Abstract: Substituted [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3 dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having antimicrobial properties and being particularly useful in the treatment of vaginal candidosis.

Abstract: Herbicidally active novel N,N'-bis-sulphonyl guanidines of the formula ##STR1## in which M is hydrogen, a metal or an ammonium radical, andR.sup.4, R.sup.5, R.sup.40 and R.sup.41 are various organic radicals.

Abstract: Sulfonamides such as N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1,3-dihydro-6-methyl-3-oxof uro[3,4-c]pyridine-4-sulfonamide are useful as herbicides and plant growth regulants.

Abstract: Thiophenesulfonamides such as N-[(4,6-dimethylpyrimidin-2-yl)aminocarbonyl]-3-(isoxazol-3-yl)-2-thiophen esulfonamide are useful as herbicides and plant growth regulants.

Abstract: A process for the preparation of a 5-acylpyrimidine of the formula ##STR1## in which R is an organic radical comprising reacting a methyl ketone of the formulaR--CO--CH.sub.3in a first stage with a formylating reagent in the presence of a base to form an enolketone of the formulaR--CO--CH.dbd.CH--OR.sup.10in which R.sup.10 represents hydrogen or a base radical, thereafter reacting the enolketone in 2nd and 3rd stages with formamidine or a formamidine salt, and with an amino-formylating agent, and, in a 4th stage heating to cyclize the compound formed.The end products, some of which are new, are intermediates for making herbicides.

Abstract: Cardiovascular activity is exhibited by compounds having the formula ##STR1## and pharmaceutically acceptable salts thereof, wherein R.sub.1 is alkyl, cycloalkyl, aryl, heterocyclo, --(CH.sub.2).sub.n --Y.sub.2, --(CH.sub.2).sub.p --Y.sub.3 or halo substituted alkyl;R.sub.2 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, aryl, --(CH.sub.2).sub.n --Y.sub.1, or halo substituted alkyl;R.sub.3 is hydrogen, alkyl, cycloalkyl, aryl, heterocyclo, --(CH.sub.2).sub.n --Y.sub.2, --(CH.sub.2).sub.p --Y.sub.3, or halo substituted alkyl;R.sub.4 is aryl or heterocyclo;R.sub.5 is hydrogen, alkyl, aryl, arylalkyl, cyano, nitro, ##STR2## Y.sub.1 is cycloalkyl, aryl, heterocyclo, hydroxyl, alkoxy, aryl-(CH.sub.2).sub.m --O--, mercapto, alkylthio, aryl-(CH.sub.2).sub.m --S--, amino, substituted amino, carbamoyl, ##STR3## Y.sub.2 is cycloalkyl, aryl, heterocyclo, carbamoyl, ##STR4## amino, or substituted amino; m is 0 or an integer of 1 to 6;n is an integer of 1 to 6; andp is an integer of 2 to 6.

Abstract: A biologically active compound can be solubilized by reaction in different sequences to form a derivative carrying the active moiety, a linking group such as an optionally substituted diisocyanate radical, a polyether moiety such as a polyoxyethylene radical, and a terminal group such as a butyl radical, e.g. ##STR1## n=1 to 400. The active materials can be agricultural chemicals, pharmaceuticals, and the like.

Abstract: Cardiovascular activity is exhibited by compounds having the formula ##STR1## and pharmaceutically acceptable salts thereof wherein X is oxygen or sulfur;R.sub.1 is alkyl, cycloalkyl, aryl, heterocyclo, --(CH.sub.2).sub.n --Y.sub.1, or halo substituted alkyl;R.sub.2 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, aryl, --(CH.sub.2).sub.n --Y.sub.1, or halo substituted alkyl;R.sub.3 is hydrogen, alkyl, cycloalkyl, aryl, heterocyclo, --(CH.sub.2).sub.n --Y.sub.2, --(CH.sub.2).sub.p --Y.sub.3, or halo substituted alkyl;R.sub.4 is aryl or heterocyclo;Y.sub.1 is cycloalkyl, aryl, heterocyclo, hydroxyl, alkoxy, aryl--(CH.sub.2).sub.m --O--, mercapto, alkylthio, aryl--(CH.sub.2).sub.m --S--, amino, substituted amino, carbamoyl, ##STR2## Y.sub.2 is cycloalkyl, aryl, heterocyclo, carbamoyl, ##STR3## Y.sub.3 is hydroxyl, alkoxy, aryl--(CH.sub.2).sub.m --O--, mercapto, alkylthio, aryl--(CH.sub.2).sub.

Abstract: A guanidine derivative of the formula I: ##STR1## in which R.sup.1, R.sup.2, R.sup.3, R.sup.4, ring X and D are a variety of radicals defined in the specification and A is a 3-8C alkylene chain which is substituted by a hydroxy radical and into which is optionally inserted, as part of the backbone of the chain, one or two groups selected from oxygen and sulphur atoms and NH and 1-6C N-alkyl radicals; and the pharmaceutically-acceptable acid additions salts thereof. Pharmaceutical compositions and methods of manufacture are also described. The compound of the formula I is a histamine H-2 antagonist and is therefore useful in ulcer therapy.

Abstract: Novel pyridinesulfonamide compounds containing ortho-heterocyclic substituents such as N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-2-(1H-1,2,4-triazol-1-yl)-3 -pyridinesulfonamide display utility as herbicides and plant growth regulants.

Abstract: Tetrahydropyridazinones of the formula I ##STR1## wherein R denotes an optionally substituted carbocyclic or heterocyclic radical, R.sup.1 denotes hydrogen; alkyl; aralkyl, which is optionally substituted in the aryl part; or acyl, and R.sup.2 denotes hydrogen; alkyl, which can optionally be substituted; or optionally substituted phenyl; and their acid addition compounds, if these can be prepared.The tetrahydropyridazinone derivatives of the formula I according to the invention and their physiologically acceptable salts exhibit useful pharmacological actions.

Abstract: This invention relates to new tetrahydropyrimidines, to a process for their production and to their use as catalysts in the production of polyurethane plastics, including polyurethane foams.

Abstract: Herbicidal compounds of the formula: ##STR1## wherein A represents R.sup.1 R.sup.2 N-- (wherein R.sup.1 represents C.sub.1-8 alkyl or C.sub.2-8 alkenyl or alkynyl unsubstituted or substituted by CN, OH, C.sub.1-6 alkoxy, carboxy, C.sub.2-9 alkoxycarbonyl, aminocarbonyl optionally substituted by C.sub.1-8 alkyl or C.sub.2-8 alkenyl, C.sub.1-8 alkoxyaminocarbonyl, C.sub.1-8 alkanesulphonamidocarbonyl, --C(.dbd.O)Het, where Het represents a nitrogen-containing heterocyclic group, or one or more halogen atoms or R.sup.1 represents C.sub.3-6 cycloalkyl optionally substituted by C.sub.1-4 alkyl and R.sup.2 represents H or R.sup.1, or R.sup.1 represents C.sub.1-4 alkylthio and R.sup.2 represents H, or A represents R.sup.p (R.sup.q)--C.dbd.N-- (wherein R.sup.p represents C.sub.1-4 alkoxy or amino substituted by one or two C.sub.1-4 alkyl groups and R.sup.q represents H or C.sub.1-4 alkyl) or A represents 2-oxo-azetidin-1-yl, 2-oxo-pyrrolidin-1-yl or 2-oxo-piperidin-1-yl optionally substituted by C.sub.

Abstract: The invention relates to novel N-phenyl-1,3,5-oxadiazine-2,4-diones of formula I ##STR1## wherein R.sub.1 is fluorine or chlorine andR.sub.2 is hydrogen, fluorine or chlorine,to the preparation thereof, to the use thereof in pest control and to pesticidal compositions which contain said oxadiazines. The preferred field of application is the control of pests of animals and plants.

Abstract: Disclosed herein are a derivative of tetrahydrobenzothiazole represented by the formula (I): ##STR1## wherein R represents a hydrogen atom, a hydroxyl group or a lower acyloxy group such as acetoxy group and propionyloxy group and X represents a methylene group, C.sub.1 to C.sub.4 -alkylamino group, benzylamino group or --O--, and a herbicidal composition containing the same as an active ingredient.

Abstract: This invention relates to a novel class of sulfonamides and their use as herbicides and plant growth regulants.

Abstract: There are disclosed novel 1,3,5-oxadiazine-2,4-diones of the formula I ##STR1## wherein R.sub.1 is halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -alkylthio,R.sub.2 is hydrogen, halogen, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy or C.sub.1 -C.sub.4 -alkylthio,R.sub.3 and R.sub.4 are each hydrogen, halogen or C.sub.1 -C.sub.4 -alkyl,R.sub.5 is hydrogen, halogen, C.sub.1 -C.sub.4 -alkyl or --COOR.sub.8,R.sub.6 is hydrogen or halogen,R.sub.7 is mono- or polyhalogenated C.sub.1 -C.sub.4 -alkyl,R.sub.8 is hydrogen or C.sub.1 -C.sub.4 -alkyl, andm is 1 or 2,the production thereof, their use for controlling pests, and pesticidal compositions containing these oxadiazines as active ingredients. The preferred field of application is the control of pests on animals and plants.

Abstract: This invention relates to new salts of 1,3,5-oxadiazines-2,4,6-triones, to new 1,3,5-oxadiazines-2,4,6-triones and to the preparation thereof.

Abstract: Disclosed is a primer composition which contains an isocyanate compound having one or more 1,3,5-oxadiazine-2,4,6-trione rings as an adhesion promoter, which is useful as a primer for bonding polyester plastics to the same or different substrates using an adhesive such as polyurethane, epoxy and polyolefin adhesives. When the surface of polyester plastics is treated with said primer prior to application of the adhesive, the bonding achieved is excellent in adhesion.

Abstract: Hexahydrotriazinones substituted by a 5-substituted-1,2-oxazol-3-yl moiety, useful for controlling the growth of unwanted plants.

Abstract: An oxidiazine derivative of the formula ##STR1## in which R.sup.1 represents halogen or alkyl,R.sup.2 represents hydrogen or halogen,R.sup.3, R.sup.5 and R.sup.6 are selected independently of one another and each represent hydrogen, halogen, alkyl or halogenoalkyl andR.sup.4 represents halogenoalkyl, halogenoalkoxy, halogenoalkylthio or tert.-alkyl, or R.sup.4, together with R.sup.3, represents dioxahalogenoalkanediyl or, in the case where at least one of the radicals R.sup.3, R.sup.5 and R.sup.6 represents halogenoalkyl, R.sup.4 may alternatively represent hydrogen or halogen, or in the case where R.sup.1 represents chlorine and at the same time R.sup.2 represents fluorine, R.sup.4 may alternatively represent halogen or alkoxy,which possesses arthropodicidal and nematicidal properties.

Abstract: Diphenyloxadiazinediones of the formula (I) ##STR1## where R.sub.1 is CH.sub.3, F, Cl or Br, R.sup.2 is H, F or Cl and R.sup.3 to R.sup.8 are H, F, Cl, Br, CH.sub.3, CF.sub.3, --OCF.sub.3, --OCHF.sub.2, OCF.sub.2 CHClF, --OCH.sub.3 or --OC.sub.2 H.sub.5, their preparation and their use, especially as insecticides and acaricides.

Abstract: Disclosed is a one-can type pressure-sensitive adhesive composition which contains a polyurethane polyol obtained by the reaction of an isocyanate component having oxadiazine-2,4,6-trione ring, other organic diisocyanate and a polyol component having a molecular weight of 400 to 50,000 at a specific proportion. This composition has an excellent heat resistance, stable pressure-sensitive adhesion, holding power and tackiness.

Abstract: Polyisocyanates having oxadiazinetrione rings obtained by reacting bis(isocyanatomethyl)cyclohexane, an oligomer thereof, an adduct thereof or a mixture of them with carbon dioxide. Said polyisocyanates have excellent properties as raw materials for the production of polyurethanes, because of their higher reactivity at lower temperature and better storage stability.

Abstract: This invention relates to novel compounds of the formula ##STR1## wherein R.sup.1 is lower alkenyl or lower alkynyl; R.sup.2 is lower alkenyl, lower alkynyl or cycloalkyl; R.sup.3 is hydrogen; R.sup.4 is alkyl, cycloalkyl or lower alkoxycarbonylalkyl or R.sup.2 and R.sup.3 are joined to form dimethyleneoxy (i.e. --CH.sub.2 OCH.sub.2 --) or R.sup.3 and R.sup.4 taken together with the nitrogen to which they are attached, form a 5- to 6- membered heterocyclic ring, compositions containing said compounds and a method of employing said compounds as arthropod repellents.

Abstract: A process for the preparation of a 1-amino-1,3,5-triazine-2,4(1H, 3H)-dione compounds comprising the steps of reacting an N-substituted imido-dicarboxylic acid diaryl ester with an isothiosemicarbazone at a temperature of between 50.degree. and 150.degree. C. to form a 1-alkylidene-amino-1,3,5-triazine-2,4(1H, 3H)-dione reaction product; and thereafter, hydrolyzing the reaction product in an acid medium. The reaction product need not be separated from the reaction mixture before the hydrolysis step. Certain novel 1-amino-1,3,5-triazine-2,4(1H, 3H)-dione compounds are provided. The compounds are useful as herbicides.

Abstract: An oxidiazine derivative of the formula ##STR1## in which R.sup.1 represents halogen or alkyl,R.sup.2 represents hydrogen or halogen,R.sup.3, R.sup.5 and R.sup.6 are selected independently of one another and each represent hydrogen, halogen, alkyl or halogenoalkyl andR.sup.4 represents halogenoalkyl, halogenoalkoxy, halogenoalkylthio or tert.-alkyl, or R.sup.4, together with R.sup.3, represents dioxahalogenoalkanediyl or, in the case where at least one of the radicals R.sup.3, R.sup.5 and R.sup.6 represents halogenoalkyl, R.sup.4 may alternatively represent hydrogen or halogen, or in the case where R.sup.1 represents chlorine and at the same time R.sup.2 represents fluorine, R.sup.4 may alternatively represent halogen or alkoxy,which possesses arthropodicidal and nematicidal properties.

Abstract: Alkylated glyoxal/cyclic urea condensates are excellent formaldehyde-free crosslinking resins for textile fabrics.

Abstract: Disclosed are new compounds of the formula ##STR1## Wherein R.sup.1 is selected from the group consisting hydrogen and alkyl; Z is selected from the group consisting of --CHR.sup.2 --, oxygen, sulfur and --NR.sup.3 --; R.sup.2 and R.sup.3 are selected from the group consisting of hydrogen and alkyl; A,C, and E are each independently selected from the group consisting of C1-C10 alkyl and hydrogen; B,D and F are each independently selected from the group consisting of C1-C10 alkyl, C3-C10 alkenyl, C4-C10 alkynyl, cycloalkyl, alkoxy, alkylthio, amino, cyano and hydrogen.These compounds are useful as herbicides.

Abstract: Alkylated glyoxal/cyclic urea condensates are excellent formaldehyde-free crosslinking resins for textile fabrics.

Abstract: Alkylated glyoxal/cyclic urea condensates are excellent formaldehyde-free crosslinking resins for textile fabrics.

Abstract: N.sup.2 -naphthalenesulfonyl-L-argininamides and the pharmaceutically acceptable salts thereof have been found to be effective as pharmaceutical agents for the inhibition and suppression of thrombosis.

Abstract: Insectically active oxadiazindione derivatives of the formula: ##STR1## wherein R.sup.1 is 2-chlorophenyl, 4-chlorophenyl, 2,6-dichlorophenyl, 3,5-dichlorophenyl, 2,6-difluorophenyl, 3-nitrophenyl, 3-trifluoromethylphenyl, 2-tolyl or 3,5-xylyl, and R.sup.2 is phenyl or phenyl substituted by methyl, methoxy, chlorine, fluorine, or nitro, provided that at least one of R.sup.1 and R.sup.2 is a chloro-or fluoro-substituted phenyl group.

Abstract: N.sup.2 -naphthalenesulfonyl-L-arginine esters and amides and the pharmaceutically acceptable acid addition salts thereof which have antithrombotic properties.

Abstract: N.sup.2 -substituted-L-arginine esters and amides, and the pharmaceutically acceptable acid addition salts thereof have been found to be effective as pharmaceutical agents for the inhibition and suppression of thrombosis.

Abstract: A novel catalyst system is described that is useful in the trimerization of organic isocyanates. The system comprises (1) N,N',N"-trisdialkylaminoalkyl-s-hexahydrotriazine and (2) a compound selected from the group consisting of 3,5-bis(N,N-dialkylaminoalkyl)-1,3,5-tetrahydrooxadiazine, 5-(N,N-dialkylaminoalkyl)-1,3,5-dihydrodioxazine and the mixtures thereof.

Abstract: Novel 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas, active as insecticides, and methods for their use as insecticides.

Abstract: New diazine derivatives corresponding to the formula ##STR1## wherein R.sub.1 denotes a heterocyclic-aromatic radical which is optionally substituted by halogen, lower alkyl, aryl, nitro, cyano, trifluoromethyl, carboxyl, R.sub.3 OOC--, (R.sub.3).sub.2 NCO--, (R.sub.3).sub.2 N--, R.sub.3 O--, R.sub.3 SO.sub.2 --, R.sub.3 SO-- or R.sub.3 S--, and R.sub.2 and R.sub.3 independently of one another denote lower alkyl, alkoxyalkyl, alkenyl or cycloalkyl which is optionally bonded via an alkylene bridge, processes for the production of the new compounds, compositions containing these compounds and a process for combating Coccidia.

Abstract: Novel ureidoalkylphosphonates, methods for their preparation as well as for their use in preparing durable, flameproof finishes for textiles are disclosed. These ureidoalkylphosphonates are found to be low in cost, readily prepared and of minimal toxicity.