Patents by Inventor Klaus Jelich

Klaus Jelich has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • Patent number: 4990622
    Abstract: A process for the preparation of 2-chloro-5-chloromethylpyridine of the formula (I) ##STR1## which is used as an intermediate for the preparation of insecticides, the process comprising (a) reacting in a first step nicotinic acid of the formula (II) ##STR2## with phosphorus pentachloride, if appropriate in the presence of thionyl chloride and if appropriate in the presence of a diluent, (b) reacting in a second step the resulting 3-trichloromethylpyridine from the first step, of the formula III, ##STR3## with an alkali metal alkoxide of the formual (IV)R--O--M (IV)in whichR represents alkyl andM represents an alkali metal cation,if appropriate in the presence of a diluent, (c) reacting in a third step the resulting pyridine ether acetal from the second step, of the formula (V), ##STR4## in which R has the abovementioned meaning with water, if appropriate in the presence of a catalyst acid, (d) hydrogenating in a fourth step the resulting pyridine aldehyde from the third step, of the formula (VI), ##STR5## in
    Type: Grant
    Filed: December 6, 1989
    Date of Patent: February 5, 1991
    Assignee: Bayer Aktiengesellschaft
    Inventor: Klaus Jelich
  • Patent number: 4988718
    Abstract: Fungicidal substituted 4-heterocyclyloximinopyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another in each case represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case unsubstituted or in each case substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an unsubstituted or substituted heterocycle.
    Type: Grant
    Filed: August 9, 1990
    Date of Patent: January 29, 1991
    Assignee: Bayer Aktiengesellschaft
    Inventors: Kurt Findeisen, Klaus Jelich, Gerd Hanssler
  • Patent number: 4981507
    Abstract: Herbicidal triazoloazines of the formula ##STR1## in which A stands for nitrogen or for a radical C--R.sup.3,R.sup.1, R.sup.2 and R.sup.3 independently of one another each stand for hydrogen, hydroxyl, halogen, for optionally substituted alkyl, for alkoxy, alkylthio or for optionally substituted aryl, or eitherR.sup.1 and R.sup.3 together or R.sup.3 and R.sup.2 together stand for a fused, optionally substituted carbocyclic or heterocyclic ring,X stands for oxygen, sulphur, a sulphinyl group, or a sulphonyl group andAr stands for in each case optionally substituted aryl or heteroaryl.
    Type: Grant
    Filed: April 5, 1989
    Date of Patent: January 1, 1991
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Hans-Joachim Santel, Robert R. Schmidt, Harry Strang
  • Patent number: 4968687
    Abstract: Fungicidal substituted 4-heterocyclyloximinopyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another in each case represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case unsubstituted or in each case substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an unsubstituted or substituted heterocycle.
    Type: Grant
    Filed: September 5, 1989
    Date of Patent: November 6, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventors: Kurt Findeisen, Klaus Jelich, Gerd Hanssler
  • Patent number: 4960455
    Abstract: Herbicidal triazolodihydropyrimidine-2-sulphonamides of the formula ##STR1## in which R.sup.1, R.sup.2 and R.sup.3 independently of one another each stand for hydrogen or for optionally substituted alkyl andR.sup.4 stands for in each case optionally substituted aryl or heteroaryl.
    Type: Grant
    Filed: March 7, 1989
    Date of Patent: October 2, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Peter Babczinski, Hans-Joachim Santel, Robert R. Schmidt, Harry Strang
  • Patent number: 4958025
    Abstract: A process for the preparation of 2-chloro-5-chloromethyl-pyridine of the formula ##STR1## which comprises reacting nicotinic acid of the formula ##STR2## with phosphorus pentachloride to produce 3-trichloromethylpyridine of the formula ##STR3## reacting the 3-trichloromethylpyridine in a 2nd step with an alkali metal alkoxide of the formulaR-O-M (IV)in whichR represents alkyl andM represaents an alkali metal cation, to produce a pyridine ether acetal of the formula ##STR4## reacting the pyridine ether acetal in a 3rd step with dilute aqueous acid to produce pyridone aldehyde of the formula ##STR5## hydrogenating the pyridone aldehyde in a 4th step with molecular hydrogen in the presence of a hydrogenation catalyst to produce the pyridylmethanol compound of the formula ##STR6## and reducing the pyridylmethanol compound in a 5th step with a chlorinating agent.
    Type: Grant
    Filed: December 4, 1989
    Date of Patent: September 18, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventor: Klaus Jelich
  • Patent number: 4929738
    Abstract: Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radial.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also new.
    Type: Grant
    Filed: May 10, 1989
    Date of Patent: May 29, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Wilhelm Brandes, Gerd Hanssler, Paul Reinecke
  • Patent number: 4921993
    Abstract: Fungicidally active substituted benzamides of the formula ##STR1## in which R.sup.1 represents alkoxy, alkenyloxy, alkinyloxy or a heterocyclyl radical,R.sup.2 represents cyano, a carbamoyl radical or a thiocarbamoyl radical,X represents an alkanoyl radical or an alkoximinoalkyl radical, andn represents a number 1, 2 or 3.Intermediates wherein R' is replaced by bromine and R.sup.2 is cyano or a carbamoyl radical are also new.
    Type: Grant
    Filed: November 23, 1987
    Date of Patent: May 1, 1990
    Assignee: Bayer Aktiengesellschaft
    Inventors: Herbert Gayer, Klaus Jelich, Wolfgang Kramer, Wilhelm Brandes
  • Patent number: 4886833
    Abstract: Novel fungicides of the formula ##STR1## in which R.sup.1 represents optionally substituted hydroxyalkyl, optionally substituted hydroxyalkoxyalkyl, optionally substituted heteroarylalkyl or optionally substituted heteroaryl, andR.sup.2 represents optionally substituted alkyl, optionally substituted alkenyl, or alkinyl.Intermediate therefor, wherein R.sup.2 is hydrogen or an alkali metal cation, are also new.
    Type: Grant
    Filed: August 24, 1987
    Date of Patent: December 12, 1989
    Assignee: Bayer Aktiengesellschaft
    Inventors: Herbert Gayer, Klaus Jelich, Winfried Lunkenheimer, Wilhelm Brandes, Gerd Hanssler
  • Patent number: 4874424
    Abstract: A method of combating unwanted vegetation which comprises applying to such vegetation or to a locus from which it is desired to exclude such vegetation a herbicidally effective amount of an alkoximinoalkylamide of the formula ##STR1## in which R represents hydrogen or alkyl,R.sup.1 represents hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy, halogenoalkylthio, phenyl, phenoxy, formyl, alkoxycarbonyl, alkanoyl or alkoximinoalkyl andR.sup.2 represents halogen, cyano, nitro, alkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy, halogenoalkylthio, phenyl phenoxy, formyl, alkoxycarbonyl, alkanoyl or alkoximinoalkyl.
    Type: Grant
    Filed: April 27, 1988
    Date of Patent: October 17, 1989
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Herbert Gayer, Wolfgang Kramer, Hans-Joachim Santel, Robert R. Schmidt, Harry Strang
  • Patent number: 4864029
    Abstract: Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkyllaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radical.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also new.
    Type: Grant
    Filed: May 11, 1988
    Date of Patent: September 5, 1989
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Wilhelm Brandes, Gerd Hanssler, Paul Reinecke
  • Patent number: 4854964
    Abstract: Novel herbicides of the formula ##STR1## in which R.sup.1 represents alkyl,R.sup.2 represents hydrogen, alkyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, alkenyl, alkinyl or optionally substituted aralkyl, andR.sup.3 represents optionally substituted aryl.Intermediates of the formula ##STR2## in which R.sup.6 is hydrogen, chlorine or hydroxyl,are also new.
    Type: Grant
    Filed: July 30, 1987
    Date of Patent: August 8, 1989
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Hans-Joachim Santel, Robert R. Schmidt, Harry Strang
  • Patent number: 4841086
    Abstract: A process for the preparation of a 2-cyano-2-oximino-acetamide derivative of the formula ##STR1## in which R.sup.I is alkyl or other organic radical,R.sup.II is hydrogen or alkyl,R.sup.III is hydrogen, alkyl or other organic radical which comprises reacting a 2-cyano-2-oximino-acetamide of the formula ##STR2## with a base B at a temperature between 0.degree. C. and 100.degree. C., to produce a salt of the formula ##STR3## in which B represents one equivalent of an organic of inorganic base,and reacting such salt with an alkylating agent of the formula ##STR4## in which X is halogen, methane- or p-toluenesulphonate or methyl sulphate, at a temperature between 0.degree. C. and 150.degree. C.
    Type: Grant
    Filed: January 20, 1988
    Date of Patent: June 20, 1989
    Assignee: Bayer Aktiengesellschaft
    Inventors: Herbert Gayer, Klaus Jelich
  • Patent number: 4767775
    Abstract: Microbicidal substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represent in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl andHet represents an optionally substituted heterocyclic radical.Intermediates therefor of the formula ##STR2## in which R is alkyl, are also disclosed.
    Type: Grant
    Filed: July 24, 1986
    Date of Patent: August 30, 1988
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Wilhelm Brandes, Gerd Hanssler, Paul Reinecke
  • Patent number: 4743615
    Abstract: Fungicidally active substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 and R.sup.2 independently of one another each represents hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkoxycarbonyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or represents in each case optionally substituted oxiranylalkyl, aralkyl, heterocyclyl or aryl, andR.sup.3 represents halogenoalkyl, halogenoalkenyl or halogenoalkinyl, or represents substituted cycloalkyl, or represents substituted cycloalkylalkyl.
    Type: Grant
    Filed: October 31, 1986
    Date of Patent: May 10, 1988
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Wilhelm Brandes, Gerd Hanssler, Paul Reinecke
  • Patent number: 4666933
    Abstract: Fungicidally active substituted pyrazolin-5-ones of the formula ##STR1## in which R.sup.1 is hydrogen or alkyl,R.sup.2 is hydrogen, alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, hydroxycarbonylalkyl or alkoxycarbonylalkyl, aminocarbonylalkyl, alkylaminocarbonylalkyl or dialkylaminocarbonylalkyl, or in each case optionally substituted oxiranylmethyl, aralkyl or aryl, andR.sup.3 is alkyl, alkenyl, alkinyl, cyanoalkyl, hydroxyalkyl, alkoxyalkyl, hydroxycarbonylalkyl, alkoxycarbonylalkyl, cycloalkyl or cycloalkylalkyl, or in each case optionally substituted aralkyl, aryloxyalkyl or arylthioalkyl, but wherein R.sup.3 is methyl or ethyl only if R.sup.1 and/or R.sup.2 is not hydrogen or methyl.
    Type: Grant
    Filed: June 17, 1986
    Date of Patent: May 19, 1987
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus Jelich, Wolfgang Kramer, Wilhelm Brandes, Gerd Hanssler, Paul Reinecke