Patents by Inventor Sylvain Celanire

Sylvain Celanire has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Fused Oxazoles & Thiazoles As Histamine H3- Receptor Ligands
    Publication number: 20100009969
    Abstract: The present invention relates to compounds comprising fused oxazole or thiazole derivatives of formula (I), processes for preparing them, pharmaceutical compositions comprising said compounds and their uses as H3-receptor ligands, wherein A is a cyclic amine which is linked to the propylene group via an amino nitrogen; B is selected from the group consisting of heteroaryl, 5-8-membered heterocycloalkyl, 5-8-membered cycloalkyl; X is either N or CH; Y is either O or S.
    Type: Application
    Filed: July 17, 2007
    Publication date: January 14, 2010
    Applicant: UCB PHARMA, S.A.
    Inventors: Frédéric Denonne, Sylvain Celanire, Laurent Provins, Sabine Defays
  • Compounds Comprising a Lactam or a Lactam Derivative Moiety, Processes for Making Them, and Their Uses
    Publication number: 20090023708
    Abstract: The present invention relates to compounds of formula (I) comprising a lactam or a lactam derivative moiety, processes for preparing them, pharmaceutical compositions comprising said compounds and their uses as pharmaceuticals.
    Type: Application
    Filed: October 25, 2006
    Publication date: January 22, 2009
    Applicant: UCB PHARMA, S.A.
    Inventors: Sylvain Celanire, Luc Quere, Frederic Denonne, Laurent Provins
  • Compounds Comprising an Oxazole or Thiazole Moiety, Processes for Making Them, and Their Uses
    Publication number: 20080275046
    Abstract: The present invention relates to compounds comprising an oxazole or thiazole moiety of formula (I), processes for preparing them, pharmaceutical compositions comprising said compounds and their uses as H3-receptor ligands, Formula (I), wherein, A1 is CH, C(alkyl), C-halogen or N; R1 is hydrogen, halogen, C1-6 alkyl or alkoxy; R2 is, Formula (II?), A3 is O or S; R3 is hydrogen, halogen, C1-6 alkyl or alkoxy; R4 is hydrogen, halogen, C1-6 alkyl, alkoxy or —O-L; R5 is hydrogen or —O-L, wherein L is an aminoalkyl group and at least one of R4 and R5 should be —O-L.
    Type: Application
    Filed: March 28, 2006
    Publication date: November 6, 2008
    Applicant: UCB PHARMA, S.A.
    Inventors: Sylvain Celanire, Frederic Denonne
  • Compounds Comprising an Oxazoline or Thiazoline Moiety, Processes for Making Them, and Their Uses
    Publication number: 20080161331
    Abstract: The present invention relates to compounds comprising an oxazoline or thiazoline moiety, processes for preparing them, pharmaceutical compositions comprising said compounds and their uses as H3-receptor ligands, (I), wherein A1 is CH C(CH3) or N; R1 is hydrogen or halogen; R2 is (II); A2 is O or S; R3 is hydrogen, halogen, C1-4 alkyl or C1-4 alkoxy; R4 is hydrogen, halogen, C1-4 alkyl, C1-4 alkoxy, trifluoromethyl or —O—(CH2)n-NR12aR each CH2 in —O—(CH2)n-NR12aR 12b being optionally substituted by one or two C1-4 alkyl; R5 is hydrogen or —O—(CH2)m—NR13aR13b, each CH2 in —O—(CH2)m—NR13aR13b being optionally substituted by one or two C1-4 alkyl, and at least one of R4 and R5 should be a —O—(CH2)n-NR12/13aR12/13b group.
    Type: Application
    Filed: March 29, 2006
    Publication date: July 3, 2008
    Applicant: UCB PHARMA, S.A.
    Inventors: Regorius Leurs, Henkdrik Timmerman, Sylvain Celanire, Patrice Talaga, Frederic Denonne, Florence Lebon