Patents by Inventor Shin Sugimoto

Shin Sugimoto has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 11759456
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition contains pemafibrate, a salt thereof or a solvate thereof in an amount of 0.017 to 4.2 mass % in terms of a free form of pemafibrate with respect to the total mass of the pharmaceutical composition.
    Type: Grant
    Filed: June 29, 2018
    Date of Patent: September 19, 2023
    Assignee: KOWA COMPANY, LTD.
    Inventors: Shin Sugimoto, Akito Minamizono
  • Patent number: 11730719
    Abstract: Provided is a pharmaceutical composition which contains pemafibrate, a salt thereof or a solvate thereof and has excellent stability. A pharmaceutical composition is provided containing pemafibrate, a salt thereof or a solvate thereof and having a moisture content of 2.4 mass % or less.
    Type: Grant
    Filed: February 2, 2022
    Date of Patent: August 22, 2023
    Assignee: KOWA COMPANY, LTD.
    Inventors: Shin Sugimoto, Akito Minamizono
  • Publication number: 20230190712
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition is provided to contain the following components (A) and (B): (A) pemafibrate, a salt thereof or a solvate thereof; and (B) one or more selected from the group consisting of the following components (B-1) to (B-6): (B-1) a cellulose ether species; (B-2) a starch species; (B-3) a povidone species; (B-4) a silicic acid compound; (B-5) a polyhydric alcohol; and (B-6) an alkyl sulfate ester.
    Type: Application
    Filed: February 22, 2023
    Publication date: June 22, 2023
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Patent number: 11419855
    Abstract: Provided is a novel technique for improving storage stability of a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and a cellulose species. A pharmaceutical preparation obtained by storing a pharmaceutical composition containing the following components (A) and (B) in a tight package: (A) pemafibrate, a salt thereof or a solvate thereof; and (B) a cellulose species.
    Type: Grant
    Filed: June 29, 2018
    Date of Patent: August 23, 2022
    Assignee: KOWA COMPANY, LTD.
    Inventors: Shin Sugimoto, Akito Minamizono
  • Patent number: 11406621
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition is provided containing the following components (A) and (B): (A) pemafibrate, a salt thereof or a solvate thereof; and (B) a disaccharide species.
    Type: Grant
    Filed: June 29, 2018
    Date of Patent: August 9, 2022
    Assignee: KOWA COMPANY, LTD.
    Inventors: Shin Sugimoto, Akito Minamizono
  • Publication number: 20220151996
    Abstract: Provided is a pharmaceutical composition which contains pemafibrate, a salt thereof or a solvate thereof and has excellent stability. A pharmaceutical composition is provided containing pemafibrate, a salt thereof or a solvate thereof and having a moisture content of 2.4 mass % or less.
    Type: Application
    Filed: February 2, 2022
    Publication date: May 19, 2022
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Patent number: 11298340
    Abstract: Provided is a pharmaceutical composition which contains pemafibrate, a salt thereof or a solvate thereof and has excellent stability. A pharmaceutical composition is provided containing pemafibrate, a salt thereof or a solvate thereof and having a moisture content of 2.4 mass % or less.
    Type: Grant
    Filed: June 29, 2018
    Date of Patent: April 12, 2022
    Assignee: KOWA COMPANY, LTD.
    Inventors: Shin Sugimoto, Akito Minamizono
  • Publication number: 20220096443
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition is provided to contain the following components (A) and (B): (A) pemafibrate, a salt thereof or a solvate thereof; and (B) one or more selected from the group consisting of the following components (B-1) and (B-7): (B-1) an alkylcellulose and a salt thereof; and a (meth)acrylic acid-based polymer.
    Type: Application
    Filed: December 27, 2019
    Publication date: March 31, 2022
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO, Chisa NISHIDA
  • Publication number: 20220047585
    Abstract: A preventing or treating agent for glaucoma is provided. This drug has a strong action of reducing intraocular pressure such that the intraocular pressure can be reduced even from the normal intraocular pressure. More specifically, a prophylactic or therapeutic agent for glaucoma, a preventing or treating agent for ocular hypertension, and eye drops containing (S)-(?)-1-(4-fluoro-5-isoquinolinesulfonyl)-2-methyl homopiperazine or its salt and phosphoric acid or its salt are provided.
    Type: Application
    Filed: November 1, 2021
    Publication date: February 17, 2022
    Applicant: KOWA CO., LTD.
    Inventors: Shin SUGIMOTO, Ken MIZUNO, Masatoshi TAKAHASHI, Makoto KANEBAKO
  • Publication number: 20200179346
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition contains pemafibrate, a salt thereof or a solvate thereof in an amount of 0.017 to 4.2 mass % in terms of a free form of pemafibrate with respect to the total mass of the pharmaceutical composition.
    Type: Application
    Filed: June 29, 2018
    Publication date: June 11, 2020
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Publication number: 20200155514
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition is provided containing the following components (A) and (B): (A) pemafibrate, a salt thereof or a solvate thereof; and (B) a disaccharide species.
    Type: Application
    Filed: June 29, 2018
    Publication date: May 21, 2020
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Publication number: 20200129483
    Abstract: Provided is a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and having excellent homogeneity. The pharmaceutical composition is provided to contain the following components (A) and (B): (A) pemafibrate, a salt thereof or a solvate thereof; and (B) one or more selected from the group consisting of the following components (B-1) to (B-6): (B-1) a cellulose ether species; (B-2) a starch species; (B-3) a povidone species; (B-4) a silicic acid compound; (B-5) a polyhydric alcohol; and (B-6) an alkyl sulfate ester.
    Type: Application
    Filed: June 29, 2018
    Publication date: April 30, 2020
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Publication number: 20200121649
    Abstract: Provided is a novel technique for improving storage stability of a pharmaceutical composition containing pemafibrate, a salt thereof or a solvate thereof and a cellulose species. A pharmaceutical preparation obtained by storing a pharmaceutical composition containing the following components (A) and (B) in a tight package: (A) pemafibrate, a salt thereof or a solvate thereof; and (B) a cellulose species.
    Type: Application
    Filed: June 29, 2018
    Publication date: April 23, 2020
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Publication number: 20200121650
    Abstract: Provided is a pharmaceutical composition which contains pemafibrate, a salt thereof or a solvate thereof and has excellent stability. Apharmaceutical composition is provided containing pemafibrate, a salt thereof or a solvate thereof and having a moisture content of 2.4 mass % or less.
    Type: Application
    Filed: June 29, 2018
    Publication date: April 23, 2020
    Applicant: KOWA COMPANY, LTD.
    Inventors: Shin SUGIMOTO, Akito MINAMIZONO
  • Publication number: 20190328730
    Abstract: A preventing or treating agent for glaucoma is provided. This drug has a strong action of reducing intraocular pressure such that the intraocular pressure can be reduced even from the normal intraocular pressure. More specifically, a prophylactic or therapeutic agent for glaucoma, a preventing or treating agent for ocular hypertension, and eye drops containing (S)-(?)-1-(4-fluoro-5-isoquinolinesulfonyl)-2-methyl homopiperazine or its salt and phosphoric acid or its salt are provided.
    Type: Application
    Filed: July 8, 2019
    Publication date: October 31, 2019
    Applicant: KOWA CO., LTD.
    Inventors: Shin SUGIMOTO, Ken MIZUNO, Masatoshi TAKAHASHI, Makoto KANEBAKO
  • Patent number: 10376523
    Abstract: An aqueous composition having an excellent antiseptic effect is provided. An aqueous composition containing: a compound represented by Formula (1), a salt thereof, or a solvate of the compound or the salt thereof, where X represents a halogen atom, and a quaternary ammonium surfactant. A method for producing an aqueous composition with an antiseptic effect, by incorporating a compound represented by Formula (1), a salt thereof, or a solvate of the compound or the salt thereof and a quaternary ammonium surfactant into the aqueous composition.
    Type: Grant
    Filed: September 25, 2015
    Date of Patent: August 13, 2019
    Assignee: KOWA COMPANY, LTD.
    Inventor: Shin Sugimoto
  • Publication number: 20170290841
    Abstract: An aqueous composition having an excellent antiseptic effect is provided. An aqueous composition comprising a compound represented by Formula (1), wherein X represents a halogen atom, or a salt thereof, or a solvate of the compound or the salt thereof, and a quaternary ammonium surfactant.
    Type: Application
    Filed: September 25, 2015
    Publication date: October 12, 2017
    Applicant: KOWA COMPANY, LTD.
    Inventor: Shin SUGIMOTO
  • Publication number: 20170266080
    Abstract: A technique is provided for suppressing discoloration of an aqueous composition containing a halogenated isoquinoline derivative during preservation at high temperature. A pharmaceutical preparation obtained by storing an aqueous composition comprising a compound represented by Formula (1), wherein X represents a halogen atom, or a salt thereof, or a solvate of the compound or the salt thereof, in a container made of polyolefin-based resin.
    Type: Application
    Filed: September 25, 2015
    Publication date: September 21, 2017
    Applicant: KOWA COMPANY, LTD.
    Inventor: Shin SUGIMOTO
  • Publication number: 20100233287
    Abstract: A preventing or treating agent for glaucoma is provided. This drug has a strong action of reducing intraocular pressure such that the intraocular pressure can be reduced even from the normal intraocular pressure. More specifically, a prophylactic or therapeutic agent for glaucoma, a preventing or treating agent for ocular hypertension, and eye drops containing (S)-(?)-1-(4-fluoro-5-isoquinolinesulfonyl)-2-methyl homopiperazine or its salt and phosphoric acid or its salt are provided.
    Type: Application
    Filed: May 24, 2010
    Publication date: September 16, 2010
    Applicant: Kowa Co., Ltd.
    Inventors: Shin Sugimoto, Ken Mizuno, Masatoshi Takahashi, Makoto Kanebako
  • Publication number: 20060142270
    Abstract: A preventing or treating agent for glaucoma is provided. This drug has a strong action of reducing intraocular pressure such that the intraocular pressure can be reduced even from the normal intraocular pressure. More specifically, a prophylactic or therapeutic agent for glaucoma, a preventing or treating agent for ocular hypertension, and eye drops containing (S)-(-)-1-(4-fluoro-5-isoquinolinesulfonyl)-2-methyl homopiperazine or its salt and phosphoric acid or its salt are provided.
    Type: Application
    Filed: December 14, 2005
    Publication date: June 29, 2006
    Applicant: Kowa Co., Ltd.
    Inventors: Shin Sugimoto, Ken Mizuno, Masatoshi Takahashi, Makoto Kanebako