Publication number: 20050038041
Abstract: Fungicidal pyrimidine derivatives and the use as a fungicide of the compounds of formula (1): wherein R1 is H, C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl, C3-C6cycloalkyl, C1-C6alkoxy, C3-C6cycloalkoxy, C1-C6alkylthio, C1-C6alkylsulfinyl, C1-C6alkylsulfonyl, phenyl, pyridinyl or azolyl groups, (being optionally substituted by one or more substituents); or N(R4)C(O)R5, R2 is polyfluoroalkyl, R3 is fluorine, chlorine, bromine or iodine; ethenyl or ethynyl (being optionally substituted by one or more of halogen), R4 and R5 are, independently, H, C1-C6alkyl, C2-C6alkenyl or C2-C6alkynyl groups, (being optionally substituted by one or more of halogen or cyano); or R4 and R5 can join together to form a 5 or 6-membered ring, Q is a heteroaromatic ring selected from the following ring system; imidazol-1-yl, pyrazol-1-yl, 1,2,3-triazol-1-yl, 1,2,3-triazol-2-yl, 1,2,4-triazol-1-yl, 1,2,4-triazol-4-yl, benzimidazol-1-yl or tetrazol-5-yl groups, (being optionally substituted by one or more of substituents).
Type:
Application
Filed:
June 4, 2004
Publication date:
February 17, 2005
Inventors:
Yuki Nakagawa, Sergey Bobrov, Charles Semer, Thomas Kucharek, Masahiro Hamamoto
Patent number: 6818631
Abstract: Fungicidal pyrimidine derivatives and the use as a fungicide of the compounds of formula (1):
wherein R1 is H, C1-C6alkyl, C2-C6alkenyl, C2-C6alkynyl C3-C6cycloalkyl, C1-C6alkoxy, C3-C6cycloalkoxy, C1-C6alylthio, C1-C6alkylsulfinyl, C1-C6alkylsulfonyl, phenyl, pyridinyl or azolyl groups, (being optionally substituted by one or more substituents); or N(R4)C(O)R5, R2 is polyfluoroalkyl, R3 is fluorine, chlorine, bromine or iodine; ethenyl or ethynyl (being optionally substituted by one or more of halogen), R4 and R5 are, independently, H, C1-C6alkyl, C2-C6alkenyl or C2-C6alkynyl groups, (being optionally substituted by one or more of halogen or cyano); or R4 and R5 can join together to form a 5 or 6-membered ring, Q is a heteroaromatic ring selected from the following ring system; imidazol-1-yl, pyrazol-1-yl, 1,2,3-triazol-1-yl, 1,2,3-triazol-2-yl, 1,2,4-triazol-1-yl, 1,2,4-triazol-1-yl, benzimidazol-1-yl or tetrazol-5-yl groups, (being optionally substituted by one or more of substituents).
Type:
Grant
Filed:
August 15, 2003
Date of Patent:
November 16, 2004
Assignee:
Nippon Soda Co. Ltd.
Inventors:
Yuki Nakagawa, Sergey Bobrov, Charles R. Semer, IV, Thomas A. Kucharek, Masahiro Haramoto
Patent number: 6713629
Abstract: Fungicidal 5,5-disubstituted thiazolidine derivatives are provided having the formula;
wherein R1 is selected from the group consisting of C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 cycloalkyl, and optionally substituted phenyl; R2 is phenyl substituted by An; A is each independently selected from the group consisting of H, halogen, C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxy, C1-C6 alkenyloxy, C1-C6 alkynyloxy, nitro, optionally substituted amino, C1-C6 alkylthio, C1-C6 alkoxycarbonyl, phenoxy, phenyl, optionally aubstituted pyridyl, optionally substituted thienyl, and optionally substituted furyl; n is 0-5; X is O; Y is selected from the group consisting of O, S, N—OH, optionally substituted arylimino, optionally substituted alkylimino, optionally substituted carbamoyloxyimino, optionally substituted sulfamoyloxyimino, optionally substituted aroyloxyimino, optionally substituted alkoxycarbonyloxyimino, optionally substituted alkylhydrazono, optionally substituted phenylhydrazono, and alkylsu
Type:
Grant
Filed:
September 11, 2002
Date of Patent:
March 30, 2004
Assignee:
Nippon Soda Co., Ltd.
Inventors:
Isao Iwataki, Vladimir F. Rudchenko, Thomas Kurz, Charles R. Semer, IV, Thomas A. Kucharek, Detlef Geffken