Patents by Inventor Willy Kinzy

Willy Kinzy has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20070031336
    Abstract: The present invention provides compounds of formula (I) wherein X and Y represent CH, CH2 or a divalent or trivalent heteroatom under the proviso that X and Y are not simultaneously CH or CH2; m and o represent independently of each other 0 or 1, with the proviso that if m is 0 then the dotted line between Y and the neighboring C atom represents a bond and Y is CH or a trivalent heteroatom, if m is 1 then the dotted line between Y and the neighboring C atom is absent and Y is CH2 or a divalent heteroatom, if o is 0 then the dotted line between X and the neighboring C atom represents a bond and X is CH or a trivalent heteroatom, if o is 1 then the dotted line between X and the neighboring C atom is absent and X is CH2 or a divalent heteroatom; A represents (CH3CR4)p and Q represents (CR9R10)n; n and p represent independently of each other 0 or 1; R6, R7, R13 and R14 denote independently of each other hydrogen, halogen, (C1-4)alkyl, (C1-4)alkylSO2, SO3H, carboxy, (C1-4)alkoxy carbonyl, (C1-4)alkoxy, OH or NR15R
    Type: Application
    Filed: August 17, 2004
    Publication date: February 8, 2007
    Inventors: Yves Auberson, Hans-Ulrich Gremlich, Martin Hintersteiner, Willy Kinzy, Rainer Kneuer
  • Patent number: 6723831
    Abstract: Polyamide conjugates comprising either (a) a xenoantigenic group; or (b) a biologically active group and a macromolecular, macro- or microscopic entity; bound to a polyamide backbone, processes for their preparation and the use of these conjugates in therapeutic compositions.
    Type: Grant
    Filed: April 16, 2002
    Date of Patent: April 20, 2004
    Assignee: Novartis AG
    Inventors: Rudolf Duthaler, Andreas Katopodis, Willy Kinzy, Reinhold Öhrlein, Gebhard Thoma
  • Publication number: 20020164347
    Abstract: Polyamide conjugates comprising either (a) a xenoantigenic group; or (b) a biologically active group and a macromolecular, macro- or microscopic entity; bound to a polyamide backbone, processes for their preparation and the use of these conjugates in therapeutic compositions.
    Type: Application
    Filed: April 16, 2002
    Publication date: November 7, 2002
    Inventors: Rudolf Duthaler, Andreas Katopodis, Willy Kinzy, Reinhold Ohrlein, Gebhard Thoma
  • Patent number: 6399071
    Abstract: Polyamide conjugates comprising either (a) a xenoantigenic group; or (b) a biologically active group and a macromolecular, macro- or microscopic entity, bound to a polyamide backbone, processes for their preparation and the use of these conjugates in therapeutic compositions.
    Type: Grant
    Filed: October 14, 1999
    Date of Patent: June 4, 2002
    Assignee: Novartis AG
    Inventors: Rudolf Duthaler, Andreas Katopodis, Willy Kinzy, Reinhold Öhrlein, Gebhard Thoma
  • Patent number: 5508390
    Abstract: Diterpenes of the formula I ##STR1## in which R.sup.1 is --CH.sub.2 --C(CH.sub.3).dbd.CH--R.sup.3 or --CH.sub.2 --CH(CH.sub.3)--CH.sub.2 --R.sup.3,R.sup.3 is --CH.sub.2 OH, --CHO, --COOH or --COOR.sup.4,R.sup.4 is alkyl having 1 to 5 C atoms,A is ##STR2## and R.sup.2 is H, pentoses, hexoses, di-/oligosaccharides or amino sugars,are suitable for production of medicaments having immunomodulatory action, in particular stimulating T-cells.
    Type: Grant
    Filed: February 15, 1991
    Date of Patent: April 16, 1996
    Assignee: Merck Patent Gesellschaft mit Beschrankter Haftung
    Inventors: Hans-Eckart Radunz, Michael Wolf, Manfred Baumgarth, Willy Kinzy, Gerd-Albrecht Luckenbach
  • Patent number: 5371203
    Abstract: The invention relates to a process for the stereoselective preparation of .beta.-L-fucopyranosyl phosphates via the trichloroacetimidates of protected L-fucose and the synthesis and purification of very pure GDP-fucose from the .beta.-L-fucopyranosyl phosphates.
    Type: Grant
    Filed: January 31, 1992
    Date of Patent: December 6, 1994
    Assignee: Merck Patent Gesellschaft mit beschrankter Haftung
    Inventors: Richard R. Schmidt, Karl-Heinz Jung, Barbara Spahngehl, Willy Kinzy, Jurgen Hemberger
  • Patent number: 5319077
    Abstract: The invention relates to a new process for the stereoselective preparation of Gal-.alpha.(1-3)/Gal-.beta.(1-4)/GlcNac trisaccharides of the formula ##STR1## and of .beta.(1-3)-linked oligolactosamines of the formula ##STR2## via partially alkylated glycals of the formula ##STR3## and other new intermediate products, wherein, depending on the formula, R is H, R'CH.sub.2 --, or allyl,R.sup.1 is H, R'CH.sub.2 --, allyl or R'CO--,R' is H, C.sub.1 to C.sub.3 -alkyl or (un)substituted phenyl,S is a spacer, preferably of the formula --(CH.sub.2).sub.n --COOR'',R'' is alkyl having 1 to 4 C atoms,X is N.sub.3 or --NHCOCH.sub.3,X is N.sub.3 or --NHCOCH.sub.3,Y is .beta.-OSiR.sub.2.sup.3 or .alpha.-OC(.dbd.NH)CCl.sub.3,R.sup.2 is C.sub.1 or C.sub.4 -alkyl or phenyl andm and n are integers from 1 to 4 or 4 to 12 respectively.
    Type: Grant
    Filed: June 12, 1992
    Date of Patent: June 7, 1994
    Assignee: Merck Patent Gesellschaft mit beschrankter Haftung
    Inventor: Willy Kinzy