1,3,4-thiadiazoles (including Hydrogenated) Patents (Class 504/263)
  • Patent number: 9722184
    Abstract: A thiadiazole contains a basic skeleton represented by any of formulae (1), (2), and (3) in the molecule.
    Type: Grant
    Filed: October 16, 2013
    Date of Patent: August 1, 2017
    Assignee: SEIKO EPSON CORPORATION
    Inventors: Tetsuji Fujita, Hidetoshi Yamamoto
  • Patent number: 9650345
    Abstract: The present invention provides a process for the preparation of N-alkylated fluorine-containing pyrazolecarboxylic acid derivatives of Formula I. The present invention further provides a pyrazole compound of formula IIIa.
    Type: Grant
    Filed: May 2, 2016
    Date of Patent: May 16, 2017
    Assignee: SRF LIMITED
    Inventors: Srikant Dakshinamoorthy, Thangaselvam Kamaraj, Sarathy Iyengar, Arumugam Nagappan, Rahul Saxena, Rajdeep Anand
  • Publication number: 20140323305
    Abstract: The present invention relates to the use of strobilurine type compounds of formula I and the N-oxides and the salts thereof for combating phytopathogenic fungi containing a mutation in the mitochondrial cytochrome b gene conferring resistance to Qo inhibitors, and to methods for combating such fungi. The invention also relates to novel compounds, processes for preparing these compounds, to compositions comprising at least one such compound, to plant health applications, and to seeds coated with at least one such compound.
    Type: Application
    Filed: December 6, 2012
    Publication date: October 30, 2014
    Applicant: BASF SE
    Inventors: Joachim Rheinheimer, Violeta Terteryan, Stefan Redlich, Doris Kremzow, Claudia Rosenbaum, Sebastian Georgios Rohrer, Wassilios Grammenos, Christian Pilger, Franz Roehl, Markus Gewehr, Gerd Stammler, Jurith Montag, Hubert Sauter
  • Patent number: 8809547
    Abstract: The present application relates to the use of heterocyclic compounds, some of which are known, for controlling animal pests, including arthropods and in particular insects, furthermore to novel heterocyclic compounds and to processes for their preparation.
    Type: Grant
    Filed: July 4, 2009
    Date of Patent: August 19, 2014
    Assignee: Bayer CropScience AG
    Inventors: Thomas Bretschneider, Eva-Maria Franken, Ulrich Görgens, Martin Füβlein, Achim Hense, Joachim Kluth, Hans-Georg Schwarz, Adeline Köhler, Olga Malsam, Arnd Voerste, Angela Becker
  • Publication number: 20140013654
    Abstract: Ready-to-use foamable pesticide compositions that contain a particulate pesticide suspended therein and applicators for dispensing such compositions. Methods for treating pests such as arthropods by contacting pests with such compositions are also provided.
    Type: Application
    Filed: September 17, 2013
    Publication date: January 16, 2014
    Inventor: Terrence R. Burke
  • Publication number: 20130324409
    Abstract: The present invention provides methods of regulating plant stress tolerance.
    Type: Application
    Filed: March 14, 2013
    Publication date: December 5, 2013
    Inventors: SEAN R. CUTLER, ANDREW DEFRIES
  • Publication number: 20120289403
    Abstract: The invention relates to alkylsulfide derivatives compounds of formula I as hereunder depicted or the enantiomers or veterinarily acceptable salts thereof which are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to methods for controlling invertebrate pests by using these compounds and to plant propagation material and to agricultural and veterinary compositions comprising said compounds. wherein U, R1, R2, R3U, X, n and p are defined as in the description.
    Type: Application
    Filed: November 11, 2010
    Publication date: November 15, 2012
    Inventors: Sebastian Soergel, Ralph Paulini, Steffen Gross, Carsten Beyer, Matthias Pohlman, Henricus Maria Martinus Bastiaans, Michael Rack, Deborah L. Culbertson, Douglas D. Anspaugh, Sarah Thompson, Vincent Salgado
  • Publication number: 20120283100
    Abstract: The invention disclosed in this document concerns controlling planthoppers.
    Type: Application
    Filed: May 4, 2012
    Publication date: November 8, 2012
    Applicant: DOW AGROSCIENCES LLC
    Inventors: Agamananda Roy, Sanjoy Kundu, Suresh Ramachandran
  • Publication number: 20110195844
    Abstract: A process for solubilizing hydrophobic active ingredients in aqueous medium, which comprises using, as an assistant, at least one hyperbranched polymer (A) which is obtainable by reacting at least one hyperbranched polymeric compound having at least one primary or secondary amino group per molecule (a), selected from (a1) hyperbranched polyamides and (a2) hyperbranched polyureas, with (b) at least one mono-, di- or oligosaccharide.
    Type: Application
    Filed: February 4, 2011
    Publication date: August 11, 2011
    Applicant: BASF SE
    Inventors: Bernd Bruchmann, Holger Türk, Daniel Schönfelder, Monika Haberecht, Dietmar Appelhans, Victor Boyko
  • Patent number: 7820595
    Abstract: Penoxsulam, 2-(2,2-difluoroethoxy)-N-(5,8-dimethoxy[1,2,4]-triazolo[1,5-c]pyrimidin-2-yl)-6-(trifluoromethyl)benzenesulfonamide, provides synergistic herbicidal control with dicamba, the mixture of 2,4-D, triclopyr and clopyralid, or the mixture of 2,4-D and mecoprop-P.
    Type: Grant
    Filed: October 15, 2008
    Date of Patent: October 26, 2010
    Assignee: Dow AgroSciences LLC
    Inventors: Daniel L. Loughner, Anita L. Alexander, Toshiya Ogawa, James M. Breuninger
  • Publication number: 20100261606
    Abstract: The use of mixtures of different plant protectant active substance granule particles which remain homogeneous upon storage, handling and application, for the stable storage of mixing-incompatible active substances, and a preparation process therefor.
    Type: Application
    Filed: October 28, 2008
    Publication date: October 14, 2010
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Smita Patel, Mohammad Atiur Rahman
  • Publication number: 20100152044
    Abstract: The present invention relates to the use of a compound for plant growth regulation, preferably by application of the compound to plants, to the seeds from which they grow or to the locus in which they grow, in an effective plant growth regulating, preferably non-phytotoxic amount, which compound is a 3,4-disubstituted maleimide derivative of formula (I) or an agriculturally acceptable salt thereof, wherein: X is aryl or heteroaryl which groups are unsubstituted or substituted; Y is NH or a covalent bond; and Z is aryl or heteroaryl which groups are unsubstituted or substituted and a method for treatment of plants with such compounds in order to induce growth regulating responses.
    Type: Application
    Filed: April 30, 2005
    Publication date: June 17, 2010
    Applicant: Bayer CropScience GmbH
    Inventors: Henricus M.M. Bastiaans, Günter Donn, Nathalie Knittel, Arianna Martelletti, Richard Rees, Michael Schwall, Ryan Whitford
  • Publication number: 20100113276
    Abstract: The use of N2-phenylamidines of formula (I) as herbicides is described. In this formula (I), R2, R3, R4, R5 and R6 are different radicals and A is a bond or various 1- or polyatomic bridging elements.
    Type: Application
    Filed: March 4, 2008
    Publication date: May 6, 2010
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Birgit Kuhn, Harald Jakobi, Thomas Mueller, Joerg Tiebes, Heinz Kehne, Dirk Schmutzler, Martin Hills, Christopher Rosinger, Klaus Kunz, Mark Wilheim Drewes, Dieter Feucht, Thomas Seitz, Benoit Hartmann, Ralf Dunkel, Joerg Nico Greul, Oliver Guth, Kerstein Ilg, Darren James Mansfeld, Wahed Ahmed Moradi, Peter Dahmen, Ulrike Wachendorf-Neumann, Arnd Voerste, Dale Robert Mitchell, Jean-Pierre Andre Vors, Dale Robert Mitchell, Tom Hough
  • Patent number: 7189679
    Abstract: 3-Amino-2-thiomethylbenzoylpyrazoles of the formula (I) and their use as herbicides are described. In this formula (I) R1 to R9 are various radicals.
    Type: Grant
    Filed: April 1, 2005
    Date of Patent: March 13, 2007
    Assignee: Bayer CropScience GmbH
    Inventors: Monika Schmitt, Andreas van Almsick, Lothar Willms, Thomas Auler, Heinz Kehne, Martin Hills, Dieter Feucht
  • Patent number: 6967188
    Abstract: The invention relates to novel herbicidal synergistic active compound combinations comprising heteroaryloxy-acetamides and known herbicidally active compounds and/or safeners described in the description and their use for the selective control of weeds in crops of various useful plants.
    Type: Grant
    Filed: May 9, 2001
    Date of Patent: November 22, 2005
    Assignee: Bayer Cropscience AG
    Inventors: Dieter Feucht, Peter Dahmen, Mark Wilhelm Drewes, Rolf Pontzen, Mathias Kremer
  • Patent number: 6878675
    Abstract: The invention relates to a composition comprising (a) 2-(2?-nitro-4?-methylsulfonylbenzoyl)-1,3-cyclohexanedione, or an agriculturally acceptable salt or metal complex thereof; and (b) N-isopropyl-(5-trifluoromethyl-1,3,4-thiadiazol-2-yl)-4-(4?-fluoro-oxycetanilide); and their use as herbicides.
    Type: Grant
    Filed: September 17, 2001
    Date of Patent: April 12, 2005
    Assignee: Bayer CropScience S.A.
    Inventors: Ken Pallett, Ashley Slater
  • Patent number: 6849579
    Abstract: A selective synergistic postemergent herbicide composition is provided for the control of undesired broadleaf vegetation and grassyweeds comprising the combination of quinclorac and a selective herbicidal protox inhibitor. About 0.05 part to about 0.1 part by weight of the protox inhibitor is provided for each part by weight of quinclorac. Better synergistic results are obtained from the combination of quinclorac, a selective herbicidal protox inhibitor, and a selective herbicidal auxinic agent. About 0.05 part to about 0.1 part by weight of the protox inhibitor is provided for each part by weight of quinclorac, and about 1 part to about 4 parts by weight of the auxinic herbicidal agent for each part by weight of quinclorac. The synergistic composition hereof has been found to provide more rapid and better control of grassy weeds such as crabgrass than presently registered herbicides.
    Type: Grant
    Filed: June 25, 2003
    Date of Patent: February 1, 2005
    Assignee: PBI Gordon Corporation
    Inventors: James A. Armbruster, Dale R. Sanson
  • Patent number: 6835694
    Abstract: A method for controlling the growth of weeds at a locus which comprises applying to the locus an effective amount of: (a) a urea herbicide of general formula (1); and (b) 2-(2′-nitro-4′-methylsulfonylbenzoyl)-1,3-cyclohexanedione or an agriculturally acceptable salt or metal complex thereof.
    Type: Grant
    Filed: October 2, 2003
    Date of Patent: December 28, 2004
    Assignee: Bayer CropScience S.A.
    Inventors: Ken Pallett, Ashley Slater
  • Publication number: 20040157740
    Abstract: The invention relates to novel heterocyclylphenyl benzyl ethers, to a process for their preparation and to their use for controlling harmful organisms.
    Type: Application
    Filed: November 12, 2003
    Publication date: August 12, 2004
    Inventors: Fritz Maurer, Ulrich Heinemann, Bernd-Wieland Kruger, Herbert Gayer, Christiane Boie, Astrid Mauler-Machnik, Ulrike Wachendorff-Neumann
  • Publication number: 20030220197
    Abstract: Novel isothiazole derivatives of the formula (I) wherein A represents a group selected from (1), (2) and (3) in which R1, R2, R3, R4 and R5 have the meanings given in the specification processes for the preparation of the novel compounds and their use as microbicides.
    Type: Application
    Filed: October 9, 2002
    Publication date: November 27, 2003
    Inventors: Yoshinori Kitagawa, Koichi Ishikawa, Haruko Sawada, Yasuo Araki, Takuma Shigyo, Lutz Assmann
  • Patent number: 6642180
    Abstract: The present invention relates to novel biphenyl-substituted cyclic ketoenols of the formula (I) in which W represents hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, Z represents hydrogen, halogen, alkyl, alkoxy, halogenoalkyl or halogenoalkoxy, CKE represents one of the groups  in which A, B, D, L, M, Q1, Q2, Q3, Q4, Q5 and Q6 are as defined in the description, to preparation and to their use as pesticides and herbicides.
    Type: Grant
    Filed: January 25, 2002
    Date of Patent: November 4, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Reiner Fischer, Alan Graff, Thomas Bretschneider, Christoph Erdelen, Mark Wilhelm Drewes, Dieter Feucht
  • Patent number: 6632775
    Abstract: A herbicidal composition, comprising: (a) at least one arylthiadiazole having the formula (I):  wherein: R represents linear or branched C1-C6 alkyl or haloalkyl; or C3-C5 cycloalkyl or halocycloalkyl; said alkyl, haloalkyl, cycloalkyl or halocycloalkyl being optionally substituted with linear or branched C1-C3 alkyl; X represents halogen; Y represents halogen; linear or branched C1-C4 alkyl or haloalkyl; linear or branched C1-C4 alkoxyl or haloalkoxyl; R1 represents hydrogen or methyl; and (b) one or more herbicidal compounds.
    Type: Grant
    Filed: December 3, 1999
    Date of Patent: October 14, 2003
    Assignee: Isagro Ricerca S.r.L.
    Inventors: Franco Bettarini, Ernesto Signorini, Piero La Porta, Sergio Massimini, Domenico Portoso
  • Publication number: 20030148890
    Abstract: The invention relate to compounds of formula (I) in which R1, R2, R1, X1, X2 and X3 are as defined in claim 1, and to any enantiomers thereof. The active substances have advantageous pesticidal properties. They are particularly suitable for controlling pests in domestic and useful animals.
    Type: Application
    Filed: May 31, 2002
    Publication date: August 7, 2003
    Inventors: Pierre Ducray, Jacques Bouvier, Maurizio Schwarzenbach
  • Patent number: 6602827
    Abstract: The invention relates to novel 5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl-oxyacetanilides of the general formula (I) in which n represents the number 0, 1, 2 or 3, R represents straight-chain or branched alkyl having 1 to 4 carbon atoms, and X represents nitro, cyano, halogen or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylthio, alkylsulphinyl or alkylsulphonyl having in each case 1 to 4 carbon atoms, except for the compounds N-methyl-5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl-oxyacetanilide, N-ethyl-5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl-oxyacetanilide, 4-chloro-N-methyl-(5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl)-oxyacetanilide and 3-trifluoromethyl-N-methyl-(5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl)-oxyacetanilide, N-i-propyl-5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl-oxyacetanilide, and 4-fluoro-N-methyl-(5-chlorodifluoromethyl-1,3,4-thiadiazol-2-yl)-oxyacetanilide and 4-fluoro-N-ethyl-(5-chlorodifluoromethyl-1
    Type: Grant
    Filed: January 24, 2002
    Date of Patent: August 5, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hans-Jochem Riebel, Heinz Förster, Mark Wilhelm Drewes, Peter Dahmen, Dieter Feucht, Rolf Pontzen
  • Patent number: 6589914
    Abstract: The dihalopropene compounds of the general formula (I) have excellent insecticidal/acaricidal activity, so that they are satisfactorily effective for the control of noxious insects, mites and ticks.
    Type: Grant
    Filed: March 4, 2002
    Date of Patent: July 8, 2003
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Noriyasu Sakamoto, Sanshiro Matsuo, Masaya Suzuki, Taro Hirose, Kazunori Tsushima, Kimitoshi Umeda
  • Patent number: 6559100
    Abstract: Substituted 2-benzoylcyclohexane-1,3-diones of the formula I where: R1 and R2 are each hydrogen, mercapto, nitro, halogen, cyano, thiocyanato, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl, C2-C6-alkynyl, —OR3, —OCOR3, —OSO2R3, —S(O)nR3, —SO2OR3, —SO2N(R3)2, —NR3SO2R3 or —NR3COR3; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, phenyl or phenyl-C1-C6-alkyl; where the abovementioned alkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups: hydroxyl, mercapto, amino, cyano, R3, —OR3, —SR3, —N(R3)2, ═NOR3, —OCOR3, —SCOR3, —NR3COR3, —CO2R3, —COSR3, —CON(R3)2, C1-C4-alkyliminooxy, C1-C4-alkoxyamino, C1-C4-alkylcarbonyl, C1-C4-alkoxy-C2-C6-alkoxycarbonyl, C1-C4-alkylsulfonyl, heterocyclyl, heterocyclyloxy, phenyl, benzyl, hetaryl, phenoxy, benzyloxy and hetaryloxy, where the eight last mentioned radic
    Type: Grant
    Filed: February 7, 2000
    Date of Patent: May 6, 2003
    Assignee: BASF Aktiengesellschaft
    Inventors: Stefan Engel, Joachim Rheinheimer, Ernst Baumann, Wolfgang von Deyn, Regina Luise Hill, Guido Mayer, Ulf Misslitz, Oliver Wagner, Matthias Witschel, Martina Otten, Helmut Walter, Karl-Otto Westphalen
  • Patent number: 6544931
    Abstract: The invention relates to novel substituted heteroaryloxyacetanilides of the general formula (I), in which n, R, X, and Z are to intermediates for their preparation and to their use as herbicides.
    Type: Grant
    Filed: January 16, 2002
    Date of Patent: April 8, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus-Helmut Müller, Lothar Rohe, Joachim Kluth, Mark Wilhelm Drewes, Peter Dahmen, Dieter Feucht, Rolf Pontzen
  • Publication number: 20020025910
    Abstract: Benzoyl derivatives of the formula I 1
    Type: Application
    Filed: December 27, 2000
    Publication date: February 28, 2002
    Inventors: Wolfgang von Deyn, Regina Luise Hill, Uwe Kardorff, Ernst Baumann, Stefan Engel, Guido Mayer, Matthias Witschel, Michael Rack, Norbert Gotz, Joachim Gebhardt, Ulf MiBlitz, Helmut Walter, Karl-Otto Westphalen, Martina Otten, Joachim Rheinheimer
  • Patent number: 6339042
    Abstract: The novel compounds of formula I: wherein Het represents an optionally substituted, optionally benzofused nitrogen containing 5- or 6-membered heteroaromatic group; R1 represents an alkyl, alkoxyalkyl or cycloalkyl group; R2 each independently represent an alkyl or alkenyl group, and m is 0 or an integer from 1 to 6, and herbicidal compositions containing such compounds as active ingredients can be utilized in various agricultural methods.
    Type: Grant
    Filed: November 29, 1999
    Date of Patent: January 15, 2002
    Assignee: American Cyanamid Co.
    Inventors: Trevor Newton, Helmut Siegfried Baltruschat
  • Patent number: 6316389
    Abstract: Compounds of the formula I in which: where: X is CH or N; Y is O; S, S═O or NR5; Z is OR2, SR2, N(R3)R4; or Y and Z together form 5- to 7-membered ring which contains, 2 or 3 hetero atoms O and/or N and which is unsubstituted or substituted by C1-C4alkyl, halo-C1-C4alkyl, halogen, ═O or cyclopropyl; V is a direct bond or C1-C6alkylene, which is unsubstituted or substituted by C1-C3alkyl, C2-C3alkylidene or C3-C6cycloalkylidene; U is O, S, NR7, SO or SO2; W is substituted or unsubstituted aryl or substituted or unsubstituted heteroaryl; R1 is cyclopropyl, C1C6alkyl or halo-C1-C6alkyl; R2 and R3 independently of one another are C1-C6alkyl or halo-C1-C6alkyl; R4 and R5 independently of one another are hydrogen, C1-C6alkyl or C1-C6alkoxy; R7 is hydrogen, C1-C6alkyl, benzyl, C1-C6alkylcarbonyl, halo-C1-C6alkylcarbonyl, halo-C2-C6alkenylcarbonyl; R21 and R22 independently of one another are hydrogen, halogen, C1-C8alkyl or C1-C8alkoxy or C1-C8alkylthio; R23, R24, R25, R26 i
    Type: Grant
    Filed: June 16, 1997
    Date of Patent: November 13, 2001
    Assignee: Bayer Aktiengesellschaft
    Inventors: Henry Szczepanski, Martin Zeller, Ottmar Franz Hüter
  • Patent number: 6265351
    Abstract: The invention relates to phenylpyrazoles having general formula (I): The compounds having formula (I) have a high herbicidal activity and are used for controlling weeds in the agronomic field.
    Type: Grant
    Filed: August 3, 2000
    Date of Patent: July 24, 2001
    Assignee: Isagro Ricerca S.r.L.
    Inventors: Piero La Porta, Franco Bettarini, Giovanni Meazza, Gregorio Valea, Ernesto Signorini, Domenico Portoso
  • Patent number: 6232470
    Abstract: Substituted Pyrazol-3-ylbenzazoles I salts thereof, and their use as herbicides or for the desiccation/defoliation of plants.
    Type: Grant
    Filed: June 16, 1999
    Date of Patent: May 15, 2001
    Assignee: BASF Aktiengesellschaft
    Inventors: Cyrill Zagar, Gerhard Hamprecht, Markus Menges, Olaf Menke, Peter Schäfer, Karl-Otto Westphalen, Ulf Misslitz, Helmut Walter
  • Patent number: 6004903
    Abstract: Benzoyl derivatives of the formula I ##STR1## where Z is a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen,Q is a cyclohexane-1, 3-dione ring bonded in the 2-position and of the formula II, ##STR2## or conventional agricultural salts of the compounds I.
    Type: Grant
    Filed: August 14, 1997
    Date of Patent: December 21, 1999
    Assignee: Basf Aktiengesellschaft
    Inventors: Wolfgang von Deyn, Regina Luise Hill, Uwe Kardorff, Stefan Engel, Martina Otten, Marcus Vossen, Peter Plath, Harald Rang, Albrecht Harreus, Franz Rohl, Helmut Walter, Karl-Otto Westphalen, Ulf Misslitz
  • Patent number: 5945379
    Abstract: Heteroaryloxy-acetamides of the general formula (I) ##STR1## in which Het represents thiadiazolyl which is substituted by halogen or by C.sub.1 -C.sub.4 -alkyl or phenyl, each of which is optionally substituted by halogen, andAr represents optionally halogen-, C.sub.1 -C.sub.4 -alkyl- or C.sub.1 -C.sub.4 -halogenoalkyl-substituted phenyl.can be used with good results as selective herbicides in rice cultivation.The novel herbicidal active compound combinations comprising (1) a heteroaryloxy-acetamide of the formula (I) above and (2) in each case one active compound from the group of already known selective rice herbicides (e.g. bensulfuron, MCPB, and thiobencarb) exhibit, at certain weight ratios, synergistic activities and can be used particularly advantageously as selective herbicides in rice crops.
    Type: Grant
    Filed: May 15, 1997
    Date of Patent: August 31, 1999
    Assignee: Bayer Aktiengesellschaft
    Inventors: Markus Dollinger, Dieter Feucht, Helmut Fursch
  • Patent number: 5888941
    Abstract: Compounds of general formula I and their salts and solvates are antifungal agents and as such are useful in the treatment of various fungal infections. Pharmaceutical compositions including these compounds and processes for their preparation are also provided.
    Type: Grant
    Filed: March 31, 1997
    Date of Patent: March 30, 1999
    Assignee: J. Uriach & Cia. S.A.
    Inventors: Javier Bartroli, Enric Turmo, Manuel Anguita
  • Patent number: 5874382
    Abstract: Compounds of Formula I and II, and their agriculturally-suitable salts, are disclosed which are useful for controlling undesired vegetation ##STR1## wherein X is a direct bond; O; S; NH; N(C.sub.1 -C.sub.3 alkyl); N(C.sub.1 -C.sub.3 haloalkyl); or N(allyl);R.sup.1 is H; F; Cl; or Br;R.sup.2 is H; F; Cl; Br; CF.sub.3 ; nitro; or cyano;R.sup.4 is H; C.sub.1 -C.sub.3 alkyl; or halogen;R.sup.5 is H; C.sub.1 -C.sub.6 alkyl; C.sub.1 -C.sub.6 haloalkyl; halogen; S(O).sub.2 (C.sub.1 -C.sub.6 alkyl); or C(.dbd.O)R.sup.8 ; orR.sup.4 and R.sup.5 are taken together along with the carbon to which they are attached to form a spiro-cyclopropane ring;and R.sup.3, R.sup.8, and J are as defined in the disclosure.Also disclosed are compositions containing the compounds of Formulae I and II and a method for controlling undesired vegetation which involves contacting the vegetation or its environment with an effective amount of a compound of Formula I or II.
    Type: Grant
    Filed: January 23, 1998
    Date of Patent: February 23, 1999
    Assignee: E. I. du Pont de Nemours and Company
    Inventors: Balreddy Kamireddy, William Mark Murray
  • Patent number: 5846906
    Abstract: Herbicidally active phenyldiketone compounds of the formula I ##STR1## in which the substituents have the following meanings: L and M are hydrogen, C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkynyl, C.sub.1 -C.sub.4 -alkoxy, it being possible for these groups to be unsubstituted or substituted by one to five halogen atoms or C.sub.1 -C.sub.4 -alkoxy, or halogen, cyano, nitro, a group --(Y).sub.n --S(O).sub.m R.sup.7 or a group --(Y).sub.n --CO--R.sup.8,Z is a 5- or 6-membered heterocyclic saturated or unsaturated radical which has one to three hetero atoms selected from the group consisting of oxygen, sulfur or nitrogen and which is unsubstituted or substituted by halogen, cyano, nitro, a group --CO--R.sup.8, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkylthio, di-C.sub.1 -C.sub.
    Type: Grant
    Filed: July 30, 1997
    Date of Patent: December 8, 1998
    Assignee: BASF Aktiengesellschaft
    Inventors: Wolfgang von Deyn, Regina Luise Hill, Uwe Kardorff, Stefan Engel, Martina Otten, Marcus Vossen, Peter Plath, Harald Rang, Albrecht Harreus, Hartmann Konig, Helmut Walter, Karl-Otto Westphalen, Ulf Misslitz
  • Patent number: 5821197
    Abstract: Arylthiadiazolones having formula (I): ##STR1## have a high herbicidal activity and are used for controlling weeds in agricultural cultivations.
    Type: Grant
    Filed: September 25, 1997
    Date of Patent: October 13, 1998
    Assignee: Isagro Ricerca S.r.l.
    Inventors: Franco Bettarini, Piero La Porta, Sergio Massimini, Ernesto Signorini, Domenico Portoso
  • Patent number: 5780392
    Abstract: This invention concerns heterocyclyl-1,3,4-thiadiazolyloxycetamides of the formula ##STR1## in which R.sup.1 is hydrogen or optionally substituted alkyl, alkenyl, alkinyl or aralkyl, R.sup.2 is optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, aralkyl, aryl, alkoxy, alkenyloxy or alkinyloxy or R.sup.1 and R.sup.2, together with the nitrogen atom to which they are bound, form an optionally substituted, saturated or unsaturated nitrogen heterocycle which may contain other hetero-atoms and to which a benzo-grouping can be fused, and Het is an optionally substituted heterocyclyl group with the exception of thienyl. The Invention also concerns a method of preparing such compounds, intermediates used in their preparation and the use of such compounds as herbicides.
    Type: Grant
    Filed: October 4, 1996
    Date of Patent: July 14, 1998
    Assignee: Bayer Aktiengesellschaft
    Inventors: Heinz Forster, Hans-Joachim Diehr, Hans-Joachim Santel, Markus Dollinger
  • Patent number: 5767041
    Abstract: The invention relates to new substituted aryliminoheterocycles of the general formula (I) ##STR1## in which A represents oxygen, sulphur or the group N--R.sup.1 whereR.sup.1 represents hydrogen or in each case optionally substituted alkyl, alkenyl or akinyl,E represents one of the following groups ##STR2## where Q represents oxygen, sulphur or the group N--R.sup.1 (where R.sup.1 has the abovementioned meaning) andR.sup.2 represents hydrogen, cyano or in each case optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl or cycloalkenyl,R represents hydrogen or in each case optionally substituted alkyl, alkenyl or alkinyl, andAr represents in each case optionally substituted monocyclic or bicyclic aryl or heteroaryl,to processes for their preparation and to their use as herbicides.
    Type: Grant
    Filed: January 7, 1997
    Date of Patent: June 16, 1998
    Assignee: Bayer Aktiengesellschaft
    Inventors: Otto Schallner, Andreas Lender, Hans-Joachim Santel, Markus Dollinger
  • Patent number: 5712225
    Abstract: The present invention relates to oxa(di)azabicyclic and thia(di)azabicyclic compounds, a method for their preparation and their use as herbicides.
    Type: Grant
    Filed: February 28, 1996
    Date of Patent: January 27, 1998
    Assignees: E. I. du Pont de Nemours and Company, Degussa Aktiengesellschaft
    Inventors: Wonpyo Hong, Matthias Schafer, Thomas Martin Stevenson
  • Patent number: 5679623
    Abstract: Compounds of the formula ##STR1## in which R.sub.l, R.sub.2, R.sub.3, R.sub.4, Y and Z are as defined in claim 1, and, if appropriate, the tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.
    Type: Grant
    Filed: June 2, 1995
    Date of Patent: October 21, 1997
    Assignee: Ciba-Geigy Corporation
    Inventors: Henry Szczepanski, Haukur Kristinsson
  • Patent number: 5591695
    Abstract: Novel herbicidal compounds of the general formula I ##STR1## wherein X represents an oxygen or sulphur atom; A represents an optionally substituted alkyl, alkenyl, cycloalkyl, cycloalkenyl, dialkylamino, aryl, heteroaryl, aralkyl or heteroalkyl group; R.sup.1 represents a hydrogen atom, an optionally substituted alkyl group or an optionally substituted acyl group; and R.sup.2 represents an optionally substituted aralkyl or heteroaralkyl group; together with their preparation, formulation and use.
    Type: Grant
    Filed: May 24, 1995
    Date of Patent: January 7, 1997
    Assignee: American Cyanamid Co.
    Inventor: Trevor W. Newton
  • Patent number: 5589439
    Abstract: Herbicidal novel tetrazolinone derivatives of the formula: ##STR1## wherein R.sup.1 is alkyl, haloalkyl, cycloalkyl, alkenyl, haloalkenyl, alkynyl, alkoxy or phenyl which is optionally substituted, andR.sup.2 is alkyl, haloalkyl, cycloalkyl, alkenyl, haloalkenyl, alkynyl, alkoxy or phenyl which is optionally substituted, orR.sup.1 and R.sup.2 form, together with the nitrogen atom to which R.sup.1 and R.sup.2 are bonded, a 5- or 6-membered heterocyclic ring, optionally fused to a carbocyclic ring optionally and independently substituted by C.sub.1-4 alkyl, andR.sup.3 is a 5-membered heterocyclic radical containing at least one hereto atom selected from the group consisting of nitrogen, oxygen, and sulfur, optionally substituted by at least one substitutent selected from the group consisting of halogen, benzyl, phenyl, halogen-substituted phenyl, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 haloalkyl, C.sub.1-4 haloalkoxy, C.sub.1-4 alkylthio, C.sub.1-4 alkyl-sulfonyl and C.sub.
    Type: Grant
    Filed: July 28, 1995
    Date of Patent: December 31, 1996
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Toshio Goto, Koichi Moriya, Fritz Maurer, Seishi Ito, Katsuaki Wada, Kazuhiro Ukawa, Ryo Watanabe, Asami Ito, Natsuko Minegishi
  • Patent number: 5573999
    Abstract: .beta.-Substituted cinnamic acid derivatives of the formula 1, ##STR1## where R.sup.1 is alkyl, chlorine or bromine, --X-- is --O--, --S--, ##STR2## m is 0 or 1, --Y is --OR.sup.4, --O--N.dbd.CR.sup.5 R.sup.6, --NR.sup.7 R.sup.8, --N(OR.sup.9)R.sup.10 or --SR.sup.11, where the above-mentioned substituents R.sup.2 to R.sup.11 are alkyl, and R.sup.2, and R.sup.3 and R.sup.5 to R.sup.11 can also be hydrogen,Z is halogen, nitro, cyano, alkyl, cycloalkyl, aralkyl, aryloxyalkyl, arylthioalkyl, hetarylalkyl, hetaryloxyalkyl, hetarylthioalkyl, alkenyl, aralkenyl, aryloxyalkenyl, arylthioalkenyl, hetarylalkenyl, hetaryloxyalkenyl, hetarylthioalkenyl, alkynyl, arylalkynyl, hetarylalkynyl, aryl, hetaryl, arylazo, acylamino, --OR.sup.12, --SR.sup.13, --SOR.sup.14, --SO.sub.2 R.sup.15, --COOR.sup.16, --CONR.sup.17 R.sup.18, --COR.sup.19, --CR.sup.20 .dbd.NR.sup.21, --N.dbd.CR.sup.22, R.sup.23, --CR.sup.24 .dbd.N--OR.sup.25, --CR.sup.25 R.sup.26 --O--, N.dbd.CR.sup.27 R.sup.28, --CH.sub.2 --OCOR.sup.39 or --NR.sup.37 R.
    Type: Grant
    Filed: May 15, 1995
    Date of Patent: November 12, 1996
    Assignee: BASF Aktiengesellschaft
    Inventors: Hubert Sauter, Herbert Bayer, Klaus Oberdorf, Horst Wingert, Wolfgang von Deyn, Wassilios Grammenos, Hartmann Koenig, Harald Rang, Franz Roehl, Gisela Lorenz, Eberhard Ammermann
  • Patent number: 5538940
    Abstract: .beta.-Substituted cinnamic acid derivatives of the formula 1, ##STR1## where R.sup.1 is substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and R.sup.1 can also be chlorine or bromine,--X-- is --O--, --S--, ##STR2## m is 0 or 1, --Y is --OR.sup.4, --O--N.dbd.CR.sup.5 R.sup.6, --NR.sup.7 R.sup.8, --NR.sup.7 R.sup.8, --N(OR.sup.9)R.sup.10 or SR.sup.11, where the abovementioned substitutes R.sup.2 to R.sup.11 are substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and R.sup.2, R.sup.3 and R.sup.5 to R.sup.11 can be hydrogen and Z, U, V, W are defined in the specification.
    Type: Grant
    Filed: May 12, 1995
    Date of Patent: July 23, 1996
    Assignee: BASF Aktiengesellschaft
    Inventors: Hubert Sauter, Herbert Bayer, Klaus Oberdorf, Horst Wingert, Wolfgang Von Deyn, Wassilios Grammenos, Hartmann Koenig, Harald Rang, Franz Roehl, Gisela Lorenz, Eberhard Ammermann
  • Patent number: 5523278
    Abstract: There are provided substituted benzisoxazole and benzisothiazole compounds having the structural formula I ##STR1## Further provided are compositions and methods comprising those compounds for the control of undesirable plant species.
    Type: Grant
    Filed: September 12, 1995
    Date of Patent: June 4, 1996
    Assignee: American Cyanamid Company
    Inventor: Peter J. Wepplo
  • Patent number: 5494889
    Abstract: Thiadiazabicyclooctanes and thiadiazabicyclooctenes of formula I ##STR1## wherein the substituents are as defined herein, having good pre- and post-emergence selective herbicidal properties.
    Type: Grant
    Filed: December 2, 1993
    Date of Patent: February 27, 1996
    Assignee: Ciba-Geigy Corporation
    Inventors: Hans-Georg Brunner, Hans Moser, Georg Pissiotas
  • Patent number: 5484763
    Abstract: There are provided substituted benzisoxazole and benzisothiazole compounds having the structural formula I ##STR1## Further provided are compositions and methods comprising those compounds for the control of undesirable plant species.
    Type: Grant
    Filed: February 10, 1995
    Date of Patent: January 16, 1996
    Assignee: American Cyanamid Company
    Inventor: Peter J. Wepplo
  • Patent number: 5424443
    Abstract: The invention relates to new substituted benzothiazole derivatives of general formula (I), in which X, Y and Z have the meanings given in the description, processes for their preparation and their use as herbicides.
    Type: Grant
    Filed: January 24, 1994
    Date of Patent: June 13, 1995
    Assignee: Schering Aktiengesellschaft
    Inventors: Michael Ganzer, Gabriele Dorfmeister, Wilfried Franke, Gerhard Johann, Richard Rees