Nitrogen Attached Directly To The Hetero Ring By Nonionic Bonding Patents (Class 549/68)
  • Patent number: 4240820
    Abstract: Novel method for regulating the growth of plants which method comprises applying to the plants or their habitat, effective amounts of heterocyclic compound of the formula ##STR1## in which R.sup.1 is alkyl or optionally substituted aryl,R.sup.2 is hydrogen, alkyl or optionally substituted aryl,R.sup.3 is hydrogen or the radical ##STR2## in which Y is oxygen or sulfur andR.sup.5 is alkyl, haloalkyl, alkoxyalkyl, aryloxyalkyl, which is optionally substituted in the aryloxy part, alkoxy, optionally substituted aryl, optionally substituted aryloxy, monoalkylamino, dialkylamino, alkenylamino, dialkenylamino, optionally substituted arylamino, a 5-membered to 7-membered heterocyclic ring, bonded via nitrogen, or the radical ##STR3## in which R.sup.6 is hydrogen or alkyl andR.sup.7 is hydrogen or alkyl, orR.sup.6 and R.sup.7, together with the adjacent nitrogen atom, are a 5-membered to 7-membered heterocyclic ring,R.sup.4 is cyano or the grouping --COR.sup.8in whichR.sup.
    Type: Grant
    Filed: April 13, 1979
    Date of Patent: December 23, 1980
    Assignee: Bayer Aktiengesellschaft
    Inventors: Karlfried Dickore, Klaus Lurssen
  • Patent number: 4234580
    Abstract: Carbamate thiosulfenylcarbamoyl fluoride compounds are insecticidal and miticidal compounds and are also useful intermediates in the preparation of pesticidally active bis-carbamate disulfide compounds.
    Type: Grant
    Filed: March 28, 1977
    Date of Patent: November 18, 1980
    Assignee: Union Carbide Corporation
    Inventor: Themistocles D. J. D'Silva
  • Patent number: 4232035
    Abstract: Novel N-dithioalkyl and N-dithioaryl substituted cyclic carbamoyloximes exhibit exceptional pesticidal activity.
    Type: Grant
    Filed: December 30, 1975
    Date of Patent: November 4, 1980
    Assignee: Union Carbide Corporation
    Inventor: Themistocles D. J. D'Silva
  • Patent number: 4230872
    Abstract: Novel 9-substituted or unsubstituted thienyl-3,7-dimethyl-nona-2,4,6,8-tetraene derivatives, useful as antitumor agents as well as processes for their preparation and novel intermediates are disclosed.
    Type: Grant
    Filed: May 11, 1978
    Date of Patent: October 28, 1980
    Assignee: Hoffmann-La Roche Inc.
    Inventors: Michael J. Klaus, Beverly A. Pawson
  • Patent number: 4230707
    Abstract: Oxo-pyrido[1,2-a]thienopyrimidine compounds, salts thereof, methods of production, intermediates in their production, pharmaceutical compositions containing said compounds and methods for treating allergies using said compositions are disclosed.
    Type: Grant
    Filed: August 27, 1979
    Date of Patent: October 28, 1980
    Assignee: Warner-Lambert Company
    Inventors: Francis J. Tinney, David T. Connor, Wiaczeslaw A. Cetenko, Joseph J. Kerbleski, Roderick J. Sorenson
  • Patent number: 4220793
    Abstract: A process for preparing 5-nitro-2-thenoic acid by oxidation of the corresponding aldehyde is described.
    Type: Grant
    Filed: November 14, 1978
    Date of Patent: September 2, 1980
    Assignee: Labaz
    Inventors: Yves Bazile, Paul de Cointet de Fillain, Charles Pigerol
  • Patent number: 4211696
    Abstract: Disperse monoazo dyestuffs, free from carboxylic and sulphonic acid groups, derived from 3,5-dinitro-2-amino thiophene as disazo component and an arylamine coupling component exhibit superior properties when used to give colorations to textile materials such as secondary cellulose acetate and cellulose triacetate, polyamide and aromatic polyester textile materials, said colorations having excellent fastness to light and to wet and dry heat treatments. The dyestuffs also have high tinctorial strength and excellent dyeing and build-up properties and produce depths of shade which are relatively independent of the dyebath pH, or the temperature of the dyebath or the liquor ratio of the dyebath.
    Type: Grant
    Filed: February 9, 1976
    Date of Patent: July 8, 1980
    Assignee: Imperial Chemical Industries Limited
    Inventors: David B. Baird, Alan T. Costello, Brian R. Fishwick, Robert D. McClelland, Peter Smith
  • Patent number: 4199588
    Abstract: Compounds of the formula ##STR1## wherein R.sub.1 is hydrogen, chlorine, bromine or alkyl of 1 to 4 carbon atoms;R.sub.2 is hydrogen, fluorine, chlorine, bromine, nitro or trifluoromethyl; andR.sub.3 is chlorine, bromine, alkoxy of 1 to 3 carbon atoms, alkylmercapto of 1 to 3 carbon atoms, cycloalkyl of 3 to 6 carbon atoms, cycloalkenyl of 3 to 6 carbon atoms, or a saturated or unsaturated 5- to 6-membered heterocycle comprising an oxygen, sulfur or nitrogen heteroatom, where a substitutable nitrogen heteroatom may optionally have a lower akyl substituent attached thereto;and non-toxic, pharmacologically acceptable acid addition salts thereof; the compounds as well as their salts are useful as tranquilizers, muscle-relaxants and anticonvulsants.
    Type: Grant
    Filed: November 30, 1977
    Date of Patent: April 22, 1980
    Assignee: Boehringer Ingelheim GmbH
    Inventors: Karl-Heinz Weber, Adolf Bauer, Peter Danneberg, Franz J. Kuhn
  • Patent number: 4198350
    Abstract: This invention relates to the intramolecular oxidation and reduction of aromatic hydrocarbons containing at least one methyl group and a nitro group ortho to the methyl group. Further, it relates to preparing methyl o-amino arylcarboxylates and aromatic amines. The process comprises reacting aromatic hydrocarbons having at least one methyl group and a nitro group ortho to the methyl group in a solvent at a temperature of about 450.degree. to 750.degree. C. When the solvent is methanol, methyl o-amino arylcarboxylates useful in anesthetics, printing inks for polyethylene, and useful in the manufacture of azo dyes are produced. Novel substituted methyl anthranilates have been produced which have the foregoing uses. When no solvent is used or the solvent is benzene, cyclohexane, toluene, hexafluorobenzene or any other non-reactive solvent, the compounds are demethylated and aromatic amines are produced.
    Type: Grant
    Filed: February 12, 1976
    Date of Patent: April 15, 1980
    Assignee: Standard Oil Company (Indiana)
    Inventor: Ellis K. Fields
  • Patent number: 4182892
    Abstract: A compound of the formula I: ##STR1## wherein: R is substituted or unsubstituted C.sub.1-6 alkyl, a substituted or unsubstituted aromatic ring, a heterocyclic ring, a cycloalkyl group or a fused ring system,R.sup.1 is hydrogen, lower alkyl, cycloaliphatic or heterocyclic ring, andX is a halogen atom.
    Type: Grant
    Filed: February 24, 1978
    Date of Patent: January 8, 1980
    Assignee: Chinoin Gyogyszer es Vegyeszeti Termekek Gyara Rt
    Inventors: Magda Huhn, Eva Somfai, Gabor Szabo, Gabor Resofszki, Livia Gneth nee Zalantai
  • Patent number: 4181806
    Abstract: Aminoalkylenephosphonic acids and their alkali metal salts prepared by a reaction utilizing a primary or secondary tetrahydrothiophenamine 1,1-dioxide or the hydrochloride thereof, an aldehyde or a ketone, and orthophosphorous acid are useful in the control of scale and sludge deposition in aqueous systems. When used in combination with known corrosion inhibitors they show synergistic results in inhibiting corrosion of metal surfaces in contact with an aqueous system that is normally corrosive to such metals.
    Type: Grant
    Filed: June 9, 1978
    Date of Patent: January 1, 1980
    Assignee: Buckman Laboratories, Inc.
    Inventors: Joseph G. E. Fenyes, John D. Pera
  • Patent number: 4179514
    Abstract: Ketoalkanesulfenyl and ketoalkanethiosulfenyl carbamates exhibit exceptional pesticidal activity.
    Type: Grant
    Filed: January 6, 1978
    Date of Patent: December 18, 1979
    Assignee: Union Carbide Corporation
    Inventor: Themistocles D. J. D'Silva
  • Patent number: 4169894
    Abstract: Unsymmetrical N-substituted bis-carbamoyloxy disulfide compounds exhibit outstanding nematocidal, miticidal and insecticidal activity, coupled with substantially reduced mammalian toxicity and phytotoxicity as compared to known pesticidal compounds having a comparable spectrum of activity against insect, arachnid and nematode pests.
    Type: Grant
    Filed: March 28, 1977
    Date of Patent: October 2, 1979
    Assignee: Union Carbide Corporation
    Inventor: Themistocles D. J. D'Silva