Abstract: A series of substituted amino ethyl meta benzoic acid amides and their salts are useful as spasmolytics, pschyotherapeutic agents and agents facilitating learning. These compounds may conveniently be prepared by hydrolysis of suitably substituted trifluoromethyl derivatives followed by amidification with a desired amine, or by a replacement reaction between a suitable ester and an appropriate amine, or by reaction of an activated form of the free acid and an appropriate amine.

Abstract: N-alkylsulfonyl and N-haloalkylsulfonyl-substituted perfluoroalkanesulfonanilides and processes for their preparation are disclosed. These compounds and their compositions are useful as herbicides and plant growth modifiers.

Abstract: The new 1-alkyl-4-(10-oxo or -hydroxy-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ylidene)-piperidine compounds are prepared from the corresponding 10-desoxy compounds having a double bond at the 10,11-position by a process involving bromination, dehydrobomination of the resulting dibromo compound, followed by enamine formation and hydrolysis to give the desired 10-oxo compound. The compounds prepared in this manner are active as antihistamines and as appetite stimulants.

Abstract: [4-(DIPHENYLMETHOXY)-1-METHYLPIPERIDINIUM]-4-[1-HYDROXY-2-(1-METHYL-3-PHENY LPROPYLAMINO)-PROPYL]PHENOLATE AND A PROCESS FOR ITS PREPARATION ARE DESCRIBED.The phenolate possesses useful anti-inflammatory activity.

Abstract: New 1,2,3,4-tetra-hydrocarbazole derivatives of the formula: ##SPC1##Wherein R.sup.1 is straight-chained or branched alkyl, and the pharmacologically compatible salts thereof, are markedly effective as inhibitors of adrogenic .beta.-receptors and thus useful for the treatment and prophylaxis of cardiac and circulatory diseases.

Abstract: Novel 3-aminocarbazole compounds of the formula: ##SPC1##WhereinX is hydrogen or halogen,Y is oxygen or represents two hydrogen atoms; andR.sub.1 and R.sub.2, which can be the same or different, are hydrogen, lower alkyl or hydroxyalkyl or amino; andn is 1 or 2, with the proviso that when n is 2, X, Y, R.sub.1 and R.sub.2 cannot all be hydrogen atoms,As well as the salts thereof with inorganic and organic acids; are outstandingly effective indicators for the determination of glucose and provide stable compositions for such glucose determination.

Abstract: N-phenylcarbamoyl-4-methylpiperidine herbicides having the formula ##SPC1##Wherein R is a member selected from the group consisting of hydrogen and fluorine, compositions containing the same and the selective herbicidal method of use as a selective preemergence herbicide toward corn and a selective postemergence herbicide toward barley and, when R is H, toward corn.

Abstract: Substituted trifluoromethanesulfonanilides wherein the anilide ring is bonded to a phenyl ring through a linking group selected from --CH.sub.2 --, --CH.sub.2 CH.sub.2 --, --CH(CH.sub.3)-- and ##EQU1## and pharmaceutically acceptable salts thereof. These compounds are active anti-microbial agents.

Abstract: The present invention relates to novel thiazolidinone acetic acid derivatives and their preparation. These derivatives show diuretic properties when used as pharmaceuticals.

Abstract: Phenylpiperidines of the formula ##SPC1##Wherein R is alkyl of 4 to 7 carbon atoms are described. The foregoing phenylpiperidines are useful as non-addicting analgesics.

Abstract: Dialkyl 1,1'-(hydrocarbylenebiscarbamoyl)bis(2-benzimidazolecarbamate) as fungicides and mite ovicides.

Abstract: The new 1-alkyl-4-(10-oxo or -hydroxy-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-ylidene)piperidine compounds are prepared from the corresponding 10-desoxy compounds having a double bond at the 10,11-position by a process involving bromination, dehydrobromination of the resulting dibromo compound, followed by enamine formation and hydrolysis to give the desired 10-oxo compound. The compounds prepared in this manner are active as antihistamines and as appetite stimulants.

Abstract: N-methyl-N-alkoxycarbonylsulphenyl-carbamates of the formula ##EQU1## in which R.sup.1 is C.sub.1.sub.-6 alkyl, andR.sup.2 is phenyl; naphthyl; indanyl; phenyl, naphthyl or indanyl substituted by trihalomethyl, halogen, nitro, nitrile, dioxanyl, dioxolanyl, methyl-dioxanyl, methyl-dioxolanyl, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, dialkoxymethyl, alkenoxy, alkynoxy, alkylmercapto, alkenylmercapto, alkynylmercapto or dialkylamino, with up to 6 carbon atoms in each alkyl, alkenyl or alkynyl group; a radical of the formula ##EQU2## in which R.sup.3 and R.sup.4 are each alkyl, alkylthio, nitrile or phenyl; or ##EQU3## in which R.sup.5 is hydrogen or C.sub.1.sub.-6 alkyl, which possess insecticidal, acaricidal, fungicidal, nematocidal and bactericidal properties.

Abstract: Novel (3-thioxo-1,2-dithiol-4-yl)substituted triaylphosphates and thiophosphates are used as additives for lubricating oils. The are prepared by reacting corresponding phosphoryl chlorides with 4-(hydroxy-aryl)-1,2-dithiole-3-thiones.

Abstract: A method for producing tetra-N-alkyl derivatives of bicyclic ureas having the general formula: ##EQU1## wherein n is 0 or 1; R and R' is H, lower alkyls, which can be the same or different, characterized in that bicyclic ureas, unsubstituted at nitrogen atoms are alkylated with alkyl halides in liquid ammonia under the action of an alkali metal amide, followed by separation of the target product.Said tetra-N-alkyl derivatives of bicyclic ureas are pharmacologically active compounds. The most active representative of said compounds, 2,4,6,8 tetramethyl-2,4,6,8-tetraazabicyclo-3,3,O-octanedi-3,7-one, is the active principle of a medicinal preparation used for treating psychic disorders.

Abstract: Polyphenolic components of coniferous tree barks are reacted with a concentrated aqueous solution containing ammonia and sulfur dioxide to produce aminated sulfite reaction products having high nitrogen contents. The products have a number of valuable applications including utility in the agricultural field. The reaction takes place at temperatures of 130.degree. - 190.degree.C., the ratio of NH.sub.3 /bark is within the range of 0.2 - 1.2 and ratio of SO.sub.2 /bark is within the range of 0.25 - 0.4, on a weight basis.

Abstract: .beta.-Ketoacyl derivatives of 6-aminopenicillanic acid of the formula: ##SPC1##Are disclosed. In the above structure R.sup.1 is hydrogen, alkyl, halogen, alkoxy, cyano, trifluoromethyl and the like; Z is CHR.sup.2 or NR.sup.2 ; R.sup.2 is hydrogen, alkyl, aralkyl; M is an alkali or alkaline earth metal such as sodium, potassium, or calcium. These compounds are useful as anti-bacterials.

Abstract: Phenyl-lower-alkylamines having anti-inflammatory activity are prepared either by reductive alkylation of an amine with a phenyl-lower-alkanaldehyde; by condensation of a phenyl-lower-alkanaldehyde with a secondary amine, conversion of the resulting phenylvinylamine to the corresponding iminium salt, and reduction of the latter with an alkali metal borohydride; or by reaction of a phenyl-lower-alkanoyl halide with an amine and reduction of the resulting amide with a reagent effective to reduce an amide to an amine.

Abstract: 1-(Substituted-aminoalkyl)-3-benzoyl-4-hydroxy-4-phenylpiperidines and related compounds having anti-arrhythmic activity are described herein. The 3-benzoyl compounds can be prepared by condensing the appropriate diamine with acetophenone and formaldehyde. The related 3-(.alpha.-hydroxybenzyl) compounds are prepared by reduction of the corresponding 3-benzoyl compounds.

Abstract: A process for preparing p-[5-chloro-2-methoxy-benzamidoethyl]-benzene sulfonamide consisting of treating 5-chlorosalicylic acid or its ester by methylating and aminolysis to form N-phenethyl-5-chloro-2-methoxybenzamide followed by chlorosulfonation and aminolysis.