Hetero Ring Is Six-membered Including Nitrogen And Oxygen Patents (Class 504/223)
  • Patent number: 9700050
    Abstract: The present invention relates to a method of controlling weeds in a crop field, the method including treating the crop field with crystal of flumioxazin described in the specification, before sowing or planting, at the same time of sowing or planting, or after sowing or planting crop seeds or vegetative organs such as tubers, bulbs, or stem fragments which are treated with one or more compounds selected from the following group B; Group B: neonicotinoid type compounds, diamide type compounds, carbamate type compounds, organic phosphorous type compounds, biological nematicidal compounds, other insecticidal compounds and nematicidal compounds, azole type compounds, strobilurin type compounds, metalaxyl type compounds, SDHI compounds, and other fungicidal compounds and plant growth regulators. According to the method of controlling pests of the present invention, weeds in clop fields can be efficiently controlled.
    Type: Grant
    Filed: December 6, 2013
    Date of Patent: July 11, 2017
    Assignee: SUMITOMO CHEMICAL COMPANY, LIMITED
    Inventor: Hajime Ikeda
  • Patent number: 9034353
    Abstract: Disclosed herein are mesocapsules that include agriculturally active ingredients. These mesocapsules are comprised of a polyurea shell and include hydrophilic groups on their surfaces and have a volume-average diameter of about 500 nm or less and some of them have a volume-average diameter on the order of about 300 nm or less. These mesocapsules are suited for delivering active ingredients that are not very soluble in water. Methods for making these mesocapsules include interfacial polycondensation reactions carried out in the presence of surfactants and other methods in which all or most of the surfactant is replaced by adding amino acids to the aqueous phase of the interfacial reaction mixture before forming the final emulsion.
    Type: Grant
    Filed: August 5, 2010
    Date of Patent: May 19, 2015
    Assignee: Dow AgroSciences LLC
    Inventors: Robert J. Ehr, Thomas H. Kalantar, Lei Liu, Dale C. Schmidt, Mike P. Tolley, Kerrm Y. Yau, Qiang Zhang, Min Zhao
  • Patent number: 8765640
    Abstract: Crystal forms of sulfonylurea compound and method for producing the same. It has been found that a sulfonylurea compound of Formula (1): has two types of crystal polymorphisms and four types of pseudo crystal polymorphisms. A production method of each crystal form of the sulfonylurea compound of Formula (1) through recrystallization or solvate has been also found. In addition, a suspension of a composition containing the crystal that is improved in storage stability is provided.
    Type: Grant
    Filed: October 25, 2010
    Date of Patent: July 1, 2014
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Yoshiyuki Kusuoka, Yoshihiko Nakaya, Nao Kitayado
  • Patent number: 8642509
    Abstract: The present invention provides a method of reducing phytotoxicity to crops (especially maize) caused by a herbicidal benzoylisoxazole and/or dione derivative of formula (I) or an agriculturally acceptable salt or metal complex thereof; which method comprises applying to the locus of the crop an antidotally effective amount of an antidote compound, optionally with a partner herbicide.
    Type: Grant
    Filed: June 27, 2006
    Date of Patent: February 4, 2014
    Assignee: Aventis Cropscience UK Limited
    Inventors: Ken Pallett, Ashley Slater
  • Patent number: 8637496
    Abstract: The invention relates to the use of compounds having a monogalactosyldiacylglycerol (MGDG) synthase inhibitory activity as herbicide or algaecide, and to herbicide and algaecide compositions containing at least one of these compounds.
    Type: Grant
    Filed: June 2, 2008
    Date of Patent: January 28, 2014
    Assignees: Commissariat a l'Energie Atomique, Centre National de la Recherche Scientifique
    Inventors: Anne-Laure Bonneau, Cyrille Botte, Michael Deligny, Nadia Saidani, Hélène Hardre, Bernard Rousseau, Roman Lopez, Eric Marechal
  • Patent number: 8629083
    Abstract: The present invention relates to mixtures of strobilurin fungicides and plant growth regulators and to the foliar application of these mixtures on crops including cotton.
    Type: Grant
    Filed: June 16, 2006
    Date of Patent: January 14, 2014
    Assignee: Syngenta Crop Protection, LLC
    Inventors: Steven Harrison, Bernd Druebbisch, Patrick Ewan
  • Publication number: 20130324412
    Abstract: N-Alkoxyamides of 4-aminopicolinic acids and 6-amino-4-pyrimidinecarboxylates are selective herbicides for corn, canola and sugar beet.
    Type: Application
    Filed: August 8, 2013
    Publication date: December 5, 2013
    Applicant: DOW AGROSCIENCES LLC
    Inventors: Joseph D. Eckelbarger, Paul R. Schmitzer, Carla N. Yerkes, Timothy A. Boebel, Norbert M. Satchivi, Gregory T. Whiteker
  • Publication number: 20120220461
    Abstract: Crystal forms of sulfonylurea compound and method for producing the same. It has been found that a sulfonylurea compound of Formula (1): has two types of crystal polymorphisms and four types of pseudo crystal polymorphisms. A production method of each crystal form of the sulfonylurea compound of Formula (1) through recrystallization or solvate has been also found. In addition, a suspension of a composition containing the crystal that is improved in storage stability is provided.
    Type: Application
    Filed: October 25, 2010
    Publication date: August 30, 2012
    Applicant: NISSAN CHEMICAL INDUSTRIES, LTD.
    Inventors: Yoshiyuki Kusuoka, Yoshihiko Nakaya, Nao Kitayado
  • Publication number: 20120088672
    Abstract: Disclosed is a method of improving the growth of plants wherein at least one compound of formula (I) wherein A is 2-chloropyrid-5-yl, 2-methylpyrid-5-yl, 1-oxido-3-pyridinio, 2-chloro-1-oxido-5-pyridinio, 2,3-dichloro-1-oxido-5-pyridinio, tetrahydrofuran-3-yl, 5-methyl-tetrahydrofuran-3-yl or 2-chlorothiazol-5-yl group, R is hydrogen, C1-C6alkyl, phenyl-C1-C4alkyl, C3-C6cycloalkyl, C2-C6alkenyl or C2-C6alkynyl; Y is —N(R)(R2) or SR2; R1 and R2 are independently of each other C1-C4-alkyl, C1-C4-alkenyl, —C(?O)—CH3 or benzyl; or together form a group —CH2—CH2—, —CH2—CH2—CH2—, —CH2—O—CH2—, —CH2—S—CH2—, —CH2—NH—CH2— or —CH2—N(CH3)—CH2—; and X is N—NO2 or N—CN or CH—NO2, or, where appropriate, a tautomer thereof, in each case in free from or in salt form; is applied to the plant or the locus thereof.
    Type: Application
    Filed: October 11, 2011
    Publication date: April 12, 2012
    Applicant: SYNGENTA CROP PROTECTION, LLC
    Inventors: Robert SENN, Dieter HOFER, Thomas Thieme, Larry Zang
  • Patent number: 8084397
    Abstract: The present invention provides a composition including a polymer nanoparticle and at least one agricultural active compound incorporated with the nanoparticle, wherein the nanoparticle are less than 100 nm in diameter, and the polymer includes a polyelectrolyte.
    Type: Grant
    Filed: May 6, 2010
    Date of Patent: December 27, 2011
    Assignee: Vive Nano, Inc.
    Inventors: Fugang Li, Hung Pham, Darren J. Anderson
  • Patent number: 8067337
    Abstract: An agricultural chemical composition which enables a wide range of herbicidal compounds including ones showing phytotoxicity to crop plants, etc. upon mere application to exhibit a sufficient herbicidal effect and to show reduced or no phytotoxicity to the crop plants. The agricultural chemical composition comprises (A) a herbicidal compound selected from the group consisting of sulfonylurea compounds, sulfonamide compounds, chloroacetanilide compounds, thiocarbamate compounds, pyrimidinyloxy(thio)benzoic acid compounds, tetrazolinone compounds, pyrazole compounds, cyclohexanedione compounds, phenoxycarboxylic acid compounds, oxazinone compounds, and difluoromethanesulfonylanilide compounds or salts thereof and (B) a compound selected among benzoic acid compounds.
    Type: Grant
    Filed: August 5, 2005
    Date of Patent: November 29, 2011
    Assignee: Kumiai Chemical Industry Co., Ltd
    Inventors: Toshihiro Ikeuchi, Tetsuo Ohkawa, Shuji Ohno, Hiroshi Kawasaki, Ryo Hanai, Yasunori Ogawa, Makoto Fujinami
  • Patent number: 8062995
    Abstract: Novel dioxazine- and oxdiazine-substituted arylamides of the formula (I) in which A1, A2, R1, R2, R3, R4 and R5 are as defined in the description, a plurality of processes for preparing these compounds and their use for controlling pests, and also novel intermediates and processes for their preparation.
    Type: Grant
    Filed: September 5, 2006
    Date of Patent: November 22, 2011
    Assignee: Bayer CropScience AG
    Inventors: Bernd-Wieland Krüger, Achim Hense, Bernd Alig, Rüdiger Fischer, Christian Funke, Ernst Rudolf Gesing, Olga Malsam, Mark Wilhelm Drewes, Christian Arnold, Peter Lümmen, Erich Sanwald
  • Patent number: 8048825
    Abstract: A haloalkylsulfonanilide derivative represented by general formula (I) or a salt thereof wherein R1 represents a halo(C1-C8)alkyl group, R2, R3, R4, R5, R6, R7, R8, R9 and R10 represent hydrogen atoms, etc., n represents 1 or 2, A represents an oxygen atom, W represents an oxygen atom, X represents a halogen atom and m represents an integer of 0 to 4, are compounds useful as herbicides having both of remarkable herbicidal effect and characteristics such as excellent crop-weed selectivity.
    Type: Grant
    Filed: November 16, 2007
    Date of Patent: November 1, 2011
    Assignee: Nihon Nohyaku Co., Ltd.
    Inventors: Tomokazu Hino, Yasuko Yamada, Toshihiko Shigenari, Koki Mametsuka
  • Publication number: 20110077157
    Abstract: The present invention relates to an oil suspension concentrate comprising a) one or more herbicidally active compounds from the group of the pyridylsulfonylureas in suspended form, and b) one or more organic solvents. The oil suspension concentrate is suitable for use in crop protection.
    Type: Application
    Filed: December 3, 2010
    Publication date: March 31, 2011
    Applicant: Bayer CropScience AG
    Inventors: Frank Sixl, Annika Schmidt
  • Publication number: 20110045975
    Abstract: Various aspects disclosed herein disclose mesocapsules that include active ingredients such as agriculturally active ingredients including various fungicides, insecticides, miticides, herbicides, safeners and modifiers of plant physiology or structure. These mesocapsules are comprised of a polyurea shell and include hydrophilic groups on their surfaces. These mesocapsules have a volume-average diameter of about 500 nm or less and some of them have a volume-average diameter on the order of about 300 nm or less. These mesocapsules are especially well suited for delivering active ingredients that are not very soluble in water, many of these compounds have solubility values in the range of 1,000 ppm or less.
    Type: Application
    Filed: August 5, 2010
    Publication date: February 24, 2011
    Applicant: Dow AgroSciences LLC
    Inventors: Robert J. Ehr, Thomas H. Kalantar, Lei Liu, Dale C. Schmidt, Mike P. Tolley, Kerrm Y. Yau, Qiang Zhang, Min Zhao
  • Publication number: 20100317523
    Abstract: A method for controlling noxious organisms in a field of soybean or corn, comprising the steps of: treating soybean or corn seeds with at least one neonicotinoid compound selected from the group consisting of clothianidin, thiamethoxam, imidacloprid, dinotefuran, nitenpyram, acetamiprid, and thiacloprid, and treating the field with at least one PPO inhibitor compound selected from the group consisting of flumioxazin, sulfentrazone, saflufenacil, oxyfluorfen, and 3-(4-chloro-6-fluoro-2-trifluoromethylbenzimidazol-7-yl)-1-methyl-6-trifluoromethyl-2,4-(1H,3H)pyrimidinedione before or after the soybean or corn seeds treated with the neonicotinoid compound are sown in the field.
    Type: Application
    Filed: September 18, 2009
    Publication date: December 16, 2010
    Applicant: SUMITOMO CHEMICAL COMPANY, LIMITED
    Inventors: Hajime Ikeda, Atsushi Iwata
  • Publication number: 20100298141
    Abstract: Disclosed are compounds of Formula 1, including N-oxides, and salts thereof, wherein W is O or NR7, n is 0 or 1, and R1, R2, R3, R4, R5, R6, R7 and m are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling undesired vegetation comprising contacting the undesired vegetation or its environment with an effective amount of a compound or a composition of the invention. Also disclosed are mixtures and compositions comprising a herbicidally effective amount of a compound of Formula 1 and an effective amount of another herbicide or herbicide safener.
    Type: Application
    Filed: February 8, 2008
    Publication date: November 25, 2010
    Applicant: E. I. DU PONT DE NEMOURS AND COMPANY
    Inventors: Thomas Paul Selby, Brenton Todd Smith, Thomas Martin Stevenson
  • Publication number: 20100279862
    Abstract: The invention relates to the use of one or more compounds of the formula (I) or salts thereof, wherein the groups R1 to R8 are defined as set forth in claim 1, optionally in the presence of additional agrochemical active ingredients, for selective weed control on turf or lawn.
    Type: Application
    Filed: April 28, 2010
    Publication date: November 4, 2010
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Udo BICKERS, Michael Kilian, Stefanie Nöding, Donald F. Myers
  • Publication number: 20100267563
    Abstract: A method of improving the growth of a plant comprising applying to a plant, plant propagation material or locus thereof a composition comprising a product, which comprises microcapsules which themselves comprise (a) a polymeric shell; and (b) a core which comprises a dispersed solid active ingredient compound wherein the compound is one or more of a neonicotinoid, fipronil, a strobilurin, carboxin, acibenzolar-S-methyl, and probenazole.
    Type: Application
    Filed: June 18, 2008
    Publication date: October 21, 2010
    Applicants: SYNGENTA CROP PROTECTION, INC., SYNGENTA LIMITED
    Inventors: Domingos Pedroni, Anke Buchholz, Anne Waller, Werner Reiner
  • Publication number: 20100210465
    Abstract: The present invention provides a composition including a polymer nanoparticle and at least one agricultural active compound incorporated with the nanoparticle, wherein the nanoparticle are less than 100 nm in diameter, and the polymer includes a polyelectrolyte.
    Type: Application
    Filed: May 6, 2010
    Publication date: August 19, 2010
    Applicant: VIVE NANO, INC.
    Inventors: Fugang LI, Hung PHAM, Darren J. ANDERSON
  • Publication number: 20100144531
    Abstract: A method of increasing plant hormone activity in a plant comprising applying to the plant, part of the plant, the plant propagation material thereof and/or a surrounding area thereof an effective amount of one or more neonicotinoid compounds selected from thianicotinyl compounds and tetrahydrofuranyl compounds.
    Type: Application
    Filed: September 28, 2007
    Publication date: June 10, 2010
    Applicant: SYNGENTA CROP PROTECTION, INC.
    Inventors: Paulo Aramaki, Joao Carlos Nunes, Andre Oliveira, Nestor Gabriel Da Silva, Domingo Pedroni, Dieter Hofer, Michael Schade
  • Patent number: 7732374
    Abstract: A fungicidal mixture comprising prothioconazole or its salts or adducts and at least one insecticide selected from the group consisting of fipronil, chlorpyrifos or thiamethoxam.
    Type: Grant
    Filed: July 17, 2007
    Date of Patent: June 8, 2010
    Assignee: BASF SE
    Inventors: Eberhard Ammermann, Reinhard Stierl, Gisela Lorenz, Siegfried Strathmann, Klaus Schelberger, V. James Spadafora, Thomas Christen
  • Patent number: 7709636
    Abstract: A pyrazole compound of the formula: where: R1 is C1-3alkyl, C1-3haloalkyl, C1-3alkoxy C1-3alkyl, phenyl or pyridyl; R2 is a hydrogen atom, C1-3alkyl, C1-3haloalkyl, C1-3alkoxy or a halogen atom; R3, R4, R5 and R6 independently of one another are a hydrogen atom, C1-3alkyl or C1-3haloalkyl, with a proviso that at least one of R3, R4, R5 and R6 is C1-3alkyl or C1-3haloalkyl; and L is a hydrogen atom, chlorine atom, SH, benzylthio, chlorosulfonyl, aminosulfonyl, SO2N?C?O, SO2NHCO2CH3 or SO2NHCONHn-C4H9. A salt of the compound that is acceptable as an agrochemical. An agrochemical containing the compound or the salt thereof as an active component. A herbicide containing the compound or the salt thereof as an active component.
    Type: Grant
    Filed: May 28, 2009
    Date of Patent: May 4, 2010
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Hiroshi Kita, Yoshitake Tamada, Yoshihiko Nakaya, Tetsuhiko Yano, Manabu Saeki
  • Publication number: 20100105559
    Abstract: An agrochemical composition includes a homogeneous single-phase liquid crystal in thermodynamic equilibrium. The agrochemical composition can be a surfactant composition or a pesticide composition. The surfactant composition is a blend of surfactants, whereas a pesticide composition has an active ingredient and one or more surfactant adjuvants. A pesticide composition, or a surfactant composition in combination with an active ingredient, may be used to control pests.
    Type: Application
    Filed: October 9, 2007
    Publication date: April 29, 2010
    Applicant: Huntsman Petrochemical Corporation
    Inventors: Curtis M. Elsik, Joe C. Arzola, Howard M. Stridde, Alan Stern
  • Publication number: 20100099561
    Abstract: Disclosed are compounds of Formula 1, N-oxides, and salts thereof, wherein J is and R1, R2, R3, R4, R5, R6, R7, R8a, R8b, R8c, G1, G2, G3, G4, G5, G6, Q1, Q2, Q3, Q4, W1, W2, Y1, Y2, Y3, m and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling undesired vegetation comprising contacting the undesired vegetation or its environment with an effective amount of a compound or a composition of the invention.
    Type: Application
    Filed: October 14, 2009
    Publication date: April 22, 2010
    Applicant: E.I. DU PONT DE NEMOURS AND COMPANY
    Inventors: THOMAS PAUL SELBY, BRENTON TODD SMITH
  • Patent number: 7655599
    Abstract: The present invention relates to novel agrochemical formulations based on ethylene diamine alkoxylate derivative emulsifiers, to a method for producing said formulations, and to the use of the same for applying the active ingredients contained therein.
    Type: Grant
    Filed: June 21, 2004
    Date of Patent: February 2, 2010
    Assignee: Bayer Cropscience AG
    Inventors: Andreas Rochling, Frank Rosenfeldt
  • Publication number: 20100016164
    Abstract: A haloalkylsulfonanilide derivative represented by general formula (I) or a salt thereof wherein R1 represents a halo(C1-C8)alkyl group, R2, R3, R4, R5, R6, R7, R8, R9 and R10 represent hydrogen atoms, etc., n represents 1 or 2, A represents an oxygen atom, W represents an oxygen atom, X represents a halogen atom and m represents an integer of 0 to 4, are compounds useful as herbicides having both of remarkable herbicidal effect and characteristics such as excellent crop-weed selectivity.
    Type: Application
    Filed: November 16, 2007
    Publication date: January 21, 2010
    Inventors: Tomokazu Hino, Yasuko Yamada, Toshihiko Shigenari, Koki Mametsuka
  • Patent number: 7648945
    Abstract: The present invention relates to a herbicide combination comprising components (A) and (B), where (A) is one or more herbicides from the group of the compounds of the formula (I) or salts thereof in which R1, R2, R3, R4, R5, R6, R7, R8 and A are as defined in claim 1; and (B) is one or more herbicides different from herbicide (A), preferably from the group of compounds consisting of (B1) herbicides which can be employed selectively and which are effective mainly against monocotyledonous and dicotyledonous harmful plants, (B2) herbicides which can be employed selectively and which are effective mainly against dicotyledonous harmful plants and (B3) herbicides which can be employed selectively and which are effective mainly against monocotyledonous harmful plants, (B4) herbicides which can be employed non-selectively and which are effective against monocotyledonous and dicotyledonous harmful plants, for example for use in the non-selective field or in crops which are specifically tolerant.
    Type: Grant
    Filed: March 25, 2005
    Date of Patent: January 19, 2010
    Assignee: Bayer CropScience AG
    Inventors: Martin Hills, Erwin Hacker, Hansjörg Krähmer, Christian Waldraff, Hansjörg Dietrich, Klaus Trabold, Dieter Feucht, Klaus-Helmut Müller, Ulrich Philipp
  • Publication number: 20090270254
    Abstract: The present invention relates to methods for increasing the stress tolerance in plants and plant cells whereby neonicotinoid compounds, such as but not limited to imidacloprid, clothianidin, thiamethoxam, dinotefuran, nitenpyram, acetamiprid or thiacloprid, are applied to plants, or cells thereof, which comprise a genome that has been modified to make the plants or their cells more stress tolerant i.e. plants engineered to be stress tolerant. Particularly effective stress tolerance synergists in combination with genetically modified stress tolerant plants or their cells are neonicotinoid compounds which comprise a chloropyridine side chain, like e.g. imidacloprid, thiacloprid, acetamiprid, nitenpyram and 6-chloronicotinic acid (6-CNA).
    Type: Application
    Filed: May 26, 2006
    Publication date: October 29, 2009
    Applicant: Bayer CropScience AG
    Inventors: Wolfgang Thielert, Michael Metzlaff, Marc De BLock
  • Patent number: 7605111
    Abstract: Compounds of formula wherein the substituents have the meanings given in claim 1, and agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides.
    Type: Grant
    Filed: March 18, 2005
    Date of Patent: October 20, 2009
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Thomas Maetzke, André Stoller, Sebastian Wendeborn, Henry Szczepanski
  • Publication number: 20090227457
    Abstract: The present invention relates to stable, agricultural oil-in-water emulsion compositions.
    Type: Application
    Filed: March 9, 2009
    Publication date: September 10, 2009
    Applicant: DOW AGROSCIENCES LLC
    Inventors: Wen Xu, Holger Tank, Joey Cobb
  • Patent number: 7563749
    Abstract: The present invention relates to a herbicide-safener combination, comprising (A) one or more compounds of the formula (I) or salts thereof as defined in the application and (B) one or more safeners.
    Type: Grant
    Filed: March 25, 2005
    Date of Patent: July 21, 2009
    Assignee: Bayer CropScience AG
    Inventors: Martin Hills, Erwin Hacker, Hansjörg Krähmer, Chris Rosinger, Udo Bickers, Frank Ziemer, Christian Waldraff, Hansjörg Dietrich, Lothar Willms, Dieter Feucht, Klaus-Helmut Müller, Ulrich Philipp
  • Patent number: 7557066
    Abstract: The invention relates to the use of compounds of the formula (I) and salts thereof, as defined in the application, for the selective control of unwanted vegetation in leguminous plants or for the non-selective control of unwanted vegetation
    Type: Grant
    Filed: March 25, 2005
    Date of Patent: July 7, 2009
    Assignee: Bayer CropScience AG
    Inventors: Martin Hills, Hansjörg Krähmer, Christian Waldraff, Hansjörg Dietrich, Dieter Feucht, Klaus-Helmut Müller, Ulrich Philipp
  • Patent number: 7557067
    Abstract: There is provided a novel herbicide. A pyrazole sulfonylurea compound of formula (1): wherein R1 is C1-3alkyl, etc., R2 is hydrogen atom, C1-3alkyl, C1-3haloalkyl, etc., R3, R4, R5 and R6 independently of one another are hydrogen atom, C1-3alkyl, etc., with a proviso that at least one of R3, R4, R5 and R6 is C1-3alkyl or C1-3haloalkyl, X and Y independently of each other are C1-3alkyl, etc., Z is nitrogen atom or methyne, and a salt thereof that is acceptable as an agrochemical; an agrochemical containing at least one of the compound and the salt thereof that is acceptable as an agrochemical as an active component, and a herbicide containing at least one of the compound and the salt thereof that is acceptable as an agrochemical as an active component.
    Type: Grant
    Filed: April 27, 2005
    Date of Patent: July 7, 2009
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Hiroshi Kita, Yoshitake Tamada, Yoshihiko Nakaya, Tetsuhiko Yano, Manabu Saeki
  • Patent number: 7494992
    Abstract: The present invention relates to novel terpene alkaloids and their use as antiparasitic agents. The present invention also relates to an antiparasitic agent which comprises a terpene alkaloid compound of this invention as an effective ingredient in an antiparasitic formulation. More particularly, the present invention relates to derivatives of the terpene alkaloid (1S,2R,4aS,5R,8R,8aR)-2-(acetyloxy)-8a-hydroxy-3,8-dimethyl-5-(1-methylethenyl)-1,2,4a,5,6,7,8,8a-octahydronaphthalen-1-yl (2S,3aR,9bR)-6-chloro-9b-hydroxy-5-methyl-1,2,3,3a,5,9b-hexahydropyrrolo[2,3-c][2,1]benzoxazine-2-carboxylate. Pharmaceutical compositions comprising the same are also disclosed.
    Type: Grant
    Filed: February 12, 2004
    Date of Patent: February 24, 2009
    Assignee: Pfizer Inc.
    Inventors: Nathan A. Chubb, Douglas J. Critcher, James J. Eshelby, Graham Lunn, Andrew J. Rudge, Nigel D. Walshe, Paul H Wiedenau, David H. Williams
  • Publication number: 20080300138
    Abstract: The invention relates to novel substituted thienylsulfonylaminocarbonyl compounds of the formula (I), in which R, Het and R5 to R8 are as defined in the description, to processes and intermediates for their preparation and to their use as herbicides.
    Type: Application
    Filed: July 13, 2005
    Publication date: December 4, 2008
    Inventors: Ernst R. F. Gesing, Dieter Feucht, Heinz Kehne, Thomas Auler, Martin Hills
  • Patent number: 7459414
    Abstract: Compounds of formula wherein the substituents have the meanings given in claim 1, and agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides.
    Type: Grant
    Filed: March 18, 2005
    Date of Patent: December 2, 2008
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Thomas Maetzke, André Stoller, Sebastian Wendeborn, Henry Szczepanski
  • Patent number: 7183238
    Abstract: The present invention relates to novel [1,2]-oxazine-3,5-dione derivatives of the formula (I) in which W, X, Y, Z, G, D, A and B are as defined in the disclosure, to a plurality of processes for their preparation, and to their use as microbicides, pesticides and herbicides.
    Type: Grant
    Filed: November 27, 2002
    Date of Patent: February 27, 2007
    Assignee: Bayer CropScience AG
    Inventors: Reiner Fischer, Thomas Schenke, Angelika Lubos-Erdelen, legal representative, Christoph Erdelen, deceased
  • Patent number: 6894005
    Abstract: Compounds of formula wherein the substituents have the meanings given in claim 1, and agronomically tolerable salts, isomers and enantiomer of those compounds, are suitable for use as herbicides.
    Type: Grant
    Filed: September 5, 2000
    Date of Patent: May 17, 2005
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Thomas Maetzke, André Stoller, Sebastian Wendeborn, Henry Szczepanski
  • Patent number: 6844339
    Abstract: There is now described a method of controlling pests with nitroimino- or nitroguanidino-compounds; more specifically a method of controlling pests in and on transgenic crops of useful plants, such as, for example, in crops of maize, cereals, soya beans, tomatoes, cotton, potatoes, rice and mustard, with a nitroimino- or nitroguanidino-compound, especially with thiamethoxam, characterized in that a pesticidal composition comprising a nitroimino- or nitroguanidino-compound in free form or in agrochemically useful salt form and at least one auxiliary is applied to the pests or their environment, in particular to the crop plant itself;
    Type: Grant
    Filed: April 18, 2002
    Date of Patent: January 18, 2005
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Bruce Lee, Marius Sutter, Hubert Buholzer
  • Patent number: 6828276
    Abstract: There are described benzoylcyclohexanediones of the formula I, their preparation, and their use as herbicides and plant growth regulators. In this formula (I), C1, C2, C3 are cyclic radicals, X1 is a hetero atom, X2 is a chain of carbon atoms, L is a chain-like element, R1, R2, R3, R4, R5 are various radicals, and Y and Z are monoatomic bridge elements.
    Type: Grant
    Filed: August 30, 2001
    Date of Patent: December 7, 2004
    Assignee: Aventis CropScience GmbH
    Inventors: Thomas Seitz, Andreas van Almsick, Lothar Willms, Hermann Bieringer, Thomas Auler, Hubert Menne
  • Publication number: 20040186021
    Abstract: The invention relates to novel substituted benzo-nitrogen heterocycles of the formula (I) 1
    Type: Application
    Filed: January 9, 2004
    Publication date: September 23, 2004
    Inventors: Otto Schallner, Dorothee Hoischen, Mark Wilhelm Drewes, Peter Dahmen, Dieter Feucht, Rolf Pontzen
  • Patent number: 6753296
    Abstract: Disclosed is a method of improving the growth of plants wherein at least one compound of formula (I) wherein A is 2-chloropyrid-5-yl, 2-methylpyrid-5-yl, 1-oxido-3-pyridinio, 2-chloro-1-oxido-5-pyridinio, 2,3-dichloro-1-oxido-5-pyridinio, tetrahydrofuran-3-yl, 5-methyl-tetrahydrofuran-3-yl or 2-chlorothiazol-5-yl group, R is hydrogen, C1-C6alkyl, phenyl-C1-C4alkyl, C3-C6cycloalkyl, C2-C6alkenyl or C2-C6alkynyl; Y is —N(R)(R2) or SR2; R1 and R2 are independently of each other C1-C4-alkyl, C1-C4-alkenyl, C1-C4-alkinyl, —C(═O)—CH3 or benzyl; or together form a group —CH2—CH2—, —CH2—CH2—CH2—, —CH2—O—CH2—, —CH2—S—CH2—, —CH2—NH—CH2— or —CH2—N(CH3)—CH2—; and X is N—NO2 or N—CN or CH—NO2; or, where appropriate, a tautomer thereof, in each case in free from or in salt form; is applied to the plant or the locus thereof.
    Type: Grant
    Filed: April 10, 2002
    Date of Patent: June 22, 2004
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Robert Senn, Dieter Hofer, Thomas Thieme, Larry Zang
  • Patent number: 6734143
    Abstract: The present invention provides 2-methoxyimino-2-(pyridinyloxymethyl) phenyl acetamides according to formula (I) as well as their use as fungicidal compounds.
    Type: Grant
    Filed: February 27, 2003
    Date of Patent: May 11, 2004
    Assignee: Dow AgroSciences LLC
    Inventors: Neil Vincent Kirby, Jenifer Lynn Adamski Butz, Brent Jeffrey Rieder, James M. Renga, Jeannie Rachel Phillips Cetusic, Irene Mae Morrison, John Todd Mathieson, Gary David Gustafson
  • Publication number: 20030236167
    Abstract: Compounds of formula I 1
    Type: Application
    Filed: June 5, 2003
    Publication date: December 25, 2003
    Inventors: Jurgen Schaetzer, Alain De Mesmaeker, Shy-Fuh Lee
  • Patent number: 6653256
    Abstract: Microcapsule formulations of A) a particulate disperse phase of a) a reaction product of at least one diamine, polyamide, dialcohol, polyalcohol and/or aminoalcohol with an isocyanate mixture characterized in the description, if appropriate as a mixture with toluylene diisocyanate, b) at least one agrochemically active compound of a particular group of substances and, c) if appropriate, additives, and B) a liquid aqueous phase, a process for the preparation of these formulations, and their use for applying the active compounds which they comprise.
    Type: Grant
    Filed: March 1, 2001
    Date of Patent: November 25, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hilmar Wolf, Joachim Weissmüller
  • Patent number: 6602823
    Abstract: Agrochemical formulations comprising a) at least one agrochemically active compound, b) 2-ethyl-hexanol alkoxylate of the formula  in which P represents E represents —CH2—CH2— and the numbers 8 and 6 are average values and c) optionally additives, a process for preparing these formulations and their use for applying the active compounds they comprise are described.
    Type: Grant
    Filed: June 8, 2001
    Date of Patent: August 5, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Andreas Röchling, Anne Suty-Heinze, Karl Reizlein, Udo Reckmann
  • Patent number: 6566306
    Abstract: Microcapsule formulations of A) a particulate disperse phase of a) a reaction product of the isocyanate of the formula if appropriate as a mixture with toluylene diisocyanate, and at least one diamine, polyamine, dialcohol, polyalcohol and/or aminoalcohol, b) at least one agrochemically active compound of a particular group of substances and, c) if appropriate, additives, and B) a liquid aqueous phase, a process for the preparation of these formulations, and their use for applying the active compounds which they comprise.
    Type: Grant
    Filed: March 1, 2001
    Date of Patent: May 20, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hilmar Wolf, Joachim Weissmüller, Maria Giuliana Cianciulli Teller
  • Patent number: 6559100
    Abstract: Substituted 2-benzoylcyclohexane-1,3-diones of the formula I where: R1 and R2 are each hydrogen, mercapto, nitro, halogen, cyano, thiocyanato, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl, C2-C6-alkynyl, —OR3, —OCOR3, —OSO2R3, —S(O)nR3, —SO2OR3, —SO2N(R3)2, —NR3SO2R3 or —NR3COR3; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, phenyl or phenyl-C1-C6-alkyl; where the abovementioned alkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups: hydroxyl, mercapto, amino, cyano, R3, —OR3, —SR3, —N(R3)2, ═NOR3, —OCOR3, —SCOR3, —NR3COR3, —CO2R3, —COSR3, —CON(R3)2, C1-C4-alkyliminooxy, C1-C4-alkoxyamino, C1-C4-alkylcarbonyl, C1-C4-alkoxy-C2-C6-alkoxycarbonyl, C1-C4-alkylsulfonyl, heterocyclyl, heterocyclyloxy, phenyl, benzyl, hetaryl, phenoxy, benzyloxy and hetaryloxy, where the eight last mentioned radic
    Type: Grant
    Filed: February 7, 2000
    Date of Patent: May 6, 2003
    Assignee: BASF Aktiengesellschaft
    Inventors: Stefan Engel, Joachim Rheinheimer, Ernst Baumann, Wolfgang von Deyn, Regina Luise Hill, Guido Mayer, Ulf Misslitz, Oliver Wagner, Matthias Witschel, Martina Otten, Helmut Walter, Karl-Otto Westphalen
  • Patent number: 6525000
    Abstract: A process for preparing fused triazoles of formula I where: X—X is C—O, C—S, C—SO, C—SO2, or C—NR1; V is C═W2, R1R2C—C(═W2)— or C(═V2)—C(═W2); W1, W2 are oxygen or sulfur; which comprises reacting substituted N-aminoureas are reacted with formaldehyde or paraformaldehyde to give the corresponding methyleneimino ureas; cyclizing these in the presence of catalytic amounts of acid or metal oxide to give tetrahydro-4H-1,3,4-oxa(or thia)diazines, and cyclizing the fused triazoles using phosgene or a phosgene substitute.
    Type: Grant
    Filed: December 18, 2000
    Date of Patent: February 25, 2003
    Assignee: BASF Aktiengesellschaft
    Inventors: Gerhard Hamprecht, Olaf Menke, Robert Reinhard, Peter Schäfer, Cyrill Zagar, Martina Otten, Karl-Otto Westphalen, Helmut Walter