Patents by Inventor Thierry F. Imbert

Thierry F. Imbert has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4657911
    Abstract: New derivatives of 3-amino quinuclidine of formula: ##STR1## in which X=sulfur or oxygen; R=H, lower alkyl or benzyl; and Ar=substituted phenyl or substituted pyrimidinyl.These new derivatives have utility in therapeutics as accelerators of the gastro-intestinal motor function and as medicament potentiators.
    Type: Grant
    Filed: June 29, 1983
    Date of Patent: April 14, 1987
    Assignee: Delalande S.A.
    Inventors: Thierry F. Imbert, Nicole A. M. Dorme, Michel Langlois
  • Patent number: 4536580
    Abstract: There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
    Type: Grant
    Filed: July 19, 1982
    Date of Patent: August 20, 1985
    Assignee: Delalande S.A.
    Inventors: Philippe L. Dostert, Thierry F. Imbert, Bernard P. Bucher
  • Patent number: 4471120
    Abstract: There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
    Type: Grant
    Filed: January 7, 1980
    Date of Patent: September 11, 1984
    Assignee: Delalande S.A.
    Inventors: Philippe L. Dostert, Thierry F. Imbert, Bernard P. Bucher
  • Patent number: 4424358
    Abstract: There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
    Type: Grant
    Filed: September 11, 1980
    Date of Patent: January 3, 1984
    Assignee: Delalande S.A.
    Inventors: Philippe L. Dostert, Thierry F. Imbert, Bernard P. Bucher
  • Patent number: 4329466
    Abstract: There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
    Type: Grant
    Filed: April 16, 1981
    Date of Patent: May 11, 1982
    Assignee: Delalande S.A.
    Inventors: Philippe L. Dostert, Thierry F. Imbert, Bernard P. Bucher
  • Patent number: 4321378
    Abstract: There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
    Type: Grant
    Filed: April 16, 1981
    Date of Patent: March 23, 1982
    Assignee: Delalande S.A.
    Inventors: Philippe L. Dostert, Thierry F. Imbert, Bernard P. Bucher
  • Patent number: 4250178
    Abstract: Compounds for the formula ##STR1## for example, ##STR2## are prepared by reacting ##STR3## with ##STR4## The compounds possess neuroleptic properties.
    Type: Grant
    Filed: February 12, 1979
    Date of Patent: February 10, 1981
    Assignee: Delalande S.A.
    Inventors: Bernard P. Bucher, Jean-Francois R. Ancher, Thierry F. Imbert
  • Patent number: 4104384
    Abstract: Compounds of the formula ##STR1## where Ar is phenyl, substituted phenyl, .alpha.-furyl or .alpha.-thienyl, andR is NH.sub.2, NHR.sup.1 wherein R.sup.1 is alkyl or cycloalkyl, or NR.sub.1 R.sub.2 whereinR.sub.1 and R.sub.2 are alkyl or --N.sub.1 R.sub.1 R.sub.2 is piperidino, pyrrolidino, morpholino or hexamethyleneimino. The compounds are prepared by reacting the corresponding Ar-substituted chloromethylated benzimadazole with the corresponding R-substituted piperazine. The compounds possess gastric antisecretory, anti-ulcerous, spasmolytic, anti-cholinergic, anti-bronchoconstrictive, analgesic, anti-inflammatory, anti-hypertensive and diuretic properties.
    Type: Grant
    Filed: November 28, 1977
    Date of Patent: August 1, 1978
    Assignee: Delalande S.A.
    Inventors: Claude P. Fauran, Michel J. Turin, Thierry F. Imbert, Guy M. Raynaud, Nicole A. M. Dorme
  • Patent number: 4072682
    Abstract: Compounds of the formula ##STR1## where Ar is phenyl, substituted phenyl, .alpha.-furyl or .alpha.-thienyl, andR is NH.sub.2, NHR.sup.1 wherein R.sup.1 is alkyl or cycloalkyl, or NR.sub.1 R.sub.2wherein R.sub.1 and R.sub.2 are alkyl or --N.sub.1 R.sub.1 R.sub.2 is piperidino, pyrrolidino, morpholino or hexamethyleneimino. The compounds are prepared by reacting the corresponding Ar-substituted chloromethylated benzimidazole with the corresponding R-substituted piperazine. The compounds possess gastric antisecretory, anti-ulcerous, spasmolytic, anti-cholinergic, anti-bronchoconstrictive, analgesic, anti-inflammatory, anti-hypertensive and diuretic properties.
    Type: Grant
    Filed: December 22, 1975
    Date of Patent: February 7, 1978
    Assignee: Delalande S.A.
    Inventors: Claude P. Fauran, Michel J. Turin, Thierry F. Imbert, Guy M. Raynaud, Nicole A. M. Dorme