Abstract: This invention relates to novel phosphonic acid esters represented by the following general formula (I) ##STR1## wherein R.sup.1 represents a lower alkyl group or an aryl group,R.sup.2 represents a lower alkyl group or a lower alkoxy-lower alkyl group,R.sup.3 represents a fluoro-substituted lower alkyl group,X represents an oxygen or sulfur atom,Y represents an oxygen or sulfur atom or a group of the formula ##STR2## in which R.sup.4 represents a hydrogen atom or a lower alkyl group, Z represents a hydrogen atom, a halogen atom or a lower alkyl group, andn represents 0 or 2,which can be used as insecticidal, miticidal and nematocidal agents.
Abstract: The invention relates to new 4-aryl-2-methyl-1,2,3,4-tetrahydro-isoquinoline derivatives of the general Formula I ##STR1## and salts thereof whereinR stands for hydrogen, lower alkyl or halogen andX represents a group of the general Formula --(CH.sub.2).sub.n --NR.sup.1 R.sup.2, --NH--R.sup.3 or --OR.sup.4, in whichR.sup.1 and R.sup.2 may be the same or different and stand for hydrogen or lower alkyl or R.sup.1 and R.sup.2 together with the adjacent nitrogen atom, they are attached to, form a 5- or 6-membered saturated heterocyclic ring which may optionally contain a further oxygen or sulfur atom or an optionally lower alkyl substituted imino group;n is an integral number 1, 2, 3 or 4;R.sup.3 stands for lower alkyl or optionally substituted phenyl andR.sup.4 is lower alkyl, halogeno lower alkyl, or phenyl lower alkyl.The compounds of the general Formula I are useful as antidepressants and antiparkinsone agents.The compounds of the general Formula I can be prepared by methods known per se.
Type:
Grant
Filed:
June 3, 1983
Date of Patent:
August 27, 1985
Assignee:
EGYT Gyogyszervegyeszeti Gyar
Inventors:
Gyula Deak, Erzsebet Zara nee Kaczian, Lajos Gyorgy, Marton Fekete, Margit Doda, Andras Seregi, Bela Kanyicska, Erzsebet Toth nee Pecsi, Maria Horvath nee Gaal, Sandor Manyai, Frigyes Gorgenyi, Gyorgyi Vaszovics nee Reichmann
Abstract: Organophosphate derivatives of the formula ##STR1## in which X is O, S or NH,Y is O or S,R.sup.1 is a lower alkyl group,R.sup.2 is a lower alkyl group or a lower alkoxy-lower alkyl group,R.sup.3 is a fluoro-substituted lower alkyl group, andn is 0 or 2.which possess pesticidal properties. The phenols of the phenyl esters are also new.
Abstract: A fungicidal composition which comprises as an active ingredient a fungicidally effective amount of a phosphoramidothionate of the formula: ##STR1## wherein R.sub.1 is a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a lower cycloalkyl group, a lower cycloalkyl(lower)alkyl group, a halogen atom-substituted lower alkyl group, a lower alkoxy(lower)alkyl group, a di(lower)alkoxy(lower)alkyl group, a cyano group-substituted lower alkyl group, a lower alkylthio(lower)alkyl group, a lower dioxothiacycloalkyl group, a lower thiacycloalkyl group, a lower oxacycloalkyl group, a furanyl(lower)alkyl group or a thiophenyl(lower)alkyl group, R.sub.2 is a lower alkyl group and R.sub.3 is a lower alkyl group or a lower alkoxy group, and an inert carrier or diluent.