Patents by Inventor Paul Martin Gore

Paul Martin Gore has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20040058923
    Abstract: Compounds of formula (I) wherein: R1 represents C1-16 alkyl, C2-6alkenyl, C2-6alkynyl, C2-6alkynyl-Y1—, aryl-Y1—, heteroaryl-Y1—, aryl-(O)t-aryl-Y1—, aryl-(O)t-heteroaryl-Y1—, heteroaryl-(O)t-aryl-Y1—, heteroaryl-(O)t-heteroaryl-Y1—, C2-6 alkenyl-Y1—, aryl-O—Y1—, heteroaryl-O—Y1—, C1-16 alkyl-SO2—Y1—,M—Y1—,J2-Y1—, —CN or C3-8 cycloalkyl-Y1— or C3-8 cycloalkenyl-Y1—, which cycloalkyl or cycloalkenyl may be optionally substituted by one or more hydroxyl or C1-16 Alkyl groups; R2 represents hydrogen or C1-16 alkyl; X represents ethylene or a group of formula CReRf wherein Re and Rf independently represent hydrogen or C1-14 alkyl or Re and Rf may together with the carbon atom to which they are attached form a C3-8 cycloalkyl group; R3 and R4 independently represent hydrogen or C1-14 alkyl; Z represents a bond, CO, SO2, CR9R6(CH2)n, (CH2)nCR9R6, CHR6(CH2)nO, CHR6(CH2)nS, CHR6(CH2)nOCO, CHR6(CH2)n
    Type: Application
    Filed: August 15, 2003
    Publication date: March 25, 2004
    Inventors: Rachael Anne Ancliff, Caroline Mary Cook, Colin David Eldred, Paul Martin Gore, Lee Andrew Harrison, Simon Teanby Hodgson, Duncan Bruce Judd, Suzanne Elaine Keeling, Xiao Qing Lewell, Graeme Michael Robertson, Stephen Swanson
  • Publication number: 20040044035
    Abstract: The present invention relates to a pharmaceutical formation which comprises an aqueous suspension of particulate (2S)-3-[4-({[4-aminocarbonyl)-1-piperidinyl]carbonyl}oxy)phenyl]-2-[((2S)-4-methyl-2-{[2-(2-methylphenoxy)acetyl]amino}pentanoyl)amino]propanoic acid or a salt or solvate thereof. Methods and uses of the formulation in the treatment of allergic rhinitis are also described, as are containers containing said formulation.
    Type: Application
    Filed: August 21, 2003
    Publication date: March 4, 2004
    Inventors: Duncan Robert Armour, David Brown, Miles Stuart Congreve, Paul Martin Gore, Darren Victor, Steven Green, Stuart Holman, Torquil Iain, Maclean Jack, Steven Philip Keeling, Andrew McMurtrie Mason, Karen Morriss, Nigel Grahame Ramsden, Marian Thomas, Peter Ward
  • Publication number: 20040037784
    Abstract: The present invention relates to a dry powder pharmaceutical formulation suitable for inhalation therapy comprising particulate (2S)-3-[4-({[4-(aminocarbonyl)-1-piperidinyl]carbonyl}oxy)phenyl]-2-[((2S)-4-methyl-2-{[2-(2-methylphenoxy)acetyl]amino}pentanoyl)amino] propanoic acid or a salt or solvate thereof and one or more suitable excipients. Methods and uses of the formulation in the treatment of inflammatory diseases are also described, as are medicament packs and inhalation devices containing said formulation.
    Type: Application
    Filed: August 21, 2003
    Publication date: February 26, 2004
    Inventors: Duncan Robert Armour, David Brown, Miles Stuart Congreve, Paul Martin Gore, Darren Victor Steven Green, Stuart Holman, Torquil Iain Maclean Jack, Steven Philip Keeling, Andrew McMurtrie Mason, Karen Morris, Nigel Grahame Ramsden, Marian Thomas, Peter Ward
  • Publication number: 20040034062
    Abstract: The present invention relates to a pharmaceutical formulation which comprises: an aqueous solution of (2S)-3-[4-({[4-(aminocarbonyl)-1-piperidinyl]carbonyl}oxy)phenyl]-2-[((2S)-4-methyl-2-{[2-(2-methylphenoxy)acetyl]amino}pentanoyl)amino] propanoic acid or a salt or solvate thereof. Methods and uses of the formulation in the treatment of allergic rhinitis are also described, as are containers containing said formulation.
    Type: Application
    Filed: August 21, 2003
    Publication date: February 19, 2004
    Inventors: Duncan Robert Armour, David Brown, Miles Stuart Congreve, Paul Martin Gore, Darren Victor Green, Stuart Holman, Andrew McMurtrie Mason, Karen Morris, Nigel Grahame Ramsden, Marian Thomas, Peter Ward