Patents by Inventor Raymond Westheim

Raymond Westheim has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Crystalline forms and processes of lenvatinib besylate
    Patent number: 12102630
    Abstract: The present invention relates to lenvatinib besylate, its crystalline forms and processes for making them. Furthermore, to a pharmaceutical composition comprising a therapeutically effective dose of lenvatinib besylate.
    Type: Grant
    Filed: October 1, 2019
    Date of Patent: October 1, 2024
    Assignee: Synthon B.V.
    Inventors: Luis Nogueiras Nieto, Lisardo Alvarez Fernandez, Raymond Westheim, Katerina Jelinkova
  • CRYSTALLINE FORM OF OZANIMOD HYDROCHLORIDE
    Publication number: 20230183194
    Abstract: The presented invention relates to crystalline form, Form A of Ozanimod hydrochloride, processes for preparation thereof and pharmaceutical compositions comprising the Ozanimod hydrochloride Form A.
    Type: Application
    Filed: March 17, 2021
    Publication date: June 15, 2023
    Inventor: Raymond WESTHEIM
  • CRYSTALLINE FORMS OF BEMPEDOIC ACID
    Publication number: 20220348531
    Abstract: The presented invention relates to crystalline Form A and Form B of Bempedoic acid, a process for preparation thereof and a composition comprising the Form A or Form B.
    Type: Application
    Filed: October 2, 2020
    Publication date: November 3, 2022
    Inventors: Michal HEGEDUS, Raymond WESTHEIM
  • CRYSTALLINE FORMS AND PROCESSES OF LENVATINIB BESYLATE
    Publication number: 20220062263
    Abstract: The present invention relates to lenvatinib besylate, its crystalline forms and processes for making them. Furthermore, to a pharmaceutical composition comprising a therapeutically effective dose of lenvatinib besylate.
    Type: Application
    Filed: October 1, 2019
    Publication date: March 3, 2022
    Inventors: Luis NOGUEIRAS NIETO, Lisardo ALVAREZ FERNANDEZ, Raymond WESTHEIM, Katerina JELINKOVA
  • Crystalline aripiprazole solvates
    Patent number: 7902198
    Abstract: Alcoholates of aripiprazole are useful as pharmaceuticals and/or as intermediates in making aripiprazole Form A or Form B.
    Type: Grant
    Filed: November 18, 2005
    Date of Patent: March 8, 2011
    Assignee: Synthon BV
    Inventors: Gerrit Jan Ettema, Raymond Westheim, Faysal Kalmoua
  • Process of making crystalline aripiprazole
    Patent number: 7642353
    Abstract: Crystalline aripiprazole Form B can be formed by crystallizing from a solvent selected from 1-propanol, 2-propanol, 1-butanol, ethyl acetate, acetonitrile or a combination thereof.
    Type: Grant
    Filed: November 18, 2005
    Date of Patent: January 5, 2010
    Assignee: Synthon BV
    Inventors: Gerrit Jan Ettema, Raymond Westheim, Faysal Kalmoua
  • CRYSTALLINE ERLOTINIB
    Publication number: 20080058355
    Abstract: Crystalline Forms of erlotinib are made. The crystalline materials are useful as pharmaceutical active agents in treating various cancers as well as in forming erlotinib salts.
    Type: Application
    Filed: July 27, 2007
    Publication date: March 6, 2008
    Inventor: Raymond Westheim
  • Process of making crystalline Type II aripiprazole
    Publication number: 20060258673
    Abstract: Crystalline aripiprazole Type II can be formed without solid state heat treatment. Instead a liquid is used such as in crystallizing from a solvent, especially 2-propanol, dimethyl sulfoxide, or a combination thereof with ethyl acetate, or in a solvent mediated solid-solid transformation, typically in ethyl acetate.
    Type: Application
    Filed: March 17, 2006
    Publication date: November 16, 2006
    Inventors: Gerrit Ettema, Raymond Westheim, Faysal Kalmoua
  • Pharmaceutical tablets of crystalline Type II aripiprazole
    Publication number: 20060257471
    Abstract: Crystalline aripiprazole Type II can be formulated into pharmaceutical tablets having reduced dissolution profile variability upon storage.
    Type: Application
    Filed: March 17, 2006
    Publication date: November 16, 2006
    Inventors: Gerrit Ettema, Raymond Westheim, Faysal Kalmoua, Korinde Jansen, Farid Dorkoosh
  • Process of making crystalline aripiprazole
    Publication number: 20060142579
    Abstract: Crystalline aripiprazole Form B can be formed by crystallizing from a solvent selected from 1-propanol, 2-propanol, 1-butanol, ethyl acetate, acetonitrile or a combination thereof.
    Type: Application
    Filed: November 18, 2005
    Publication date: June 29, 2006
    Inventors: Gerrit Ettema, Raymond Westheim, Faysal Kalmoua
  • Crystalline aripiprazole solvates
    Publication number: 20060142299
    Abstract: Alcoholates of aripiprazole are useful as pharmaceuticals and/or as intermediates in making aripiprazole Form A or Form B.
    Type: Application
    Filed: November 18, 2005
    Publication date: June 29, 2006
    Inventors: Gerrit Ettema, Raymond Westheim, Faysal Kalmoua