The Polycyclo Ring System Contains At Least Four Cyclos Patents (Class 552/220)
  • Patent number: 8119804
    Abstract: An organic semiconducting layer formulation containing an organic binder which has a permittivity, ?, at 1,000 Hz of 3.3 or less and a polyacene compound of Formula A: and processes for the preparation thereof and uses thereof in various electronic devices.
    Type: Grant
    Filed: March 8, 2010
    Date of Patent: February 21, 2012
    Assignee: Merck Patent GmbH
    Inventors: Beverley Anne Brown, Janos Veres, Remi Manouk Anemian, Richard Williams, Simon Dominic Ogier, Stephen William Leeming
  • Publication number: 20120012822
    Abstract: An aromatic compound represented by the following formula (1). [In the formula, ring A and ring B each represent a benzene ring, an aromatic fused ring composed of 2-4 rings, a heteroaromatic ring or a heterocyclic aromatic fused ring composed of 2-4 rings, R1a represents a group —CHR2a—CHR2bR2c, and R1b, R1c and R1d each represent hydrogen, aryl or a group —CHR2d—CHR2eR2f. This is with the proviso that at least 2 of R1b, R1c and R1d are not hydrogen. R2a, R2b and R2c each represent hydrogen, alkyl, aryl or a substituted silyl group, and R2a and R2b may be bonded together to form a ring. R2d, R2e and R2f each represent hydrogen, alkyl, aryl or a substituted silyl group, and R2d and R2e may be bonded together to form a ring.
    Type: Application
    Filed: January 22, 2010
    Publication date: January 19, 2012
    Applicants: KEIO UNIVERSITY, SUMITOMO CHEMICAL COMPANY, LIMITED
    Inventors: Fumitoshi Kakiuchi, Hiroki Terai
  • Patent number: 8071575
    Abstract: Bone targeted compounds and methods are provided. Compounds can include a Bone Targeting Portion (RT), having an affinity for bone; a Bone Active Portion (RA) for interacting with and affecting bone; and a Linking Portion (RL) connecting the Bone Targeting Portion and the Bone Active Portion.
    Type: Grant
    Filed: February 22, 2008
    Date of Patent: December 6, 2011
    Assignee: University of Louisville Research Foundation
    Inventors: William M. Pierce, Jr., K. Grant Taylor, Leonard C. Waite
  • Patent number: 7576208
    Abstract: A compound of formula 9 and uses thereof in various electronic devices and in a formulation for ink jet printing and in an organic semiconducting layer formulation.
    Type: Grant
    Filed: July 9, 2007
    Date of Patent: August 18, 2009
    Assignee: Merck Patent GmbH
    Inventors: Beverley Anne Brown, Janos Veres, Remi Manouk Anemian, Richard Williams, Simon Dominic Ogier, Stephen William Leeming
  • Publication number: 20080061287
    Abstract: The present invention provides an organic semiconductor material which exhibits a high mobility, and excellent solubility in solvents and oxidation resistance. The present invention also provides an organic semiconductor thin film exhibiting a high mobility, and an organic semiconductor device exhibiting excellent electronic characteristics. A transistor structure is formed by coating the silicon substrate with a thin film of pentacene compound substituted halogens at 6 and 13 positions and aliphatic hydrocarbons at 2, 3, 9 and 10 positions, wherein the substrate is patterned beforehand with gold to have a source and drain electrodes.
    Type: Application
    Filed: February 25, 2005
    Publication date: March 13, 2008
    Inventors: Kazuto Nagata, Yoshinori Naruta, Masatoshi Yakiyama
  • Patent number: 6747163
    Abstract: The invention provides a process for the preparation and isolation of compound of formula 2, comprising the following steps: oxidizing Flumethasone dissolved in a tetrahydrofuran-water mixture with periodic acid at a temperature lower than 30° C.; cooling the reaction mixture to a temperature lower than 10° C.; adding an antisolvent precooled to a temperature lower than 10° C.; and separating the precipitated crystal by filtration, whereby there is obtained a compound of formula 2 in a yield of at least 98% and of a chromatographic purity of at least 99%.
    Type: Grant
    Filed: April 4, 2003
    Date of Patent: June 8, 2004
    Assignee: Chemagis Ltd.
    Inventors: Yaacov Rubinsztain, Ariana Segal, Joseph Kaspi, Ori Lerman
  • Patent number: 5587495
    Abstract: 4-substituted anthracyclinones of formula (I): ##STR1## wherein R represents a straight or branched alkyl, alkenyl or alkynyl group of up to 16 carbon atoms optionally substituted by (a) an aryl group which is unsubstituted or substituted by an inert group such as an alkyl, alkoxy or nitro group; (b) an alkoxy group; (c) a trialkylsilyl group, (d) an ester group or (e) an amido group, are intermediates in the preparation of antitumor anthracycline glycosides of formula (IX): ##STR2## wherein R is as defined above and R.sub.1 is a hydrogen atom or a hydroxy group, and pharmaceutically acceptable salts thereof.
    Type: Grant
    Filed: April 25, 1991
    Date of Patent: December 24, 1996
    Assignee: Farmitalia Carlo Erba Srl
    Inventors: Walter Cabri, Silvia De Bernardinis, Franco Francalanci, Sergio Penco
  • Patent number: 5405979
    Abstract: A process for the production of 10.beta.-H-11.beta.-(substituted phenyl) steroids of the formulae Ia or Ib set forth in the claims by reduction of a compound of the formula III: ##STR1## followed by cleaving with a strong acid or partial cleaving with a less strong acid. Reduction with an electropositive metal in an electron-solvating solvent is preferred.
    Type: Grant
    Filed: November 30, 1992
    Date of Patent: April 11, 1995
    Assignee: Schering Aktiengesellschaft
    Inventors: Eckhard Ottow, Gunter Neef, Arwed Cleve, Rudolf Wiechert
  • Patent number: 5274141
    Abstract: Quinone- and hydroquinone-containing cyclic enediyneols and enediyneones having 10-carbon atoms in the enediyne-containing ring that cleave DNA are disclosed, as are methods of making and using the same.
    Type: Grant
    Filed: September 1, 1992
    Date of Patent: December 28, 1993
    Assignee: The Scripps Research Institute
    Inventors: Kyriacos C. Nicolaou, Aijun Liu
  • Patent number: 5187195
    Abstract: Anthraquinone compounds of the formula: ##STR1## wherein: R.sup.1 is hydrogen, hydroxy or acyloxy,R.sup.2 is hydrogen or acyl,R.sup.3 is acyl,R.sup.4 is hydrogen or acyl,R.sup.5 is hydrogen or acyl,R.sup.6 is hydrogen or acyl, andR.sup.7 is hydrogen or acylhave been found to possess endothelin antagonistic properties and are producible by various synthetic and fermentation processes.
    Type: Grant
    Filed: June 26, 1990
    Date of Patent: February 16, 1993
    Assignee: Fujisawa Pharmaceutical Co., Ltd.
    Inventors: Nobutaka Oohata, Motoaki Nishikawa, Sumio Kiyoto, Shigehiro Takase, Keiji Hemmi, Hidetsugu Murai, Masakuni Okuhara
  • Patent number: 5162545
    Abstract: Malonic acid dyes capable of forming polycondensation products have the formula ##STR1## where R.sup.1 and R.sup.2 are each independently of the other hydroxyl, C.sub.1 -C.sub.6 -alkoxy, chlorine or bromine,R.sup.3 is hydrogen or C.sub.1 -C.sub.6 -alkyl,A is C.sub.1 -C.sub.20 -alkylene which may be interrupted by oxygen atoms or by imino or C.sub.1 -C.sub.4 -alkylimino groups, andChr is the radical of a chromophore derived from an anthraquinone, perylene, disazo or trisazo dye or else, when R.sup.3 is C.sub.1 -C.sub.6 -alkyl, from a monoazo dye.
    Type: Grant
    Filed: October 12, 1990
    Date of Patent: November 10, 1992
    Assignee: BASF Aktiengesellschaft
    Inventors: Karl-Heinz Etzbach, Karin H. Beck, Gerhard Wagenblast
  • Patent number: 5110960
    Abstract: Novel antibiotic herein designated as BU-3608, BU-3608 B, and BU-3608 C are produced by fermentation of Actinomadura hibisca Strain No. P157-2, ATCC 53557, and Strain No. Q278-4, ATCC 53646. The antibiotics possess antifungal and antiviral activities.
    Type: Grant
    Filed: October 1, 1990
    Date of Patent: May 5, 1992
    Assignee: Bristol-Myers Company
    Inventors: Toshikazu Oki, Kyoichiro Saitoh, Kozo Tomatsu, Koji Tomita, Masataka Konishi, Takeo Miyaki, Mitsuaki Tsunakawa, Maki Nishio
  • Patent number: 5091418
    Abstract: The present invention relates to a novel .alpha.-glucosidase inhibitor, pradimicin Q, having the following formula ##STR1## and its pharmaceutically acceptable base salts.
    Type: Grant
    Filed: September 28, 1990
    Date of Patent: February 25, 1992
    Assignee: Bristol-Myers Squibb Company
    Inventors: Yosuke Sawada, Tomokazu Ueki, Takashi Tsuno, Toshikazu Oki