Abstract: An object of the present invention is to provide a novel tetrahydroazepine compound and a process for producing the same. The present invention relates to a tetrahydroazepine compound represented by the formula (10) or a salt thereof, and a process for producing the said compound or a salt thereof. (In the formula, R1 is an optionally substituted alkyl group, R2 is an optionally substituted alkyl group and one of the X—Y bond and the Y—Z bond is a carbon-carbon double bond and the other is a carbon-carbon single bond).

Abstract: An object of the present invention is to provide a novel tetrahydroazepine compound and a process for producing the same. The present invention relates to a tetrahydroazepine compound represented by the formula (10) or a salt thereof, and a process for producing the said compound or a salt thereof. (In the formula, R1 is an optionally substituted alkyl group, R2 is an optionally substituted alkyl group and one of the X—Y bond and the Y—Z bond is a carbon-carbon double bond and the other is a carbon-carbon single bond.

Abstract: A power supply device includes: an oscillation unit for outputting a high frequency signal; a modulation unit for outputting a pulsed high frequency signal; a level adjustment unit for adjusting and outputting a level of the pulsed high frequency signal; a power amplifier for amplifying a power outputted from the level adjustment unit; an output power detection unit for detecting an output power value from the power amplifier; and a control unit. The control unit corrects and outputs a level control signal for controlling the level of the pulsed high frequency signal based on a corresponding correction factor at each of elapsed times in an on state of the pulsed high frequency signal, and compares comparison values in a current pulse and a previous pulse to update the correction factor such that comparison result between the set power value and the output power value becomes smaller at each reflection coefficient.

Abstract: A power supply device includes: an oscillation unit for outputting a high frequency signal; a modulation unit for outputting a pulsed high frequency signal; a level adjustment unit for adjusting and outputting a level of the pulsed high frequency signal; a power amplifier for amplifying a power outputted from the level adjustment unit; an output power detection unit for detecting an output power value from the power amplifier; and a control unit. The control unit corrects and outputs a level control signal for controlling the level of the pulsed high frequency signal based on a corresponding correction factor at each of elapsed times in an on state of the pulsed high frequency signal, and compares comparison values in a current pulse and a previous pulse to update the correction factor such that comparison result between the set power value and the output power value becomes smaller at each reflection coefficient.

Abstract: A power supply circuit includes: a push-pull amplifier unit which amplifies an input signal with a push-pull amplification protocol; a variable power supply unit which varies, with a control signal, the voltage level of a power supply voltage which is supplied to the push-pull amplifier; a switch control unit which, on the basis of the input signal, outputs the control signal which controls the voltage level of the power supply voltage; and a timing control unit which applies a specified time delay to the input signal. When the control signal rises, the switch control unit causes the control signal to rise at a faster timing, according to the voltage level switch transition timing, than a delay time upon the timing control unit, and when the control signal falls, the switch control unit causes the control signal to fall at the timing of the delay time.

Abstract: A power supply circuit includes: a push-pull amplifier unit which amplifies an input signal with a push-pull amplification protocol; a variable power supply unit which varies, with a control signal, the voltage level of a power supply voltage which is supplied to the push-pull amplifier; a switch control unit which, on the basis of the input signal, outputs the control signal which controls the voltage level of the power supply voltage; and a timing control unit which applies a specified time delay to the input signal. When the control signal rises, the switch control unit causes the control signal to rise at a faster timing, according to the voltage level switch transition timing, than a delay time upon the timing control unit, and when the control signal falls, the switch control unit causes the control signal to fall at the timing of the delay time.

Abstract: An aminopropylidene derivative having excellent histamine receptor antagonistic action, a compound which is useful as a pharmaceutical composition, especially as an active ingredient, having alleviated side effects in the central nervous system is described. In the aminopropylidene derivative, R1 and R2, which may be identical or different, stand for a hydrogen, a substituted carbonyl, a substituted carbonylalkyl, and acrylic acid, excluding a case where both are hydrogen; R3 and R4, which may be identical or different, stand for hydrogen, an alkyl which may be substituted with phenyl, or the like; A stands for unsubstituted or an oxo; B stands for a carbon or an oxygen; one of X and Y stands for a carbon and the other stands for a sulfur, a broken line part stands for a single bond or a double bond, and a wavy line stands for cis-form and/or trans-form.

Abstract: Disclosed is a process for producing a thiabenzoazulene-propionic acid derivative which is useful as an active ingredient of an antihistaminic agent or the like. According to the producing process of the present invention, it is possible to produce a thiabenzoazulene-propionic acid derivative where the 2-position of the thiabenzoazulene skeleton is substituted with propionic acid. The thiabenzoazulene propionic-acid derivative thus synthesized has excellent antagonistic action to histamine H1 receptor and low intracerebral transmigration and, therefore, is useful as an active ingredient of the pharmaceutical composition such as an antihistaminic agent.

Abstract: The present invention provides a compound a piperidine derivative having excellent histamine receptor antagonistic action, which is useful as active ingredients of a pharmaceutical composition, especially an antihistamine. The piperidine derivative of the present invention has a potent histamine receptor antagonistic action. Further, the compound of the present invention shows low brain transfer even in a cerebral receptor binding test where a mouse is orally administered with the compound, so that the compound has preferred properties of alleviating side effects in the central nervous system, such as drowsiness. The piperidine derivative of the present invention is very useful as a novel antihistamine having smaller side effects in the central nervous system, such as drowsiness.

Abstract: Disclosed is a process for producing a thiabenzoazulene-propionic acid derivative which is useful as an active ingredient of an antihistaminic agent or the like. According to the producing process of the present invention, it is possible to produce a thiabenzoazulene-propionic acid derivative where the 2-position of the thiabenzoazulene skeleton is substituted with propionic acid. The thiabenzoazulene propionic-acid derivative thus synthesized has excellent antagonistic action to histamine H1 receptor and low intracerebral transmigration and, therefore, is useful as an active ingredient of the pharmaceutical composition such as an antihistaminic agent.

Abstract: An amplifier capable of lowering an electrical current flowing in a peak amplifier before a carrier amplifier becomes saturated to thereby improve the efficiency of an entirety of the amplifier is provided. The amplifier includes a carrier amplifier circuit having an amplifying element operable in class-AB or class-B, and a plurality of peak amplifier circuits which have amplifying elements operating in class-B or class-C and which are arranged to start an operation in stages in response to an input level. An output of the carrier amplifier circuit and outputs of the peak amplifier circuits are combined together for signal output. One of the peak amplifier circuits which is rendered operative at the lowest input level is smaller in saturation output than the carrier amplifier circuit.

Abstract: A power circuit used for an amplifier, which includes an amplifier provided with a linear amplifier serving as a voltage source, a DC/DC converter serving as a current source, a hysteresis comparator controlling the DC/DC converter, and a current detector detecting output current from the linear amplifier to output the detected output current to the hysteresis comparator; and a switching restricting device for restricting a switching interval in the DC/DC converter such that the switching interval is not equal to or less than a constant time or is not shorter than the constant time.

Abstract: An aminopropylidene derivative having excellent histamine receptor antagonistic action, a compound which is useful as a pharmaceutical composition, especially as an active ingredient, having alleviated side effects in the central nervous system is described. In the aminopropylidene derivative, R1 and R2, which may be identical or different, stand for a hydrogen, a substituted carbonyl, a substituted carbonylalkyl, and acrylic acid, excluding a case where both are hydrogen; R3 and R4, which may be identical or different, stand for hydrogen, an alkyl which may be substituted with phenyl, or the like; A stands for unsubstituted or an oxo; B stands for a carbon or an oxygen; one of X and Y stands for a carbon and the other stands for a sulfur, a broken line part stands for a single bond or a double bond, and a wavy line stands for cis-form and/or trans-form.

Abstract: The present invention provides a compound a piperidine derivative having excellent histamine receptor antagonistic action, which is useful as active ingredients of a pharmaceutical composition, especially an antihistamine. The piperidine derivative of the present invention has a potent histamine receptor antagonistic action. Further, the compound of the present invention shows low brain transfer even in a cerebral receptor binding test where a mouse is orally administered with the compound, so that the compound has preferred properties of alleviating side effects in the central nervous system, such as drowsiness. The piperidine derivative of the present invention is very useful as a novel antihistamine having smaller side effects in the central nervous system, such as drowsiness.

Abstract: A power circuit used for an amplifier, which includes an amplifier provided with a linear amplifier serving as a voltage source, a DC/DC converter serving as a current source, a hysteresis comparator controlling the DC/DC converter, and a current detector detecting output current from the linear amplifier to output the detected output current to the hysteresis comparator; and a switching restricting means for restricting a switching interval in the DC/DC converter such that the switching interval is not equal to or less than a constant time or is not shorter than the constant time.

Abstract: A high frequency power amplifier includes an amplifying device for amplifying an input high frequency signal, a harmonic reflection circuit for reflecting a harmonic outputted from the amplifying device, and a harmonic generating circuit provided at an input terminal of the amplifying device, the harmonic generating circuit including a divider for dividing an input signal of a fundamental wave into two parts, a harmonic generator for generating a second harmonic from one part of the fundamental wave signal, and a combiner for combining the second harmonic generated from the harmonic generator with the other part of the fundamental wave signal to offer a combined signal to the amplifying device, wherein the harmonic reflection circuit reflects the second harmonic.

Abstract: An amplifying apparatus includes a splitting unit for splitting an input signal into a first split signal and a second split signal; phase-shifting unit for phase-shifting the first split signal and the second split signal, respectively; a first amplifying unit for amplifying a first phase-shifted signal and outputting the signal as a first output signal; a second amplifying unit for amplifying, in a substantially identical manner to the first amplifying unit, a second phase-shifted signal and outputting the signal as a second output signal; and a matching unit for matching the first output signal and the second output signal to a first transmission unit and a second transmission unit, respectively. The first transmission unit is for transmitting the first output signal from the matching unit to a load resistor, and the second transmission unit is for transmitting the second output signal from the matching unit to the load resistor.

Abstract: An amplifier capable of lowering an electrical current flowing in a peak amplifier before a carrier amplifier becomes saturated to thereby improve the efficiency of an entirety of the amplifier is provided. The amplifier includes a carrier amplifier circuit having an amplifying element operable in class-AB or class-B, and a plurality of peak amplifier circuits which have amplifying elements operating in class-B or class-C and which are arranged to start an operation in stages in response to an input level. An output of the carrier amplifier circuit and outputs of the peak amplifier circuits are combined together for signal output. One of the peak amplifier circuits which is rendered operative at the lowest input level is smaller in saturation output than the carrier amplifier circuit.

Abstract: A distortion compensation apparatus includes distortion generating means for generating distortions to compensate for a distortion generated in an amplifier 2. The distortion generating means includes a nonlinear circuit 13 having an input/output expansion characteristic as a circuit which generates a distortion of the lowest odd order as a compensation target and also includes a nonlinear circuit 18 having an input/output saturation characteristic as a circuit which generates a distortion of another odd order as a compensation target.

Abstract: An amplifying apparatus includes a splitting unit for splitting an input signal into a first split signal and a second split signal; phase-shifting unit for phase-shifting the first split signal and the second split signal, respectively; a first amplifying unit for amplifying a first phase-shifted signal and outputting the signal as a first output signal; a second amplifying unit for amplifying, in a substantially identical manner to the first amplifying unit, a second phase-shifted signal and outputting the signal as a second output signal; and a matching unit for matching the first output signal and the second output signal to a first transmission unit and a second transmission unit, respectively. The first transmission unit is for transmitting the first output signal from the matching unit to a load resistor, and the second transmission unit is for transmitting the second output signal from the matching unit to the load resistor.