Ring Attached Directly To Oxygen Of N-c(=0)-0 Patents (Class 514/490)
  • Patent number: 4985413
    Abstract: A composition which comprises (a) at least one insecticide selected from the group consisting of organic phosphorous insecticides, carbamate insecticides and pyrethroid insecticide, (b) crystalline cellulose and (c) crop product powders evaporated with (d) an essential oil and (e) a saccharide respectively in amounts of 0.1 to 10.0% by weight and 10.0 to 40.0% by weight based on the total weight of the composition, which is useful as a bait for the control of noxious insects.
    Type: Grant
    Filed: March 4, 1988
    Date of Patent: January 15, 1991
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Takuji Kohama, Fumiyasu Minagawa, Goro Shinjo, Kazuyuki Maeda
  • Patent number: 4963583
    Abstract: Novel 3-acyloxy-4-keto-.beta.-ionone derivatives of the formula I ##STR1## wherein Z is either the radical ##STR2## in which R.sub.1 represents C.sub.2 -C.sub.5 alkyl, C.sub.1 -C.sub.5 alkoxy-C.sub.1 -C.sub.5 alkyl having a maximum number of 6 carbon atoms, cyclopropyl or cyclopropyl which is substituted by methyl or by halogen or represents the radical ##STR3## wherein R.sub.2 represents C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 alkoxy-C.sub.1 -C.sub.5 alkyl having a maximum number of 6 carbon atoms, cyclopropyl or cyclopropyl which is substituted by methyl or by halogen and X represents either oxygen or sulphur, and ##STR4## display very effective microbicidal activity. They can especially be used in microbicidal compositions to control plant-pathogenic microorganisms, preferably fungi of the order Oomycetes.
    Type: Grant
    Filed: September 28, 1988
    Date of Patent: October 16, 1990
    Assignee: Ciba-Geigy Corporation
    Inventor: Walter Kunz
  • Patent number: 4948807
    Abstract: Phenyl carbamates of the general formula ##STR1## wherein R.sub.1 to R.sub.5 are as defined in the claims, are useful as pharmaceuticals.
    Type: Grant
    Filed: March 8, 1989
    Date of Patent: August 14, 1990
    Assignee: Proterra AG
    Inventors: Marta W. Rosin, Michael Chorev, Zeev Tashma
  • Patent number: 4939170
    Abstract: Fungicidal substituted aminophenyl carbamates of the formula ##STR1## in which X represents --CO--NR.sup.8 R.sup.9 ; --CO--OR.sup.9 ; --CO--SR.sup.9 ; --CO.sup.R.sup.10 ; --SO.sub.2 R.sup.9 or hydrogen, in whichR.sup.8 represents hydrogen or alkyl,R.sup.9 represents optionally substituted aryl, optionally substituted aralkyl, optionally substituted alkyl, alkenyl, halogenoalkenyl, or in each case optionally substituted cycloalkyl, cycloalkenyl or cycloalkylalkyl, andR.sup.10 has the meaning of R.sup.9 or represents an optionally substituted heterocyclic ring,Y.sup.1 to Y.sup.4 are identical or different and represent hydrogen, halogen, nitro, cyano, alkyl, halogenoalkyl, alkoxy, halogenoalkoxy, alkylthio, alkylsulfonyl or halogenoalkythio,R.sup.1 to R.sup.7 are identical or different and represent hydrogen, alkyl, halogenoalkyl or alkoxyalkyl,n represents 0 or 1, andZ represents alkyl, halogenoalkyl or a ##STR2## radical, in which R.sup.11 to R.sup.
    Type: Grant
    Filed: May 20, 1988
    Date of Patent: July 3, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventors: Bernd-Wieland Kruger, Klaus Sasse, Peter Heitkamper, Klaus Konig, Wilhelm Brandes, Gerd Hanssler, Albrecht Marhold
  • Patent number: 4935413
    Abstract: A physical property-improving reagent which comprises an alkenoylcarbamate compound of the formula: ##STR1## wherein R is a hydrogen atom or a lower alkyl group, X is an oxygen atom (--O--), a sulfur atom (--S--) or a substituted or unsubstituted imino group (--NR'--), R' being a hydrogen atom or a lower alkyl group, and Y is the residue of an active hydrogen atom-containing compound excluding --X-H therefrom dissolved in an organic solvent having a solubility parameter of not less than 8, which can impact excellent physical properties to a polymer produced with the same.
    Type: Grant
    Filed: June 5, 1987
    Date of Patent: June 19, 1990
    Assignee: Nippon Paint Co., Ltd.
    Inventors: Satoshi Urano, Ryuzo Mizuguchi, Noriyuki Tsuboniwa, Kei Aoki, Yuji Suzuki, Takeyasu Itoh
  • Patent number: 4933329
    Abstract: Novel bis-S-alkylbenzene derivatives capable of inhibiting lipoxygenase, inparticular, 5-lipoxygenase are disclosed. It is expected that the compounds, which are hardly metabolized in vivo, are highly useful in the treatment and/or prevention of various diseases, including allergic diseases such as asthma, inflammation, myocardial infarction, nephritis, scabies and gout.
    Type: Grant
    Filed: December 6, 1988
    Date of Patent: June 12, 1990
    Assignee: Green Cross Corporation
    Inventors: Youichiro Naito, Yasunari Yamaura, Masanori Sugiura, Chikara Fukaya, Kazumasa Yokoyama
  • Patent number: 4931466
    Abstract: A compound of the chemical formula (I) ##STR1## in a specific crystalline form, processes for its preparation, and its use for pest control.
    Type: Grant
    Filed: February 15, 1989
    Date of Patent: June 5, 1990
    Assignee: BASF Aktiengesellschaft
    Inventors: Siegfried Kersten, Karl-Friedrich Jaeger, Karl-Heinz Koenig, Albrecht Mueller, Josef B. Pawliczek, Hans-Gert Recker, Wolfgang Rohr, August Wigger
  • Patent number: 4925657
    Abstract: The invention provides insecticidal compositions for combatting aphids, which compositions contain an aphid insecticide in an amount lower than the minimum usual percentage for said insecticide in an aphicidal composition and an alarm pheromone for aphids. The compositions of the invention are less toxic because of the reduced insecticide content but they are not less effective than the insecticidal compositions which do not contain an alarm pheromone.
    Type: Grant
    Filed: June 29, 1987
    Date of Patent: May 15, 1990
    Assignee: Denka International B.V.
    Inventors: Antonie A. Den Braber, Evert R. Slootweg
  • Patent number: 4914124
    Abstract: A method of combating endoparasites which comprises applying thereto or to an endoparasite habitat an endoparasiticidally effective amount of an N-organooxycarbamic acid ester of the formula ##STR1## in which R.sup.1 represents alkyl, cycloalkyl, alkenyl, alkinyl or aryl, which can optionally be substituted,R.sup.2 represents alkyl, alkenyl or alkinyl, which can optionally be substituted, andR.sup.3 represents alkyl, alkenyl or alkinyl, which can optionally be substituted.Those compounds wherein one of R.sup.2 and R.sup.3 is alkinyl are new.
    Type: Grant
    Filed: January 25, 1988
    Date of Patent: April 3, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventors: Nikolaus Muller, Peter Andrews
  • Patent number: 4906653
    Abstract: A method for controlling molluscs with 2-(2-chloro-1-methoxyethoxy)phenyl methylcarbamate of the formula ##STR1## and molluscicides containing a mixture of 2-(2-chloro-1-methoxyethoxy)phenyl methylcarbamate with methyl benzimidazol-2-ylcarbamate is described.
    Type: Grant
    Filed: February 10, 1988
    Date of Patent: March 6, 1990
    Assignee: BASF Aktiengesellschaft
    Inventors: Karl Kiehs, Christoph Kuenast
  • Patent number: 4891385
    Abstract: Sprayable aqueous insecticidal solutions are disclosed based on a mixture of fatty acid amide emulsifiers which have been acidified to a pH of less than about 7 with a water soluble acid and thickening agents which are preferably cellulose based together with an active known insecticidal ingredient propoxur, the solutions having a final pH in the range of about 3.5 to 7.
    Type: Grant
    Filed: November 23, 1981
    Date of Patent: January 2, 1990
    Assignee: Mobay Corporation
    Inventor: Joseph Synek
  • Patent number: 4871766
    Abstract: An oil-in-water pesticidal emulsion which comprises one or more of hydrocarbons represented by the formula, ##STR1## wherein X.sub.1, X.sub.2, Y.sub.1, Y.sub.2, Z.sub.1 and Z.sub.2, which may be the same or different, represent a hydrogen atom or an alkyl group having two or less carbon atoms, R.sub.1 and R.sub.2, which may be the same or different, represent a hydrogen atom or a methyl group, and n represents 0 or 1, in an oil-in-water pesticidal emulsion containing an active ingredient having a pesticidal activity, of which the melting point is 0.degree. C. or higher and the solubility at 0.degree. C. in the hydrocarbons represented by the above formula is 10 wt. % or more (when two or more active ingredients are used together, said melting point and solubility shall be those of a mixture of these active ingredients).
    Type: Grant
    Filed: December 29, 1986
    Date of Patent: October 3, 1989
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Shigenori Tsuda, Yukio Manabe, Kozo Tsuji
  • Patent number: 4863909
    Abstract: New arthropodicidal synergistic mixtures comprising the known active compounds (I) the pyrethroid: .alpha.-cyano-3-phenoxy-4-fluoro-benzyl 2,2-dimethyl-3-dichlorovinyl-cyclopropanecarboxylate or .alpha.-cyano-3-phenoxybenzyl 2,2-dimethyl-3-dibromovinyl-cyclopropanecarboxylate (decamethrine) and (II) 0,0-dimethyl 0-2,2-dichlorovinyl phosphate (dichlorvos) and (III), if desired, 0-isopropoxyphenyl N-methylcarbamate (propoxur). The novel mixtures are particularly suitable for use in aerosols and oil sprays.
    Type: Grant
    Filed: February 13, 1985
    Date of Patent: September 5, 1989
    Assignee: Bayer Aktiengesellschaft
    Inventors: Wolfgang Behrenz, Manfred Schutte
  • Patent number: 4855140
    Abstract: O-(O-ethyl-S-alkylphosphoryl)-O-(carbamoyl)-pyrocatechol derivatives of the formula I ##STR1## where R.sup.1 is C.sub.1 -C.sub.4 -alkyl, R.sup.2 is hydrogen, C.sub.1 -C.sub.4 -alkyl or C.sub.1 -C.sub.4 -alkoxy, R.sup.3 is hydrogen or C.sub.1 -C.sub.4 -alkyl, and X is oxygen or sulfur, and methods of combating pests with effective amounts of I.
    Type: Grant
    Filed: September 26, 1988
    Date of Patent: August 8, 1989
    Assignee: BASF Aktiengesellschaft
    Inventors: Wolfgang Seppelt, Linhard Sproesser, Siegfried Kersten, Peter Hofmeister, Christoph Kuenast
  • Patent number: 4755528
    Abstract: Disclosed are 2,3-diamino-1,4-butanedithiol; 4,5-diamino-1,2-dithiane; and their N-acyl and N-alkyl derivatives. Also disclosed are processes for preparing the disclosed compounds; pharmaceutical compositions comprising such compounds; and a method of treatment comprising administering such compounds and compositions when an antihypertensive effect or radioprotective effect is indicated.
    Type: Grant
    Filed: April 17, 1987
    Date of Patent: July 5, 1988
    Assignee: Alcon Laboratories, Inc.
    Inventors: Mark T. DuPriest, Billie M. York, Jr.
  • Patent number: 4745233
    Abstract: Antitumor compounds corresponding to the following formula: ##STR1## in which the substituents R.sub.1 and R.sub.2 may be the same or different and represent hydrogen, an aminocarbonyl group, a C.sub.1 -C.sub.6 alkylaminocarbonyl group, a di-C.sub.1 -C.sub.6 -alkylaminocarbonyl group, the group PO(OH).sub.2, a C.sub.2 -C.sub.8 alkanoyl group, a C.sub.2 -C.sub.8 halogen alkanoyl group or a C.sub.3 -C.sub.8 alkenoyl group, a process for their preparation, and their use in treating oestrogen-receptor-positive-tumors as well as the prostate carcinoma.
    Type: Grant
    Filed: June 9, 1986
    Date of Patent: May 17, 1988
    Assignee: Asta-Werke Aktiengesellschaft
    Inventors: Helmut Schonenberger, Rolf W. Hartmann, Martin Schneider, Walter Schwarz, Jurgen Engel
  • Patent number: 4698362
    Abstract: The present disclosure is concerned with a technique for producing storage stable, non-caking, low viscosity pesticidal concentrates and the compositions so obtained. The technique involves milling a solid biologically active compound in a low viscosity aliphatic petroleum fraction in which it is slightly soluble until it has an average particle size of less than about 10 microns at a temperature in excess of about 40.degree. C. in the presence of a high or ultra-high surface area silica and lecithin. The milling is conducted in such a manner as to avoid melting any significant portion of the biologically active compound undergoing milling. The concentrate so obtained, typically display room temperature viscosities between about 20 and 2,000 cps and contain between about 120 and 480 grams per liter of biologically active compound.
    Type: Grant
    Filed: March 14, 1985
    Date of Patent: October 6, 1987
    Assignee: Mobay Corporation
    Inventor: Jimmie G. Shafer
  • Patent number: 4656163
    Abstract: The present invention relates to the use of the sulphenic acid amides of the general formula (I) ##STR1## in which X represents identical or different halogen atoms,Y.sup.1 and Y.sup.2 are identical or different and represent hydrogen, halogen, alkyl, alkoxy, halogenoalkyl or NO.sub.2 andZ represents halogen, --OH, --NHOH or the group --OR.sup.1,in whichR.sup.1 denotes optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aryl, aralkyl and heterocyclyl, orZ represents the group ##STR2## in which R.sup.2 and R.sup.3 are identical or different and denote hydrogen or a heterocyclic radical, orZ represents the group --OMin which M denotes ammonium or the equivalent of an alkali metal, alkaline earth metal or heavy metal cation, for prolonging the duration of a high activity in agents for combating soil pests.
    Type: Grant
    Filed: November 14, 1985
    Date of Patent: April 7, 1987
    Assignees: Bayer Aktiengesellschaft, Mobay Corporation
    Inventors: John Anderson, Bernhard Homeyer, Engelbert Kuhle, Hans Scheinpflug, Walter M. Zeck, Donald E. Simonet
  • Patent number: 4656188
    Abstract: Angiotensin converting enzyme inhibitors are useful in the treatment of senile macular degeneration.
    Type: Grant
    Filed: October 9, 1985
    Date of Patent: April 7, 1987
    Assignee: Merck & Co., Inc.
    Inventors: Daniel F. Veber, John J. Baldwin
  • Patent number: 4632936
    Abstract: The persistance of bendiocarb and propoxur deposited on both porous and non-porous surfaces is increased by the addition of silica to formulations, in which the insecticides are dissolved in organic solvent.
    Type: Grant
    Filed: June 10, 1985
    Date of Patent: December 30, 1986
    Assignee: FBC Limited
    Inventors: Clive J. Boase, Howard B. Dawson
  • Patent number: 4605667
    Abstract: Pesticidal water-soluble aminoacid sulfenylated carbamates useful as broad spectrum insecticides and miticides, particularly useful as systemic insecticides.
    Type: Grant
    Filed: March 29, 1985
    Date of Patent: August 12, 1986
    Assignee: Union Carbide Corporation
    Inventors: Chennupati K. Rao, Themistocles D. D'Silva
  • Patent number: 4602033
    Abstract: Aryl N-oxalyl-N-methyl-carbamates of the general formula ##STR1## in which X represents an alkoxy, alkenoxy, alkinoxy, aryloxy, alkylthio, alkenylthio, alkinylthio or arylthio radical, each of which may be optionally substituted or represents a radical of the general formula --N R.sup.3 R.sup.4, wherein R.sup.3 and R.sup.4 are identical or different and represent a hydrogen atom or an alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl or aryl radical, each of which may be optionally substituted, or the radicals R.sup.3 and R.sup.4, together with the N atom to which they are bonded, form an optionally substituted heterocyclic ring, andR.sup.1 represents an aryl radical which is optionally substituted,are novel and find use as pesticides, especially for combating insects, acarids and nematodes.
    Type: Grant
    Filed: January 3, 1985
    Date of Patent: July 22, 1986
    Assignee: Bayer Aktiengesellschaft
    Inventors: Gerhard Heywang, Engelbert Kuhle, Wolfgang Behrenz, Ingeborg Hammann, Bernhard Homeyer
  • Patent number: 4584318
    Abstract: A method is described for the control of nematodes in agricultural crops which comprises applying to the situs of infestation of a nematicidal composition containing as active ingredient a compound of the formula ##STR1## wherein Q is hydroxy, carbamoyloxy, or acyloxy, R is alkyl, alkenyl, alkynyl, X is halogen or methyl, n is 1 or 2. Preparation of active ingredient compounds is described, and nematicidal utility of compositions is exemplified.
    Type: Grant
    Filed: June 20, 1983
    Date of Patent: April 22, 1986
    Assignee: FMC Corporation
    Inventors: Clinton J. Peake, Carmine P. DiSanzo, John F. Engel
  • Patent number: 4564630
    Abstract: The invention relates to new carbamyloxybenzhydrol derivatives of the formula (I) ##STR1## wherein R.sub.1 is hydrogen, halogen, trihalomethyl, alkyl having from one to 4 carbon atoms or alkoxy having from one to 4 carbon atoms;R.sub.2 is hydrogen or an R.sub.3 --NH--COO-- group;R.sub.3 is alkyl having from one to 6 carbon atoms, cycloalkyl having up to 7 carbon atoms, or phenyl, optionally substituted with one or more halogen(s).The compounds of the formula (I) show antilipaemic activity and can therefore be used in therapy for treating hyperlipaemia and coronary diseases. Pharmaceutical compositions containing them as active ingredient are also within the scope of the invention.
    Type: Grant
    Filed: December 27, 1983
    Date of Patent: January 14, 1986
    Assignee: Richter Gedeon Vegyeszeti Gyar Rt
    Inventors: Edit Toth, Jozsef Torley, Istvan Hajdu, Sander Gorog, Andrea Maderspach, Gyorgy Hajos, Laszlo Szporny, Andras Javor
  • Patent number: 4543362
    Abstract: p-Alkyl or cycloalkyl phenoxy alkanols and esters are provided having the structure: ##STR1## in which: R.sub.1 is an alkyl group having from one to six carbon atoms, preferably tertiary, and still more preferably tertiary-butyl; or a bivalent cycloalkylene group condensed with the phenyl group at adjacent ring carbons thereof, such as in indane;R.sub.2 is lower alkyl having from one to three carbon atoms or hydrogen;R.sub.3 is hydroxyl or an ester group selected from the group consisting of COOR.sub.4 and OOCR.sub.4 derived from unsubstituted and hydroxy-substituted monocarboxylic acids and COOR.sub.5 OOC and OOCR.sub.
    Type: Grant
    Filed: January 13, 1984
    Date of Patent: September 24, 1985
    Assignee: Frank M. Berger
    Inventors: Frank M. Berger, Joseph I. DeGraw, Jr., Howard L. Johnson
  • Patent number: 4532256
    Abstract: N-Methyl-carbamic acid esters of the formula ##STR1## wherein R.sub.1 is unsubstituted or substituted 2,3-dihydrobenzofuranyl, phenyl, naphthyl or ##STR2## R.sub.2 is hydroxyl, halogen, --OR.sub.1, C.sub.1 -C.sub.10 -alkoxy, C.sub.2 -C.sub.10 -alkenyloxy, C.sub.1 -C.sub.10 -dialkylamino or ##STR3## R.sub.3 is hydrogen, C.sub.1 -C.sub.6 -alkyl or C.sub.2 -C.sub.3 -alkenyl, R.sub.4 is C.sub.1 -C.sub.6 -alkyl, --SR.sub.5, ##STR4## R.sub.5 is C.sub.1 -C.sub.6 -alkyl or C.sub.2 -C.sub.3 -alkenyl, R.sub.6 and R.sub.7 are each hydrogen or C.sub.1 -C.sub.6 -alkyl, andn is zero or 1.A process for producing these compounds and their use for combating pests are described.
    Type: Grant
    Filed: December 12, 1983
    Date of Patent: July 30, 1985
    Assignee: Ciba-Geigy Corporation
    Inventor: Jozef Drabek
  • Patent number: 4511579
    Abstract: Substituted aryl alkylcarbamates have been found to provide outstanding pest repellancy when applied to desirable foliage or agronomic crops.
    Type: Grant
    Filed: November 8, 1983
    Date of Patent: April 16, 1985
    Assignee: Union Carbide Corporation
    Inventors: George L. Rotramel, Daniel P. Veilleux, Joseph L. Allen