Patents by Inventor Timothy D. Cutarelli

Timothy D. Cutarelli has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Process and intermediates for the synthesis of 2-(quinolin-5-yl)-4,5 disubstituted-azole derivatives
    Patent number: 7985860
    Abstract: This application discloses a novel process to synthesize 2-(Quinolin-5yo)-4,5-Disubstituted-Azole derivatives, which may be used, for example, as PDE IV inhibitor compounds in pharmaceutical preparations.
    Type: Grant
    Filed: August 10, 2007
    Date of Patent: July 26, 2011
    Assignee: Schering Corporation
    Inventors: Timothy D. Cutarelli, Xiaoyong Fu, Timothy L. McAllister, Michael R. Reeder, Jianguo Yin, Kelvin H. Yong, Shuyi Zhang
  • Process and intermediates for the Synthesis of heterocyclic Substituted Piperazines with CXCR3 Antagonist Activity
    Publication number: 20110124867
    Abstract: The present invention relates to novel processes for the preparation of the compound of the Formula A45: or a physiologically acceptable salt, solvate or prodrug thereof, which has utility, for example, as a pharmaceutically active compound with CXCR3 antagonist activity, and to novel intermediates useful in the synthesis thereof.
    Type: Application
    Filed: December 16, 2008
    Publication date: May 26, 2011
    Applicant: Schering Corporation
    Inventors: Frank Xing Chen, Timothy D. Cutarelli, Xiayong Fu, Xian Liang, Timothy L. McAllister, Robert K. Orr, Jianguo Yin, Kelvin H. Yong, Man Zhu
  • PROCESS FOR THE PRODUCTION OF SUBSTITUTED 5-QUINOLYL-OXAZOLES AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
    Publication number: 20100324295
    Abstract: The present invention relates a process for the preparation of a compound of the formula: wherein R1, R2, R6, R9 and R10 are as described herein. The compounds are inhibitors of phosphodiesterase 4 (PDE4).
    Type: Application
    Filed: July 3, 2008
    Publication date: December 23, 2010
    Inventors: Timothy D. Cutarelli, Dimitar L. Filipov, Christopher Stanley Pridgen, Michael R. Reeder, Kelvin H. Yong, Dimitrios N. Zarkadas