Patents by Inventor Shotaro Tsunoda

Shotaro Tsunoda has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 11453632
    Abstract: Provided is a novel compound having a selective activating effect on ER?. The present invention provides a compound represented by the following formula (1) wherein R1 represents a cycloalkyl group having 3 to 8 carbon atoms, an alkenyl group having 2 to 6 carbon atoms and optionally substituted with a halogen atom, a 5-membered nitrogen-containing heteroaryl group, a 4- to 6-membered cyclic amino group, an alkanoylamino group having 2 to 6 carbon atoms and optionally substituted with a halogen atom, a 1-trifluoromethyl-1-hydroxymethyl group, or a 1-methylpropyl group; R2 to R5 are the same or different and each represent a hydrogen atom or a fluorine atom; and R6 represents a hydrogen atom or an alkanoyl group having 2 to 5 carbon atoms, or a salt thereof.
    Type: Grant
    Filed: October 23, 2019
    Date of Patent: September 27, 2022
    Assignee: KAO CORPORATION
    Inventors: Kensuke Misawa, Takayoshi Inoue, Shotaro Tsunoda
  • Publication number: 20220009869
    Abstract: Provided is a novel compound having a selective activating effect on ER?. The present invention provides a compound represented by the following formula (1) wherein R1 represents a cycloalkyl group having 3 to 8 carbon atoms, an alkenyl group having 2 to 6 carbon atoms and optionally substituted with a halogen atom, a 5-membered nitrogen-containing heteroaryl group, a 4- to 6-membered cyclic amino group, an alkanoylamino group having 2 to 6 carbon atoms and optionally substituted with a halogen atom, a 1-trifluoromethyl-1-hydroxymethyl group, or a 1-methylpropyl group; R2 to R5 are the same or different and each represent a hydrogen atom or a fluorine atom; and R6 represents a hydrogen atom or an alkanoyl group having 2 to 5 carbon atoms, or a salt thereof.
    Type: Application
    Filed: October 23, 2019
    Publication date: January 13, 2022
    Applicant: KAO CORPORATION
    Inventors: Kensuke MISAWA, Takayoshi INOUE, Shotaro TSUNODA
  • Patent number: 10329558
    Abstract: An object of the present invention is to provide a method of stably introducing a heterocycle into a substrate peptide by using an azoline backbone introducing enzyme. The present invention provides a method of introducing a heterocycle into a leader-sequence-free substrate peptide by using an azoline backbone introducing enzyme to which a leader sequence of the substrate has been bound.
    Type: Grant
    Filed: March 7, 2014
    Date of Patent: June 25, 2019
    Assignee: The University of Tokyo
    Inventors: Hiroaki Suga, Yuki Goto, Shotaro Tsunoda
  • Publication number: 20160083719
    Abstract: An object of the present invention is to provide a method of stably introducing a heterocycle into a substrate peptide by using an azoline backbone introducing enzyme. The present invention provides a method of introducing a heterocycle into a leader-sequence-free substrate peptide by using an azoline backbone introducing enzyme to which a leader sequence of the substrate has been bound.
    Type: Application
    Filed: March 7, 2014
    Publication date: March 24, 2016
    Inventors: Hiroaki Suga, Yuki Goto, Shotaro Tsunoda