Patents by Inventor Mauro GABOARDI

Mauro GABOARDI has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • PROCESS FOR THE PREPARATION OF ERLOTINIB
    Publication number: 20160115137
    Abstract: A process for the preparation of Erlotinib is disclosed in which the compound of formula (II) Is reacted with the compound of formula (III) and the reaction product is subsequently treated with a source of hydrochloric acid in a suitable solvent to give Erlotinib hydrochloride.
    Type: Application
    Filed: October 27, 2015
    Publication date: April 28, 2016
    Inventors: Marco BARATELLA, Giuseppe PALLANZA, Mauro GABOARDI, Graziano CASTALDI
  • INTERMEDIATES USEFUL FOR THE PREPARATION OF SAXAGLIPTIN
    Publication number: 20160107992
    Abstract: Intermediates useful for the synthesis of saxagliptin and their preparationare described.
    Type: Application
    Filed: June 18, 2014
    Publication date: April 21, 2016
    Inventors: Graziano CASTALDI, Giuseppe PALLANZA, Mauro GABOARDI, Marta CASTALDI
  • PROCESS AND INTERMEDIATES FOR THE PREPARATION OF DASATINIB
    Publication number: 20150259337
    Abstract: The present invention relates to a process for the synthesis of dasatinib and to intermediates useful for its preparation.
    Type: Application
    Filed: February 26, 2015
    Publication date: September 17, 2015
    Inventors: Alessandro BARUTO, Mauro GABOARDI, Marta CASTALDI, Graziano CASTALDI
  • Process and intermediates for the preparation of dasatinib
    Patent number: 9115124
    Abstract: The present invention relates to a process for the synthesis of dasatinib and to intermediates useful for its preparation.
    Type: Grant
    Filed: February 26, 2015
    Date of Patent: August 25, 2015
    Assignee: CERBIOS-PHARMA SA
    Inventors: Alessandro Baruto, Mauro Gaboardi, Marta Castaldi, Graziano Castaldi
  • INTERMEDIATES USEFUL FOR THE SYNTHESIS OF FEXOFENADINE, PROCESSES FOR THEIR PREPARATION AND FOR THE PREPARATION OF FEXOFENADINE
    Publication number: 20130237709
    Abstract: Intermediates useful for the synthesis of fexofenadine, processes for their preparation and processes for the synthesis of fexofenadine are described.
    Type: Application
    Filed: February 21, 2013
    Publication date: September 12, 2013
    Applicant: CHEMELECTIVA S.r.l.
    Inventors: Graziano CASTALDI, Marco BARATELLA, Mauro GABOARDI
  • PROCESS FOR THE PREPARATION OF CROSS-LINKED POLYALLYLAMINES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF
    Publication number: 20120196988
    Abstract: The present invention relates to a process for the preparation of cross-linked polyallylamines or pharmaceutically acceptable salts thereof. The invention further relates to a process for the preparation of Sevelamer or pharmaceutically acceptable salts thereof, preferably hydrochloride or carbonate salts, used in the treatment of hyperphosphatemia, and having good flowability, low porosity and/or a swelling index of between 7 and 9.
    Type: Application
    Filed: January 31, 2012
    Publication date: August 2, 2012
    Applicant: CHEMI SPA
    Inventors: Mauro GABOARDI, Erminio OLDANI