Hetero Ring Containing Patents (Class 504/195)
  • Patent number: 11647751
    Abstract: The invention primarily relates to the use of phosphorus containing herbicidal active ingredients (herbicides) as desiccant for (parts of) plants of the genus Saccharum, and to corresponding methods for desiccation, i.e. for the desiccating treatment. In another aspect the present invention relates to a method for increasing the amount of saccharose (sucrose) obtainable from (aerial parts of) plants of the genus Saccharum officinarum, and to a method for producing saccharose from (aerial parts of) plants of the genus Saccharum officinarum.
    Type: Grant
    Filed: December 16, 2014
    Date of Patent: May 16, 2023
    Assignee: BASF SE
    Inventors: Luis Eduardo Alves Corrêa, Paulo Cesar Idalgo Donadoni, Thiago De OLIVIERA, Juliano Negrisido Della Valle, Rodolfo Carvalho César De San Juan
  • Patent number: 9556121
    Abstract: The present application relates to novel pyridyloxyalkylcarboxamides of the formula (I) and to their use as endoparasiticides against endoparasites in animals or humans, and to their use as nematicides for controlling phytopathogenic nematodes, and furthermore to endoparasiticides and nematicides comprising pyridyloxyalkylcarboxamides.
    Type: Grant
    Filed: November 8, 2013
    Date of Patent: January 31, 2017
    Assignee: BAYER CROPSCIENCE AG
    Inventors: Joerg Nico Greul, Hans-Georg Schwarz, Bernd Alig, Angela Becker, Daniela Portz, Kerstin Ilg, Ulrich Goergens, Claudia Welz
  • Patent number: 9346839
    Abstract: Benzothiazole phosphonate analogs and methods of using the same to inhibit the activity of Amyloid Binding Alcohol Dehydrogenase and in the amelioration or treatment of Alzheimer's disease are provided.
    Type: Grant
    Filed: November 12, 2014
    Date of Patent: May 24, 2016
    Assignee: University of Kansas
    Inventors: ShiDu Yan, Koteswara Rao Valasani
  • Patent number: 9221853
    Abstract: This invention provides the herbicidal active ingredient, a dimethylamine salt crystal of N-phosphonomethyl glycine (glyphosate), its preparation process and a solid formulation containing the crystalline dimethylamine salt of glyphosate as well as its application. Said preparation process comprises adding glyphosate and a suitable amount of solvent into a conventional reactor and introducing a dimethylamine gas for reaction, wherein the reaction temperature is controlled between 5 and 90° C. After the completion of the reaction, the temperature is reduced slowly to a certain value, a crystalline dimethylamine salt of glyphosate is precipitated (or precipitated after a crystal seed is added).
    Type: Grant
    Filed: October 25, 2010
    Date of Patent: December 29, 2015
    Assignee: ZHEJIANG WYNCA CHEMICAL INDUSTRY GROUP CO., LTD.
    Inventors: Wei Wang, Shuguang Zhou, Long Qin, Bufan Ren, Zhigang Qian, Tao Liu, Huiling She, Yaxian Zhang
  • Patent number: 9212140
    Abstract: The invention relates to (5s,8s)-3-(4?-chloro-3?-fluoro-4-methylbiphenyl-3-yl)-4-hydroxy-8-methoxy-1-azaspiro[4.5]dec-3-en-2-one for therapeutic purposes, to pharmaceutical compositions and to their use in therapy, in particular for the prophylaxis and therapy of tumour disorders.
    Type: Grant
    Filed: February 3, 2012
    Date of Patent: December 15, 2015
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Ningshu Liu, Kai Thede, Philip Lienau, Arne Scholz, Christoph-Stephan Hilger, Ulf Bömer, Maher Najjar, Knut Eis, Reiner Fischer, Wahed Ahmed Moradi
  • Publication number: 20150141251
    Abstract: The present disclosure relates to a pesticidal formulation including i) at least one pesticide, typically an organophosphate compound in an amount between 5.0% w/w and 40.0% w/w, preferably between 15.0% w/w and 30.0% w/w, ii) Solvent system comprising at least one glycol ether and at least one lactone in an amount between 10.0% to 80.0% w/w, preferably between 30.0% w/w and 55% w/w, with ratio of the glycol ether and the lactone is the in the range of 1:9 and 9:1, preferably in the range of 2:8 and 4:6, iii) Surfactant system containing at least two nonionic surfactants where the primary surfactant has an HLB range of 10 to 20 and the co-surfactant has a HLB range 1 to 5, in an amount ranging between 0.1% w/w to 60.0% w/w preferably in the range of 20.0% w/w to 40.0% w/w, and iv) at least one excipient in the range of 0.1% w/w to 10% w/w and preferably 0.5% w/w to 5.0% w/w.
    Type: Application
    Filed: October 15, 2013
    Publication date: May 21, 2015
    Applicant: GOWAN COMERCIO INTERNACIONAL E SERVICOS LIMIADA
    Inventors: Howard Bernard DAWSON, Rachel BRANAGHAN, Eric James MCEWEN, Sandra ALCARAZ, Tak Wai CHEUNG
  • Patent number: 9012365
    Abstract: The present invention generally relates to a method for minimizing the formation of insoluble salts of phenoxy herbicides. The method comprises (1) mixing a compatibility agent, amine salts of phenoxy acid herbicides, and a chemical containing non-amine cations in a aqueous system to form a stable and non-nozzle plugging solution; and (2) application of said stable and non-nozzle plugging solution onto target plants.
    Type: Grant
    Filed: March 30, 2007
    Date of Patent: April 21, 2015
    Assignee: Akzo Nobel N.V.
    Inventors: Jinxia Susan Sun, Shawn Zhu, Shuaib A. Khan
  • Publication number: 20140274688
    Abstract: This disclosure relates to the field of molecules having pesticidal utility against pests in Phyla Nematoda, Arthropoda, and/or Mollusca, processes to produce such molecules and intermediates used in such processes, compositions containing such molecules, and processes of using such molecules against such pests. These molecules may be used, for example, as nematicides, acaricides, insecticides, miticides, and/or molluscicides. This document discloses molecules having the following formula (“Formula One”).
    Type: Application
    Filed: March 13, 2014
    Publication date: September 18, 2014
    Applicant: DOW AGROSCIENCES LLC
    Inventors: Lindsey G. Fischer, Erich W. Baum, Gary D. Crouse, Carl DeAmicis, Beth Lorsbach, Jeff Petkus, Thomas C. Sparks, Gregory T. Whiteker
  • Publication number: 20140249029
    Abstract: Suggested are solid agricultural compositions, comprising: (a1) at least one alkoxylated alcohol according to general formula (I) R1O(AO)nH, wherein R1 stands for an unsaturated, linear hydrocarbon residue having 12 to 22 carbon atoms and 1, 2, or 3 double bonds, AO comprises an ethylene oxide, propylene oxide, and/or butylene oxide unit, and n comprises an integer of from 1 to 60; (a2) at least one alkoxylated alcohol according to general formula (II) R2O(AO)mH, wherein R2 comprises a saturated, branched hydrocarbon residue having 8 to 36 carbon atoms, AO comprises an ethylene oxide, propylene oxide, and/or butylene oxide unit, and m comprises an integer of from 1 to 60; (b) at least one biocide, and optionally (c) at least one inert Broenstedt base and/or (d) at least one solvent, emulsifier, polymer or filler, therein the compositions are granules with a water content of less than 10% b.w.
    Type: Application
    Filed: September 27, 2011
    Publication date: September 4, 2014
    Applicant: Cognis IP Management GmbH
    Inventors: Jianhua Mao, Anbao Zuo
  • Publication number: 20140206541
    Abstract: Suggested are agricultural compositions, comprising one or more esters of C6-C22 monocarboxylic acids or C2-C20 dicarboxylic acids and polyhydric alcohols selected from the group consisting of diglycerol, triglycerol, oligo- or polyglycerol and their respective alkylene oxide adducts, one or more biocides, and optionally, one or more oil components or solvents and/or one or more emulsifiers, wherein the esters are essentially free of esters of monomeric glycerol and esters of alkylene oxide adducts of monomeric glycerol. The esters are useful for forming agricultural compositions using hard water.
    Type: Application
    Filed: January 24, 2013
    Publication date: July 24, 2014
    Inventors: Dean Oester, Mike White, Timothy H. Anderson
  • Patent number: 8748346
    Abstract: The present invention relates to the blending of key nutritional and hormonal components for successful application through a controlled drop applicator to satisfy plant requirements for growth. More specifically this invention provides a micronutrient composition for enhancing plant growth made of a mixture of gibberellic acid dissolved in triethanolamine. The gibberellic acids are: Gibberellic acid 4, Gibberellic acid 7, Gibberellic acid 9, Gibberellic acid 12. The gibberellic acids are mixed with kinetin dissolved in an alcohol; tryptophan dissolved in a humic acid solution; and a sufficient amount of a chelating agent.
    Type: Grant
    Filed: April 17, 2012
    Date of Patent: June 10, 2014
    Assignee: Floratine Products Group, Inc.
    Inventors: Kevin Cavanaugh, Timothy B. Cartwright
  • Publication number: 20140128265
    Abstract: The invention relates to compositions that contain A) one or more copolymers, said copolymers containing one or more structural units obtained from a) 19.9 to 75.9 wt. % glycerin, b) 0.1 to 30 wt. % at least one dicarboxylic acid, and c) 24 to 80 wt. % at least one monocarboxylic acid according to formula (I) R1—COOH (I), in which R1 is (C5-C29)-alkyl; (C7-C29)-alkenyl; phenyl; or naphthyl, and B) one or more solvents that are not miscible with water. The invention is characterized in that said compounds either do not contain water or contain water in a quantity less than or equal to 1.0 wt. % with respect to the total weight of the respective composition. The compositions are advantageously suitable for producing pesticide compositions for example.
    Type: Application
    Filed: March 8, 2012
    Publication date: May 8, 2014
    Applicant: CLARIANT FINANCE (BVI) LIMITED
    Inventor: Andreas Wacker
  • Patent number: 8541343
    Abstract: Compounds of the formula (I), wherein the substituents are as defined in claim 1, are useful as a pesticides.
    Type: Grant
    Filed: November 29, 2010
    Date of Patent: September 24, 2013
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Thomas Pitterna, Michel Muehlebach, Jurgen Harry Schaetzer
  • Publication number: 20130012384
    Abstract: The present invention relates to novel compounds of the formula (I), in which W, X, Y, Z, G, A and t have the meanings given above, to a plurality of processes and intermediates for their preparation and to their use as pesticides and/or herbicides. Moreover, the invention relates to selective herbicidal compositions comprising, firstly, the spiroheterocyclic tetronic acid derivates and, secondly, a crop plant compatibility-improving compound. The present invention furthermore relates to increasing the activity of crop protection compositions comprising in particular phenyl-substituted bicyclooctane-1,3-dione derivates by adding ammonium salts or phosphonium salts and, if appropriate, penetrants, to the corresponding compositions, to processes for their preparation and to their use in crop protection as insecticides and/or acaricides and/or for preventing unwanted plant growth.
    Type: Application
    Filed: September 14, 2012
    Publication date: January 10, 2013
    Applicant: Bayer CropScience AG
    Inventors: Thomas BRETSCHNEIDER, Reiner Fischer, Stefan Lehr, Olga Malsam, Arnd Voerste
  • Publication number: 20120283099
    Abstract: The invention disclosed in this document concerns controlling planthoppers.
    Type: Application
    Filed: May 4, 2012
    Publication date: November 8, 2012
    Applicant: DOW AGROSCIENCES LLC
    Inventors: Agamananda Roy, Sanjoy Kundu, Suresh Ramachandran
  • Publication number: 20120108431
    Abstract: The present invention relates to a method and composition for improving the efficacy of a plant growth regulator by the use of, particularly but not exclusively, anthranilic acid in combination with an additional agrochemically acceptable additive.
    Type: Application
    Filed: April 7, 2010
    Publication date: May 3, 2012
    Applicant: TAMINCO, NAAMLOZE VENNOOTSCHAP
    Inventors: Richard Williams, Peter Roose, Johan Josef De Saegher
  • Patent number: 7732374
    Abstract: A fungicidal mixture comprising prothioconazole or its salts or adducts and at least one insecticide selected from the group consisting of fipronil, chlorpyrifos or thiamethoxam.
    Type: Grant
    Filed: July 17, 2007
    Date of Patent: June 8, 2010
    Assignee: BASF SE
    Inventors: Eberhard Ammermann, Reinhard Stierl, Gisela Lorenz, Siegfried Strathmann, Klaus Schelberger, V. James Spadafora, Thomas Christen
  • Patent number: 7041625
    Abstract: The present invention generally relates to methods of inhibiting ethylene responses in plants and plant materials, and particularly relates to methods of inhibiting various ethylene responses including plant maturation and degradation, by exposing plants to cyclopropene derivatives and compositions thereof wherein the cyclopropene is associated with another ring system.
    Type: Grant
    Filed: August 21, 2003
    Date of Patent: May 9, 2006
    Assignee: Rohm and Haas Company
    Inventors: Richard Martin Jacobson, Martha Jean Kelly, Fiona Linette Wehmeyer, Edward C. Sisler
  • Patent number: 6653256
    Abstract: Microcapsule formulations of A) a particulate disperse phase of a) a reaction product of at least one diamine, polyamide, dialcohol, polyalcohol and/or aminoalcohol with an isocyanate mixture characterized in the description, if appropriate as a mixture with toluylene diisocyanate, b) at least one agrochemically active compound of a particular group of substances and, c) if appropriate, additives, and B) a liquid aqueous phase, a process for the preparation of these formulations, and their use for applying the active compounds which they comprise.
    Type: Grant
    Filed: March 1, 2001
    Date of Patent: November 25, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hilmar Wolf, Joachim Weissmüller
  • Patent number: 6566306
    Abstract: Microcapsule formulations of A) a particulate disperse phase of a) a reaction product of the isocyanate of the formula if appropriate as a mixture with toluylene diisocyanate, and at least one diamine, polyamine, dialcohol, polyalcohol and/or aminoalcohol, b) at least one agrochemically active compound of a particular group of substances and, c) if appropriate, additives, and B) a liquid aqueous phase, a process for the preparation of these formulations, and their use for applying the active compounds which they comprise.
    Type: Grant
    Filed: March 1, 2001
    Date of Patent: May 20, 2003
    Assignee: Bayer Aktiengesellschaft
    Inventors: Hilmar Wolf, Joachim Weissmüller, Maria Giuliana Cianciulli Teller
  • Publication number: 20020160916
    Abstract: The invention pertains to new composition and a method for increasing the solubility of various agricultural compounds in water at a low pH. The compounds included in this patent are typically not soluble at pH ranges less than 7 to produce commercially viable liquid concentrates. This method requires the use of amine-containing surfactants and organic acids to lower the pH of various compounds and also keep them soluble in water.
    Type: Application
    Filed: February 20, 2002
    Publication date: October 31, 2002
    Inventors: Greg Volgas, Johnnie R. Roberts, Amanda Hayes
  • Patent number: 6100218
    Abstract: 2-Phenylpyridines I ##STR1## wherein X is a chemical bond, 1,2-ethynediyl or optionally substituted --(CH.sub.2).sub.1-3 --, --O--(CH.sub.2).sub.1-2 --, --s--(CH.sub.2).sub.1-2 --, --CH.sub.2 --O--CH.sub.2 --, --CH.sub.2 --S--CH.sub.2 -- or --CH.dbd.CH--;Y is oxygen or sulfur;Z.sup.1 is oxygen, sulfur or --N(R.sup.7)--;Z.sup.2 is oxygen, sulfur or --N(R.sup.8)--;R.sup.1, R.sup.2, R.sup.7 and R.sup.8 independently of one another are hydrogen, optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, phenyl or heterocyclyl; orR.sup.1 and R.sup.2 or R.sup.7, or R.sup.2 and R.sup.8 together are optionally substituted --(CH.sub.2).sub.2-5 -- or --(CH.sub.2).sub.2 --O--(CH.sub.2).sub.2 --, orR.sup.1 and R.sup.2 together are optionally substituted 1,2-phenylene;R.sup.3 is cyano, halogen, alkyl, haloalkyl, alkoxy or haloalkoxy;R.sup.4 and R.sup.5 are hydrogen or halogen;R.sup.
    Type: Grant
    Filed: August 4, 1998
    Date of Patent: August 8, 2000
    Assignee: BASF Aktiengesellschaft
    Inventors: Cyrill Zagar, Peter Schafer, Gerhard Hamprecht, Elisabeth Heistracher, Markus Menges, Olaf Menke, Karl-Otto Westphalen, Ulf Misslitz, Helmut Walter
  • Patent number: 6039966
    Abstract: A low volatile organic compound co-solvent system is disclosed for preparing emulsion concentrates of water-insoluble pesticides having a melting point of less than about 110.degree. C. The co-solvent system comprises a water-soluble ethoxylated fatty acid/rosin acid-nonionic surfactant composition.
    Type: Grant
    Filed: December 16, 1998
    Date of Patent: March 21, 2000
    Assignee: Aquatrols Corporation of America, Inc.
    Inventors: Stanley J. Kostka, Rennan Pan
  • Patent number: 5830826
    Abstract: The present invention relates to novel 1H-3-aryl-pyrrolidine-2,4-dione derivatives of the formula (I) ##STR1## in which A, B, G, X, Y and Z have the meaning given in the description, to processes for their preparation and to intermediates for this purpose. The compounds of the formula (I) are used as pesticides and herbicides.
    Type: Grant
    Filed: September 27, 1996
    Date of Patent: November 3, 1998
    Assignee: Bayer Aktiengesellschaft
    Inventors: Reiner Fischer, Thomas Bretschneider, Bernd-Wieland Kruger, Michael Ruther, Christoph Erdelen, Ulrike Wachendorff-Neumann, Hans-Joachim Santel, Markus Dollinger
  • Patent number: 5811374
    Abstract: New 3-arylpyrrolidine-2,4-dione derivatives of the formula (I): ##STR1## in which the variables A, B, E, R, X, Y, Z and n are set forth in the specification, are useful as insecticides, acaricides, and herbicides.
    Type: Grant
    Filed: June 7, 1995
    Date of Patent: September 22, 1998
    Assignee: Bayer Aktiengesellschaft
    Inventors: Heinz-Jurgen Bertram, Reiner Fischer, Bernd-Wieland Kruger, Christoph Erdelen, Klaus Lurssen, Robert R. Schmidt, Hans-Joachim Santel
  • Patent number: 5728650
    Abstract: Herbicidal compositions containing a bisphosphonic acid compound of the formula ##STR1## wherein n is 0, 1, 2, 3, 4, 5 or 6, or an agrochemically acceptable salt or hydrolyzable ester thereof and methods of controlling undesirable plant growth using these bisphosphonic acid containing compositions. The herbicidal compositions exhibit desirable efficacy when applied to plants post-emergence, but exhibit little significant activity when applied to plants pre-emergence. Novel aza-bisphosphonic acid compounds are also disclosed.
    Type: Grant
    Filed: April 7, 1995
    Date of Patent: March 17, 1998
    Assignee: Zeneca Limited
    Inventors: Karl J. Fisher, Frank X. Woolard, Michael R. Leadbetter, John M. Gerdes
  • Patent number: 5693590
    Abstract: This invention pertains to compositions comprising herbicidal phosphosulfonates, having the general formula ##STR1## wherein Y is an optionally substituted phenyl, naphthyl, benzyl, a (C.sub.5 -C.sub.8)cycloalkyl, a 5-membered heteroaromatic ring, a 6-membered heteraromatic ring, a fused 5,6-membered heteroaromatic ring, or a fused 6,6-membered heteroaromatic ring;X is an oxygen or a sulfur atom; andR.sup.1 and R.sup.2 are each independently selected from substituted or unsubstituted alkyl, alkoxy, alkylthio, alkenyloxy, alkynyloxy, haloalkoxy, cyanoalkoxy, alkoxyalkoxy, cycloalkyloxy, cycloalkylalkoxy, alkylideneiminooxy, chloro, amino, phenyl or phenoxy; or R.sup.1 and R.sup.2 are both alkoxy, taken together with the phosphorus atom to form a 6-membered oxygen-containing ring; anddichloroacetamide safeners having the general formula ##STR2## wherein R.sup.a and R.sup.b are each independently selected from alkyl, alkenyl, or alkyl or alkenyl substituted with halo, or R.sup.a and R.sup.
    Type: Grant
    Filed: July 20, 1995
    Date of Patent: December 2, 1997
    Assignee: Rohm and Haas Company
    Inventors: James Delbert Fisher, Ernest Leroy Burdge, Vincent Angelo Musco, Jr., Lori Ann Spangler
  • Patent number: 5622917
    Abstract: The invention relates to new 1H-3-aryl-pyrrolidine-2,4-dione derivatives of the formula (I) ##STR1## in which A, B, X, Y and G have the meanings given in the description, to a plurality of processes for their preparation, and to their use as pesticides.
    Type: Grant
    Filed: January 3, 1995
    Date of Patent: April 22, 1997
    Assignee: Bayer Aktiengesellschaft
    Inventors: Reiner Fischer, Thomas Bretschneider, Bernd-Wieland Kr uger, Michael Ruther, Christoph Erdelen, Ulrike Wachendorff-Neumann, Hans-Joachim Santel, Markus Dollinger
  • Patent number: 5500405
    Abstract: This invention pertains to phosphosulfonates, having the general formula ##STR1## wherein Y is phenyl, naphthyl, benzyl, a (C.sub.5 -C.sub.8)cycloalkyl, a 5-membered heteroaromatic ring, a 6-membered heteraromatic ring, a fused 5,6-membered heteroaromatic ring, or a fused 6,6-membered heteroaromatic ring; andX is oxygen or sulfur; andR.sup.1 and R.sup.2 are each independently selected from substituted or unsubstituted alkyl, alkoxy, alkylthio, alkenyloxy, alkynyloxy, haloalkoxy, cyanoalkoxy, alkoxyalkoxy, cycloalkyloxy, cycloalkylalkoxy, alkylideneiminooxy, chloro, amino, phenyl or phenoxy; or R.sup.1 and R.sup.2 are both alkoxy, taken together with the phosphorus atom to form a 6-membered oxygen-containing ring; compositions containing these compounds and their use as herbicides.
    Type: Grant
    Filed: September 22, 1993
    Date of Patent: March 19, 1996
    Assignee: Rohm and Haas Company
    Inventors: Robert E. Rosen, Damian G. Weaver, Jane W. Cornille, Lori A. Spangler
  • Patent number: 5272128
    Abstract: This invention pertains to phosphosulfonates, having the general formula ##STR1## wherein Y is phenyl, naphthyl, benzyl, a (C.sub.5 -C.sub.8)cycloalkyl, a 5-membered heteroaromatic ring, a 6-membered heteraromatic ring, a fused 5,6-membered heteroaromatic ring, or a fused 6,6-membered heteroaromatic ring; andX is oxygen or sulfur; andR.sup.1 and R.sup.2 are each independently selected from substituted or unsubstituted alkyl, alkoxy, alkylthio, alkenyloxy, alkynyloxy, haloalkoxy, cyanoalkoxy, alkoxyalkoxy, cycloalkyloxy, cycloalkylalkoxy, alkylideneiminooxy, chloro, amino, phenyl or phenoxy; or R.sup.1 and R.sup.2 are both alkoxy, taken together with the phosphorus atom to form a 6-membered oxygen-containing ring; compositions containing these compounds and their use as herbicides.
    Type: Grant
    Filed: April 1, 1992
    Date of Patent: December 21, 1993
    Assignee: Rohm and Haas Company
    Inventors: Robert E. Rosen, Damian G. Weaver, Jane W. Cornille, Lori A. Spangler
  • Patent number: 5216171
    Abstract: 2-Amino-4-trichloromethylpyridines of the general formula I ##STR1## where R.sup.1 is hydrogen or C.sub.1 -C.sub.8 -alkyl,R.sup.2 is C.sub.1 -C.sub.8 -alkyl, C.sub.5 -C.sub.8 -cycloalkyl, C.sub.2 -C.sub.4 -alkenyl or phenyl, benzyl or phenylsulfonyl,--CX--R.sup.3, --SO.sub.2 R.sup.3 or --PX(OR.sup.4).sub.2 orR.sup.1 and R.sup.2 together form .dbd.CR.sup.5 R.sup.6 or --CO--Z--CO--,X is oxygen or sulfur,R.sup.3 is C.sub.1 -C.sub.20 -alkyl, C.sub.2 -C.sub.6 -alkenyl, amino, C.sub.1 -C.sub.6 -alkylamino, di-C.sub.1 -C.sub.6 -alkylamino, morpholino, piperidino, pyrazolidino or C.sub.1 -C.sub.8 -alkylcarbonylamino, substituted or unsubstituted phenylamino or benzylamino,R.sup.4 is C.sub.1 -C.sub.8 -alkyl, C.sub.1 -C.sub.8 -haloalkyl or substituted or unsubstituted phenyl,R.sup.5 is hydrogen, C.sub.1 -C.sub.4 -alkyl, or substituted or unsubstituted phenyl,R.sup.
    Type: Grant
    Filed: April 8, 1991
    Date of Patent: June 1, 1993
    Assignee: BASF Aktiengesellschaft
    Inventors: Helmut Hagen, Hans Ziegler, Juergen Pfister, Gerhard Nilz, Gisela Lorenz, Juergen Dressel
  • Patent number: 5205852
    Abstract: Herbicidal compounds have the formula ##STR1## in which R is C.sub.3 -C.sub.6 alkyl or C.sub.3 -C.sub.6 cycloalkyl;X is oxygen or sulfur;R.sub.1 is C.sub.1 -C.sub.12 alkyl, C.sub.3 -C.sub.6 cycloalkyl optionally substituted with up to two C.sub.1 -C.sub.3 alkyl groups, phenyl, or substituted phenyl having from 1 to 2 substituents selected from halo, nitro, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 thioalkyl, C.sub.3 -C.sub.4 alkenyl, C.sub.1 -C.sub.4 alkoxycarbonyl, and phenyl;R.sub.2 is hydrogen, C.sub.1 -C.sub.6 alkyl or C.sub.3 -C.sub.6 cycloalkyl; andR.sub.3 is C.sub.2 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, phenyl or substituted phenyl having from 1 to 2 substituents selected from C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkyl and halogen;provided that if R.sub.2 is hydrogen, R.sub.3 is not phenyl or substituted phenyl;or R.sub.2 and R.sub.3 taken together with the nitrogen atom form a 4-8 membered ring, optionally including an oxygen heteroatom.
    Type: Grant
    Filed: November 12, 1991
    Date of Patent: April 27, 1993
    Assignee: Imperial Chemical Industries PLC
    Inventors: Michael D. Broadhurst, Tsze H. Tsang
  • Patent number: 5188642
    Abstract: This invention involves a cloning or expression vector comprising a gene which encodes 5-enolpyruvylshikimate-3-phosphate synthase (EPSPS) polypeptide which, when expressed in a plant cell contains a chloroplast transit peptide which allows the polypeptide, or an enzymatically active portion thereof, to be transported from the cytoplasm of the plant cell into a chloroplast in the plant cell, and confers a substantial degree of glyphosate resistance upon the plant cell and plants regenerated therefrom.The EPSPS coding sequence may be ligated to a strong promoter, such as the 35S promoter from cauliflower mosaic virus, to create a chimeric gene. Such genes can be inserted into plant transformation vectors, and subsequently introduced into plant cells. Plant cells transformed using such genes and plants regenerated therefrom have been shown to exhibit a substantial degree of glyphosate resistance.
    Type: Grant
    Filed: February 12, 1990
    Date of Patent: February 23, 1993
    Assignee: Monsanto Company
    Inventors: Dilip M. Shah, Stephen G. Rogers, Robert B. Horsch, Robert T. Fraley
  • Patent number: 5186733
    Abstract: Herbicides have the formula ##STR1## in which R is hydrogen, mono- or poly-halo, mono- or di-(C.sub.1 -C.sub.4 alkyl), C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkoxy, phenoxy or nitro;R.sub.1 is hydrogen or C.sub.1 -C.sub.4 alkyl;R.sub.3 is C.sub.1 -C.sub.6 alkyl;R.sub.2 is C.sub.2 -C.sub.4 alkyl, C.sub.3 -C.sub.6 cycloalkyl, phenyl, optionally substituted by C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkoxy, one or more halogens, or two C.sub.1 -C.sub.4 alkoxy groups, or one C.sub.1 -C.sub.4 alkyl and one C.sub.1 -C.sub.4 alkoxy group, phenyl-(C.sub.1 -C.sub.2)alkyl or pyridyl; orR.sub.1 and R.sub.2, and/or R.sub.3 and R.sub.4 respectively, taken together with the nitrogen atom, form a 4-8 member ring, optionally including an oxygen heteroatom;and R.sub.4 is C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, phenyl, optionally substituted by C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkoxy, one or more halogens, or two C.sub.1 -C.sub.
    Type: Grant
    Filed: November 12, 1991
    Date of Patent: February 16, 1993
    Assignee: Imperial Chemical Industries PLC
    Inventors: Michael D. Broadhurst, Tsze H. Tsang, John Tomko