Publication number: 20050009704
Abstract: The invention relates to novel substituted aryl ketones of the general formula (I) in which n represents the number 0, 1 or 2, A represents alkanediyl (alkylene), R1 represents one of the groupings below where m, R5, R6, R7, R8, R9, R10, R11, R12 and R13 each have one of the meanings given in the description, R2 represents hydrogen, nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or dialkylaminosulphenyl, R3 represents nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkyl-sulphinyl, alkylsulphonyl, alkylamino, dialkylamino or dialkylaminosulphonyl, and R4 represents an optionally substituted 4- to 12-membered, saturated or unsaturated, monocyclic or bicyclic heterocyclic grouping, and to processes for their preparation, to intermediates and to the use of these compound
Type:
Application
Filed:
July 26, 2004
Publication date:
January 13, 2005
Inventors:
Otto Schallner, Stefan Lehr, Hans-Georg Schwarz, Klaus-Helmut Muller, Dorothee Hoischen, Mark Drewes, Peter Dahmen, Dieter Feucht, Rolf Pontzen, Akihiko Yanagi, Shinichi Narabu, Toshio Goto
Patent number: 6838415
Abstract: The invention relates to novel substituted benzoylisoxazoles of the general formula (I), in which n represents the number 0, 1, 2 or 3, A represents a single bond or represents alkanediyl (alkylene), R1 represents hydrogen or represents in each case optionally substituted alkyl, alkenyl or cycloalkyl, R2 represents hydrogen, cyano, carbamoyl, halogen, or represents in each case optionally substituted alkyl, alkylcarbonyl, alkoxy, alkoxycarbonyl or alkylthio, alkylsulphinyl or alkylsulphonyl, R3 represents hydrogen, nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or dialkylaminosulphonyl, R4 represents nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino or dialkylaminosulphonyl, and Z represents an optionally substituted 4-
Type:
Grant
Filed:
April 20, 2000
Date of Patent:
January 4, 2005
Assignee:
Bayer Aktiengesellschaft
Inventors:
Klaus-Helmut Müller, Stefan Lehr, Otto Schallner, Hans-Georg Schwarz, Heinz-Jürgen Wroblowsky, Mark Wilhelm Drewes, Dieter Feucht, Rolf Pontzen, Ingo Wetcholowsky
Patent number: 6815398
Abstract: Novel substituted phenyluracils of the general formula (I)
in which
n represents 0, 1 or 2,
R1 represents hydrogen, amino or optionally substituted alkyl,
R2 represents carboxyl, cyano, carbamoyl, thiocarbamoyl or in each case optionally substituted alkyl or alkoxycarbonyl,
X represents hydroxyl, mercapto, amino, nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkylcarbonyloxy, alkoxycarbonyloxy, alkylaminocarbonyloxy, dialkylaminocarbonyloxy, phenylcarbonyloxy, alkylcarbonylamino, alkoxycarbonylamino, alkylsulphonylamino, alkenyl, alkenyloxy, alkenyloxycarbonyl, alkinyl, alkinyloxy or alkinyloxycarbonyl, where in the case that n is greater than 1, X in the individual possible compounds may also have meanings other than those given.
Type:
Grant
Filed:
May 7, 2002
Date of Patent:
November 9, 2004
Assignee:
Bayer Aktiengesellschaft
Inventors:
Roland Andree, Hans-Georg Schwarz, Mark Wilhelm Drewes, Dieter Feucht, Rolf Pontzen, Ingo Wetcholowsky
