Abstract: New .alpha.-(cyclic tert. aminophenyl)-aliphatic acids, e.g. those of the formula ##STR1## AND FUNCTIONAL DERIVATIVES THEREOF, ARE ANTI-INFLAMMATORY AGENTS.

Abstract: The present invention relates to dialkyl ({[3-(alkoxy-carbonyl)-1,4-dihydro-4-oxo-8-quinolinyl]amino}methylene)-pro panedioates having the following structural formula: ##STR1## wherein R.sub.1 is lower alkyl; and R.sub.2 is hydrogen, halogen, lower alkyl or nitro.These compounds exhibit antibacterial activity against gram positive and gram negative bacteria and are therefore useful in the treatment of bacterial infections caused by these organisms.

Abstract: Biphenyltetrayltetrakis(sulfonylimino)tetrabenzene dicarboxyic acid alkali metal salts, useful as complement inhibitors, and a biphenyltetrayltetrakis(sulfonylimino)tetrabenzene dicarboxylic acid octakis methoxyethyl ester that is a new intermediate for the preparation of the active salts.

Abstract: s-Phenenyltris(ureylene)triisophthalic acid salts useful as complement inhibitors.

Abstract: Anionic substituted benzenetetrayltetrakis-(carbonylimino)tetraisophthalic acid salts, useful as complement inhibitors, and a methoxyethyl substituted benzenetetrayltetrakis(carbonylimino)tetraisophthalic acid ester that is a new intermediate for the preparation of the active salts.

Abstract: Novel quinoline-3-carboxamides of the formula ##STR1## wherein R.sub.1 is in the 5,6,7 or 8-position and is selected from the group consisting of hydrogen, halogen, --CF.sub.3, --OCF.sub.3, --SCF.sub.3, straight chain alkyl of 1 to 4 carbon atoms, branched alkyl of 3 to 5 carbon atoms and alkoxy of 1 to 4 carbon atoms, R.sub.2 is selected from the group consisting of hydrogen and methyl, R.sub.3 is selected from the group consisting of thiazolyl, 4,5-dihydrothiazolyl, pyridinyl, oxazolyl and imidazolyl and R.sub.4 is selected from the group consisting of hydrogen, hydroxyl, alkyl of 1 to 4 carbon atoms, phenyl and benzyl with the proviso that when R.sub.1 is in the 7 or 8-position and is halogen, --CH.sub.3, --OCF.sub.3 or --SCF.sub.3 and R.sub.4 is hydrogen, R.sub.3 is not thiazolyl, pyridinyl or oxazolyl and the non-toxic, pharmaceutically acceptable acid addition salts when R.sub.3 is imidazolyl or 4,5-dihydrothiazolyl having analgesic activity and their preparation and novel intermediates therefore.

Abstract: Chlorine-substituted vinylaminobenzoic acid compounds of the formula ##STR1## in which R is hydroxyl, alkoxy of from 1 to 4 carbon atoms or monoalkylamino of from 1 to 3 carbon atoms,R.sup.1, r.sup.4 and R.sup.5 are individually selected from hydrogen and chlorine, provided that at least one of R.sup.1, R.sup.4 and R.sup.5 is chlorine,R.sup.2 is alkylcarbonyl of from 1 to 4 carbon atoms in the alkyl moiety or carbalkoxy of from 1 to 4 carbon atoms in the alkoxy moiety; andR.sup.3 is cyano, alkylcarbonyl of from 1 to 4 carbon atoms in the alkyl moiety or carbalkoxy of from 1 to 4 carbon atoms in the alkoxy moietyExhibit outstanding plate growth regulating effects, e.g., the inhibition of vegetative plant growth.

Abstract: An antioxidant useful for stabilizing polyesters having the formula ##STR1## where R.sub.1 is hydrogen or a lower alkyl radical; R.sub.2 is a monovalent radical containing carbon, hydrogen, and oxygen, free of ethylenic or acetylenic unsaturation, and having a molecular weight between about 99-300 and, further, containing two carboxyl groups or their ester forming equivalents; R.sub.3 and R.sub.4 are tertiary alkyl radicals each containing not more than 8 carbon atoms; and x is an integer of from 0-4.

Abstract: Compounds represented below ##STR1## and pharmaceutical compositions thereof, the compositions including the non-substituted phenylene dioxamates are useful in the prophylactic treatment of sensitized mammals for allergy and all anaphylactic reactions of a reagin or non-reagin mediated nature.

Abstract: New carboxylic acid derivatives are proposed for use as agents in the treatment of prevention of arteriosclerosis. 1-(p-chlorophenoxy)-3-(N-phenyl-N-carbomethoxymethylamino)-2-propanol is a typical compound.

Abstract: Novel imide carboxylates, O-carboxylates thereof, and amide carboxylates are useful as intermediates for preparation of sequestrant compounds.

Abstract: Anti-allergic agents of aromatic oxamic acid derivation present the following formula: ##STR1## in which A is a member selected from the group consisting of .alpha.-naphthyl, .beta.-naphthyl, phenyl, 2,6-dichlorophenyl, and substituted phenyl moieties containing from one to three substituents in any of the 2,3,4 and 5 positions of the phenyl ring, independently selected from the group consisting of lower alkyl, lower alkylthio, lower alkylsulfinyl, lower alkoxy, hydroxy (lower)alkoxy, 2-(oxalyloxy) ethoxy, benzyloxy, N-mono- and di-lower alkylamino(lower)alkoxy, halo, sulfamyl, polyhalo(lower)alkyl, carbamyl, N-lower alkylcarbamyl, nitro, mono and di lower alkylamino, carboxy, lower alkylcarbonyl, carb(lower)alkoxy, phenoxy(lower)alkoxy, and oxalamidophenoxy radicals;And pharmaceutically acceptable salts thereof.

Abstract: New 1-aza-4-thiacyclohexane-4,4-dioxide derivatives are used alone or in combination with other stabilizers for stabilizing organic materials. The new compounds are prepared by reacting substituted diallylsulfides with ammonia, amines or hydrazines.

Abstract: Novel imide carboxylates, O-carboxylates thereof, and amide carboxylates are useful as intermediates for preparation of sequestrant compounds.

Abstract: Novel polyfunctional compounds which may be hydrolyzed to the corresponding salts, which in turn are metal sequestering agents, are disclosed, as well as a novel method for their preparation. The compounds are the reaction product obtained from the reaction of selected salts of monoalkyl esters of maleic acid with selected active hydrogen containing compounds. These products are prepared by a reaction of the starting materials in preferably a substantially anhydrous medium at an elevated temperature.

Abstract: Compounds of the general formula I ##STR1## in which R represents hydrogen or a lower alkyl radical which may be further substituted, n is an integer of from 1 to 4, and which may contain further non-chromophoric substituents. They are prepared by reaction of the dichloride of naphthalene-1,4-dicarboxylic acid with an o-aminophenol and subsequent ring closure. These compounds can be used as optical brighteners.

Abstract: Disclosed is a process for making a C.sub.1 -C.sub.7 aliphatic hydrocarbyl ester of an N-[2,6-(C.sub.1 -C.sub.7 alkyl)phenyl] .alpha.-amino-carboxylic acid from the corresponding 2,6-di(C.sub.1 -C.sub.7 alkyl)aniline and the corresponding chlorocarboxylic acid ester, which comprises effecting with a catalytic quantity of di(C.sub.1 -C.sub.7 alkyl)aniline hydrochloride the reaction of said aniline and said ester.