Patents by Inventor Toshiaki Yanai

Toshiaki Yanai has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 6506913
    Abstract: A dimethylfurancarboxyanilide compound of the formula (I): wherein R1 and R2 are the same or different and each is hydrogen, (C2-C6)-alkyl, (C3-C6)-cycloalkyl, (C3-C6)-alkenyl, (C2-C6) alkynyl, (C1-C3)-halogenoalkyl, (C2-C6)-alkoxy, (C1-C6)-alkoxy-(C1-C6)-alkyl, cyano, substituted amide, (C1-C6)-alkoxy-carbonyl, benzoyl which is unsubstituted or has 1 to 2 substituents, benzoylamino which is unsubstituted or has 1 to 2 substituents; (C2-C6)-alkanoylamino, (C3-C6)-cycloalkylcarbonylamino, benzyl which is unsubstituted or has 1 to 2 substituents, phenyl which is unsubstituted or has 1 to 2 substituents, or (C1-C6)-alkoxycarbonyl-(C2-C5)-alkenylene; and R1 and R2 do not both represent hydrogen at the same time. A wood preservative containing the dimethylfurancarboxyanilide compound as an active ingredient. A method of preserving wood by applying the dimethylfurancarboxyanilide compound to wood.
    Type: Grant
    Filed: October 24, 2001
    Date of Patent: January 14, 2003
    Assignee: Sankyo Company, Limited
    Inventors: Kiyoshi Konishi, Toshiaki Yanai, Akio Saito
  • Publication number: 20020091154
    Abstract: A dimethylfurancarboxyanilide compound of the formula (I): 1
    Type: Application
    Filed: October 24, 2001
    Publication date: July 11, 2002
    Applicant: SANKYO COMPANY LIMITED
    Inventors: Kiyoshi Konishi, Toshiaki Yanai, Akio Saito
  • Patent number: 6380247
    Abstract: A dimethylfurancarboxyanilide compound of the formula (I): wherein R1 and R2 are the same or different and each is hydrogen, (C2-C6)-alkyl, (C3-C6)-cycloalkyl, (C3-C6)-alkenyl, (C2-C6) alkynyl, (C1-C3)-halogenoalkyl, (C2-C6)-alkoxy, (C1-C6)-alkoxy-(C1-C6)-alkyl, cyano, substituted amide, (C1-C6)-alkoxy-carbonyl, benzoyl which is unsubstituted or has 1 to 2 substituents, benzoylamino which is unsubstituted or has 1 to 2 substituents; (C2-C6)-alkanoylamino, (C3-C6)-cycloalkylcarbonylamino, benzyl which is unsubstituted or has 1 to 2 substituents, phenyl which is unsubstituted or has 1 to 2 substituents, or (C1-C6)-alkoxycarbonyl-(C2-C5)-alkenylene; and R1 and R2 do not both represent hydrogen at the same time. A wood preservative containing the dimethylfurancarboxyanilide compound as an active ingredient. A method of preserving wood by applying the dimethylfurancarboxyanilide compound to wood.
    Type: Grant
    Filed: December 4, 2000
    Date of Patent: April 30, 2002
    Assignee: Sankyo Company, Limited
    Inventors: Kiyoshi Konishi, Toshiaki Yanai, Akio Saito
  • Publication number: 20010000184
    Abstract: A dimethylfurancarboxyanilide compound of the formula (I): 1
    Type: Application
    Filed: December 4, 2000
    Publication date: April 5, 2001
    Applicant: Sankyo Company, Limited
    Inventors: Kiyoshi Konishi, Toshiaki Yanai, Akio Saito
  • Patent number: 5977168
    Abstract: A dimethylfurancarboxyanilide compound of the formula (I): ##STR1## wherein R.sup.1 and R.sup.2 are the same or different and each is hydrogen, (C.sub.2 -C.sub.6)-alkyl, (C.sub.3 -C.sub.6)-cycloalkyl, (C.sub.3 -C.sub.6)-alkenyl, (C.sub.2 -C.sub.6) alkynyl, (C.sub.1 -C.sub.3)-halogenoalkyl, (C.sub.2 -C.sub.6)-alkoxy, (C.sub.1 -C.sub.6)-alkoxy- (C.sub.1 -C.sub.6)-alkyl, cyano, substituted amide, (C.sub.1 -C.sub.6)-alkoxy-carbonyl, benzoyl which is unsubstituted or has 1 to 2 substituents, benzoylamino which is unsubstituted or has 1 to 2 substituents; (C.sub.2 -C.sub.6)-alkanoylamino, (C.sub.3 -C.sub.6)-cycloalkylcarbonylamino, benzyl which is unsubstituted or has 1 to 2 substituents, phenyl which is unsubstituted or has 1 to 2 substituents, or (C.sub.1 -C.sub.6)-alkoxycarbonyl-(C.sub.2 -C.sub.5)-alkenylene; and R.sup.1 and R.sup.2 do not both represent hydrogen at the same time. A wood preservative containing the dimethylfurancarboxyanilide compound as an active ingredient.
    Type: Grant
    Filed: December 29, 1997
    Date of Patent: November 2, 1999
    Assignee: Sankyo Company, Limited
    Inventors: Kiyoshi Konishi, Toshiaki Yanai, Akio Saito
  • Patent number: 5614470
    Abstract: 13-Substituted milbemycin derivatives having the formula (I): ##STR1## wherein: R.sup.1 is methyl, ethyl, isopropyl or sec-butyl;R.sup.2 is hydrogen or alkyl;X is (.alpha.-hydroxyimino- or .alpha.-alkoxyimino-substituted)-arylmethyl or (.alpha.-hydroxyimino- or .alpha.-alkoxyimino-substituted)-heterocyclylmethyl, N-substituted-aminophenyl or N-substituted-aminophenoxy;m is 0 or 1; and n is 0 or 1;are valuable as agricultural and horticultural anthelmintic, acaricidal and insecticidal agents.
    Type: Grant
    Filed: March 29, 1995
    Date of Patent: March 25, 1997
    Assignee: Sankyo Company, Limited
    Inventors: Hideo Takeshiba, Kazuo Sato, Toshiaki Yanai, Shinji Yokoi, Reiji Ichinose, Kinji Tanizawa
  • Patent number: 5530021
    Abstract: A novel hydrazine derivative and a pesticidal composition containing the hydrazine derivative as the effecting ingredient. The hydrazine derivative show high pesticidal activity against harmful pests which are resistant to known pesticides such as organophosphorus pesticides, pyrethroids, etc., especially against Lepidoptera harmful pests such as Plutella xylostella, Spodoptera litura, Cnaphalocrocis medinalis, Adoxophyes orana, etc., and is effective for controlling harmful pests in paddy field, upland field, orchard, forest or places to be kept environmentally hygienic.
    Type: Grant
    Filed: September 19, 1994
    Date of Patent: June 25, 1996
    Assignees: Nippon Kayaku Kabushiki Kaisha, Sankyo Company, Limited
    Inventors: Mikio Yanagi, Hiroyasu Sugizaki, Tetsuya Toya, Yasuhito Kato, Hidetoshi Shirakura, Tetsuo Watanabe, Yoshimi Yajima, Seiichirou Kodama, Akio Masui, Toshiaki Yanai, Yoshihisa Tsukamoto, Yoshihiro Sawada, Shinji Yokoi
  • Patent number: 5405867
    Abstract: Compounds having a 16-membered macrolide ring, and related to the milbemycins and avermectins, with substituents at positions 5.13, 25 and optionally also 23, have acaricidal, insecticidal and anthelmintic properties. They are useful for treating various pests in plants and animals.
    Type: Grant
    Filed: October 8, 1993
    Date of Patent: April 11, 1995
    Assignee: Sankyo Company, Limited
    Inventors: Kazuo Sato, Toshiaki Yanai, Takao Kinoto, Keiji Tanaka, Akira Nishida, Toshimitsu Toyama, Bruno Frei, Anthony O'Sullivan
  • Patent number: 5378726
    Abstract: A novel hydrazine derivative and a pesticidal composition containing the hydrazine derivative as the effecting ingredient. The hydrazine derivative show high pesticidal activity against harmful pests which are resistant to known pesticides such as organophosphorus pesticides, pyrethroids, etc., especially against Lepidopters harmful pests such as Plutella xylostella, Spodoptera litura, Cnaphalocrocis medinalis, Adoxophyes orana, etc., and is effective for controlling harmful pests in paddy field, upland field, orchard, forest or places to be kept environmentally hygienic.
    Type: Grant
    Filed: November 15, 1993
    Date of Patent: January 3, 1995
    Assignees: Nippon Kayaku Kabushiki Kaisha, Sankyo Company, Limited
    Inventors: Mikio Yanagi, Hiroyasu Sugizaki, Tetsuya Toya, Yasuhito Kato, Hidetoshi Shirakura, Tetsuo Watanabe, Yoshimi Yajima, Seiichirou Kodama, Akio Masui, Toshiaki Yanai, Yoshihisa Tsukamoto, Yoshihiro Sawada, Shinji Yokoi
  • Patent number: 5276033
    Abstract: Compounds having the formula (I) ##STR1## wherein: R.sup.1 is methyl, ethyl or isopropyl; R.sup.2 is alkyl, aralkyl, cycloalkyl, cycloalkylmethyl, aryl, heterocyclic, or heterocyclic-substituted thio; R.sup.3 is hydrogen, methyl or ethyl; or R.sup.2 together with R.sup.3 is --(CH.sub.2).sub.n --, wherein n is 3,4 or 5; and A is aromatic heterocyclic; and salts thereof, are valuable agricultural and horticultural anthelmintic, acaricidal and insecticidal agents.
    Type: Grant
    Filed: December 17, 1992
    Date of Patent: January 4, 1994
    Assignee: Sankyo Company, Limited
    Inventors: Toshiaki Yanai, Soji Sugai, Hideo Takeshiba, Junzo Tobitsuka, Kazuo Sato, Shinji Yokoi, Shinya Niimi, Akio Saito
  • Patent number: 5212322
    Abstract: Compounds with acaricidal, insecticidal and anthelmintic activities have the formula: ##STR1## wherein: --X--Y-- is selected from the group consisting of --CH.sub.2 --CH.sub.2 --, --CH.sub.2 --CHOH--, --CH.dbd.CH--, and --CH.sub.2 --C(.dbd.O)--;R.sup.1 is selected from the group consisting of a methyl group, an ethyl group, an isopropyl group, a sec-butyl group and groups of formula --C(CH.sub.3).dbd.CHR.sup.5 in which R.sup.5 is selected from the group consisting of a methyl group, an ethyl group and an isopropyl group;R.sup.2 represents a group of formula --(CH.sub.2).sub.n --C(R.sup.6).dbd.C(R.sup.7)(R.sup.8) in which n is 0, 1 or 2, R.sup.6 and R.sup.7 each is selected from the group consisting of a hydrogen atom and a methyl group and R.sup.8 is selected from the group consisting of a hydrogen atom, a C.sub.1-4 alkyl group, a phenyl group and a phenyl group substituted with at least one substituent selected from the group consisting of halogen, methyl and nitro substituents;R.sup.
    Type: Grant
    Filed: January 22, 1991
    Date of Patent: May 18, 1993
    Assignee: Sankyo Company, Limited
    Inventors: Takao Okazaki, Shuji Takahashi, Seigo Iwado, Keiji Tanaka, Toshiaki Yanai, Hisaki Kajino
  • Patent number: 5208349
    Abstract: 13-Hydroxy-5-ketomilbemycin derivatives are prepared by oxidizing a 5-ketomilbemycin with selenium dioxide in the presence of a lower aliphatic carboxylic acid. A range of new 13-acyloxy-5-ketomilbemycins and a method of preparing them are also disclosed.
    Type: Grant
    Filed: January 24, 1991
    Date of Patent: May 4, 1993
    Assignee: Sankyo Company, Limited
    Inventors: Kazuo Sato, Takao Kinoto, Shigeru Mio, Toshiaki Yanai
  • Patent number: 5008191
    Abstract: Compounds with acaricidal, insecticidal and anthelmintic activities have the formula: ##STR1## wherein: --X--Y-- is selected from the group consisting of --CH.sub.2 --CH.sub.2 --, --CH.sub.2 --CHOH--, --CH.dbd.CH--, and --CH.sub.2 --C(.dbd.O)--;R.sup.1 is selected from the group consisting of a methyl group, an ethyl group, an isopropyl group, a sec-butyl group and groups of formula --C(CH.sub.3).dbd.CHR.sup.5 in which R.sup.5 is selected from the group consisting of a methyl group, an ethyl group and an isopropyl group;R.sup.2 represents a group of formula --(CH.sub.2).sub.n --C(R.sup.6).dbd.C(R.sup.7)(R.sup.8) in which n is 0, 1 or 2, R.sup.6 and R.sup.7 each is selected from the group consisting of a hydrogen atom and a methyl group and R.sup.8 is selected from the group consisting of a hydrogen atom, a C.sub.1-4 alkyl group, a phenyl group and a phenyl group substituted with at least one substituent selected from the group consisting of halogen, methyl and nitro substitutents;R.sup.
    Type: Grant
    Filed: December 10, 1987
    Date of Patent: April 16, 1991
    Assignee: Sankyo Company Limited
    Inventors: Takao Okazaki, Shuji Takahashi, Seigo Iwado, Keiji Tanaka, Toshiaki Yanai, Hisaki Kajino
  • Patent number: 4963582
    Abstract: Compounds having a 16-membered macrolide ring, and related to the milbemycins and avermectins, with substituents at positions 5, 13, 25 and optionally also 23, have acaricidal, insecticidal and anthelmintic properties. They are useful for treating various pests in plants and animals.
    Type: Grant
    Filed: March 24, 1987
    Date of Patent: October 16, 1990
    Assignee: Sankyo Company Limited
    Inventors: Kazuo Sato, Toshiaki Yanai, Takao Kinoto, Keiji Tanaka, Akira Nishida, Toshimitsu Toyama, Bruno Frei, Anthony O'Sullivan
  • Patent number: 4959386
    Abstract: The present invention relates to novel compounds of the formula ##STR1## wherein R.sub.1 is hydrogen, a silyl group or an acyl group,R.sub.2 is methyl, ethyl, is propyl or sec-butyl, and R is hydrogen, unsubstituted or substituted straight chain or branched C.sub.1 -Cl.sub.18 alkyl, an unsubstituted or substituted cycloaliphatic group containing 3 to 10 carbon atoms, unsubstituted or substituted C.sub.2 -C.sub.6 alkenyl, unsubstituted or substituted C.sub.2 -C.sub.6 -alkynyl, unsubstituted or substituted phenyl or unsubstituted or substituted benzyl. These compounds posseses advantageous pesticidal properties and are suitable in particular for controlling pests in agriculture and the storage sector.
    Type: Grant
    Filed: September 28, 1988
    Date of Patent: September 25, 1990
    Assignee: Ciba-Geigy Corporation
    Inventors: Bruno Frei, Hari B. Mereyala, Anthony C. O'Sullivan, Kazuo Sato, Toshiaki Yanai
  • Patent number: 4945105
    Abstract: Derivatives of milbemycins D, A.sub.3 and A.sub.4 and of the corresponding sec-butyl compound have a halogen atom at the 13-position; at the 5-position, they have an oxygen (keto) atom, an oxime group or a substituted oxime group. They may be prepared from known compounds by any appropriate combination of halogenation, ketonization and oximation.
    Type: Grant
    Filed: December 28, 1988
    Date of Patent: July 31, 1990
    Assignee: Sankyo Company Limited
    Inventors: Kazuo Sato, Toshiaki Yanai, Noritoshi Kitano, Akira Nishida, Bruno Frei, Anthony O'Sullivan
  • Patent number: 4912090
    Abstract: 8,9 and/or 14,15 epoxidized and 5-acylated milbemycins and avermectins are prepared from the parent milbemycins and avermectins by epoxidation and acylation (in either order). They have enhanced anthelmintic, acaricidal and insecticidal activities.
    Type: Grant
    Filed: December 30, 1986
    Date of Patent: March 27, 1990
    Assignee: Sankyo Company Limited
    Inventors: Toshiaki Yanai, Kazuo Sato, Akira Nishida, Keiji Tanaka
  • Patent number: 4835290
    Abstract: 13-Hydroxy-5-ketomilbemycin derivatives are prepared by oxidizing a 5-ketomilbemycin with selenium dioxide in the presence of a lower aliphatic carboxylic acic. A range of new 13-acyloxy-5-ketomilbemycins and a method or preparing them are also disclosed.
    Type: Grant
    Filed: October 26, 1987
    Date of Patent: May 30, 1989
    Assignee: Sankyo Company, Limited
    Inventors: Kazuo Sato, Takao Kinoto, Shigeru Mio, Toshiaki Yanai
  • Patent number: 4460597
    Abstract: Pyrazole derivatives of formula (I): ##STR1## (R.sup.1 is methyl, halogen or nitro; n is 2 or 3; R.sup.2 is hydrogen, C.sub.1-4 alkyl, C.sub.3-4 alkenyl or aralkyl; R.sup.3 is C.sub.1-4 alkyl, C.sub.3-4 alkenyl or phenyl; A is C.sub.1-5 alkylene) are of use as herbicides.
    Type: Grant
    Filed: May 23, 1983
    Date of Patent: July 17, 1984
    Assignee: Sankyo Company, Limited
    Inventors: Toshiaki Yanai, Teruomi Jojima, Katsuhiko Kawakubo, Toyokuni Honma, Masahiro Shindo