Patents Represented by Attorney, Agent or Law Firm William A. Teoli, Jr.
  • Patent number: 6133447
    Abstract: 2-chloro-3-hydroxypyridine is prepared by reacting 3-hydroxypyridine with aqueous sodium hypochlorite.
    Type: Grant
    Filed: February 17, 1999
    Date of Patent: October 17, 2000
    Assignee: Novartis Crop Protection, Inc.
    Inventors: Dominik Faber, Denis Blaser, Thierry Bourquard, Andrea Rolf Sting, Dean Kent Hoglen
  • Patent number: 6121455
    Abstract: The invention relates to a process for the preparation of a compound of the formula ##STR1## and, where applicable, its E/Z-isomers, mixtures of E/Z-isomers and/or tautomers, in each case in free form or in salt form, whereinQ is CH or N,Y is NO.sub.2 or CN,Z is CHR.sub.3, O, NR.sub.3 or S,R.sub.1 and R.sub.2 are either each independently of the other hydrogen or unsubstituted or R.sub.4 -substituted C.sub.1 -C.sub.8 alkyl, or together form an alkylene bridge having two or three carbon atoms, and said alkylene bridge may additionally contain a hetero atom selected from the group consisting of NR.sub.5, O and S,R.sub.3 is H or unsubstituted or R.sub.4 -substituted C.sub.1 -C.sub.12 alkyl,R.sub.4 is unsubstituted or substituted aryl or heteroaryl, andR.sub.5 is H or C.sub.1 -C.sub.
    Type: Grant
    Filed: August 13, 1999
    Date of Patent: September 19, 2000
    Assignee: Novartis Crop Protection, Inc.
    Inventors: Thomas Pitterna, Henry Szczepanski, Peter Maienfisch, Ottmar Franz Huter, Thomas Rapold, Marcel Senn, Thomas Gobel, Anthony Cornelius O'Sullivan, Gottfried Seifert
  • Patent number: 6103667
    Abstract: Compounds of formula I ##STR1## wherein the substituents R.sub.1 and R.sub.6 and n are as defined in claim 1, and the salts and stereoisomers of the compounds of formula I have good pre- and post-emergence selective herbicidal properties.The preparation of those compounds and their use as herbicidal active ingredients are described.
    Type: Grant
    Filed: December 12, 1996
    Date of Patent: August 15, 2000
    Assignee: Novartis Corporation
    Inventors: Hans-Georg Brunner, Milan Karvas, Kurt Nebel, Georg Pissiotas
  • Patent number: 6090750
    Abstract: The invention discloses a novel method for reducing phytotoxicity of Dicamba to crop plants, which comprises co-applying to the crop plants or to the locus thereof a phytotoxicity reducing effective amount of a quinolinyloxy alkanoic acid derivative together with a herbicidally effective amount of Dicamba and salt forms thereof.
    Type: Grant
    Filed: March 10, 1997
    Date of Patent: July 18, 2000
    Assignee: Novartis AG
    Inventors: Reynold Chollet, Luke L. Bozeman
  • Patent number: 6083881
    Abstract: Compounds of formula (I) ##STR1## in which the substituents W, R.sub.100, R.sub.101 and R.sub.102 are as defined 1; and the pyrazole N-oxides, salts, complexes and stereoisomer of the compounds of (I) have good pre- and post-emergence selective herbicidal properties. The preparation compounds and their use as herbicidal active compounds are described.
    Type: Grant
    Filed: January 6, 1997
    Date of Patent: July 4, 2000
    Assignee: Novartis Corporation
    Inventors: Kurt Nebel, Hans-Georg Brunner, Georg Pissiotas
  • Patent number: 6071857
    Abstract: A liquid pesticidal composition, which is substantially free of water, comprising a hydrophobic pesticide or mixture of pesticides dissolved in an organic solvent and comprising as surfactants(1) a butanol-ethoxyate/propoxylate-blockcopolymer having 12-30 mol ethoxylate and 16-48 mol propoxylate, in combination with(2) a branched C.sub.8 -C.sub.18 alcohol ethoxylate having 5-10 mol ethoxylate, and/or(3) a tristyrenephenol-ethoxylate having 8-30 mol ethoxylate, or its phosphate or salt thereof.The compositions include also gels having a viscosity of 500 to 20,000 mPas and comprising additionally a gelling agent.
    Type: Grant
    Filed: December 22, 1998
    Date of Patent: June 6, 2000
    Assignee: Novartis Crop Protection, Inc.
    Inventors: Manfred Vogt, William Baettig
  • Patent number: 6066596
    Abstract: A herbicidal synergistic composition, comprising, besides customary inert formulation auxiliaries, a compound of formula I ##STR1## and a synergistically active amount of at least one active ingredient selected from among the compounds of formula II ##STR2## and of formula III ##STR3## and of formula V ##STR4##
    Type: Grant
    Filed: October 11, 1996
    Date of Patent: May 23, 2000
    Assignee: Novartis Corporation
    Inventors: Jean Louis Allard, Manfred Hudetz
  • Patent number: 6063732
    Abstract: The invention relates to compositions comprising: (a) a 4-benzoylisoxazole of formula (I), wherein R, R.sup.1, R.sup.2 and n are as defined in the description and (b) a chloroacetamide herbicide; and their use as herbicides.
    Type: Grant
    Filed: September 3, 1998
    Date of Patent: May 16, 2000
    Assignee: Novartis Crop Protection, Inc.
    Inventor: Willy T. Ruegg
  • Patent number: 6048824
    Abstract: Compounds of formula (I), wherein A is an unsubstituted or substituted aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical wherein a ring nitrogen atom may have been replaced by a group ##STR2## R.sub.1 is hydrogen or C.sub.1 -C.sub.3 alkyl; R.sub.2 is hydrogen or C.sub.1 -C.sub.3 alkyl; R.sub.3 is hydrogen, an unsubstituted or substituted C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl C.sub.2 -C.sub.6 alkenyl or C.sub.2 -C.sub.6 alkynyl group, or C(.dbd.O)--R.sub.5, R.sub.5 is C.sub.1 -C.sub.4 alkyl C.sub.1 -C.sub.4 alkoxy, an unsubstituted or substituted phenyl, phenoxy or benzyloxy group, or N(R.sub.6).sub.2, each R.sub.6, independently of the other, is hydrogen, C.sub.1 -C.sub.4 alkyl or unsubstituted or substituted phenyl, X is CH--NO.sub.2, N--CN or N--NO.sub.2 and n is from 1 to 3, in free form or in salt form, and, where appropriate, tautomers of those compounds and the salts thereof, can be used as agrochemical active ingredients and can be prepared in a manner known per se.
    Type: Grant
    Filed: November 22, 1995
    Date of Patent: April 11, 2000
    Assignee: Novartis Corporation
    Inventors: Peter Maienfisch, Jozef Gonda, Olivier Jacob, Laurenz Gsell
  • Patent number: 6034083
    Abstract: Compounds of formula ##STR1## wherein n and Z are as defined in claim 1, and, where appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.
    Type: Grant
    Filed: July 20, 1998
    Date of Patent: March 7, 2000
    Assignee: Novartis Corp.
    Inventors: Henry Szczepanski, Haukur Kristinsson, Peter Maienfisch, Josef Ehrenfreund
  • Patent number: 6022871
    Abstract: Compounds of the formula ##STR1## in which A is an unsubstituted or mono- to tetrasubstituted, aromatic or non-aromatic, monocyclic or bicyclic heterocyclic radical, where one to two of the substituents of A can be selected from the group consisting of halo-C.sub.1 -C.sub.3 alkyl, cyclopropyl, halocyclopropyl, C.sub.2 -C.sub.3 alkenyl, C.sub.2 -C.sub.3 alkynyl, halo-C.sub.2 -C.sub.3 alkenyl, halo-C.sub.2 -C.sub.3 alkynyl, halo-C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylthio, halo-C.sub.1 -C.sub.3 alkylthio, allyloxy, propargyloxy, allylthio, propargylthio, haloallyloxy, haloallylthio, cyano and nitro, and one to four of the substituents of A can be selected from the group consisting of C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 alkoxy and halogen;R is hydrogen, C.sub.1 -C.sub.6 alkyl, phenyl-C.sub.1 -C.sub.4 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.2 -C.sub.6 alkenyl or C.sub.2 -C.sub.6 alkynyl; andX is N--NO.sub.
    Type: Grant
    Filed: February 18, 1999
    Date of Patent: February 8, 2000
    Assignee: Novartis Corporation
    Inventors: Peter Maienfisch, Laurenz Gsell
  • Patent number: 6017850
    Abstract: A herbicidal composition comprising, in addition to customary inert formulation adjuvants, as active ingredienta) an antagonistically active amount of at least one compound A selected from the group of compounds of formula A.sub.1 ##STR1## and compounds of formula A.sub.2 ##STR2## compounds of formula A.sub.3 ##STR3## b) a herbicidally effective amount of at least one compound G selected from the group of compounds, preferably having the 2R-configuration, of formula G.sub.1 ##STR4## compounds of formula G.sub.2 ##STR5## c) an acid the pK value of which is smaller than the pK values of compounds G and A.
    Type: Grant
    Filed: December 6, 1996
    Date of Patent: January 25, 2000
    Assignee: Novartis Finance Corporation
    Inventors: Michael Donald Johnson, Cheryl Lynn Dunne, Manfred Hudetz, Daniel Worden Kidder
  • Patent number: 5998636
    Abstract: Substituted N-phenyl- and N-heteroarylalkylcarbamates of the formula I ##STR1## in which Q is a group ##STR2## R is halogen, trifluoromethyl, cyano, nitro or C.sub.1 -C.sub.3 haloalkoxy;Z is hydrogen or halogen; orZ and R together in the 2- and 3-position of the phenyl ring form a group --OCF.sub.2 O--;R.sub.1 is C.sub.1 -C.sub.5 alkyl;R.sub.2, R.sub.3, R.sub.4 and R.sub.5, independently of one another, are hydrogen, methyl or ethyl;X is oxygen, sulfur, --SO-- or --SO.sub.2 --;Y is hydrogen, halogen, C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.3 haloalkyl, C.sub.1 -C.sub.3 alkoxy or cyano;n is 0, 1 or 2;n.sub.1 is 0 or 1; andm is 0 or 1,with the proviso that m is 1 if Q is group (1) or (2);and the diastereomers and enantiomers thereof,exhibit pre- and post-emergence herbicidal properties. The preparation of these compounds and their use as herbicidally active ingredients are described.
    Type: Grant
    Filed: August 4, 1998
    Date of Patent: December 7, 1999
    Assignee: Novartis Finance Corporation
    Inventors: Hermann Rempfler, Fredrik Cederbaum, Felix Spindler, Willy Urs Lottenbach
  • Patent number: 5994395
    Abstract: The present invention relates to a composition for controlling parasites, in and on animals, which comprises, as active ingredient, a combination, in variable proportions, of at least one parasiticidally active compound, in free form or in salt form, selected from the N-phenyl-N'-benzoyl-urea class of substances, and at least one parasiticidally active compound, in free form or in salt form, selected from the milbemycin, avermectin, milbemycin oxime, moxidectin, ivermectin, abamectin and doramectin classes of substances; to a method of controlling these parasites; to a process for the preparation of this composition; and to the use of this composition.
    Type: Grant
    Filed: January 23, 1998
    Date of Patent: November 30, 1999
    Assignee: Novartis Animal Health US, Inc.
    Inventors: Philip Anthony Lowndes, Stefan Kemmethmuller, Steven Craig Parks, Douglas Irvin Hepler
  • Patent number: 5986139
    Abstract: A process for the preparation of primary or secondary amines by hydrogenation of imines with hydrogen at elevated pressure and in the presence of a dinuclear Ir(III) complex having ditertiary diphosphine ligands, halide bridges, halide and hydride ligands, or an Ir(III) halide complex salt containing ditertiary diphosphine ligands, as catalyst, wherein the catalyst corresponds to formula I or Ia or to mixtures of at least two compounds of formula I, at least two compounds of formulae I and Ia, or at least two compounds of formula Ia[(DIP)IrX.sub.q Y.sub.r ].sub.2 (I),[(DIP)X.sub.4 ].sup..crclbar. Me.sup..sym. (Ia),whereinDIP is the ditertiary diphosphine ligand of a ferrocenyldiphosphine the phosphine groups of which are either bonded directly or via a bridge group --CR.sub.v R.sub.w -- to the ortho positions of a cyclopentadienyl ring or are each bonded to a cyclopentadienyl ring of a ferrocenyl, so that a 5-, 6- or 7-membered ring is formed together with the Ir atom;R.sub.v and R.sub.
    Type: Grant
    Filed: January 26, 1998
    Date of Patent: November 16, 1999
    Assignee: Novartis Crop Protection, Inc.
    Inventors: Rafael Sablong, John Anthony Osborn, Felix Spindler
  • Patent number: 5985921
    Abstract: Compounds of the formula ##STR1## in which n, q, A, X, G, Y, Z, R, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.7 and R.sub.9 are as defined in claim 1, and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers thereof, in each case in the free form or in an agrochemically suitable salt form, can be used as agrochemical active compounds and can be prepared in a manner known per se.
    Type: Grant
    Filed: December 6, 1996
    Date of Patent: November 16, 1999
    Assignee: Novartis Corporation
    Inventors: Saleem Farooq, Stephen Trah, Hugo Ziegler, Rene Zurfluh, Alfons Pascual, Henry Szczepanski, Roger Graham Hall
  • Patent number: 5981432
    Abstract: Herbicidal compositions comprising S-metolachlor and at least one additional herbicide selected from atrazine, terbuthylazine, flumetsulan, pendimethalin, metosulam, pyridate, glyphosate, glufosinate, cyanazine, dicamba, halosulfuron, prosulfuron, primisulfuron, sulcotrione, metribuzin, BAY FOE 5043, and salts thereof. The compositions may also contain the safener benoxacor.
    Type: Grant
    Filed: February 2, 1998
    Date of Patent: November 9, 1999
    Assignee: Novartis Crop Protection
    Inventors: Manfred Hudetz, Dan Worden Kidder, Robert Franklin Milliken, Norbert Nelgen
  • Patent number: 5965486
    Abstract: The invention relates to a herbicidal composition, comprising a compound of formula I ##STR1## and a compound of formula II ##STR2## and/or of formula III ##STR3## or an agriculturally acceptable salt of the compound of formula II and/or III in admixture.
    Type: Grant
    Filed: October 15, 1998
    Date of Patent: October 12, 1999
    Assignee: Novartis Crop Protection, Inc.
    Inventor: Willy Ruegg
  • Patent number: 5962371
    Abstract: A herbicidal composition comprising at least one compound of formula I ##STR1## R.sub.2 is methyl, methoxy or --OCHF.sub.2, R.sub.3 is methyl or --OCHF.sub.2 andE is .dbd.C-- or .dbd.N--, with E being .dbd.N-- when R.sub.2 is methoxy,or an agrochemically acceptable salt of at least one of the compounds of formula I, and a compound of formula II ##STR2## or an agrochemically acceptable salt of the compound of formula II and/or III, in admixture with one another.
    Type: Grant
    Filed: December 12, 1997
    Date of Patent: October 5, 1999
    Assignee: Novartis Crop Protection, Inc.
    Inventors: Manfred Hudetz, Karl Gutbrod
  • Patent number: D419076
    Type: Grant
    Filed: November 10, 1998
    Date of Patent: January 18, 2000
    Assignee: Novartis Crop Protection
    Inventor: Lawrence Clifford Dull