Patents by Inventor Stanislaw Sobiak

Stanislaw Sobiak has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 10065935
    Abstract: The present invention relates to the new chemical compounds containing (Z)-1,2-diphenylethene moiety in the structures, particularly the new derivatives of cis-stilbene, the new derivatives of 4,5-diphenyl-1,3-oxazole, the new derivatives of 1-methyl-4,5-diphenyl-1H-imidazole and pharmaceutically acceptable salts thereof. The invention relates also to the application of aforementioned compounds as a microtubule-interfering agents (MIAs). The new derivatives, because of their potential antimitotic and antiangio-genic activity, can be used as ingredients in the preparations used in the treatment of cancer.
    Type: Grant
    Filed: March 28, 2013
    Date of Patent: September 4, 2018
    Assignee: Uniwersytet Medyczny IM. Karola Marcinkowskiego
    Inventors: Tomasz Stefański, Jakub Różański, Renata Mikstacka, Stanislaw Sobiak
  • Patent number: 9169267
    Abstract: The invention relates to a novel class of quaternary ammonium salts containing tetra-hydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium moiety in the structure, in particular the new derivatives of 4-methyltetrahydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium, 4-(2-oxoethyl)tetrahydro[1,3]oxazolo[2,3-6][1,3]oxazol-4-ium, bis{4-methyltetrahydro[1,3]oxazoio[2,3-6][1,3]oxazol-4-ium}, bis{4-(2-oxoethyl)tetrahydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium} and tris{4-methyltetrahydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium} salts, process for the preparation of a novel class of quaternary ammonium salts and applications thereof.
    Type: Grant
    Filed: January 31, 2013
    Date of Patent: October 27, 2015
    Assignee: Uniwersytet Medyczny IM. Karola Marcinkowskiego
    Inventors: Jakub Różański, Agnieszka Gielara-Korzańska, Stanislaw Sobiak, Marcelina Maria Kubicka, Helena Kukuła
  • Publication number: 20150080583
    Abstract: The invention relates to a novel class of quaternary ammonium salts containing tetra-hydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium moiety in the structure, in particular the new derivatives of 4-methyltetrahydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium, 4-(2-oxoethyl)tetrahydro[1,3]oxazolo[2,3-6][1,3]oxazol-4-ium, bis{4-methyltetrahydro[1,3]oxazoio[2,3-6][1,3]oxazol-4-ium}, bis{4-(2-oxoethyl)tetrahydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium} and tris{4-methyltetrahydro[1,3]oxazolo[2,3-b][1,3]oxazol-4-ium} salts, process for the preparation of a novel class of quaternary ammonium salts and applications thereof.
    Type: Application
    Filed: January 31, 2013
    Publication date: March 19, 2015
    Applicant: UNIWERSYTET MEDYCZNY IM. KAROLA MARCINKOWSKIEGO
    Inventors: Jakub Rózanski, Agnieszka Gielara-Korzanska, Stanislaw Sobiak, Marcelina Maria Kubicka, Helena Kukula
  • Publication number: 20150065727
    Abstract: The present invention relates to the new chemical compounds containing (Z)-1,2-diphenylethene moiety in the structures, particularly the new derivatives of cis-stilbene, the new derivatives of 4,5-diphenyl-1,3-oxazole, the new derivatives of 1-methyl-4,5-diphenyl-1H-imidazole and pharmaceutically acceptable salts thereof. The invention relates also to the application of aforementioned compounds as a microtubule-interfering agents (MIAs). The new derivatives, because of their potential antimitotic and antiangio-genic activity, can be used as ingredients in the preparations used in the treatment of cancer.
    Type: Application
    Filed: March 28, 2013
    Publication date: March 5, 2015
    Inventors: Tomasz Stefanski, Jakub Rózanski, Renata Mikstacka, Stanislaw Sobiak