Patents by Inventor Tobias Kapferer
Tobias Kapferer has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).
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Patent number: 10774036Abstract: The invention relates to a new enantioselective process for producing useful intermediates for the manufacture of NEP inhibitors or prodrugs thereof, in particular NEP inhibitors comprising a ?-amino-?-biphenyl-?-methylalkanoic acid, or acid ester, backbone.Type: GrantFiled: December 20, 2017Date of Patent: September 15, 2020Assignee: Novartis AGInventors: Florian Karl Kleinbeck-Riniker, Tobias Kapferer, Hongyong Kim, Jie Ku, Kurt Laumen, Yunzhong Li, Wei Peng, Thomas Ruch, Thierry Schlama, Yao Yang
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Publication number: 20200039935Abstract: The present disclosure relates to a method of synthesizing 5-chloro-N2-(2-isopropoxy-5-methyl-4-(piperidin-4-yl)phenyl)-N4-[2-(propane-2-sulfonyl)-phenyl]-pyrimidine-2,4-diamine (ceritinib) and/or intermediates thereof, their use as pharmaceuticals and pharmaceutical compositions and the use of intermediates for preparing ceritinib.Type: ApplicationFiled: October 8, 2019Publication date: February 6, 2020Inventors: Mark Clinton Davis, Baoqing Gong, Denis Har, Tobias Kapferer, Xuchun Zheng
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Publication number: 20180057457Abstract: The present disclosure relates to a method of synthesizing 5-chloro-N2-(2-isopropoxy-5-methyl-4-(piperidin-4-yl)phenyl)-N4-[2-(propane-2-sulfonyl)-phenyl]-pyrimidine-2,4-diamine (ceritinib) and/or intermediates thereof, their use as pharmaceuticals and pharmaceutical compositions and the use of intermediates for preparing ceritinib.Type: ApplicationFiled: March 4, 2015Publication date: March 1, 2018Applicant: Novartis AGInventors: Mark Clinton Davis, Baoqing Gong, Denis Har, Tobias Kapferer, Xuchun Zheng
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Patent number: 9375000Abstract: Arylpyrrolidines of Formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal parasite-controlling agents.Type: GrantFiled: September 13, 2011Date of Patent: June 28, 2016Assignee: Bayer Intellectual Property GmbHInventors: Jun Mihara, Mamoru Hatazawa, Daiei Yamazaki, Hidetoshi Kishikawa, Kei Domon, Hidekazu Watanabe, Norio Sasaki, Tetsuya Murata, Koichi Araki, Eiichi Shimojo, Teruyuki Ichihara, Tadashi Ishikawa, Katsuhiko Shibuya, Ulrich Görgens, Peter Bruechner, Reiner Fischer, Johannes-Rudolf Jansen, Tobias Kapferer, Simon Maechling, Michael Maue, Arnd Voerste
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Patent number: 9204645Abstract: The invention relates to compounds of the general formulae (I) and (II) in which the radicals A1, A2, A3, A4, M1, M2, M3, Q, R1, T, W1 and W2 have the meaning given in the description and to the use of the compounds for controlling animal pests. The invention furthermore relates to processes and intermediates for preparing the compounds of formula (I).Type: GrantFiled: December 17, 2012Date of Patent: December 8, 2015Assignee: BAYER INTELLECTUAL PROPERTY GMBHInventors: Michael Maue, Tobias Kapferer, Friedrich August Muehlthau, Olga Malsam
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Patent number: 9206122Abstract: Arylpyrrolidines of formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal parasite-controlling agents.Type: GrantFiled: March 12, 2013Date of Patent: December 8, 2015Assignee: BAYER INTELLECTUAL PROPERTY GMBHInventors: Reiner Fischer, Peter Bruechner, Tobias Kapferer, Kerstin Ilg, Ulrich Goergens, Arnd Voerste, Mamoru Hatazawa, Eiichi Shimojo
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Patent number: 9126945Abstract: The invention relates to compounds of the general formula (I) in which the radicals A1, A2, A3, A4, L, Q, R1, T and W have the meaning given in the description and to the use of the compounds for controlling animal pests. The invention furthermore relates to processes and intermediates for preparing the compounds of formula (I).Type: GrantFiled: March 12, 2012Date of Patent: September 8, 2015Assignee: BAYER INTELLECTUAL PROPERTY GMBHInventors: Michael Maue, Isabelle Adelt, Markus Heil, Peter Jeschke, Tobias Kapferer, Friedrich August Mühlthau, Alexander Sudau, Olga Malsam, Peter Lösel, Arnd Voerste, Ulrich Görgens
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Patent number: 9107411Abstract: The present invention relates to compounds of the general formula (I) in which R1 to R6, A, Y, X, G, n and m are each as defined in the description—and to a process for preparation thereof and to the use thereof as insecticides and acaricides.Type: GrantFiled: March 5, 2012Date of Patent: August 18, 2015Assignee: BAYER INTELLECTUAL PROPERTY GMBHInventors: Markus Heil, Eike Kevin Heilmann, Graham Holmwood, Peter Jeschke, Michael Maue, Tobias Kapferer, Matthias Riedrich, Angela Becker, Olga Malsam, Peter Lösel, Arnd Voerste, Ulrich Görgens, Roland Andree
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Patent number: 8946234Abstract: The invention relates to compounds of the general formula (I), in which the radicals A1, A2, A3, A4, Lm, Q, R1, T and U have the meaning given in the description and to the use of the compounds for controlling animal pests. In addition, the invention relates to processes and intermediates for the preparation of the compounds according to formula (I).Type: GrantFiled: October 27, 2009Date of Patent: February 3, 2015Assignee: Bayer CropScience AGInventors: Michael Maue, Isabelle Adelt, Wolfgang Giencke, Markus Heil, Peter Jeschke, Bernd-Wieland Krüger, Friedrich August Mühlthau, Alexander Sudau, Klaus Raming, Ulrich Ebbinghaus-Kintscher, Martin Adamczewski, Arnd Voerste, Ulrich Görgens, Tobias Kapferer, Mark Wilhelm Drewes, Angela Becker, Eva-Maria Franken
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Publication number: 20150025253Abstract: Arylpyrrolidines of formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal parasite-controlling agents.Type: ApplicationFiled: March 12, 2013Publication date: January 22, 2015Applicant: BAYER INTELLECTUAL PROPERTY GMBHInventors: Reiner Fischer, Peter Bruechner, Tobias Kapferer, Kerstin Ilg, Ulrich Goergens, Arnd Voerste, Mamoru Hatazawa, Eiichi Shimojo
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Publication number: 20140371240Abstract: The invention relates to compounds of the general formulae (I) and (II) in which the radicals A1, A2, A3, A4, M1, M2, M3, Q, R1, T, W1 and W2 have the meaning given in the description and to the use of the compounds for controlling animal pests. The invention furthermore relates to processes and intermediates for preparing the compounds of formula (I).Type: ApplicationFiled: December 17, 2012Publication date: December 18, 2014Inventors: Michael Maue, Tobias Kapferer, Friedrich August Muehlthau, Olga Malsam
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Patent number: 8889878Abstract: The present invention relates to halogen-substituted amide derivatives of the general formula (I) in which R1 to R6, Q1 to Q8, A, V, W, X, Y, n and m are each defined as described in the description—and to a process for preparation thereof and to the use thereof as insecticides and acaricides.Type: GrantFiled: October 27, 2010Date of Patent: November 18, 2014Assignee: Bayer CropScience AGInventors: Markus Heil, Eike Kevin Heilmann, Alexander Sudau, Tobias Kapferer, Friedrich August Mühlthau, Peter Jeschke, Arnd Voerste, Ulrich Görgens, Klaus Raming, Ulrich Ebbinghaus-Kintscher, Mark Drewes, Martin Adamczewski, Angela Becker
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Patent number: 8710242Abstract: The present invention relates to halogen-substituted amide derivatives of the general formula (I) in which R1 to R6, Q1 to Q8, A, V, W, X, Y, n and m are each defined as described in the description—and to a process for preparation thereof and to the use thereof as insecticides and acaricides.Type: GrantFiled: September 14, 2012Date of Patent: April 29, 2014Assignee: Bayer CropScience AGInventors: Markus Heil, Eike Kevin Heilmann, Alexander Sudau, Tobias Kapferer, Friedrich August Mühlthau, Peter Jeschke, Arnd Voerste, Ulrich Görgens, Klaus Raming, Ulrich Ebbinghaus-Kintscher, Mark Drewes, Martin Adamczewski, Angela Becker
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Publication number: 20140088167Abstract: The present invention relates to compounds of the general formula (I) in which R1 to R6, A, Y, X, G, n and m are each as defined in the description—and to a process for preparation thereof and to the use thereof as insecticides and acaricides.Type: ApplicationFiled: March 5, 2012Publication date: March 27, 2014Applicant: Bayer Intellectual Property GmbHInventors: Markus Heil, Eike Kevin Heilmann, Graham Holmwood, Peter Jeschke, Michael Maue, Tobias Kapferer, Matthias Reidrich, Angela Becker, Olga Malsam, Peter Losel, Arnd Voerste, Ulrich Görgens, Roland Andree
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Publication number: 20140088153Abstract: The invention relates to compounds of the general formula (I) in which the radicals A1, A2, A3, A4, L, Q, R1, T and W have the meaning given in the description and to the use of the compounds for controlling animal pests. The invention furthermore relates to processes and intermediates for preparing the compounds of formula (I).Type: ApplicationFiled: March 12, 2012Publication date: March 27, 2014Applicant: BAYER INTELLECTUAL PROPERTY GMBHInventors: Michael Maue, Isabelle Adelt, Markus Heil, Peter Jeschke, Tobias Kapferer, Friedrich August Muehlthau, Alexander Sudau, Olga Malsam, Peter Loesel, Arnd Voerste, Ulrich Goergens
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Publication number: 20140046069Abstract: Arylpyrrolidines of Formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal paracite-controlling agents.Type: ApplicationFiled: September 13, 2011Publication date: February 13, 2014Applicant: BAYER INTELLECTUAL PROPERTY GMBHInventors: Jun Mihara, Mamoru Hatazawa, Daiei Yamazaki, Hidetoshi Kishikawa, Kei Domon, Hidekazu Watanabe, Norio Sasaki, Tetsuya Murata, Koichi Araki, Eiichi Shimojo, Teruyuki Ichihara, Tadashi Ishikawa, Katsuhiko Shibuya, Ulrich Goergens, Peter Bruechner, Reiner Fischer, Johannes-Rudolf Jansen, Tobias Kapferer, Simon Maechling, Michael Maue, Arnd Voerste
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Publication number: 20130172390Abstract: The present invention relates to halogen-substituted amide derivatives of the general formula (I) in which R1 to R6, Q1 to Q8, A, V, W, X, Y, n and m are each defined as described in the description—and to a process for preparation thereof and to the use thereof as insecticides and acaricides.Type: ApplicationFiled: September 14, 2012Publication date: July 4, 2013Applicant: Bayer Intellectual Property GmbHInventors: Markus Heil, Eike Kevin Heilmann, Alexander Sudau, Tobias Kapferer, Friedrich August Mühlthau, Peter Jeschke, Arnd Voerste, Ulrich Görgens, Klaus Raming, Ulrich Ebbinghaus-Kintscher, Mark Drewes, Martin Adamczewski, Angela Becker
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Publication number: 20110301181Abstract: The invention relates to compounds of the general formula (I), in which the radicals A1, A2, A3, A4, Lm, Q, R1, T and U have the meaning given in the description and to the use of the compounds for controlling animal pests. In addition, the invention relates to processes and intermediates for the preparation of the compounds according to formula (I).Type: ApplicationFiled: October 27, 2009Publication date: December 8, 2011Applicant: Bayer CropScience AGInventors: Michael Maue, Isabelle Adelt, Wolfgang Giencke, Markus Heil, Peter Jeschke, Bernd-Wieland Krüger, Friedrich August Mühlthau, Alexander Sudau, Klaus Raming, Ulrich Ebbinghaus-Kintscher, Martin Adamczewski, Arnd Voerste, Ulrich Görgens, Tobias Kapferer, Mark Wilhelm Drewes, Angela Becker, Eva-Maria Franken
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Publication number: 20110184188Abstract: The present invention relates to a novel benzenedicarboxamide derivative and the use thereof as an insecticide having the formula (I) wherein the chemical groups W1 to W9, and R1 to R3 are as defined here-in.Type: ApplicationFiled: July 28, 2009Publication date: July 28, 2011Applicant: Bayer CropScience AGInventors: Katsuaki Wada, Yasushi Yoneta, Takuya Gomibuchi, Tetsuya Murata, Sachio Kudo, Hidetoshi Kishikawa, Katsuhiko Shibuya, Eiichi Shimojo, Akira Emoto, Yoshitaka Sato, Rüdiger Fisher, Christian Funke, Christian Arnold, Eva-Maria Franken, Olga Malsam, Erich Sanwald, Ulrich Görgens, Masashi Ataka, Udo Reckmann, Christian Paulitz, Tobias Kapferer
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Publication number: 20110105532Abstract: The present invention relates to halogen-substituted amide derivatives of the general formula (I) in which R1 to R6, Q1 to Q8, A, V, W, X, Y, n and m are each defined as described in the description—and to a process for preparation thereof and to the use thereof as insecticides and acaricides.Type: ApplicationFiled: October 27, 2010Publication date: May 5, 2011Applicant: Bayer CropScience AGInventors: Markus HEIL, Eike Kevin Heilmann, Alexander Sudau, Tobias Kapferer, Friedrich August Mühlthau, Peter Jeschke, Arnd Voerste, Ulrich Görgens, Klaus Raming, Ulrich Ebbinghaus-Kintscher, Mark Drewes, Martin Adamczewski, Angela Becker