Abstract: The present invention provides compounds which show high effectiveness against positive symptoms, negative symptoms and cognitive dysfunction in schizophrenia and reduce conventional side-effect risks as well as have remarkable effects for central neurological diseases associated with cognitive dysfunction other than schizophrenia. N-Acyl cyclic amine derivatives of formula (1): wherein Ar1 and Ar2 are aryl or heteroaryl; V is nitrogen, or CR3; W1 is a single bond, —C(O)—, etc.; W2 is C1-alkylene; W3 is a single bond, methylene, —NH—, —CR4?CR5—, etc.; Ring Q is a group of formula (a) in which n is 0 or 1; m is 0 to 2; k is 1 to 3; Z is a single bond, methylene, oxygen, etc.; R1a, R1b and R1c are each, same or different, hydrogen, hydroxyl, halogen, cyano, C1-6 alkyl, etc.; or pharmaceutically acceptable salts thereof are provided.

Abstract: The present invention provides compounds which show high effectiveness against positive symptoms, negative symptoms and cognitive dysfunction in schizophrenia and reduce conventional side-effect risks as well as have remarkable effects for central neurological diseases associated with cognitive dysfunction other than schizophrenia. N-Acyl cyclic amine derivatives of formula (1): wherein Ar1 and Ar2 are aryl or heteroaryl; V is nitrogen, or CR3; W1 is a single bond, —C(O)—, etc.; W2 is C1-alkylene; W3 is a single bond, methylene, —NH—, —CR4?CR5—, etc.; Ring Q is a group of formula (a) in which n is 0 or 1; m is 0 to 2; k is 1 to 3; Z is a single bond, methylene, oxygen, etc.; R1a, R1b and R1c are each, same or different, hydrogen, hydroxyl, halogen, cyano, C1-6 alkyl, etc.; or pharmaceutically acceptable salts thereof are provided.

Abstract: The present invention relates to a compound of the formula (1): wherein R1 is group of the formula (2): (wherein X is nitrogen atom or C(R5), Y is nitrogen atom or C(R6), R5 and R6 are each independently hydrogen atom, etc.) etc., m is 1 to 6, L1 is single bond, etc., R2 is hydrogen atom, substituted or unsubstituted alkyl group, etc., R3 is hydrogen atom, etc., L2 is single bond, etc., R4 is hydrogen atom, substituted or unsubstituted aryl group, etc., or pharmaceutically acceptable salt thereof, being useful for preventing or treating Alzheimer's disease.

Abstract: The present invention relates to a compound of the formula (1): wherein R1 is group of the formula (2): (wherein X is nitrogen atom or C(R5), Y is nitrogen atom or C(R6), R5 and R6 are each independently hydrogen atom, etc.) etc., m is 1 to 6, L1 is single bond, etc., R2 is hydrogen atom, substituted or unsubstituted alkyl group, etc., R3 is hydrogen atom, etc., L2 is single bond, etc., R4 is hydrogen atom, substituted or unsubstituted aryl group, etc., or pharmaceutically acceptable salt thereof, being useful for preventing or treating Alzheimer's disease.

Abstract: In a relay device or the like in which a speed changes from a high speed to a low speed, a packet residence (packet transfer wait) occurs when a packet string in which packet intervals are shortened arrives. When a packet discard occurs before passing through the relay device or the like, a packet interval having been lengthened by the packet discard is shortened by the relay device or the like for transferring packets. When a packet discard occurs after passing through the relay device or the like, a packet interval having been lengthened by the packet discard remains unshortened for transferring packets. Therefore, by observing at terminals the packet discard and the packet interval on the occasion of the packet discard, whether the packet discard has occurred in the high speed section or the low speed section is specified.

Abstract: A computer-readable recording medium recording a program capable of accurately analyzing the cause of a performance fault at the very end point of a client system, server system, etc. Outgoing and incoming packets are captured during execution of a communication application to measure a round trip time, and a communication window size of the transmitting source is estimated based on the captured incoming packets. A throughput estimate is calculated from the round trip time and the communication window size, and the estimated value and actual measured value of the throughput are displayed on, for example, a display, together with various other communication parameters including the communication window size and the round trip time, whereby the cause of a performance fault can be accurately located by quantitative analysis.

Abstract: A compound of the formula I where R represents unsubstituted or substituted, alkyl, cycloalkyl, alkenyl, alkynyl, or aryl, and X represents where R1 and R2 are each H or alkyl, is disclosed. Compounds of formula I are particularly useful as an attractant for cockroaches, namely, Blattella germanica. Synthesis of the compounds, methods of controlling cockroach populations, and of disrupting cockroach mating are also disclosed.

Abstract: A computer-readable recording medium recording a program capable of accurately analyzing the cause of a performance fault at the very end point of a client system, server system, etc. Outgoing and incoming packets are captured during execution of a communication application to measure a round trip time, and a communication window size of the transmitting source is estimated based on the captured incoming packets. A throughput estimate is calculated from the round trip time and the communication window size, and the estimated value and actual measured value of the throughput are displayed on, for example, a display, together with various other communication parameters including the communication window size and the round trip time, whereby the cause of a performance fault can be accurately located by quantitative analysis.

Abstract: In a relay device or the like in which a speed changes from a high speed to a low speed, a packet residence (packet transfer wait) occurs when a packet string in which packet intervals are shortened arrives. When a packet discard occurs before passing through the relay device or the like, a packet interval having been lengthened by the packet discard is shortened by the relay device or the like for transferring packets. When a packet discard occurs after passing through the relay device or the like, a packet interval having been lengthened by the packet discard remains unshortened for transferring packets. Therefore, by observing at terminals the packet discard and the packet interval on the occasion of the packet discard, whether the packet discard has occurred in the high speed section or the low speed section is specified.

Abstract: A novel dipeptide compound inhibiting the enzymatic activity of HIV protease and an anti-AIDS medicine comprising this dipeptide compound as an effective component represented by formula (I) wherein R1, R2, and R3 independently represent C1-4 alkyl, alkoxyl, hydrogen etc . . . (provided that not all of the R1, R2, and R3 are hydrogen), R2 and R3 may form a ring together, R4 represents C1-4 alkyl or hydrogen; X is a methylene group or a sulfur atom; Y represents e.g., a five or six member monocycle or aryloxyalkyl having up to 12 carbon atoms (provided that the aromatic ring may be substituted by alkyl etc . . . ); and Z represents a C1-6 aliphatic hydrocarbon or an aromatic hydrocarbon having up to 12 carbon atoms (provided that this aromatic ring may be substituted by alkyl etc . . . , or at least one carbon atom in the aromatic hydrocarbon may be replaced by a hereto atom).

Abstract: An end equipment (including a terminal equipment and a router) executes a destination address resolution of a data packet. In a network layer, when a packet transmitter detects that a direct route of an input packet is not registered in a routing table a path manager transmits an inquiry packet, demands a preparation of a point-to-point logical interface of the direct route based on a data link layer address of the destination included in the received response packet, and registers the prepared logical interface in the routing table.

Abstract: A novel dipeptide compound inhibiting the enzymatic activity of HIV protease, an anti-AIDS medicine comprising this dipeptide compound as an effective component.

Abstract: A novel tripeptide compound represented by the following general formula (I) exhibiting superior HIV protease inhibition activity, and an anti-AIDS medicine comprising this compound as an effective component and a pharmaceutically acceptable salt thereof. (R)-N-(2-methylbenzyl)-3-{(2S,3S)-3-[N-(2-chromonecarbonyl)-L-asparaginyl]amino-2-hydroxy-4-phenylbutanoyl}-5,5-dimethyl-1,3-thiazolidine-4-carboxamide can be given as a typical example of this compound.

Abstract: A signal from an input terminal (1) is supplied to a video signal processing circuit (2) which derives a carrier chrominance signal. The carrier chrominance signal is supplied through a low-pass filter (3) to an A/D converter circuit (4). A signal converted by the A/D converter circuit (4) is supplied to a bandpass filter (5) which limits the band of the chrominance signal. A signal from the bandpass filter (5) is supplied to a decoder circuit (6) which alternately derives color difference signals (R-Y) and (B-Y). The signal from the decoder circuit (6) is supplied to a decimation filter (7) which effects a decimation. The signal thus decimated is supplied to a multiplexer (8) and thereby generated as 2-bit series data. A signal from the multiplexer (8) is supplied to a CNR (chroma noise reducer) circuit (9). Thus, the number of bits can be reduced without reducing the number of lines of a chroma signal and data gradation.

Abstract: An adaptively controlled noise reduction device in which an input video signal is supplied to first, second, and third adders and in which an output of the first adder is supplied to the second adder via a memory responsive to a controller whereby the memory provides a controllable delay. An output of the second adder is supplied via a first coefficient multiplication unit having variable attenuation that is controlled by the controller to the first adder as well as via a second coefficient multiplication unit having variable attenuation that is controlled by the controller to the third adder. A change-over switch responsive to the controller outputs either a signal from the third adder or from the memory. Therefore, a signal is output even during the delay period produced by the memory when the signal is delayed between the first and second adders.

Abstract: In a network, a route which can be uniquely identified is constructed by selecting an arbitrary packet-switching node and an arbitrary transmission line in an arbitrary order from the network. A route memory unit stores data indicating which route is involved in which transmission line within the network. A congested state detecting unit detects a congested state of a transmission line accommodated within its own node. The detected congested state is transmitted to another node by a congested state informing unit as congested state information. A route identifying unit receives the congested state information from the other node and retrieves a route within a corresponding transmission line from the route memory unit to thereby identify the route accommodated within its node. A route control unit carries out control of the congested state of the identified route on the basis of the received congested state information.

Abstract: A packet switching system having a matrix switch including input packet transfer buses and output packet transfer buses. Transfer buffers or gates are provided at cross points of the input and output packet transfer buses. An input packet is supplied to the matrix switch through a transfer control circuit, and an output packet from the matrix switch is output through the transfer control circuit. The input packet is permitted to be applied to the matrix switch so that each of the output packet transfer buses has only one packet during one packet transfer cycle.

Abstract: A data transfer system having a transfer discrimination circuit for discriminating the type of data transfer between an input/output channel device and I/O devices for a computer includes a transfer discrimination circuit. This circuit includes a edge detection unit operating in response to a tag signal supplied to the edge detection unit for detecting the trailing edge of the tag signal after a leading edge of the tag signal has passed. The edge detection unit having a leading edge detector, a trailing edge detector, a storage element, and logic gate circuits. A timing unit is included operating in response to the output of the edge detection unit for counting a predetermined time, along with a discrimination storage unit operating in response to the output of the timing unit for delivering an output indicating an interlock data transfer or an output indicating a data streaming feature data transfer.

Abstract: A loop transmission system and a method of controlling the loop-back condition thereof. The loop transmission system comprises a plurality of node stations, a supervisory station, and two duplicate loop transmission lines which transmit signals in opposite directions. In the loop transmission system, the supervisory station first sends out loop-back commands via both of the duplicate loop transmission lines when faults are detected on both of the duplicate loop transmission lines at the same time. Each of the node stations establishes a loop-back path while retaining a connection path to a succeeding node station upon the receipt of a loop-back command. The loop-back path is released only in the node stations which receive signals normally from both of the duplicate loop transmission lines when the supervisory station sends release commands to the node stations after sending the loopback commands.