Patents by Inventor Stephen Antonelli

Stephen Antonelli has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • BIPHENYLAZETIDINONE CHOLESTEROL ABSORPTION INHIBITORS
    Publication number: 20090131395
    Abstract: The invention relates to a chemical genus of 4-biphenyl-1-phenylazetidin-2-ones useful in the treatment of hypercholesterolemia and other disorders. The compounds have the general formula I: Pharmaceutical compositions and methods for treating cholesterol- and lipid-associated diseases are also disclosed.
    Type: Application
    Filed: May 5, 2006
    Publication date: May 21, 2009
    Applicant: MICROBIA, INC.
    Inventors: Stephen Antonelli, Regina Lundrigan, Eduardo J. Martinez, Wayne C. Schairer, John J. Talley, Timothy C. Barden, JingJing Yang, Daniel P. Zimmer
  • Processes for Production of 4-(Biphenylyl)Azetidin-2-One Phosphonic Acids
    Publication number: 20090099355
    Abstract: The present invention relates to processes for the production of 4-(biphenylyl)azetidin-2-one phosphonic acid derivatives of formula
    Type: Application
    Filed: May 25, 2006
    Publication date: April 16, 2009
    Applicant: MICROBIA, INC.
    Inventors: Stephen Antonelli, Timothy C. Barden, Peter Lee, Eduardo J. Martinez, Wayne C. Schairer, John J. Talley
  • Process For Production Of 4-Biphenylyazetidin-2-Ones
    Publication number: 20080287663
    Abstract: The present invention relates to processes for the production of 4-biphenylylazetidin-2-one derivatives of formula
    Type: Application
    Filed: May 8, 2006
    Publication date: November 20, 2008
    Applicant: MICROBIA, INC.
    Inventors: Peter Lee, Stephen Antonelli, Regina Lundrigan, Eduardo J. Martinez, Wayne C. Schairer, John J. Talley
  • 4-BIARYLYL-1-PHENYLAZETIDIN-2-ONES
    Publication number: 20080167255
    Abstract: 4-Biarylyl-1-phenylazetidin-2-ones useful for the treatment of hypercholesterolemia are disclosed. The compounds are of the general formula in which represents an aryl or heteroaryl residue; Ar represents an aryl residue; U is a two to six atom chain; and the R's represent substituents.
    Type: Application
    Filed: December 11, 2007
    Publication date: July 10, 2008
    Applicant: MICROBIA, INC.
    Inventors: Eduardo J. Martinez, John J. Talley, Stephen Antonelli, Timothy C. Barden, Regina Lundrigan-Soucy, Wayne C. Schairer, Jing-Jing Yang, Daniel P. Zimmer, Brian Cali, Mark G. Currie, Peter S. Yorgey
  • 4-Biarylyl-1-phenylazetidin-2-ones
    Patent number: 7320972
    Abstract: 4-Biarylyl-1-phenylazetidin-2-ones useful for the treatment of hypercholesterolemia are disclosed. The compounds are of the general formula in which represents an aryl or heteroaryl residue; Ar represents an aryl residue; U is a two to six atom chain; and the R's represent substituents.
    Type: Grant
    Filed: November 10, 2004
    Date of Patent: January 22, 2008
    Assignee: Microbia, Inc.
    Inventors: Eduardo Martinez, John J. Talley, Stephen Antonelli, Timothy C. Barden, Regina Lundrigan-Soucy, Wayne C. Schairer, Jing-Jing Yang, Daniel P. Zimmer, Brian Cali, Mark G. Currie, Peter S. Yorgey
  • 4-Biarylyl-1-phenylazetidin-2-ones
    Publication number: 20050209165
    Abstract: 4-Biarylyl-1-phenylazetidin-2-ones useful for the treatment of hypercholesterolemia are disclosed. The compounds are of the general formula in which represents an aryl or heteroaryl residue; Ar represents an aryl residue; U is a two to six atom chain; and the R's represent substituents.
    Type: Application
    Filed: November 10, 2004
    Publication date: September 22, 2005
    Inventors: Eduardo Martinez, John Talley, Stephen Antonelli, Timothy Barden, Regina Lundrigan-Soucy, Wayne Schairer, Jing-Jing Yang, Daniel Zimmer