Patents by Inventor Yolanda Cancho-Grande

Yolanda Cancho-Grande has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Publication number: 20250099600
    Abstract: The present invention relates to active metabolites of inactive precursor compounds of kinesin spindle protein inhibitors having at least one —COOH group.
    Type: Application
    Filed: August 29, 2024
    Publication date: March 27, 2025
    Inventors: Hans-Georg LERCHEN, Anne-Sophie REBSTOCK, Yolanda CANCHO GRANDE, Leo MARX, Beatrix STELTE-LUDWIG, Carsten TERJUNG, Christoph MAHLERT, Simone GREVEN, Anette SOMMER, Sandra BERNDT
  • Publication number: 20250066332
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3a, R3b, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: November 13, 2024
    Publication date: February 27, 2025
    Inventors: Alexander Arlt, Werner Hallenbach, Hans-Georg Schwarz, Martin Fuesslein, Heinz-Juergen Wroblowsky, Marc Linka, Sascha Eilmus, Kerstin Ilg, Ulrich Goergens, Arunas Jonas Damijonaitis, Yolanda Cancho Grande, Ulrich Ebbinghaus-Kintscher, Peter Jeschke, Weijie Ha, Iring Heisler, Andreas Turberg
  • Patent number: 12187705
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3a, R3b, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Grant
    Filed: April 10, 2019
    Date of Patent: January 7, 2025
    Assignee: BAYER AKTIENGESELLSCHAFT
    Inventors: Alexander Arlt, Werner Hallenbach, Hans-Georg Schwarz, Martin Fuesslein, Heinz-Juergen Wroblowsky, Marc Linka, Sascha Eilmus, Kerstin Ilg, Ulrich Goergens, Arunas Jonas Damijonaitis, Yolanda Cancho Grande, Ulrich Ebbinghaus-Kintscher, Peter Jeschke, Weijie Ha, Iring Heisler, Andreas Turberg
  • Patent number: 12171229
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Grant
    Filed: August 11, 2023
    Date of Patent: December 24, 2024
    Assignee: BAYER AKTIENGESELLSCHAFT
    Inventors: Alexander Arlt, Werner Hallenbach, Hans-Georg Schwarz, Martin Fuesslein, Heinz-Juergen Wroblowsky, Estella Buscato Arsequell, Marc Linka, Kerstin Ilg, Arunas Jonas Damijonaitis, Ulrich Ebbinghaus-Kintscher, Ulrich Goergens, Yolanda Cancho Grande, Peter Jeschke, Joachim Telser, Iring Heisler, Andreas Turberg
  • Publication number: 20240417391
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3a, R3b, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: August 28, 2024
    Publication date: December 19, 2024
    Inventors: Alexander ARLT, Werner HALLENBACH, Hans-Georg SCHWARZ, Martin FUESSLEIN, Heinz-Juergen WROBLOWSKY, Marc LINKA, Ulrich GOERGENS, Kerstin ILG, Ulrich EBBINGHAUS-KINTSCHER, Yolanda CANCHO GRANDE, Arunas Jonas DAMIJONAITIS, Sascha EILMUS, Andreas TURBERG, Iring HEISLER
  • Patent number: 12144865
    Abstract: The present invention relates to novel binder-prodrug conjugates (APDCs) where binders are conjugated with inactive precursor compounds of kinesin spindle protein inhibitors, and to antibody-drug conjugates ADCs and to processes for producing these APDCs and ADCs.
    Type: Grant
    Filed: July 13, 2021
    Date of Patent: November 19, 2024
    Assignee: BAYER PHARMA AKTIENGESELLSCHAFT
    Inventors: Hans-Georg Lerchen, Anne-Sophie Rebstock, Yolanda Cancho Grande, Leo Marx, Beatrix Stelte-Ludwig, Carsten Terjung, Christoph Mahlert, Simone Greven, Anette Sommer, Sandra Berndt
  • Publication number: 20240368125
    Abstract: The present invention relates to novel pyrazinyl-triazole compounds of the general formula (I), in which the structural elements X, R1, R2, R31, R31 and R4 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: August 19, 2022
    Publication date: November 7, 2024
    Inventors: Robin Maximilian BAER, Yolanda CANCHO GRANDE, Martin FÙßLEIN, Peter JESCHKE, Hans-Georg SCHWARZ, Joachim TELSER, Philipp WINTER, Ulrich EBBINGHAUS-KINTSCHER, Peter LOESEL, Marc LINKA, Arunas DAMIJONAITIS, Andreas TURBERG, Iring HEISLER
  • Patent number: 12116357
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3a, R3b, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Grant
    Filed: April 15, 2019
    Date of Patent: October 15, 2024
    Assignee: Bayer Aktiengesellschaft
    Inventors: Alexander Arlt, Werner Hallenbach, Hans-Georg Schwarz, Martin Fuesslein, Heinz-Juergen Wroblowsky, Marc Linka, Ulrich Goergens, Kerstin Ilg, Ulrich Ebbinghaus-Kintscher, Yolanda Cancho Grande, Arunas Jonas Damijonaitis, Sascha Eilmus, Andreas Turberg, Iring Heisler
  • Publication number: 20240294533
    Abstract: The invention relates to novel compounds of the formula (I) in which A1, A3, X, R1, R3, R4, R6, R7, R8 and n have the definitions given above, to the use thereof as acaricides and/or insecticides for controlling animal pests and to processes and intermediates for preparation thereof.
    Type: Application
    Filed: May 10, 2022
    Publication date: September 5, 2024
    Inventors: Ruediger FISCHER, Steffen MUELLER, Matthieu WILLOT, Elke HELLWEGE, Marc LINKA, Peter LOESEL, Nina KAUSCH-BUSIES, Yolanda CANCHO GRANDE, Yeshua SEMPERE MOLINA, Sascha EILMUS, Kerstin ILG, Ulrich GOERGENS
  • Publication number: 20240254121
    Abstract: The present invention relates to novel alkylamide substituted, annulated imidazole derivatives of the general formula (I), in which the structural elements A1; A2, A3, A4, R1, R2, R3 and R4 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: May 2, 2022
    Publication date: August 1, 2024
    Inventors: Yolanda Cancho Grande, Martin Füßlein, Peter Jeschke, Steffen Müller, Hans-Georg Schwarz, Joachim Telser, Philipp Winter, Ulrich Ebbinghaus-Kintscher, Peter Lösel, Andreas Turberg, Iring Heisler, Robin Maximilian Bär, Arunas Jonas Damijonaitis
  • Patent number: 11864557
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Grant
    Filed: September 29, 2022
    Date of Patent: January 9, 2024
    Assignee: BAYER AKTIENGESELLSCHAFT
    Inventors: Alexander Arlt, Werner Hallenbach, Hans-Georg Schwarz, Martin Fuesslein, Heinz-Juergen Wroblowsky, Estella Buscato Arsequell, Marc Linka, Kerstin Ilg, Arunas Jonas Damijonaitis, Ulrich Ebbinghaus-Kintscher, Ulrich Goergens, Yolanda Cancho Grande, Peter Jeschke, Joachim Telser, Iring Heisler, Andreas Turberg
  • Publication number: 20230399411
    Abstract: The invention relates to specific Antibody-Drug-Conjugates (ADCs) with KSP inhibitors and anti-CD123-antibodies, to the use of these conjugates for the treatment and/or prophylaxis of diseases and to the use of these conjugates for preparing medicaments for treatment and/or prevention of diseases, in particular hyperproliferative and/or angiogenic disorders such as, for example, cancer diseases. Such treatments can be carried out as monotherapy or else in combination with other medicaments or further therapeutic measures.
    Type: Application
    Filed: June 16, 2023
    Publication date: December 14, 2023
    Inventors: Hans-Georg LERCHEN, Anne-Sophie REBSTOCK, Yolanda CANCHO GRANDE, Sven WITTROCK, Beatrix STELTE-LUDWIG, Dennis KIRCHHOFF, Christoph MAHLERT, Simone GREVEN, Stephan MÄRSCH
  • Publication number: 20230389550
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: August 11, 2023
    Publication date: December 7, 2023
    Inventors: Alexander ARLT, Werner HALLENBACH, Hans-Georg SCHWARZ, Martin FUESSLEIN, Heinz-Juergen WROBLOWSKY, Estella BUSCATO ARSEQUELL, Marc LINKA, Kerstin ILG, Arunas Jonas DAMIJONAITIS, Ulrich EBBINGHAUS-KINTSCHER, Ulrich GOERGENS, Yolanda CANCHO GRANDE, Peter JESCHKE, Joachim TELSER, Iring HEISLER, Andreas TURBERG
  • Patent number: 11806404
    Abstract: The invention relates to site specific homogeneous binder drug conjugates of kinesin spindle protein inhibitors, to active metabolites of these conjugates, to processes for preparing these conjugates, to the use of these conjugates for the treatment and/or prophylaxis of diseases and to the use of these conjugates for preparing medicaments for treatment and/or prevention of diseases, in particular hyperproliferative and/or angiogenic disorders such as, for example, cancer diseases. Such treatments can be carried out as monotherapy or else in combination with other medicaments or further therapeutic measures.
    Type: Grant
    Filed: February 3, 2021
    Date of Patent: November 7, 2023
    Assignee: BAYER PHARMA AKTIENGESELLSCHAFT
    Inventors: Hans-Georg Lerchen, Yolanda Cancho Grande, Beatrix Stelte-Ludwig, Anette Sommer, Christoph Mahlert, Anne-Sophie Rebstock, Simone Greven, Nils Griebenow, Jan Tebbe, Oliver Kensch
  • Publication number: 20230348432
    Abstract: The present invention relates to novel heteroaryl-triazole compounds of the general formula (I), in which the structural elements X, R1, R2, R3 and R4 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: May 5, 2021
    Publication date: November 2, 2023
    Inventors: Peter JESCHKE, Martin FUESSLEIN, Hans-Georg SCHWARZ, Joachim TELSER, Yolanda CANCHO GRANDE, Alexander ARLT, Steffen MUELLER, Ulrich EBBINGHAUS-KINTSCHER, Peter LOESEL, Marc LINKA, Arunas Jonas DAMIJONAITIS, Iring HEISLER, Andreas TURBERG, Oleksandr MANDZHULO
  • Publication number: 20230247994
    Abstract: The invention relates to novel compounds of the formula (I) in which R1, R2, R3, R4, R5, R6, R7, Y, Z, n and m have the definitions given above, to the use thereof as acaricides and/or insecticides for controlling animal pests, and to methods and intermediates for the preparation thereof.
    Type: Application
    Filed: June 28, 2021
    Publication date: August 10, 2023
    Inventors: Ruediger FISCHER, Steffen MUELLER, Yeshua SEMPERE MOLINA, Yolanda CANCHO GRANDE, Matthieu WILLOT, Elke HELLWEGE, Marc LINKA, Peter LOESEL, Olga MALSAM
  • Publication number: 20230242513
    Abstract: The present invention relates to novel heteroaryl-substituted pyrazine derivatives of the general formula (I), in which the structural elements R1, R2, R3, R4, R5 and R6 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: June 23, 2021
    Publication date: August 3, 2023
    Inventors: Iring HEISLER, Andreas TURBERG, Joachim TELSER, Alexander ARLT, Peter JESCHKE, Hans-Georg SCHWARZ, Martin FUESSLEIN, Yolanda CANCHO-GRANDE, Peter LOESEL, Ulrich EBBINGHAUS-KINTSCHER, Bing Ashley Liang O'DOWD, Melanie ARMENAT
  • Publication number: 20230148601
    Abstract: The present invention relates to novel heteroaryl-triazole compounds of the general formula (I), in which the structural elements X, Y, R1, R2, R3a, R3b, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: February 15, 2021
    Publication date: May 18, 2023
    Inventors: Alexander ARLT, Yolanda CANCHO GRANDE, Martin FUESSLEIN, Martin HAHN, Peter JESCHKE, Steffen MUELLER, Hans-Georg SCHWARZ, Joachim TELSER, Ulrich EBBINGHAUS-KINTSCHER, Marc LINKA, Peter LOESEL, Arunas Jonas DAMIJONAITIS, Iring HEISLER, Andreas TURBERG
  • Patent number: 11643469
    Abstract: The invention relates to specific Antibody-Drug-Conjugates (ADCs) with KSP inhibitors and anti-CD123-antibodies, to the use of these conjugates for the treatment and/or prophylaxis of diseases and to the use of these conjugates for preparing medicaments for treatment and/or prevention of diseases, in particular hyperproliferative and/or angiogenic disorders such as, for example, cancer diseases. Such treatments can be carried out as monotherapy or else in combination with other medicaments or further therapeutic measures.
    Type: Grant
    Filed: April 29, 2022
    Date of Patent: May 9, 2023
    Assignee: BAYER PHARMA AKTIENGESELLSCHAFT
    Inventors: Hans-Georg Lerchen, Anne-Sophie Rebstock, Yolanda Cancho Grande, Sven Wittrock, Beatrix Stelte-Ludwig, Dennis Kirchhoff, Christoph Mahlert, Simone Greven, Stephan Märsch
  • Publication number: 20230063447
    Abstract: The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements Y, Q1, Q2, R1, R2, R3, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.
    Type: Application
    Filed: September 29, 2022
    Publication date: March 2, 2023
    Inventors: Alexander ARLT, Werner HALLENBACH, Hans-Georg SCHWARZ, Martin FUESSLEIN, Heinz-Juergen WROBLOWSKY, Estella BUSCATO ARSEQUELL, Marc LINKA, Kerstin ILG, Arunas Jonas DAMIJONAITIS, Ulrich EBBINGHAUS-KINTSCHER, Ulrich GOERGENS, Yolanda CANCHO GRANDE, Peter JESCHKE, Joachim TELSER, Iring HEISLER, Andreas TURBERG