Patents by Inventor Simon James Shaw

Simon James Shaw has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • 7-quinolyl ketolide antibacterial agents
    Patent number: 7595300
    Abstract: 15-fluoroketolides of the formula having improved activity and safety, compositions comprising them, and methods for their preparation and use in the treatment of bacterial infections.
    Type: Grant
    Filed: December 7, 2006
    Date of Patent: September 29, 2009
    Assignee: Kosan Biosciences Incorporated
    Inventors: Simon James Shaw, Gary W Ashley, Mark A. Burlingame
  • Motilide compounds
    Patent number: 7582611
    Abstract: Compounds having a structure according to formula (I) where RA, RB, RC, RD, RE, and RF are as defined herein, are useful as prokinetic agents.
    Type: Grant
    Filed: May 2, 2006
    Date of Patent: September 1, 2009
    Assignee: Pfizer Inc.
    Inventors: Yaoquan Liu, Christopher Carreras, David C. Myles, Yong Li, Simon James Shaw, Hong Fu, Yue Chen, Hao Zheng, Yandong Li, Mark A. Burlingame
  • Compounds useful for the synthesis of (+)-discodermolide and methods thereof
    Patent number: 7348436
    Abstract: Compounds and methods useful for the synthesis of (+)-discodermolide, a naturally occurring microtubule stabilizing agent useful as an anti-cancer agent.
    Type: Grant
    Filed: March 1, 2005
    Date of Patent: March 25, 2008
    Assignee: Kosan Biosciences Incorporated
    Inventors: David C. Myles, Simon James Shaw, Kurt F. Sundermann
  • Synthetic techniques and intermediates for polyhydroxy dienyl lactones and mimics thereof
    Patent number: 7342124
    Abstract: Synthetic methods and intermediates useful in the preparation of lactone containing compounds such as discodermolide and compounds which mimic the chemical or biological activity of discodermolide are provided.
    Type: Grant
    Filed: April 2, 2004
    Date of Patent: March 11, 2008
    Assignees: The Trustees Of The University Of Pennsylvania, Kosan Biosciences, Inc.
    Inventors: David C. Myles, Mark Burlingame, Simon James Shaw, Kurt F. Sundermann, Brian Scott Freeze, Ignació Brouard Martin, Tomoyasu Hirose, Amos B. Smith, III
  • Synthetic discodermolide analogs
    Patent number: 7214708
    Abstract: Synthetic discodermolide analogs having utility as antiproliferative agents, having a structure represented by formula A where RA through RE and XA are as defined herein.
    Type: Grant
    Filed: October 28, 2005
    Date of Patent: May 8, 2007
    Assignee: Kosan Biosciences Incorporated
    Inventors: Kurt F. Sundermann, Simon James Shaw, Daniel V. Santi
  • Amido macrolides
    Patent number: 6939861
    Abstract: Various macrolide compounds such as those having the following formulas are provided where the variables have the values provided herein.
    Type: Grant
    Filed: January 17, 2003
    Date of Patent: September 6, 2005
    Assignee: Kosan Biosciences, Inc.
    Inventors: Gary Ashley, Simon James Shaw, Yandong Li, David C. Myles
  • Amido macrolides
    Publication number: 20030199458
    Abstract: Various macrolide compounds such as those having the following formulas are provided where the variables have the values provided herein.
    Type: Application
    Filed: January 17, 2003
    Publication date: October 23, 2003
    Applicant: Kosan Biosciences, Inc.
    Inventors: Gary Ashley, Simon James Shaw, Yandong Li