Abstract: Substituted phenyl azabicyclohexanones, their method of preparation, and their conversion into substituted phenyl azabicyclohexanes which are active anxiolytic and analgesic agents.
Type:
Grant
Filed:
June 23, 1977
Date of Patent:
October 3, 1978
Assignee:
American Cyanamid Company
Inventors:
William Joseph Fanshawe, Sidney Robert Safir, Lantz Stephen Crawley
Abstract: A method for resolving racemic substituted cyclopropanedicarboxylic acids which are useful as intermediates for the preparation of substituted phenyl azabicyclohexanes which possess anxyolitic and analgesic activity.
Abstract: Substituted benzenesulfonic acid salts and amides of naphthalenetrisulfonamides and salts thereof useful as complement inhibitors, as well as triphenyl and hexaphenyl esters of substituted benzenesulfonic acid-naphthalenetrisulfonanilides which are new intermediates for the preparation of the active naphthalenetrisulfonamides and the process for their preparation.