Patents by Inventor Yasuaki ANAMI

Yasuaki ANAMI has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • LINKERS FOR ANTIBODY DRUG CONJUGATES
    Publication number: 20240059647
    Abstract: In one aspect, the present disclosure provides compounds of the formula: wherein the variables are as defined herein. In another aspect, the present disclosure provides compounds of the formula: wherein the variables are as defined herein. In another aspect, the present disclosure also provides methods of preparing the compounds disclosed herein. In another aspect, the present disclosure provides antibody drug conjugates comprising compounds of the present disclosure. In another aspect, the present disclosure also provides pharmaceutical compositions and methods of use of the compounds and anti-body drug conjugates disclosed herein.
    Type: Application
    Filed: February 23, 2023
    Publication date: February 22, 2024
    Inventors: Kyoji TSUCHIKAMA, Yasuaki ANAMI, Chisato TSUCHIKAMA, Ningyang ZHANG, Zhiqiang AN
  • Linkers for antibody drug conjugates
    Patent number: 11629122
    Abstract: In one aspect, the present disclosure provides compounds of the formula (I): wherein the variables are as defined herein. In another aspect, the present disclosure provides compounds of the formula (V): wherein the variables are as defined herein. In another aspect, the present disclosure also provides methods of preparing the compounds disclosed herein. In another aspect, the present disclosure provides antibody drug conjugates comprising compounds of the present disclosure. In another aspect, the present disclosure also provides pharmaceutical compositions and methods of use of the compounds and anti-body drug conjugates disclosed herein.
    Type: Grant
    Filed: May 24, 2018
    Date of Patent: April 18, 2023
    Assignee: THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM
    Inventors: Kyoji Tsuchikama, Yasuaki Anami, Chisato Tsuchikama, Ningyang Zhang, Zhiqiang An
  • LINKERS FOR ANTIBODY DRUG CONJUGATES
    Publication number: 20200115326
    Abstract: In one aspect, the present disclosure provides compounds of the formula (I): wherein the variables are as defined herein. In another aspect, the present disclosure provides compounds of the formula (V): wherein the variables are as defined herein. In another aspect, the present disclosure also provides methods of preparing the compounds disclosed herein. In another aspect, the present disclosure provides antibody drug conjugates comprising compounds of the present disclosure. In another aspect, the present disclosure also provides pharmaceutical compositions and methods of use of the compounds and anti-body drug conjugates disclosed herein.
    Type: Application
    Filed: May 24, 2018
    Publication date: April 16, 2020
    Inventors: Kyoji TSUCHIKAMA, Yasuaki ANAMI, Chisato TSUCHIKAMA, Ningyang ZHANG, Zhiqiang AN