Four Or More Ring Nitrogens In The Tricyclo Ring System Patents (Class 544/251)
  • Patent number: 4091094
    Abstract: The novel compound 9-azariboflavin is prepared. This compound has anticoccidial, antiprotozoal and antiparasitic activity. It is particularly useful for controlling cecal and/or intestinal coccidiosis when administered in minor quantities to animals, in particular to poultry, usually in admixture with animal sustenance.
    Type: Grant
    Filed: August 23, 1976
    Date of Patent: May 23, 1978
    Assignee: Merck & Co., Inc.
    Inventors: Donald W. Graham, Edward F. Rogers
  • Patent number: 4087423
    Abstract: New pyrazolo[4,3-e][1,2,4]triazolo[4,3-c]pyrimidines have the general formula ##STR1## They are useful as antiinflammatory agents.
    Type: Grant
    Filed: July 20, 1977
    Date of Patent: May 2, 1978
    Assignee: E. R. Squibb & Sons, Inc.
    Inventors: Uwe D. Treuner, Hermann Breuer
  • Patent number: 4087422
    Abstract: Dihydrotetrazolo [1,5-a] quinazolines having the formula: ##STR1## wherein (a) n is 0, X is oxygen, and R is optionally unsubstituted alkyl, alkenyl of at least 4 carbon atoms, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, amino or substituted aryl; or (b) n is 1 or 2, X is oxygen, R is hydrogen, or optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy or (c) n is 0, 1 or 2, X is sulphur, R is hydrogen, or optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy; or (d) n is 0, 1 or 2, X is NR.sub.2 where R.sub.2 is hydrogen, alkyl having 1 to 10 carbon atoms, benzyl or hydroxyalkyl, R is optionally-substituted alkyl, alkenyl, alkynyl, aryl, aralkyl, alkylthio, cycloalkyl, or amino, and R.sup.1 is hydroxy, halogen, nitro, alkyl or alkoxy; and salts thereof. These compounds demonstrate pesticidal activity.
    Type: Grant
    Filed: June 13, 1977
    Date of Patent: May 2, 1978
    Assignee: Imperial Chemical Industries Limited
    Inventors: Raymond Alexander Bowie, John Michael Cox, Gordon Michael Farrell, Margaret Claire Shephard