Abstract: This invention relates to novel 1-[4-(R.sub.1 R.sub.2 N-C.sub.n H.sub.2n -O)phenyl]-5-R.sub.4 -2-(4-R.sub.3 -phenyl)indoles having antifertility and hypocholesterolemic activities and to novel intermediates for their preparation.

Abstract: Novel 2-(aminoalkyl)-6,7-dihydroindolo[1,7-ab][1]benzazepines and acid-addition salts thereof having antibacterial activity, and intermediate and process for the preparation thereof are disclosed.

Abstract: Novel 2-(aminoalky)-6,7-dihydroindolo[1,7-ab] 1,7-ab][1]benzazepines and acid-addition salts thereof having antibacterial activity, and intermediate and process for the preparation thereof are disclosed.

Abstract: The compounds of this invention are novel 1-phenyl-3-azacarbocyclic-ureas having anthelmintic activity which are prepared by the reaction of azacarbocyclicamines or azacarbocyclicimines with appropriate phenyl isocyanates.

Abstract: 3-(Substituted-amino)-1,2,3,4-tetrahydrocarbazoles are prepared by reacting appropriate 4-substituted-aminocyclohexanones with a phenylhydrazine, by reacting a 3-(sulfonyloxy)-1,2,3,4-tetrahydrocarbazole with an appropriate substituted amine, or by reduction of an appropriate 3-(acylamino)-1,2,3,4-tetrahydrocarbazole. The 3-(substituted-amino)-1,2,3,4-tetrahydrocarbazoles of this invention have analgetic and psychotropic activities. Moreover, certain of these compounds also have antihistaminic activity.

Abstract: Novel 9-aroyl-1,2,3,4-tetrahydrocarbazoles bearing a carboxy substituent at position 3 or 4 and corresponding esters having antiinflammatory activity, the preparation thereof and novel intermediates therefor are described.

Abstract: The invention relates to novel tetrahydro-2H-1,3,5-thiadiazine-2-thiones substituted at the 3 and 5 positions by R--O--A or R--O--benzyl, wherein R is alkyl and A is alkylene, having antimicrobial activity.

Abstract: Novel 3-Z-9-benzoyl-1,2,3,4-tetrahydrocarbazoles, wherein Z is CONR.sub.5 R.sub.6, CONHOH, CN, or COCH.sub.2 X, where X is chloro or bromo, having antimicrobial and/or anti-inflammatory activity are disclosed. Compounds wherein Z is CONR.sub.5 R.sub.6 and CONHOH are prepared from the corresponding 3-carboxylic acids by conversion to the corresponding acid chlorides and subsequent reaction with the appropriate amines and hydroxylamine respectively; compounds where Z is CN are prepared by the dehydration of the corresponding compounds where Z is CONH.sub.2 ; and the compounds where Z is COCH.sub.2 X are prepared by reacting hydrogen chloride or bromide with the corresponding compounds where Z is COCHN.sub.2 which in turn is prepared from the corresponding 3-carboxylic acid chloride by reaction with diazomethane.

Abstract: Novel 4-R.sub.1 R.sub.2 NCH.sub.2 -9-benzyl-6-R.sub.3 -7-R.sub.4 -1,2,3,4-tetrahydrocarbazoles having antibacterial activity are disclosed. The compounds are prepared by the chemical reduction of the corresponding 4-R.sub.1 R.sub.2 NCO-9-benzyl-6-R.sub.3 -7-R.sub.4 -1,2,3,4-tetrahydrocarbazoles.

Abstract: 3-(Dimethylamino)-1,2,3,4,8,9-hexahydro-1H[1]benzazepino[1,2,3-k,j]carbazol e and acid-addition salts thereof having anti-bacterial activity, and process for the preparation thereof are disclosed.