharmaceutical compositions in which they are present.According to the invention, these derivatives have the general formula ##STR1## in which n is equal to 0 or 1 and R.sub.1 and R.sub.2, which are identical or different, are selected from a hydrogen atom, a halogen, a hydroxyl group, a trifluoromethyl group, an alkyl group having from 1 to 4 carbon atoms and an alkoxy group having from 1 to 5 carbon atoms and are useful in the treatment of cardiovascular diseases associated with hyperactivity of the sympathetic nervous system.
    Type: Grant
    Filed: October 19, 1992
    Date of Patent: June 21, 1994
    Assignee: Institut de Recherches Chimiques et Biologiques Appliquees (I.R.C.E.B.A.)
    Inventors: Fabienne Jobard-Rouppert, Patrick Houziaux, Jean-Pierre Riffaud, Jean-Yves Lacolle, Patrick Saur, Bernard Danree
  • Patent number: 5212161
    Abstract: The present invention relates to novel derivatives of 2'-deoxyuridine substituted in the 5-, 3'- or 5'-position by .alpha.-aminoacyl groups, to a process for their preparation and the drugs in which they are present.These derivatives have the following general formula: ##STR1## in which R is selected from an alkyl or alkenyl radical having from 1 to 4 carbon atoms, an aryl radical or a halogen, it being possible for said alkyl, alkenyl and aryl radicals to contain at least one halogen substituent, and a radical of the formula --NH--R.sub.1, in which R.sub.1 is an amino acid residue or a peptide residue containing from 2 to 6 amino acids; andR' and R" are selected from a hydroxyl radical and a radical of the formula --NH--R.sub.1, in which R.sub.1 is as defined above,with the proviso that R' and R" are not simultaneously --NH--R.sub.1 and that, when R is --NH--R.sub.1, R' and R" are simultaneously a hydroxyl group.Application: treatment of cancers and viral infections.
    Type: Grant
    Filed: August 17, 1990
    Date of Patent: May 18, 1993
    Assignee: Institut de Recherches Chimiques et Biologiques Appliquees (I.R.C.E.B.A.)
    Inventors: Jean-Luc Moriniere, Michelle Faulques, Claude Rousseau, Bernard Danree, Claude Marquer, Patrick Saur, Jean Lemoine, Jean-Yves Lacolle