Plural Ring Nitrogens In The Hetero Ring Patents (Class 504/168)
  • Patent number: 10501435
    Abstract: Disclosed are new small molecules having a substituted quinazoline core structure and the uses thereof for modulating glucocerebrosidase activity. Also disclosed are pharmaceutical compositions comprising the small molecules or activated glucocerebrosidase conjugated to the small molecules, which compositions may be administered in methods of treating diseases or disorders associated with glucocerebrosidase activity, including neurological diseases and disorders such as Gaucher's disease and Parkinson's disease.
    Type: Grant
    Filed: October 30, 2018
    Date of Patent: December 10, 2019
    Assignee: Northwestern University
    Inventors: Dimitri Krainc, Richard B. Silverman, Jianbin Zheng
  • Patent number: 10167270
    Abstract: Disclosed are new small molecules having a substituted quinazoline core structure and the uses thereof for modulating glucocerebrosidase activity. Also disclosed are pharmaceutical compositions comprising the small molecules or activated glucocerebrosidase conjugated to the small molecules, which compositions may be administered in methods of treating diseases or disorders associated with glucocerebrosidase activity, including neurological diseases and disorders such as Gaucher's disease and Parkinson's disease.
    Type: Grant
    Filed: June 30, 2016
    Date of Patent: January 1, 2019
    Assignee: Northwestern University
    Inventors: Dimitri Krainc, Richard B. Silverman, Jianbin Zheng
  • Patent number: 10015967
    Abstract: A crystalline form of isoxadifen-ethyl of formula (I), the crystal preparation process, the analyses of the crystal through various analytical methods and using the crystal to prepare stable agrochemical formulation. The invention also describes the use of various solvents towards the crystalline form preparation conditions.
    Type: Grant
    Filed: October 29, 2015
    Date of Patent: July 10, 2018
    Assignee: Rotam Agrochem International Company Limited
    Inventor: James Timothy Bristow
  • Patent number: 9434695
    Abstract: The present invention relates to the field of medicine, provided herein are novel nitrogenous heterocyclic compounds, their preparation methods and their uses as drugs, especially for treatment and prevention of tissue fibrosis. Also provided herein are pharmaceutically acceptable compositions comprising the nitrogenous heterocyclic compounds and the uses of the compositions in the treatment of human or animal tissue fibrosis, especially for human or animal renal interstitial fibrosis, glomerular sclerosis, liver fibrosis, pulmonary fibrosis, peritoneal fibrosis, myocardial fibrosis, dermatofibrosis, postsurgical adhesion, benign prostatic hyperplasia, skeletal muscle fibrosis, scleroderma, multiple sclerosis, pancreatic fibrosis, cirrhosis, myosarcoma, neurofibroma, pulmonary interstitial fibrosis, diabetic nephropathy, alzheimer disease or vascular fibrosis.
    Type: Grant
    Filed: July 18, 2013
    Date of Patent: September 6, 2016
    Assignee: SUNSHINE LAKE PHARMA CO., LTD
    Inventors: Yingjun Zhang, Jiancun Zhang, Xiaojun Wang, Runfeng Lin, Shengtian Cao, Zhaohe Wang, Jing Li
  • Patent number: 9334246
    Abstract: Disclosed herein are triazine compounds and methods of making and using thereof to treat malaria, provide chemoprophylaxis, and/or treat or inhibit infection by one or more Plasmodium spp.
    Type: Grant
    Filed: March 13, 2014
    Date of Patent: May 10, 2016
    Assignee: The United States of America, as represented by the Secretary of the Army, on behalf of the Walter Reed Army Institute of Research
    Inventors: Richard J. Sciotti, Gregory A. Reichard, Kristina M. Pannone, Victor E. Zottig
  • Patent number: 9066516
    Abstract: There is a need for a selective, low-risk herbicide that can be used to control weeds in cereal cultures and turf. The present invention discloses that a bacterial secondary metabolite, thaxtomin and optionally another herbicide is an effective herbicide on broadleaved, sedge and grass weeds. Thaxtomin A and structurally similar compounds can be used as natural herbicides to control the germination and growth of weeds in cereal, turf grass, Timothy grass and pasture grass cultures with no phytotoxicity to these crops. As a natural, non-toxic compound, thaxtomin can be used as a safe alternative for weed control in both conventional and organic farming and gardening systems.
    Type: Grant
    Filed: March 15, 2013
    Date of Patent: June 30, 2015
    Assignee: Marrone Bio Innovations, Inc.
    Inventors: Marja Koivunen, Pamela Marrone, Louis Boddy
  • Publication number: 20150119239
    Abstract: The present invention related to an agrochemical composition comprising at least one protoporphyrinogen-IX oxidase inhibitor as defined in the claims and description and at least one inhibitor of complex II of the respiratory chain as defined in the claims and description. The invention further relates to the use of this composition for controlling undesired vegetation, for the desiccation and/or defoliation of plants, for controlling phytopathogenic fungi and for increasing the health of plants. The invention further relates to a method for controlling undesired vegetation, to a method for the desiccation and/or defoliation of plants, to a method for controlling phytopathogenic fungi and to a method for increasing the health of plants by using said composition.
    Type: Application
    Filed: February 27, 2013
    Publication date: April 30, 2015
    Inventors: Markus Gewehr, Cyrill Zagar, Scott Peoples
  • Publication number: 20150051075
    Abstract: The present invention relates to the use of an agrochemical composition comprising at least one specific herbicide and at least one specific fungicide for controlling undesired vegetation in soybean cultures and for the desiccation and/or defoliation of soybeans. The invention further relates to a method for controlling undesired vegetation in soybean cultures and to a method for the desiccation and/or defoliation of soybean plants.
    Type: Application
    Filed: February 27, 2013
    Publication date: February 19, 2015
    Inventors: Markus Gewehr, Cyrill Zagar, Scott Peoples, Aldo Merotto, JR., Ribas Vidal, Sebastiao Carneiro Guimaraes, Michelangelo Muzell Trezzi, Fabiane Pinto Lamego
  • Publication number: 20150018215
    Abstract: The present invention relates to the use of an agrochemical composition comprising at least one specific herbicide and at least one specific fungicide for controlling undesired vegetation in cereal cultures and for the desiccation and/or defoliation of cereals. The invention further relates to a method for controlling undesired vegetation in cereal cultures and to a method for the desiccation and/or defoliation of cereal plants.
    Type: Application
    Filed: February 27, 2013
    Publication date: January 15, 2015
    Inventors: Markus Gewehr, Cyrill Zagar, Scott Peoples, Aldo Merotto, JR., Ribas Vidal, Sebastiao Carneiro Guimaraes, Michelangelo Muzell Trezzi, Fabiane Pinto Lamego
  • Patent number: 8722580
    Abstract: Disclosed are: a substance which has an activity of inhibiting the intracellular signaling from a plant-derived cytokinin receptor and which can control the growth or differentiation of a plant. Also, disclose is a method for searching for a chemical substance capable of promoting the growth of a root of a plant, which comprises measuring the level of intracellular signaling from the receptor in a system where a cell having the receptor is contacted with a chemical substance having an agonistic activity on the receptor and a substance to be tested, comparing the level of intracellular signaling measured in the preceding step with a level of intracellular signaling measured in the absence of the chemical substance, and determining the chemical substance as being a chemical substance capable of promoting the growth of a root of a plant based on the difference obtained by the comparison; and others.
    Type: Grant
    Filed: November 22, 2007
    Date of Patent: May 13, 2014
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Asako Nagasawa, Yuto Arata, Hideki Uneme
  • Publication number: 20110224081
    Abstract: The invention relates to compositions useful in the field of agricultural chemistry and methods for making and using the compositions. The compositions include (i) a permeabilizing agent, and (ii) a active component, for example, a pesticide or plant growth regulator, and can include additional components as well, for example, flow agents. The permeabilizing agent, or a mixture of permeabilizing agents, acts as an adjuvant to the active component or chemicals to improve the degree of efficacy of the active component or speed of action of the active component. The permeabilizing agents are typically one or more chelating agents, cationic materials, anionic materials, and zwitterionic materials, and include polyphosphate salts. Examples of cationic materials include polyamines such as ethylenediamine and quaternary ammonium salts. The active components can be pesticides, herbicides, insecticides, fungicides, virucides, bacteriocides, and acaricides.
    Type: Application
    Filed: April 11, 2011
    Publication date: September 15, 2011
    Applicant: CJB INDUSTRIES
    Inventor: David Miles
  • Patent number: 7407914
    Abstract: The present invention relates to an herbicide composition comprising, as active ingredients, a uracil compound represented by the following formula (I): wherein Z represents halogen or cyano; A represents oxygen, sulfur or NH; R1 represents hydroxyl, C1-C7 alkoxy or others, and R2 represents hydrogen or methyl, and one or more compounds selected from the group consisting of N-(7-fluoro-3,4-dihydro-3-oxo-4-prop-2-ynyl-2H-1,4-benzoxazin-6-yl)cyclohex-1-ene-1,2-dicarboxamide and N-[2,4-dichloro-5-[4-(difluoromethyl)-4,5-dihydro-3-methyl-5-oxo-1H-1,2,4-triazol-1-yl]phenyl]methanesulfonamide; and a method for controlling weeds which comprises applying an effective amounts of said herbicide composition to weeds. According to the invention, particularly weeds in orchards, soybean fields and non-crop lands can be effectively controlled.
    Type: Grant
    Filed: October 23, 2006
    Date of Patent: August 5, 2008
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Nobuaki Mito, Shinsuke Shibuya
  • Patent number: 7205260
    Abstract: The present invention relates to an herbicide composition comprising, as active ingredients, a uracil compound represented by the following formula (I): wherein Z represents halogen or cyano; A represents oxygen, sulfur or NH; R1 represents hydroxyl, C1–C7 alkoxy or others, and R2 represents hydrogen or methyl, and one or more compounds selected from the group consisting of N-(7-fluoro-3,4-dihydro-3-oxo-4-prop-2-ynyl-2H-1,4-benzoxazin-6-yl)cyclohex-1-ene-1,2-dicarboxamide and N-[2,4-dichloro-5-[4-(difluoromethyl)-4,5-dihydro-3-methyl-5-oxo-1H-1,2,4-triazol-1-yl]phenyl]methanesulfonamide; and a method for controlling weeds which comprises applying an effective amounts of said herbicide composition to weeds. According to the invention, particularly weeds in orchards, soybean fields and non-crop lands can be effectively controlled.
    Type: Grant
    Filed: April 26, 2002
    Date of Patent: April 17, 2007
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Nobuaki Mito, Shinsuke Shibuya
  • Publication number: 20040138063
    Abstract: A stem/leaf desiccant for crop plants which comprises as an active ingredient, a compound of formula (I): 1
    Type: Application
    Filed: November 3, 2003
    Publication date: July 15, 2004
    Inventor: Nobuaki Mito
  • Patent number: 6683028
    Abstract: The invention relates to novel guanidine derivatives of the formula (I) in which A, R1, R2, R3 and Z are as defined in the description, to a process for their preparation and to their use for controlling animal pests.
    Type: Grant
    Filed: August 17, 2001
    Date of Patent: January 27, 2004
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Wagner, Christoph Erdelen, Andreas Turberg, Norbert Mencke, Olaf Hansen
  • Patent number: 6544927
    Abstract: The invention provides methods and compositions for reducing defoliation of plants and trees. Preferably, the methods and compositions of the invention reduce defoliation associated with the application of abscission agents or herbicides to plants and trees.
    Type: Grant
    Filed: June 29, 2001
    Date of Patent: April 8, 2003
    Assignee: University of Florida
    Inventor: Jacqueline Kay Burns
  • Patent number: 6239074
    Abstract: A substituted 3-phenyluracil of the formula I where X1 and X2 are each oxygen; W is —C(R8)=X5, where X5 is oxygen, sulfur, or a radical —NR14; R14 is hydroxyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, cycloalkenyloxy, haloalkoxy, haloalkenyloxy, hydroxyalkoxy, cyanoalkoxy, cycloalkylalkoxy, alkoxyalkoxy, alkoxyalkenyloxy, alkylcarbonyloxy, haloalkylcarbonyloxy, alkylcarbamoyloxy, haloalkylcarbamoyloxy, alkoxycarbonylalkoxy, alkylthioalkoxy, dialkylaminoalkoxy, R8 is hydrogen, cyano or alkyl; R1 is halogen or cyano; R2 is hydrogen or halogen; R3 is hydrogen or alkyl; R4 is cyano, alkyl or haloalkyl; R5 is hydrogen, halogen or alkyl; or a salt or enol ether of a compound I wherein R3 is hydrogen, or its tautomeric forms, for the desiccation and defoliation of plants or as an insecticide or herbicide.
    Type: Grant
    Filed: January 3, 1997
    Date of Patent: May 29, 2001
    Assignee: BASF Aktiengesellschaft
    Inventors: Ralf Klintz, Peter Schaefer, Gerhard Hamprecht, Elisabeth Heistracher, Hans-Josef Wolf, Karl-Otto Westphalen, Matthias Gerber, Uwe Kardorff, Helmut Walter, Klaus Grossmann
  • Patent number: 6150301
    Abstract: The harvesting of fruit, in particular olives and citrus fruit, is aided by inducing abscission by applying to fruit-bearing parts of the plant certain imidazolinone or sulfonylurea compounds. The compounds are applied in aqueous solution or in extremely low concentration in amounts ranging from 15 to 200 ppm, preferably from 20 to 70 ppm, by spraying to the point of incipient run-off.
    Type: Grant
    Filed: October 27, 1998
    Date of Patent: November 21, 2000
    Inventors: Merrill Wilcox, John B. Taylor
  • Patent number: 6057269
    Abstract: Benzylhydroxylamines I ##STR1## (X=--N(R.sup.7)--O--; Y=O, S; R.sup.1 =halogen, CN, NO.sub.2, CF.sub.3 ; R.sup.2 =H, halogen; R.sup.3 =H, NH.sub.2, CH.sub.3 ;R.sup.4 =H, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.1 -C.sub.6 -alkylthio, C.sub.1 -C.sub.6 -alkylsulfinyl or C.sub.1 -C.sub.6 -alkylsulfonyl;R.sup.5 =H, halogen, C.sub.1 -C.sub.6 -alkyl;R.sup.6 =H, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.2 -C.sub.6 -alkenyl;R.sup.7 =H, C.sub.1 -C.sub.6 -alkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.1 -C.sub.6 -alkylcarbonyl, C.sub.3 -C.sub.6 -alkenylcarbonyl, C.sub.3 -C.sub.6 -alkynylcarbonyl, C.sub.1 -C.sub.6 -alkoxycarbonyl, C.sub.2 -C.sub.8 -alkenyloxycarbonyl, C.sub.2 -C.sub.6 -alkynyloxycarbonyl, C.sub.1 -C.sub.6 -alkylthiocarbonyl, C.sub.1 -C.sub.6 -alkylsulfonyl, C.sub.1 -C.sub.
    Type: Grant
    Filed: January 5, 1998
    Date of Patent: May 2, 2000
    Assignee: BASF Aktiengesellschaft
    Inventors: Ralf Klintz, Gerhard Hamprecht, Elisabeth Heistracher, Peter Schafer, Cyrill Zagar, Karl-Otto Westphalen, Helmut Walter, Ulf Misslitz, Olaf Menke, Markus Menges
  • Patent number: 6022830
    Abstract: Described herein is a method for defoliating a crop plant or desiccating a crop vine plant to aid in harvesting the crop which comprises the step of applying to the plant an effective amount of a composition comprising a benzyloxyphenyluracil having the formula ##STR1## where R is an alkyl group of one to six carbons, in admixture with an agriculturally suitable carrier. The method is particularly effective at low use rates as an aid for harvesting potatoes and cotton.
    Type: Grant
    Filed: July 14, 1997
    Date of Patent: February 8, 2000
    Assignee: FMC Corporation
    Inventors: Mario S. Marquez, Frederick W. Hotzman, James T. Bahr
  • Patent number: 6013606
    Abstract: Substituted cinnamic oxime derivatives I and cinnamic hydroxamide derivatives II ##STR1## (R.sup.1= halogen, NO.sub.2, CN, CF.sub.3 ; R.sup.2 =H, halogen; R.sup.3= H, halogen, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, hydroxy-C.sub.1 -C.sub.6 -alkyl;R.sup.4= H, halogen, CN, C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl orR.sup.3 +R.sup.4 =chemical bond;Y=--O--, --S--, --O--CO--, --O--SO.sub.2 -- or chemical bond;Y'=--O-- or --S--;R.sup.5= unsubst. or subst. C.sub.1 -C.sub.6 -alkyl or C.sub.1 -C.sub.6 -haloalkyl; C.sub.3 -C.sub.6 -cycloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubst. or subst. phenyl or phenyl-C.sub.1 -C.sub.6 -alkyl, or, if Y is --O--, --S-- or a chemical bond, is (C.sub.1 -C.sub.6 -alkyl)carbonyl or (C.sub.1 -C.sub.6 -alkoxy)carbonyl; or, if Y is a chemical bond, is hydrogen or halogen;R.sup.5 '=R.sup.5, H or (C.sub.1 -C.sub.6 -haloalkyl)carbonyl;R.sup.6= H, C.sub.1 -C.
    Type: Grant
    Filed: June 30, 1997
    Date of Patent: January 11, 2000
    Assignee: BASF Akteingesellschaft
    Inventors: Ralf Klintz, Gerhard Hamprecht, Elisabeth Heistracher, Peter Schafer, Christoph-Sweder von dem Bussche-Hunnefeld, Peter Munster, Reinhard Kirstgen, Albrecht Harreus, Karl-Otto Westphalen, Matthias Gerber, Helmut Walter
  • Patent number: 5856273
    Abstract: A compound of formula (I): ##STR1## where E is oxygen or sulphur; A is CR.sup.3 or N where R.sup.3 is hydrogen or hydrocarbyl; D completes a 5 or 6-membered non-aromatic heterocyclic ring which optionally contains additional heteroatoms selected from oxygen, nitrogen or sulphur and which is optionally substituted by an optionally substituted lower hydrocarbyl group, or an optionally substituted heteroaryl group; R.sup.1 and R.sup.2 are each independently hydrogen; optionally substituted lower hydrocarbyl, or optionally substituted heteroaryl, or R.sup.1 and R.sup.2 together with the nitrogen atom to which they are attached, form a heterocyclic ring; Z represents halogen optionally substituted lower hydrocarbyl, optionally substituted lower hydocarbyloxy, optionally substituted lower hydrocarbylthio, hydrocarbylsulphinyl or hydrocarbylsulphonyl, cyano, nitro, CHO, NHOH, ONR.sup.7' R.sup.7", SF.sub.5 ; CO (optionally substituted lower hydrocarbyl), acylamino, COOR.sup.7, SO.sub.2 NR.sup.8 R.sup.9, CONR.sup.
    Type: Grant
    Filed: October 6, 1995
    Date of Patent: January 5, 1999
    Assignee: Zeneca Limited
    Inventors: Ian Trevor Kay, John Edward Duncan Barton, David John Collins, Bogdan Kowalczyk, Glynn Mitchell, John Martin Shribbs, John Micheal Cox, Nigel John Barnes, Stephen Christopher Smith
  • Patent number: 5773388
    Abstract: Novel pyrimidine derivatives of the formula (I): ##STR1## wherein R1 is a C.sub.1 -C.sub.6 haloalkyl group, a C.sub.1 -C.sub.6 alkyl group, a C.sub.3 -C.sub.6 cycloalkyl group or the like, R2 is a hydrogen atom, a C.sub.1 -C.sub.6 alkyl group, a C.sub.3 -C.sub.6 cycloalkyl group or the like, and X is a carbonyl group or --C(R3)OH (wherein R3 is a hydrogen atom, a C.sub.1 -C.sub.6 alkyl group or the like).
    Type: Grant
    Filed: February 9, 1996
    Date of Patent: June 30, 1998
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Jun Satow, Yasuo Kondo, Yoshihiro Kudo, Takumi Mikashima, Tsutomu Nawamaki, Yoichi Ito, Kazuhisa Sudo, Kunimitsu Nakahira, Shigeomi Watanabe, Kimihiro Ishikawa
  • Patent number: 5741755
    Abstract: This invention is related to herbicidal compositions comprising derivatives of benzenesulfonylurea and 2-methoxy-3,6-dichlorobenzoic acid for control of undesired vegetation by treating said vegetation and locus to be protected by said compositions.To eliminate the detrimental effects on crop rotation by lowering dosage of herbicide and to widen its activity spectrum a herbicidal composition is proposed comprising a mixture of ammonium salts of benzenesulfonylurea derivatives and of 2-methoxy-3,6-dichlorobenzoic acid with additives.The treatment of the vegetation and locus is performed by water solution of the disclosed composition with the dosage in the range of 50-500 g/ha of composition.
    Type: Grant
    Filed: June 22, 1995
    Date of Patent: April 21, 1998
    Assignee: Kare Ltd.
    Inventor: Vladimir Iosifovich Sorokin
  • Patent number: 5527764
    Abstract: Compounds having the structural formula ##STR1## wherein R.sub.1 is C.sub.1 -C.sub.4 alkyl, R.sub.2 is C.sub.1 -C.sub.4 alkyl or haloalkyl, R.sub.3 and R.sub.4 are hydrogen or halogen, and R.sub.5 is hydrogen or COOR.sub.6 wherein R.sub.6 is C.sub.1 -C.sub.8 linear or branched alkyl, alkenyl, or alkynyl, and compositions comprising the compounds. The compounds and compositions are useful as herbicides, desiccants and defoliants.
    Type: Grant
    Filed: September 15, 1994
    Date of Patent: June 18, 1996
    Assignees: Uniroyal Chemical Company, Inc., Uniroyal Chemical Ltd./Ltee
    Inventors: Dong Dao-cong, Alan W. Dalrymple
  • Patent number: 5518989
    Abstract: An increase in the quality of maize seed, especially with respect to improved seed vigor, is achieved by defoliating maize plants during a specific period after pollination. A maize seed assemblage then is obtained that is characterized by an enhanced seed vigor.
    Type: Grant
    Filed: January 31, 1994
    Date of Patent: May 21, 1996
    Assignee: Pioneer Hi-Bred International
    Inventors: Barry Martin, John Schoper, Laurie Carrigan
  • Patent number: 5223017
    Abstract: Compounds of formula (I) or salts thereof, ##STR1## in which J is a radical of the formula R.sup.1 SO.sub.2 --CR.sup.2 R.sup.3 --, R.sup.4 R.sup.5 N--SO.sub.2 --CR.sup.2 R.sup.3 --, or ##STR2## and wherein the radicals R.sup.1, R.sup.2, R.sup.3, R.sup.6, R.sup.7, R.sup.8, R.sup.*, A, W, m, n and 0 are defined as set forth in the specification, are suitable as selective herbicides and plant growth regulators.
    Type: Grant
    Filed: July 3, 1991
    Date of Patent: June 29, 1993
    Assignee: Hoechst Aktiengesellschaft
    Inventors: Heinz Kehne, Lothar Willms, Klaus Bauer, Hermann Bieringer
  • Patent number: 5221317
    Abstract: Herbicidally active sulphonylamino guanidinoazines of the formula ##STR1## in which R.sup.1 stands for an optionally substituted radical from the series comprising alkyl, aralkyl, aryl and hetaryl,R.sup.2 stands for an optionally substituted radical from the series comprising alkyl, aralkyl, aryl, hetaryl and dialkylamino,R.sup.3 stands for hydrogen, halogen, hydroxyl, alkyl, halogenaoalkyl, alkoxyalkyl, alkoxy, halogenoalkoxy, alkylthio, halogenoalkylthio, amino, alkylamino or dialkylamino,R.sup.5 stands for hydrogen, halogen, hydroxyl, alkyl, alkoxy, halogenoalkoxy, alkylthio, alkylamino or dialkylamino, andM stands for hydrogen, a metal equivalent, an ammonium equivalent, an alkylammonium equivalent, a dialkylammonium equivalent, or a trialkylammonium equivalent.
    Type: Grant
    Filed: June 28, 1991
    Date of Patent: June 22, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus-Helmut Muller, Christa Fest, Rolf Kirsten, Theodor Pfister, Hans-Jochem Riebel, Hans-Joachim Santel, Robert R. Schmidt, Harry Strang, Joachim Kluth, Klaus Lurssen, Ernst R. Gesing
  • Patent number: 5217522
    Abstract: Herbicidal sulphonylguanidinoazines of the formula ##STR1## in which n represents the numbers 1 or 2,A represents nitrogen or a C-X group, where X represents hydrogen or halogen.
    Type: Grant
    Filed: March 27, 1992
    Date of Patent: June 8, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hans-Jochem Riebel, Christa Fest, Ernst R. F. Gesing, Rolf Kirsten, Joachim Kluth, Klaus-Helmut Muller, Klaus Lurssen, Hans-Joachim Santel, Robert E. Schmidt
  • Patent number: 5215569
    Abstract: Substituted pyridines of the formula ##STR1## in which A represents nitrogen or a C-X group where X represents hydrogen or halogen,Q represents oxygen or sulphur,R.sup.1 and R.sup.2 are identical or different and represent hydrogen, halogen, alkyl, halogenoalkyl, alkoxyalkyl, alkoxy, halogenoalkoxy, alkylthio, alkylamino or dialkylamino,R.sup.3 represents hydrogen, amino, nitro, hydroxyl, halogen, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylamino, dialkylamino, alkylcarbonylamino, alkoxycarbonylamino or alkysulphonylamino,R.sup.4 represents hydrogen or alkyl andZ represents oxygen or one of the groups below: ##STR2## where R.sup.5, R.sup.6 and R.sup.7 are defined herein and their use in herbicide compositions.
    Type: Grant
    Filed: July 31, 1991
    Date of Patent: June 1, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Mark W. Drewes, Peter Muller, Hans-Joachim Santel, Klaus Lurssen, Robert R. Schmidt
  • Patent number: 5201937
    Abstract: Salicylic acid derivatives of the formula I ##STR1## (R.sup.1 is succinimidoxy; unsubstituted or substituted hetaryl; OR.sup.5 where R.sup.5 is substituted or unsubstituted cycloalkyl, alkyl, alkenyl, alkynyl, phenyl or substituted methyleneamino; OR.sup.8 where R.sup.8 is hydrogen, alkali metal or alkaline earth metal cation, ammonium or organic ammonium;R.sup.2 and R.sup.3 are each C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.2 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.2 -haloalkoxy and/or C.sub.1 -C.sub.4 -alkylthio;R.sup.4 is ethynyl or unsubstituted or substituted vinyl;X is oxygen or sulfur;Z is nitrogen or methine)are used as herbicides and bioregulators.
    Type: Grant
    Filed: October 16, 1991
    Date of Patent: April 13, 1993
    Assignee: BASF Aktiengesellschaft
    Inventors: Joachim Rheinheimer, Karl Eicken, Uwe J. Vogelbacher, Karl-Otto Westphalen, Matthias Gerber, Helmut Walter
  • Patent number: 5194084
    Abstract: Herbicidal substituted triazolones of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkylalkyl or cycloalkyl, or represents in each case optionally substituted aralkyl or aryl,R.sup.2 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, alkoxy, cycloalkyl or cycloalkylalkyl, or represents in each case optionally substituted aryl, aralkyl or heteroaryl,R.sup.3 and R.sup.4 independently of one another each represent hydrogen or an organic radical, or together with the nitrogen atom to which they are bonded represent an optionally substituted heterocycle,X represents oxygen or sulphur andY represents oxygen or sulphur.
    Type: Grant
    Filed: July 15, 1992
    Date of Patent: March 16, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Kurt Findeisen, Markus Lindig, Hans-Joachim Santel, Robert R. Schmidt, Klaus Lurssen
  • Patent number: 5194085
    Abstract: Herbicidally active substituted triazolinones of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, alkoxyalkyl, cycloalkyl, cycloalkylalkyl, or represents tetrahydrofuranyl, tetrahydrofuranylalkyl, or represents in each case optionally substituted aralkyl or aryl,R.sup.2 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, halogenoalkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkoxycarbonylalkyl, alkoxycarbonylalkenyl, alkylaminoalkyl, dialkylaminoalkyl, or represents in each case optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkenyl or cycloalkenylalkyl, or represents optionally substituted heterocyclylalkyl, or represents in each case optionally substituted aralkyl, aroyl, aryl, aralkyloxy or aryloxy, or represents alkoxy, alkenyloxy or alkinyloxy,X represents oxygen or sulphur andY represents oxygen or sulphur.New intermediates therefor are also shown.
    Type: Grant
    Filed: February 22, 1991
    Date of Patent: March 16, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Markus Lindig, Kurt Findeisen, Klaus-Helmut Muller, Hans-Joachim Santel, Robert R. Schmidt, Harry Strang, Dieter Feucht, Klaus Konig, Klaus Lurssen
  • Patent number: 5191089
    Abstract: Herbicidal 4-alkoxy- and 4-(substituted)amino-arylpyrrolinone derivatives of the formula ##STR1## in which X and Y independently of one another represent hydrogen, halogen, alkyl, alkoxy, halogenoalkyl or in each case unsubstituted or substituted aryloxy or arylthio,Z represents halogen, alkyl or alkoxy,n represents the number 0, 1, 2 or 3,A represents in each case unsubstituted or in each case halogen-substituted alkyl, alkenyl, alkynyl, alkoxyalkyl, polyalkoxyalkyl or alkylthioalkyl, cycloalkyl which is optionally interrupted by hetero atoms, arylalkyl which is unsubstituted or substituted by halogen, alkyl, halogenoalkyl, alkoxy and/or nitro, unsubstituted aryl or aryl substituted by a member selected from the group consisting of halogen, alkyl, alkoxy, halogenoalkyl, halogenoalkoxy and phenoxy or phenylthio which are in each case unsubstituted or substituted by halogen, alkyl, alkoxy, halogenoalkyl and/or halogenoalkoxy,B represents hydroxyl, alkoxy, halogenoalkoxy or cycloalkoxy, the cycloalkyl radical b
    Type: Grant
    Filed: August 9, 1990
    Date of Patent: March 2, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Bernd Baasner, Reiner Fischer, Klaus Lurssen, Hans-Joachim Santel, Robert R. Schmidt
  • Patent number: 5188657
    Abstract: Substituted sulfonylureas of the formula I ##STR1## where n and m are each 0 or 1, R.sup.1 is hydrogen, alkyl alkenyl or alkynyl, R.sup.2 is halogen or trifluoromethyl when m is 0, or is alkyl, alkenyl or alkynyl when m is 1, or is trifluoromethyl or chlorodifluoromethyl when X is O or S and m is 1, X is O, S or N-R.sup.4, R.sup.4 is hydrogen or alkyl, R.sup.3 is hydrogen, halogen, alkyl, haloalkyl or alkoxy, A is haloalkyl, halogen, cyano, nitro, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl or a radical ##STR2## B is oxygen or an alkylimino group N-R.sup.6 ; R.sup.5 is hydrogen, unsubstituted or substituted alkyl or unsubstituted or substituted cycloalkyl or is alkenyl or alkynyl and R.sup.6 is hydrogen or alkyl or, together with R.sup.5, forms a C.sub.4 -C.sub.6 -alkylene chain in which a methylene group may be replaced by an oxygen atom or a C.sub.1 -C.sub.
    Type: Grant
    Filed: August 2, 1991
    Date of Patent: February 23, 1993
    Assignee: BASF Aktiengesellschaft
    Inventors: Gerhard Hamprecht, Horst Mayer, Karl-Otto Westphalen, Helmut Walter, Matthias Gerber, Klaus Grossmann, Wilhelm Rademacher
  • Patent number: 5186734
    Abstract: Herbicidal bisazinyl compounds of the formula ##STR1## in which A.sup.1 and A.sup.2 are identical or different and represent nitrogen or a C--X group, X representing hydrogen, halogen, alkyl or alkoxy, andQ.sup.1 and Q.sup.2 are identical or different and represent oxygen, sulphur, NH or N-alkyl,(the substituents R, X.sup.1, X.sup.2, Y.sup.1, Y.sup.2 and Z representing a variety of organic radicals).The compounds of the formulas ##STR2## are also new.
    Type: Grant
    Filed: September 11, 1991
    Date of Patent: February 16, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Roland Andree, Mark W. Drewes, Hans-Joachim Santel, Klaus Lurssen, Robert R. Schmidt
  • Patent number: 5185026
    Abstract: Herbicidal naphthalene derivatives of the formula ##STR1## in which Q represents oxygen, sulphur or the group NR, where R represents hydrogen or alkyl,R.sup.1 represents hydrogen or alkylR.sup.2, R.sup.3 and R.sup.4 are identical or different and in each case represent hydrogen or another radical,R.sup.5 represents hydrogen or halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylamino or dialkylamino,R.sup.6 represents hydrogen or halogen, or represents in each case optionally substituted alkyl or alkoxy, andR.sup.7 represents hydrogen or halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylamino or dialkylamino, andZ represents N--R.sup.
    Type: Grant
    Filed: April 4, 1991
    Date of Patent: February 9, 1993
    Assignee: Bayer Aktiengesellschaft
    Inventors: Mark W. Drewes, Michael Haug, Klaus Lurssen, Hans-Joachim Santel, Robert R. Schmidt
  • Patent number: 5176735
    Abstract: A method of desiccating plants, which method involves the application of a desiccatingly effective amount of certain 3-carbonylphenyl uracil compounds to the locus of the plants to be treated. Such application will act as a harvest aid for field crops.
    Type: Grant
    Filed: June 28, 1990
    Date of Patent: January 5, 1993
    Assignee: Uniroyal Chemical Company, Inc.
    Inventor: Allyn R. Bell