Patents by Inventor Volker Schulze

Volker Schulze has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Anti-androgenic pyrrolidines with tumor-inhibiting action
    Patent number: 7601748
    Abstract: This invention relates to anti-androgenic N-[?-[3-[4-cyano-3-(trifluoromethyl)-phenyl]-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl]alkyl]-substituted pyrrolidines of general formula I, with a strongly pronounced antiproliferative profile of action; process for the production of the compounds of general formula I, pharmaceutical preparations and the use for the production of pharmaceutical agents.
    Type: Grant
    Filed: August 9, 2006
    Date of Patent: October 13, 2009
    Assignee: Bayer Schering Pharma AG
    Inventors: Arwed Cleve, Volker Schulze, Dieter Zopf, Jens Hoffmann, Andreas Reichel, Karsten Parczyk
  • Thiazolidinones, their production and use as pharmaceutical agents
    Patent number: 7511059
    Abstract: The invention relates to thiazolidinones of general formula (I) their production and use as inhibitors of polo-like kinases (Plk) for treating various diseases.
    Type: Grant
    Filed: February 2, 2006
    Date of Patent: March 31, 2009
    Assignee: Schering Ag
    Inventors: Volker Schulze, Knut Eis, Lars Wortmann, Dirk Kosemund, Olaf Prien, Gerhard Siemeister, Holger Hess-Stumpp, Uwe Eberspaecher, Damian O Arnaiz
  • Thiazolidinones, their production and use as pharmaceutical agents
    Publication number: 20070037862
    Abstract: Thiazolidinones of general formula I in which Q, A, B, X, R1 and R2 have the meanings that are indicated in the description, as well as those of general formula IA in which Q, A, B, X, R1 and R2a have the meanings that are indicated in the description, their production and use as inhibitors of the polo-like kinase (PLK) for treating various diseases as well as intermediate products for the production of thiazolidinones are described.
    Type: Application
    Filed: November 1, 2004
    Publication date: February 15, 2007
    Inventors: Gerhard Siemeister, Hans Briem, Volker Schulze, Knut Eis, Lars Wortmann, Wolfgang Schwede, Herbert Schneider, Uwe Eberspaecher, Holger Hess-Stumpp
  • Anti-androgenic pyrrolidines with tumor-inhibiting action
    Publication number: 20070021481
    Abstract: This invention relates to anti-androgenic N-[?-[3-[4-cyano-3-(trifluoromethyl)-phenyl]-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl]alkyl]-substituted pyrrolidines of general formula I, with a strongly pronounced antiproliferative profile of action; process for the production of the compounds of general formula I, pharmaceutical preparations and the use for the production of pharmaceutical agents.
    Type: Application
    Filed: August 9, 2006
    Publication date: January 25, 2007
    Inventors: Arwed Cleve, Volker Schulze, Dieter Zopf, Jens Hoffmann, Andreas Reichel, Karsten Parczyk
  • Metasubstituted thiazolidinones, their manufacture and use as a drug
    Publication number: 20070015759
    Abstract: This invention involves thiazolidinone of general formula (I) and its creation and use as inhibitors of polo like kinase (PLK) for the treatment of various diseases.
    Type: Application
    Filed: December 14, 2005
    Publication date: January 18, 2007
    Inventors: Volker Schulze, Knut Eis, Lars Wortmann, Dirk Kosemund, Olaf Prien, Gerhard Siemeister, Holger Hess-Stumpp, Uwe Eberspaecher, Dominic Brittain, Imadul Islam
  • New thiazolidinones without basic nitrogen, their production and use as pharmaceutical agents
    Publication number: 20070010565
    Abstract: The invention relates to thiazolidones of general formula (I): to their production and to their use as inhibitors of the polo-like kinase (Plk) for treating various diseases.
    Type: Application
    Filed: April 25, 2006
    Publication date: January 11, 2007
    Inventors: Olaf Prien, Volker Schulze, Knut Eis, Lars Wortmann, Dirk Kosemund, Gerhard Siemeister, Uwe Eberspaecher, Judith Guenther, Dominic Brittain
  • Thiazolidinones without basic nitrogen, their production and use as pharmaceutical agents
    Publication number: 20070010566
    Abstract: The invention relates to thiazolidones of general formula (I) as welt as to their production and to their use as inhibitors of the polo-like kinase (Plk) for treating various diseases, as welt as to intermediate products for the production of the compounds according to the invention.
    Type: Application
    Filed: April 25, 2006
    Publication date: January 11, 2007
    Inventors: Olaf Prien, Volker Schulze, Knut Eis, Lars Wortmann, Dirk Kosemund, Gerhard Siemeister, Uwe Eberspaecher, Judith Guenther, Dominic Brittain
  • Anti-androgenic pyrrolidines with tumor-inhibiting action
    Patent number: 7138421
    Abstract: This invention relates to anti-androgenic N-[?-[3-[4-cyano-3-(trifluoromethyl)-phenyl]-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl]alkyl]-substituted pyrrolidines of general formula I, with a strongly pronounced antiproliferative profile of action; process for the production of the compounds of general formula I, pharmaceutical preparations and the use for the production of pharmaceutical agents.
    Type: Grant
    Filed: May 10, 2004
    Date of Patent: November 21, 2006
    Assignee: Schring Aktiengesellschaft
    Inventors: Arwed Cleve, Volker Schulze, Dieter Zopf, Jens Hoffmann, Andreas Reichel, Karsten Parczyk
  • Thiazolidinones, their production and use as pharmaceutical agents
    Publication number: 20060223833
    Abstract: The invention relates to thiazolidinones of general formula (I) their production and use as inhibitors of polo-like kinases (Plk) for treating various diseases.
    Type: Application
    Filed: February 2, 2006
    Publication date: October 5, 2006
    Inventors: Volker Schulze, Knut Eis, Lars Wortmann, Dirk Kosemund, Olaf Prien, Gerhard Siemeister, Holger Hess-Stumpp, Uwe Eberspaecher, Damian Arnaiz
  • Thiazolidinones and the use therof as polo-like kinase inhibitors
    Publication number: 20060079503
    Abstract: Thiazolidones of general formula I in which R1, R2, R3, X and Y have the meanings that are indicated in the description, their production and use as inhibitors of polo-like kinases (PLK) for treating various diseases as well as intermediate products for the production of thiazolidones are described.
    Type: Application
    Filed: April 29, 2003
    Publication date: April 13, 2006
    Inventors: Wolfgang Schwede, Volker Schulze, Knut Eis, Bernd Buchmann, Hans Briem, Gerhard Siemeister, Ulf Boemer, Karsten Parczyk
  • Anti-androgenic pyrrolidines with tumor-inhibiting action
    Publication number: 20050159468
    Abstract: This invention relates to anti-androgenic N-[?-[3-[4-cyano-3-(trifluoromethyl)-phenyl]-5,5-dimethyl-4-oxo-2-thioxoimidazolidin-1-yl]alkyl]-substituted pyrrolidines of general formula I, with a strongly pronounced antiproliferative profile of action; process for the production of the compounds of general formula I, pharmaceutical preparations and the use for the production of pharmaceutical agents.
    Type: Application
    Filed: May 10, 2004
    Publication date: July 21, 2005
    Inventors: Arwed Cleve, Volker Schulze, Dieter Zopf, Jens Hoffmann, Andreas Reichel, Karsten Parczyk
  • Piperazine derivatives that destabilize androgen receptors
    Patent number: 6861432
    Abstract: This invention relates to new piperazine derivatives of general formula I, in which V, W, n, R, R?, i, j, Y and Z have the meaning that is indicated in the description. The compounds according to the invention are distinguished by a diazacycloalkane substituent. They have at their disposal a special action with respect to the action that destabilizes the androgen receptor and can be used, for example, for treating prostrate cancer.
    Type: Grant
    Filed: November 22, 2002
    Date of Patent: March 1, 2005
    Assignee: Schering Aktiengesellschaft
    Inventors: Arwed Cleve, Christoph Huwe, Volker Schulze, Helmut Morack, Dieter Zopf, Jens Hoffmann, Andreas Reichel
  • Piperazine derivatives that destabilize androgen receptors
    Publication number: 20040009969
    Abstract: This invention relates to new piperazine derivatives of general formula I, 1
    Type: Application
    Filed: November 22, 2002
    Publication date: January 15, 2004
    Applicant: Schering AG
    Inventors: Arwed Cleve, Christoph Huwe, Volker Schulze, Helmut Morack, Dieter Zopf, Jens Hoffmann, Andreas Reichel
  • Fairy tale figure
    Patent number: D275090
    Type: Grant
    Filed: May 18, 1982
    Date of Patent: August 14, 1984
    Inventor: Volker Schulze-Wechsungen