Hetero Ring Is Five-membered Having Two Or More Ring Hetero Atoms Of Which At Least One Is Nitrogen Patents (Class 504/261)
  • Publication number: 20100113276
    Abstract: The use of N2-phenylamidines of formula (I) as herbicides is described. In this formula (I), R2, R3, R4, R5 and R6 are different radicals and A is a bond or various 1- or polyatomic bridging elements.
    Type: Application
    Filed: March 4, 2008
    Publication date: May 6, 2010
    Applicant: BAYER CROPSCIENCE AG
    Inventors: Birgit Kuhn, Harald Jakobi, Thomas Mueller, Joerg Tiebes, Heinz Kehne, Dirk Schmutzler, Martin Hills, Christopher Rosinger, Klaus Kunz, Mark Wilheim Drewes, Dieter Feucht, Thomas Seitz, Benoit Hartmann, Ralf Dunkel, Joerg Nico Greul, Oliver Guth, Kerstein Ilg, Darren James Mansfeld, Wahed Ahmed Moradi, Peter Dahmen, Ulrike Wachendorf-Neumann, Arnd Voerste, Dale Robert Mitchell, Jean-Pierre Andre Vors, Dale Robert Mitchell, Tom Hough
  • Patent number: 7655600
    Abstract: The present invention relates to 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the general formula (I) wherein A is a radical of the formulae A? or A2: NRA?A2 and wherein m is 0, 1, 2, 3, 4 or 5, n is 0, 1, 2, 3, 4 or 5, X is sulfur or oxygen, and wherein the variables R1, R2, R3, R4, R5a, R5b, R5c, R5d are as defined in the claims, and to the agriculturally acceptable salts thereof. The invention relates also to a method of combating animal pests, selected from insects, arachnids and nematodes and to a method for protecting crops from attack or infestation by insects, arachnids or nematodes, which comprises contacting a crop with a pesticidally effective amount of a 1-(azolin-2-yl)amino-1,2-diphenylethane compounds of the general formula I and/or at least one salt thereof.
    Type: Grant
    Filed: December 22, 2004
    Date of Patent: February 2, 2010
    Assignee: BASF Aktiengesellschaft
    Inventors: Markus Kordes, Michael Hofmann, Michael Puhl, Norbert Götz, Michael Rack, Ernst Baumann, Wolfgang von Deyn, Thomas Schmidt, Livio Tedeschi, Michael F. Treacy, Deborah L. Culbertson, Toni Bucci, David G. Kuhn
  • Publication number: 20100009853
    Abstract: Parasitic plants parasitizing on crops can be controlled effectively, by providing an agent for controlling parasitic plants, which comprises tiadinil or the like as the active ingredient and a method for using an agent for controlling parasitic plants, which comprises treating a parasitized plant or soil with an effective amount of agent for controlling parasitic plants. As a result, the yield of crops can be recovered to the level of parasitism-free crops. Additionally, by inhibiting parasitism of parasitic plants strongly, development of the next generation can be inhibited so that the level of pollution with parasitic plants on agricultural land can be lowered with cultivating sensitive crops.
    Type: Application
    Filed: July 13, 2007
    Publication date: January 14, 2010
    Applicant: Nihon Nohyaku Co., Ltd
    Inventors: Osamu Ikeda, Ken Kuriyama, Miyako Aoki, Masao Yamashita
  • Patent number: 7598395
    Abstract: The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R8, R9 and R10; X is a single or double bond; Y is O, S, N(R11) or (CR12R13)(CR14R15)m(CR16R17)n; m is 0 or 1; n is 0 or 1; and R1 to R17 each, independently, have a range of values; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
    Type: Grant
    Filed: October 14, 2003
    Date of Patent: October 6, 2009
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Josef Ehrenfreund, Hans Tobler, Harald Walter
  • Patent number: 7582589
    Abstract: The invention also relates to novel compounds of formula (1) where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to three groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(?O), optionally substituted (C1-4)alkylC(?O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is either at position 2 or at position 4 of the thiophene ring and is an organic group containing three to thirteen carbon atoms and at least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to fou
    Type: Grant
    Filed: April 21, 2004
    Date of Patent: September 1, 2009
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Josef Ehrenfreund, Harald Walter, Hans Tobler, Clemens Lamberth
  • Patent number: 7572753
    Abstract: The use of certain tetrazole compounds as fungicides is disclosed wherein said compounds are of the structural formula: wherein: R is selected from the group consisting of phenyl groups of the structural formula: and thienyl groups of the structural formula: and X and Y are each selected from the group consisting of hydrogen, haloalkyl, halogen, and nitro. Novel compounds wherein X is selected from the group consisting of haloalkyl, halogen, and nitro and Y is selected from the group consisting of hydrogen, haloalkyl, halogen, and nitro are also disclosed.
    Type: Grant
    Filed: September 15, 2005
    Date of Patent: August 11, 2009
    Assignee: Chemtura Corporation
    Inventors: Mark A. Dekeyser, Ahmad Ghavami, Robert G. Davis, Sheldon B. Park, Steven J. Hobbs, Clifford Pratt, Gaik-Lean Chee, Daniel Walther
  • Patent number: 7566683
    Abstract: Ethylene derivatives of formula (I): where Q is an unsubstituted or substituted phenyl or heterocyclic group, especially a 4-thiazolyl, 1- or 3-pyrazolyl, 1,3-oxazol-4-yl, phenyl or pyridyl group; E is a substituent such as a cyano group; A is a substituent such as a 4-pyrazolyl or thiazolyl group; and B is a substituent such as an alkylcarbonyl group. Agricultural chemicals and agents for preventing the attachment of aquatic organisms containing one or more such ethylene derivatives.
    Type: Grant
    Filed: August 15, 2005
    Date of Patent: July 28, 2009
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Tomoyuki Ogura, Hiroshi Murakami, Akira Numata, Rika Miyachi, Toshiro Miyake, Norihiko Mimori, Shinji Takii
  • Publication number: 20080276329
    Abstract: A rice cultivar designated CL171-AR is disclosed. The invention relates to the seeds of rice cultivar CL171-AR, to the plants of rice CL171-AR, to methods for producing a rice plant produced by crossing the cultivar CL171-AR with itself or another rice variety, and to methods for controlling weeds in the vicinity of plants of rice cultivar CL171-AR, which comprises increased resistance to acetohydroxyacid synthase-inhibiting herbicides. The invention further relates to hybrid rice seeds and plants produced by crossing the cultivar CL171-AR with another rice cultivar.
    Type: Application
    Filed: May 2, 2007
    Publication date: November 6, 2008
    Inventor: Karen A.K. Moldenhauer
  • Publication number: 20080234130
    Abstract: Methods and compositions are provided related to improved plants that are tolerant to more than one herbicide. Particularly, the invention provides plants that are tolerant of glyphosate and are tolerant to at least one ALS inhibitor, and methods of use thereof. The glyphosate/ALS inhibitor-tolerant plants comprise a polynucleotide that encodes a polypeptide that confers tolerance to glyphosate and a polynucleotide that encodes an ALS inhibitor-tolerant polypeptide. In specific embodiments, a plant of the invention expresses a GAT polypeptide and an HRA polypeptide. Methods to control weeds, improve plant yield, and increase transformation efficiencies are provided.
    Type: Application
    Filed: August 22, 2006
    Publication date: September 25, 2008
    Applicants: Pioneer Hi-Bred International, Inc., E.I. du Pont de Nemours and Company
    Inventors: Billy Fred McCutchen, Linda A. Castle, Timothy K. Chicoine, Hyeon-Je Cho, Jon S. Claus, Jerry M. Green, Anthony D. Guida, Christine B. Hazel, Matthew J. Heckert, Jeffrey M. Hegstad, James M. Hutchison, Donglong Liu, Albert L. Lu, Wayne J. Mehre, York Moy, Paul D. Olson, Kenneth A. Peeples, David W. Saunders, Mark D. Vogt, Jack Q. Wilkinson, James F. H. Wong
  • Publication number: 20080176746
    Abstract: The present invention relates to an oil suspension concentrate comprising microencapsulated agrochemically active compounds. The inventive oil suspension concentrate advantageously comprises (a) one or more agrochemically active compounds in the aqueous phase, which is present in encapsulated form in the oil phase, and (b) one or more agrochemically active compounds in the oil phase, and also if desired, any customary auxiliaries and/or additives.
    Type: Application
    Filed: January 22, 2008
    Publication date: July 24, 2008
    Applicant: Bayer CropScience AG
    Inventors: Ralph GROHS, Roland Deckwer, Frank Rosenfeldt
  • Patent number: 7358214
    Abstract: This invention relates to novel pyrazolylcarboxanilides of the formula (I) in which R1, G and n are as defined in the disclosure, to a plurality of processes for preparing these substances, to their use for controlling unwanted microorganisms, and to novel intermediates and their preparation.
    Type: Grant
    Filed: January 19, 2004
    Date of Patent: April 15, 2008
    Assignee: Bayer CropScience AG
    Inventors: Ralf Dunkel, Hans-Ludwig Elbe, Heiko Rieck, Peter Dahmen, Ulrike Wachendorff-Neumann, Karl-Heinz Kuck
  • Patent number: 7323433
    Abstract: The invention relates to R-(?)-1-[2-(7-Chloro-benzo[b]thiophen-3-yl-methoxy)-2-(2,4-dichloro-phenyl)-ethyl]-1H-imidazole and the salts thereof. The invention also relates to compositions thereof and their use either for treating fungal infections in humans and animals or combating crop diseases. A process for their preparation is also described.
    Type: Grant
    Filed: August 5, 2004
    Date of Patent: January 29, 2008
    Assignee: Ferrer Internacional, S.A.
    Inventors: Rafael Foguet, Jorge Ramentol, Lluis Anglada, Celia Palacin, Antonio Guglietta
  • Patent number: 7250436
    Abstract: The invention relates to compounds of the general formula wherein Ar1, Ar2, R4, R5, R6, R7, R8, W, X, a and b have the significances given in the specification, and optionally the enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are especially suitable for controlling parasites on warm-blooded animals.
    Type: Grant
    Filed: June 6, 2003
    Date of Patent: July 31, 2007
    Assignee: Novartis Animal Health US, Inc.
    Inventors: Pierre Ducray, Thomas Goebel, Jorg Fruchtel
  • Patent number: 7192906
    Abstract: Substituted pyrazole compounds of the formula (1). The compounds are synthesized from a pyrazole derivative and a haloalkyleneoxime ester derivative, and have excellent herbicidal effects.
    Type: Grant
    Filed: December 18, 2002
    Date of Patent: March 20, 2007
    Assignee: SDS Biotech K.K.
    Inventors: Yoji Hirohara, Eiji Ikuta, Sayo Osanai, Hideki Nakashima, Teruhiko Ishii
  • Patent number: 7176164
    Abstract: A process for preparing novel 1,3-selanazolin derivatives represented by chemical formula 1 at high yield.
    Type: Grant
    Filed: December 13, 2002
    Date of Patent: February 13, 2007
    Assignee: Gifu University
    Inventors: Mamoru Koketsu, Hideharu Ishihara
  • Patent number: 7112553
    Abstract: A compound of formula (I) wherein G is either (i) or (ii), where M1 or M2 is bonded to A; n is 0 or 1; when G is (i), D is S, NR7, CR8?CR9, CR8?N, CR8?N(O), N?CR9 or N(O)?CR9; when G is (ii), D is S or NR7; E is N, N-oxide or CR10; M1 is OC(?Y), N(R11)C(?Y), N?C(OR12), N?C(SR13) or N?C(NR14R15) where O or N is the atom of attachment to the ring containing D and E; M2 is N—C(?Y) where N is the atom of attachment to the ring containing D and E; Y is O, S or NR16; J is N or CR17; and A, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11, R12, R13, R14 and R15 are each certain organic or inorganic groups. These compounds are useful in fungicidal, insecticidal, acaricidal, molluscicidal and hematicidal compositions.
    Type: Grant
    Filed: April 4, 2000
    Date of Patent: September 26, 2006
    Assignee: Syngenta Limited
    Inventors: Sarah Armstrong, Nigel John Barnes, Susan Patricia Barnett, Eric Daniel Clarke, Patrick Jelf Crowley, Torquil Eoghan Macleod Fraser, David John Hughes, Christopher John Mathews, Joan Pilkington, legal representative, Roger Salmon, Stephen Christopher Smith, Russell Viner, William Guy Whittingham, John Williams, Alan John Whittle, Brian Leslie Pilkington, deceased
  • Patent number: 7105471
    Abstract: The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, Z represents hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups ?in which A, B, D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides.
    Type: Grant
    Filed: February 12, 2004
    Date of Patent: September 12, 2006
    Assignee: Bayer Aktiengesellschaft
    Inventors: Folker Lieb, Reiner Fischer, Alan Graff, Udo Schneider, Thomas Bretschneider, Christoph Erdelen, Wolfram Andersch, Mark-Wilhelm Drewes, Markus Dollinger, Ingo Wetcholowsky, Randy Allen Myers
  • Patent number: 6911416
    Abstract: The present invention relates to new substituted N-benzoyl-N?-(tetrazolylphenyl)-ureas of the formula (I) in which R1, R2, R3, R4 and n are as stated in the description, to processes for their preparation, and to their use as pesticides.
    Type: Grant
    Filed: May 2, 2001
    Date of Patent: June 28, 2005
    Assignee: Bayer Aktiengesellschaft
    Inventors: Fritz Maurer, Christoph Erdelen
  • Publication number: 20040242895
    Abstract: The invention relates to novel tetrazolinone derivatives of general formula (I) wherein R1 represents halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, C1-4 alkylthio, C1-4 alkylsulfonyl, C1-4 alkylsulfonyloxy, C2-5 alkoxycarbonyl, C2-6 alkoxyalkyl, C2-6 alkylthioalkyl, nitro or cyano, R2 represents a hydrogen atom, C1-6 alkyl, C3-6 cycloalkyl which may be optionally substituted with halogen or C1-3 alkyl, C1-4 haloalkyl, or phenyl which may be optionally substituted with halogen, C1-3 alkyl, C1-3 haloalkyl or nitro, m represents 0, 1 or 2, n represents 0 or 1, Q represents one of the groups which are mentioned in the description. The invention further relates to their use as herbicides and a process together with the intermediates for their preparation.
    Type: Application
    Filed: June 21, 2004
    Publication date: December 2, 2004
    Inventors: Akihiko Yanagi, Shinichi Narabu, Toshio Goto, Seishi Ito, Chieko Ueno
  • Patent number: 6790810
    Abstract: The invention relates to novel tetrazolinone derivatives of general formula (I) wherein R1 represents halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy, C1-4 alkylthio, C1-4 alkylsulfonyl, C1-4 alkylsulfonyloxy, C2-5 alkoxycarbonyl, C2-6 alkoxyalkyl, C2-6 alkylthioalkyl, nitro or cyano, R2 represents a hydrogen atom, C1-6 alkyl, C3-6 cycloalkyl which may be optionally substituted with halogen, or C1-3 alkyl, C1-4 haloalkyl or phenyl which may be optionally substituted with halogen, or C1-3 aklyl, C1-4 haloalkyl or nitro, m represents 0, 1 or 2, n represents 0 or 1, Q represents one of the groups which are mentioned in the description. The invention further relates to their use as herbicides and a process together with the intermediates for their preparation.
    Type: Grant
    Filed: June 30, 2003
    Date of Patent: September 14, 2004
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Akihiko Yanagi, Shinichi Narabu, Toshio Goto, Seishi Ito, Chieko Ueno
  • Patent number: 6770599
    Abstract: The instant invention relates to novel tetrazole derivatives of the formula (I) wherein R1 represents halogen, methyl, ethyl, halomethyl, methoxy, ethoxy, C1-2 haloalkoxy, methylthio, ethylthio, C1-3 alkylsulfonyl, methylsulfonyloxy, ethylsulfonyloxy, nitro or cyano, R2 represents C1-6 alkyl, C3-6 cycloalkyl which may be optionally substituted with halogen or C1-3 alkyl, C1-4 haloalkyl, C2-6 alkenyl, or phenyl which may be optionally substituted with halogen, C1-3 alkyl, C1-4 haloalkyl, C2-6 alkenyl, or phenyl which may be optionally substituted with halogen, C1-3 alkyl, C1-2 haloalkyl or nitro, m represents 0, 1 or 2, two R1 s may be identical or different, in case m represents 2, n represents 1 or 2, Q represents one the cyclic groups which are mentioned in the specification, to intermediates and several processes for their preparation, to their use as herbicides and to novel compositions containing them.
    Type: Grant
    Filed: February 20, 2003
    Date of Patent: August 3, 2004
    Assignee: Bayer CropScience KK
    Inventors: Akihiko Yanagi, Shinichi Narabu, Toshio Goto, Chieko Ueno, Shinichi Shirakura
  • Patent number: 6746989
    Abstract: The invention relates to novel substituted benzoylpyrazoles of the general formula (I), in which n represents the numbers 0, 1, 2 or 3, A represents a single bond or represents alkanediyl(alkylene), R1 represents in each case optionally substituted alkyl, alkenyl, alkinyl or cycloalkyl, R2 represents hydrogen, cyano, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkoxycarbonyl or cycloalkyl, R3 represents hydrogen, nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, dialkylamino or dialkylaminosulfonyl, R4 represents nitro, cyano, carboxyl, carbamoyl, thiocarbamoyl, halogen, or represents in each case optionally substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, dialkylamino or dialkylaminosulfonyl, Y represents hydrogen or represents in each case optionally substituted
    Type: Grant
    Filed: September 26, 2001
    Date of Patent: June 8, 2004
    Assignee: Bayer Aktiengesellschaft
    Inventors: Klaus-Helmut Müller, Stefan Lehr, Otto Schallner, Hans-Georg Schwarz, Heinz-Jürgen Wroblowsky, Mark Wilhelm Drewes, Dieter Feucht, Rolf Pontzen, Ingo Wetcholowsky
  • Publication number: 20040077500
    Abstract: A pest control agent composition having a synergistic effect which contains as the active ingredients one or more compounds selected among phthalamide derivatives represented by the general formula (I), which are useful as an insecticide or acaricide, and one or more compounds selected among compounds having insecticidal activity, acaricidal activity, or nematicidal activity. (I) In the formula (I), R1, R2, and R3 may be the same or different and each represents hydrogen, C3-6 cycloalkyl, -A1-Qp, etc.; X and Y may be the same or different and each represents hydrogen, halogeno, etc.; n is an integer of 1 to 4; m is an integer of 1 to 5; and Z1 and Z2 each represents oxygen or sulfur.
    Type: Application
    Filed: October 16, 2003
    Publication date: April 22, 2004
    Inventors: Kazuyuki Sakata, Masayuki Morimoto, Hiroshi Kodama, Tetsuyosi Nishimatsu
  • Patent number: 6660690
    Abstract: A method of preventing damage to the seed and/or shoots and foliage of a plant by a pest includes treating the seed from which the plant grows with a composition that includes a combination of at least one pyrethrin or synthetic pyrethroid and at least one other insecticide selected from the group consisting of an oxadiazine derivative, a chloronicotinyl, a nitroguanidine, a pyrrol, a pyrazone, a diacylhydrazine, a triazole, a biological/fermentation product, a phenyl pyrazole, an organophosphate and a carbamate. It is preferred that when the other insecticide is an oxadiazine derivative, the pyrethroid is selected from the group consisting of taufluvalinate, flumethrin, trans-cyfluthrin, kadethrin, bioresmethrin, tetramethrin, phenothrin, empenthrin, cyphenothrin, prallethrin, imiprothrin, allethrin and bioallethrin. The treatment is applied to the unsown seed.
    Type: Grant
    Filed: October 1, 2001
    Date of Patent: December 9, 2003
    Assignee: Monsanto Technology, L.L.C.
    Inventors: Jawed Asrar, Frank C. Kohn
  • Publication number: 20030224943
    Abstract: The instant invention relates to novel tetrazole derivatives of the formula (I) wherein R1 represents halogen, methyl, ethyl, halomethyl, methoxy, ethoxy, C1-2 haloalkoxy, methylthio, ethylthio, C1-3 alkylsulfonyl, methylsulfonyloxy, ethylsulfonyloxy, nitro or cyano, R2 represents C1-6 alkyl, C3-6 cycloalkyl which may be optionally substituted with halogen or C1-3 alkyl, C1-4 haloalkyl, C2-6 alkenyl, or phenyl which may be optionally substituted with halogen, C1-3 alkyl, C1-4 haloalkyl, C2-6 alkenyl, or phenyl which may be optionally substituted with halogen, C1-3 alkyl, C1-2 haloalkyl or nitro, m represents 0, 1 or 2, two R1 s may be identical or different, in case m represents 2, n represents 1 or 2, Q represents one the cyclic groups which are mentioned in the specification, to intermediates and several processes for their preparation, to their use as herbicides and to novel compositions containing them.
    Type: Application
    Filed: February 20, 2003
    Publication date: December 4, 2003
    Inventors: Akihiko Yanagi, Shinichi Narabu, Toshio Goto, Chieko Ueno, Shinichi Shirakura
  • Patent number: 6624121
    Abstract: Novel tetrazolinones with herbicidal activity are disclosed. The tetrazolinones of the present invention are represented by the general formula (I) wherein R1, R2, m, n and Q are as defined in the specification. A process for making the tetrazolinones of the present invention is also disclosed.
    Type: Grant
    Filed: February 5, 2002
    Date of Patent: September 23, 2003
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Akihiko Yanagi, Shinichi Narabu, Toshio Goto, Seishi Ito, Chieko Ueno
  • Patent number: 6610319
    Abstract: Immune response modifier compounds—imidazoquinoline amines, imidazopyridine amines, 6,7-fused cycloalkylimidazopyridine amines, and 1,2-bridged imidazoquinoline amines—are useful for the treatment of TH2 mediated diseases by administering a therapeutically effective amount of such compounds in order to inhibit TH2 immune response, suppress IL-4/IL-5 cytokine induction and eosinophilia, as well as enhance TH1 immune response.
    Type: Grant
    Filed: December 19, 2000
    Date of Patent: August 26, 2003
    Assignee: 3M Innovative Properties Company
    Inventors: Mark A. Tomai, David M. Hammerbeck, Karl F. Swingle
  • Patent number: 6589914
    Abstract: The dihalopropene compounds of the general formula (I) have excellent insecticidal/acaricidal activity, so that they are satisfactorily effective for the control of noxious insects, mites and ticks.
    Type: Grant
    Filed: March 4, 2002
    Date of Patent: July 8, 2003
    Assignee: Sumitomo Chemical Company, Limited
    Inventors: Noriyasu Sakamoto, Sanshiro Matsuo, Masaya Suzuki, Taro Hirose, Kazunori Tsushima, Kimitoshi Umeda
  • Patent number: 6559100
    Abstract: Substituted 2-benzoylcyclohexane-1,3-diones of the formula I where: R1 and R2 are each hydrogen, mercapto, nitro, halogen, cyano, thiocyanato, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C2-C6-alkenyl, C2-C6-alkynyl, —OR3, —OCOR3, —OSO2R3, —S(O)nR3, —SO2OR3, —SO2N(R3)2, —NR3SO2R3 or —NR3COR3; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, phenyl or phenyl-C1-C6-alkyl; where the abovementioned alkyl radicals may be partially or fully halogenated and/or may carry one to three of the following groups: hydroxyl, mercapto, amino, cyano, R3, —OR3, —SR3, —N(R3)2, ═NOR3, —OCOR3, —SCOR3, —NR3COR3, —CO2R3, —COSR3, —CON(R3)2, C1-C4-alkyliminooxy, C1-C4-alkoxyamino, C1-C4-alkylcarbonyl, C1-C4-alkoxy-C2-C6-alkoxycarbonyl, C1-C4-alkylsulfonyl, heterocyclyl, heterocyclyloxy, phenyl, benzyl, hetaryl, phenoxy, benzyloxy and hetaryloxy, where the eight last mentioned radic
    Type: Grant
    Filed: February 7, 2000
    Date of Patent: May 6, 2003
    Assignee: BASF Aktiengesellschaft
    Inventors: Stefan Engel, Joachim Rheinheimer, Ernst Baumann, Wolfgang von Deyn, Regina Luise Hill, Guido Mayer, Ulf Misslitz, Oliver Wagner, Matthias Witschel, Martina Otten, Helmut Walter, Karl-Otto Westphalen
  • Patent number: 6548450
    Abstract: According to the instant invention there have been found novel tetrazolinone derivatives represented by the general formula (I) wherein R1 represents methyl or ethyl, R2 represents halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, phenyl, phenoxy, alkoxycarbonyl, nitro or cyano, and n represents 0, 1, 2, 3, 4 or 5, processes and intermediates for their preparation and their use as herbicides.
    Type: Grant
    Filed: November 15, 2001
    Date of Patent: April 15, 2003
    Assignee: Nihon Bayer Agrochem, K.K.
    Inventors: Yukiyoshi Watanabe, Toshio Goto, Seishi Ito, Chieko Ueno
  • Patent number: 6521649
    Abstract: A method for using a compound represented by the general formula: (wherein R1 and R2 are the substituents, respectively, defined in the specification) for agricultural and horticultural disease control, and a composition used in said method.
    Type: Grant
    Filed: September 20, 2000
    Date of Patent: February 18, 2003
    Assignee: Nihon Nohayku Co., Ltd.
    Inventors: Kiyoshi Kuroda, Toru Uchikurohane, Sokichi Tajima, Kenji Tsubata
  • Publication number: 20020028748
    Abstract: There are provided 3-heterocyclic substituted benzisothiazole and benzisoxazole compounds having the structural formula I 1
    Type: Application
    Filed: April 17, 2001
    Publication date: March 7, 2002
    Applicant: Intellectual Property Department BASF Aktiengesellschaft
    Inventors: Peter John Wepplo, Richard Anthony Rampulla, Gavin David Heffernan, Michael Vernie Cossette, Charles Malcolm Langevine, Venkataraman Kameswaran, Robert Eugene Diehl, James Joseph Fiordeliso, Gregory Jay Haley, Michael Anthony Guaciaro
  • Patent number: 6294504
    Abstract: The present invention relates to new compounds of formula (I) wherein R1 to R3, U, V, W, Z and m have the significances given in the description, their use as antidotes, in herbicidal compositions for the control of weeds and plants in useful plant cultivation.
    Type: Grant
    Filed: June 24, 1999
    Date of Patent: September 25, 2001
    Assignee: Syngenta Crop Protection, Inc.
    Inventors: Hans Tobler, Henry Szczepanski, Werner Föry
  • Patent number: 6277790
    Abstract: Tetrazolinonecarboxamides of formula I wherein Het is oxetan-3-yl, thietan-3-yl, tetrahydrofuran-3-yl, furan-3-yl, tetrahydrothiophen-3-yl, thiophen-3-yl, tetrahydro-2H-pyran-3-yl, tetrahydro-2H-thiopyran-3-yl, tetrahydro-2H-pyran-4-yl or tetrahydro-2H-thiopyran-4-yl, in each case with or without substitution; R1 is optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl, or 3- to 7-membered heterocyclyl; R2 is hydrogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, or is optionally substituted cycloalkyl, cycloalkylalkyl, phenyl, phenylalkyl, 3- to 7-membered heterocyclyl, or 3- to 7-membered heterocyclylalkyl, their preparation and herbicidal compositions comprising them.
    Type: Grant
    Filed: February 1, 2000
    Date of Patent: August 21, 2001
    Assignee: BASF Aktiengesellschaft
    Inventors: Cyrill Zagar, Gerhard Hamprecht, Markus Menges, Olaf Menke, Robert Reinhard, Peter Schäfer, Karl-Otto Westphalen, Martina Otten, Helmut Walter
  • Patent number: 6174839
    Abstract: The invention is related to a novel phenylacetylene derivates of formula: wherein X represents hydrogen, halogen, optionally substituted C1-6 alkyl; Y represents hydrogen, halogen, cyano, nitro, optionally substituted C1-6 alkyl, C1-6 alkoxy, C3-8 cycloalkoxy, optionally substituted C1-6 alkylthio, C3-8 cycloalkylthio, C1-6 alkylsulfinyl, optionally substituted C1-6 alkylsulfonyl, C3-8 cycloalkylsulfonyl, C1-6 alkylsulfonyloxy, optionally substituted sulfonamide, optionally substituted carboxamide, etc., or Y may form together with Z which is bonded to the vicinal carbon atom a 5- or 6-membered ring; n is 0 or 1; Z represents hydrogen or halogen; m is 1 or 2; R represents hydrogen, halogen, C1-6 alkyl, tri(C1-6 alkyl)silyl, COORc or CONRdRe; Q represents a heterocyclic group, and their use as herbicid.
    Type: Grant
    Filed: February 23, 1999
    Date of Patent: January 16, 2001
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Akihiko Yanagi, Shin-ichi Narabu, Toshio Goto, Seishi Ito, Natsuko Minegishi, Tatsuya Yamaoka, Chieko Ueno
  • Patent number: 6063734
    Abstract: Ethylene derivatives of formula (I): ##STR1## where Q is an unsubstituted or substituted phenyl or heterocyclic group, especially a 4-thiazolyl, 1- or 3-pyrazolyl, 1,3-oxazol-4-yl, phenyl or pyridyl group; E is a substituent such as a cyano group; A is a substituent such as a 4-pyrazolyl or thiazolyl group; and B is a substituent such as an alkylcarbonyl group. Agricultural chemicals and agents for preventing the attachment of aquatic organisms containing one or more such ethylene derivatives.
    Type: Grant
    Filed: October 23, 1998
    Date of Patent: May 16, 2000
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Tomoyuki Ogura, Hiroshi Murakami, Akira Numata, Rika Miyachi, Toshiro Miyake, Norihiko Mimori, Shinji Takii
  • Patent number: 6048984
    Abstract: The invention relates to compounds of formula (I): and to their use as herbicides, and to intermediates useful in their preparation.
    Type: Grant
    Filed: August 19, 1999
    Date of Patent: April 11, 2000
    Assignee: Rhone-Poulenc Agriculture Limited
    Inventors: Kouichi Araki, Takako Brett, Kei Domom, Atsushi Go, Masahito Ito, Hideshi Mukaida, Yukiko Oe
  • Patent number: 5981438
    Abstract: The present invention relates to novel 1-Phenyl-5-anilinotetrazoles of the formula (I): ##STR1## wherein, R.sup.1, R.sup.2, R.sup.3, R.sup.4, m and n have the meaning provided in the specification, precesses for their preparation and their use as microbiocides, insecticides and/or herbicides.
    Type: Grant
    Filed: January 22, 1998
    Date of Patent: November 9, 1999
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Fritz Maurer, Kaori Kido, Yoshio Kurahashi, Haruko Sawada, Keiko Tanaka, Yuichi Otsu, Yumi Hattori, Katsuhiko Shibuya, Takahisa Abe, Toshio Goto, Seishi Ito
  • Patent number: 5977376
    Abstract: The invention relates to compounds of formula (I): ##STR1## and to their use as herbicides.
    Type: Grant
    Filed: July 17, 1998
    Date of Patent: November 2, 1999
    Assignee: Rhone-Poulenc Agriculture Limited
    Inventors: Kouichi Araki, Takako Brett, Kei Domom, Atsushi Go, Masahito Ito, Hideshi Mukaida, Yukiko Oe
  • Patent number: 5922881
    Abstract: The invention relates to novel heterocyclic imino derivatives, several processes for their preparation and their use for controlling pests.
    Type: Grant
    Filed: November 27, 1996
    Date of Patent: July 13, 1999
    Assignee: Bayer Aktiengesellschaft
    Inventors: Lutz Assmann, Thomas Seitz, Ralf Tiemann, Heinz-Wilhelm Dehne, Klaus Stenzel
  • Patent number: 5846906
    Abstract: Herbicidally active phenyldiketone compounds of the formula I ##STR1## in which the substituents have the following meanings: L and M are hydrogen, C.sub.1 -C.sub.6 -alkyl, C.sub.2 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -alkynyl, C.sub.1 -C.sub.4 -alkoxy, it being possible for these groups to be unsubstituted or substituted by one to five halogen atoms or C.sub.1 -C.sub.4 -alkoxy, or halogen, cyano, nitro, a group --(Y).sub.n --S(O).sub.m R.sup.7 or a group --(Y).sub.n --CO--R.sup.8,Z is a 5- or 6-membered heterocyclic saturated or unsaturated radical which has one to three hetero atoms selected from the group consisting of oxygen, sulfur or nitrogen and which is unsubstituted or substituted by halogen, cyano, nitro, a group --CO--R.sup.8, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.3 -C.sub.8 -cycloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy, C.sub.1 -C.sub.4 -alkylthio, C.sub.1 -C.sub.4 -haloalkylthio, di-C.sub.1 -C.sub.
    Type: Grant
    Filed: July 30, 1997
    Date of Patent: December 8, 1998
    Assignee: BASF Aktiengesellschaft
    Inventors: Wolfgang von Deyn, Regina Luise Hill, Uwe Kardorff, Stefan Engel, Martina Otten, Marcus Vossen, Peter Plath, Harald Rang, Albrecht Harreus, Hartmann Konig, Helmut Walter, Karl-Otto Westphalen, Ulf Misslitz
  • Patent number: 5814629
    Abstract: The invention relates to novel microbicidal and plant-immunising compounds of formula I ##STR1## wherein: X is hydrogen, halogen, C.sub.1 -C.sub.4 alkyl, SR.sub.8, N(R.sub.9)R.sub.10, CH.sub.2 OH, CHO or COOR.sub.8 ;R.sub.8 to R.sub.10 are hydrogen, C.sub.1 -C.sub.4 alkyl, benzyl, C.sub.1 -C.sub.4 acyl or benzoyl;Z is hydrogen, halogen, or a methyl group that is unsubstituted or to which from 1 to 3 unsubstituted or substituted hetero atoms O, S and/or N are bonded; in free form or in the form of salts. They can be used in crop protection for controlling and preventing disease infestation.
    Type: Grant
    Filed: December 19, 1996
    Date of Patent: September 29, 1998
    Assignee: Novartis Finance Corporation
    Inventors: Peter Stanetty, Walter Kunz
  • Patent number: 5786301
    Abstract: This invention relates to substituted N-benzotriazoles of the formula ##STR1## in which: R.sup.1, R.sup.2, R.sup.3,R.sup.4, R.sup.5,R.sup.6, R.sup.7, X are as defined in the specification. The compounds exhibit herbicidal activity.
    Type: Grant
    Filed: August 8, 1996
    Date of Patent: July 28, 1998
    Assignee: Zeneca Limited
    Inventors: Donald R. James, Raymond A. Felix
  • Patent number: 5747420
    Abstract: Novel herbicidal tetrazolinone derivatives of the formula ##STR1## and intermediates therefor of the formula ##STR2## wherein R.sup.1 is alkyl substituted by halogen, andR.sup.2 and R.sup.3 each independently is alkyl, alkenyl, alkynyl, cycloalkyl, phenyl or substituted phenyl, orR.sup.2 and R.sup.3 together with the N-atom to which they are attached, which may form a 5- or 6-membered heterocyclic ring.
    Type: Grant
    Filed: November 3, 1995
    Date of Patent: May 5, 1998
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Toshio Goto, Seishi Ito, Kazuhiro Ukawa, Yukiyoshi Watanabe, Shin-ichi Narabu, Akihiko Yanagi
  • Patent number: 5719104
    Abstract: Bicyclic imides of formulae (I) and (II) and their agriculturally-suitable salts, are disclosed which are useful for controlling undesirable vegatation, wherein G is O or S; n and m are each independently 0; 1; 2; or 3; provided that m+n is 2 or 3; q is 1 or 2; X is CH.sub.2 ; CH(halogen); CF.sub.2 ; CHOCH.sub.2 F; CHOCF.sub.3 ; CHOCH.sub.2 CF.sub.3 ; O; S(O).sub.0-2 ; NH; N(C.sub.1 -C.sub.4 alkyl); or N(C.sub.1 -C.sub.4 haloalkyl); and R.sup.1. R.sup.2, and Q are as defined in the disclosure. Also disclosed are compositions containing the bicyclic imides of formulae (I) and (II) and a method for controlling growth of undesired vegetation comprising applying to the locus to be protected an effective amount, of the bicyclic imides formulae (I) and (II).
    Type: Grant
    Filed: October 3, 1996
    Date of Patent: February 17, 1998
    Assignee: E. I. du Pont de Nemours and Company
    Inventors: John J. Kilama, Karlheinz Drauz, Wonpyo Hong, Matthias Schafer
  • Patent number: 5686392
    Abstract: The herbicidally active substituted N-carbamoyl-tetrazolinones of the formula (I) ##STR1## in which R.sup.1 represents, inter alia, an (optionally substituted) phenyl radical,R.sup.2 represents, inter alia, an alkyl radical, andR.sup.3 represents, inter alia, a cycloalkyl radical,are obtained in very good yields and at high purity--i.e. free from the isomeric O-carbamoyloxytetrazoles (Ia)--by reacting tetrazolinones of the formula (II) with carbamoyl halides of the formula (III) (X=halogen) ##STR2## in the presence of an acid acceptor and in the presence of a diluent, at temperatures of between 0.degree. C. and 200.degree. C., and either isomerizing the O-carbamoylation product of the formula (Ia), which is formed under these circumstances as a byproduct, into the desired product of the formula (I) by heating, or else converting it by hydrolysis or alcoholysis into water-soluble, and thus readily separable, components (variable (a)).
    Type: Grant
    Filed: February 1, 1996
    Date of Patent: November 11, 1997
    Assignee: Bayer Aktiengesellschaft
    Inventors: Uwe Stelzer, Wolfgang Gau, Karl-Julius Reubke
  • Patent number: 5679623
    Abstract: Compounds of the formula ##STR1## in which R.sub.l, R.sub.2, R.sub.3, R.sub.4, Y and Z are as defined in claim 1, and, if appropriate, the tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.
    Type: Grant
    Filed: June 2, 1995
    Date of Patent: October 21, 1997
    Assignee: Ciba-Geigy Corporation
    Inventors: Henry Szczepanski, Haukur Kristinsson
  • Patent number: 5674811
    Abstract: A cyanoketone derivatives of the following formula (1) ##STR1## which are characterized by excellent herbicidal activity and effectiveness against a variety of broad leafed weeds, including barnyard grass, green foxtail, velvet leaf, livid amaranth and hairy beggar ticks.
    Type: Grant
    Filed: October 6, 1994
    Date of Patent: October 7, 1997
    Assignee: Tokuyama Corporation
    Inventors: Toshio Kitajima, Tadashi Kobutani, Shozo Kato, Masao Yamaguchi, Masahiko Ishizaki, deceased
  • Patent number: 5668087
    Abstract: Herbicidal 1-alkenyltetrazolinones of the formula: ##STR1## wherein R.sup.1 represents the group: ##STR2## or the group: ##STR3## R.sup.2 and R.sup.3, independently of one another, represent C.sub.1-6 alkyl, C.sub.3-7 cycloalkyl which may optionally be substited by methyl, C.sub.2-4 alkenyl, C.sub.2-5 alkynyl, phenyl which may optionally be substituted or aralkyl which may optionally be substituted, orR.sup.2 and R.sup.3 may optionally form, together with the N-atom to which they are bonded, a heterocyclic ring which may optionally be substituted, and novel intermediates therefor.
    Type: Grant
    Filed: March 15, 1996
    Date of Patent: September 16, 1997
    Assignee: Nihon Bayer Agrochem K.K.
    Inventors: Toshio Goto, Yoshinori Kitagawa, Seishi Ito, Katsuhiko Shibuya, Kazuhiro Ukawa, Yoshiko Kyo, Natsuko Minegishi
  • Patent number: RE38188
    Abstract: Ethylene derivatives of formula (I): where Q is an unsubstituted or substituted phenyl or heterocyclic group, especially a 4-thiazolyl, 1- or 3-pyrazolyl, 1,3-oxazol-4-yl, phenyl or pyridyl group; E is a substituent such as a cyano group; A is a substituent such as a 4-pyrazolyl or thiazolyl group; and B is a substituent such as an alkylcarbonyl group. Agricultural chemicals and agents for preventing the attachment of aquatic organisms containing one or more such ethylene derivatives.
    Type: Grant
    Filed: October 24, 2001
    Date of Patent: July 15, 2003
    Assignee: Nissan Chemical Industries, Ltd.
    Inventors: Tomoyuki Ogura, Hiroshi Murakami, Akira Numata, Rika Miyachi, Toshiro Miyake, Norihiko Mimori, Shinji Takii