Patents Assigned to Bayer Intellectual Property GmbH
  • Substituted benzimidazoles
    Patent number: 9388140
    Abstract: The present invention relates to substituted benzimidazole compounds of general formula (I) in which R3, R5 and A are as defined in the claims, to methods of preparing said compounds, to pharmaceutical compositions and combinations comprising said compounds and to the use of said compounds for manufacturing a pharmaceutical composition for the treatment or prophylaxis of a disease, in particular of a hyper-proliferative and/or angiogenesis disorder, as a sole agent or in combination with other active ingredients.
    Type: Grant
    Filed: March 28, 2012
    Date of Patent: July 12, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Ulrich Klar, Marcus Koppitz, Duy Nguyen, Dirk Kosemund, Roland Neuhaus, Gerhard Siemeister
  • Fused bicyclic imidazoles
    Patent number: 9387204
    Abstract: Compounds of formula (I) a tautomer or stereoisomer thereof, or a salt thereof, wherein ring B and the imidazole to which it is fused, R4, R6 and R7 have the meanings as given in the description and the claims, are effective inhibitors of the Pi3K/Akt pathway.
    Type: Grant
    Filed: November 26, 2013
    Date of Patent: July 12, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Swen Hölder, Armin Zülch, Thomas Bär, Thomas Maier, Astrid Zimmermann, Thomas Beckers, Volker Gekeler, Hemant Joshi, Yogesh Munot, Umesh Bhise, Sunil Chavan, Sachin Shivatare, Sarvesh Patel, Vikas Gore
  • Liquid distributor and liquid collector for chromatography columns
    Patent number: 9383344
    Abstract: The present application relates to a liquid distributor and collector for columns for liquid chromatography with preferably round cross section, which is particularly suitable for columns with large diameter in relation to the packing height.
    Type: Grant
    Filed: August 26, 2005
    Date of Patent: July 5, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Georg-Heinrich Klepp, Sebastian Böcker, Jochen Strube, Heinz Kansy, Hendrik Schmale
  • Pesticidal arylpyrrolidines
    Patent number: 9375000
    Abstract: Arylpyrrolidines of Formula (I): wherein each substituent is as defined in the specification, and use thereof as pesticides and animal parasite-controlling agents.
    Type: Grant
    Filed: September 13, 2011
    Date of Patent: June 28, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Jun Mihara, Mamoru Hatazawa, Daiei Yamazaki, Hidetoshi Kishikawa, Kei Domon, Hidekazu Watanabe, Norio Sasaki, Tetsuya Murata, Koichi Araki, Eiichi Shimojo, Teruyuki Ichihara, Tadashi Ishikawa, Katsuhiko Shibuya, Ulrich Görgens, Peter Bruechner, Reiner Fischer, Johannes-Rudolf Jansen, Tobias Kapferer, Simon Maechling, Michael Maue, Arnd Voerste
  • 5-halogenopyrazolecarboxamides
    Patent number: 9375004
    Abstract: The present invention relates to novel 5-halogenopyrazole(thio)carboxamides, their process of preparation, their use as fungicide active agents, particularly in the form of fungicide compositions, and methods for the control of phytopathogenic fungi, notably of plants, using these compounds or compositions.
    Type: Grant
    Filed: November 14, 2011
    Date of Patent: June 28, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Jürgen Benting, Pierre-Yves Coqueron, Pierre Cristau, Peter Dahmen, Philippe Desbordes, Christophe Dubost, Stephanie Gary, Jörg Greul, Hiroyuki Hadano, Jean-Pierre Vors, Ulrike Wachendorff-Neumann
  • Process for preparing aryl- and heteroarylacetic acid derivatives
    Patent number: 9376417
    Abstract: The invention relates to a process for preparing aryl- and heteroarylacetic acids and derivatives thereof by reaction of aryl or heteroaryl halides with malonic diesters in the presence of a palladium catalyst, of one or more bases and optionally of a phase transfer catalyst. This process enables the preparation of a multitude of functionalized aryl- and heteroarylacetic acids and derivatives thereof, especially also the preparation of arylacetic acids with sterically demanding substituents.
    Type: Grant
    Filed: April 15, 2015
    Date of Patent: June 28, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Thomas Himmler, Lukas J. Goossen, Felix Rudolphi, Bingrui Song
  • Process for preparing cis-alkoxy-substituted spirocyclic phenylacetylamino acid esters and cis- alkoxy-substituted spirocyclic 1H- pyrrolidine-2,4-dione derivatives
    Patent number: 9376374
    Abstract: The present invention relates to a novel process for preparing cis-alkoxy-substituted spirocyclic phenylacetylamino acid esters and cis-alkoxy-substituted spirocyclic 1H-pyrrolidine-2,4-dione derivatives, and also to novel intermediates and starting materials which are produced and/or used in the process according to the invention.
    Type: Grant
    Filed: March 25, 2013
    Date of Patent: June 28, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Taraneh Farida, Berndt Maiwald, Martin Littmann, Winfried Etzel, Rafael Warsitz, Nicolas Henck, Michael Esser
  • 5-aminopyrimidine derivatives and use thereof for combating undesired plant growth
    Patent number: 9375002
    Abstract: What is described are compounds of the general formula (I) and agrochemically acceptable salts thereof and their use in the field of crop protection.
    Type: Grant
    Filed: March 27, 2013
    Date of Patent: June 28, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Klemens Minn, Michael Gerhard Hoffmann, Elmar Gatzweiler, Ines Heinemann, Isolde Haeuser-Hahn, Christopher Hugh Rosinger
  • Heteroarylpiperidine and piperazine derivatives as fungicides
    Patent number: 9375009
    Abstract: Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols RA1, RA2, X, Y, L1, L2, RB1, RB2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).
    Type: Grant
    Filed: December 21, 2012
    Date of Patent: June 28, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Tomoki Tsuchiya, Pierre Wasnaire, Sebastian Hoffmann, Thomas Seitz, Stefan Hillebrand, Juergen Benting, Jan Peter Schmidt, Pierre Cristau
  • Active compound combinations
    Patent number: 9370186
    Abstract: The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) ethaboxam and (B) fenamidone. Moreover, the invention relates to a method for curatively or preventively controlling the phytopathogenic fungi of plants or crops, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.
    Type: Grant
    Filed: January 30, 2013
    Date of Patent: June 21, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Albert Schirring, Ulrike Wachendorff-Neumann, Sylvain Tafforeau, Marie-Pascale Latorse
  • Use of ALS inhibitor herbicides for control of unwanted vegetation in ALS inhibitor herbicide tolerant , such as , plants
    Patent number: 9370183
    Abstract: The present invention relates to the use of the ALS inhibitor herbicides for controlling unwanted vegetation in ALS inhibitor herbicide tolerant Brassica plants, more especially, the present invention relates to the use of ALS inhibitor herbicides for control of unwanted vegetation in Brassica growing areas which Brassica plants comprise non-transgenic mutations of their endogenous acetolactate synthase (ALS) genes I and III.
    Type: Grant
    Filed: May 4, 2012
    Date of Patent: June 21, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Ruediger Hain, Gerhard Johann, Udo Bickers
  • Substituted pyrazolopyrimidines as Akt kinase inhibitors
    Patent number: 9370517
    Abstract: Compounds of formula (I) which are effective inhibitors of the Pi3K/Akt pathway, processes for their production and their use as pharmaceuticals.
    Type: Grant
    Filed: January 8, 2013
    Date of Patent: June 21, 2016
    Assignees: Bayer Intellectual Property GmbH, Bayer Pharma Aktiengesselschaft
    Inventors: Lars Bärfacker, William Scott, Andrea Hägebarth, Hartmut Rehwinkel, Oliver Politz, Roland Neuhaus, Ulf Bömer
  • Method for producing dithiine tetracarboximides
    Patent number: 9365586
    Abstract: The present invention relates to a process for preparing dithiinetetracarboximides by reaction of succinic monoamides with thionyl chloride, with continuous performance of at least one of the process steps.
    Type: Grant
    Filed: March 18, 2013
    Date of Patent: June 14, 2016
    Assignees: Bayer Cropscience AG, Bayer Intellectual Property GmbH
    Inventors: Thomas Himmler, Thomas Geller, Lars Rodefeld, Mark James Ford, Guenter Hoemberger, Dieter Heinz
  • Triazolo and tetrazolo pyrimidine derivatives as HNE inhibitors for treating COPD
    Patent number: 9359362
    Abstract: The present invention relates to novel heterocyclically fused diaryldihydropyrimidine derivatives, to processes for their preparation, to their use alone or in combination for the treatment and/or prevention of diseases and also to their use for preparing medicaments for the treatment and/or prevention of diseases, in particular for the treatment and/or prevention of disorders of the lung and the cardiovascular system.
    Type: Grant
    Filed: October 7, 2013
    Date of Patent: June 7, 2016
    Assignee: Bayer Intellectual Property Gmbh
    Inventors: Franz Von Nussbaum, Dagmar Karthaus, Sonja Anlauf, Martina Delbeck, Volkhart Min-Jian Li, Daniel Meibom, Klemens Lustig
  • Ketoheteroarylpiperdine and -piperazine derivatives as fungicides
    Patent number: 9357779
    Abstract: Ketoheteroarylpiperidine and -piperazine derivatives of the formula (I), in which the symbols A, L1, G, X, Y, T and R1 have the meanings given in the description and agrochemically active salts thereof and their use for controlling phytopathogenic harmful fungi and also processes for preparing compounds of the formula (I).
    Type: Grant
    Filed: March 13, 2013
    Date of Patent: June 7, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Pierre Cristau, Sebastian Hoffmann, Joachim Kluth, Thomas Seitz, Tomoki Tsuchiya, Pierre Wasnaire, Jürgen Benting, Ulrike Wachendorff-Neumann
  • Process for preparing pan-CDK inhibitors of the formula (I), and intermediates in the preparation
    Patent number: 9359306
    Abstract: The invention relates to a novel process for the preparation of pan-CDK inhibitors of the formula (I), and intermediates of the preparation.
    Type: Grant
    Filed: September 20, 2011
    Date of Patent: June 7, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Joachim Krüger, Jörg Gries, Kai Lovis, Jorma Haβfeld
  • Antibiotic formulations, unit doses, kits, and methods
    Patent number: 9351930
    Abstract: An aqueous or powder composition includes anti-gram-negative antibiotic or salt thereof being present at an amount ranging from about 100 mg/ml to about 200 mg/ml. Another aqueous or powder composition includes anti-gram-positive antibiotic or salt thereof being present at a concentration ranging from about 0.6 to about 0.9 of the water solubility limit, at 25° C. and 1.0 atmosphere, of the anti-gram-positive antibiotic or salt thereof. Other embodiments include unit doses, kits, and methods.
    Type: Grant
    Filed: June 12, 2012
    Date of Patent: May 31, 2016
    Assignee: Bayer Intellectual Property GMBH
    Inventors: Chatan Charan, Sarvajna Dwivedi
  • Cyanoenamines and their use as fungicides
    Patent number: 9351489
    Abstract: The present invention relates to cyanoenamine derivatives, their process of preparation, intermediate compounds, their use as fungicide active agents, particularly in the form of fungicide compositions, and methods for the control of phytopathogenic fungi, notably of plants and in material protection, using these compounds or compositions.
    Type: Grant
    Filed: November 11, 2011
    Date of Patent: May 31, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Jürgen Benting, Ulrike Wachendorff-Neumann, Philippe Desbordes, Christophe Dubost, Pierre Genix, Shinichi Narabu, Jean-Pierre Vors
  • Antibiotic formulations, unit doses, kits, and methods
    Patent number: 9351929
    Abstract: An aqueous or powder composition includes anti-gram-negative antibiotic or salt thereof being present at an amount ranging from about 100 mg/ml to about 200 mg/ml. Another aqueous or powder composition includes anti-gram-positive antibiotic or salt thereof being present at a concentration ranging from about 0.6 to about 0.9 of the water solubility limit, at 25° C. and 1.0 atmosphere, of the anti-gram-positive antibiotic or salt thereof. Other embodiments include unit doses, kits, and methods.
    Type: Grant
    Filed: May 14, 2012
    Date of Patent: May 31, 2016
    Assignee: Bayer Intellectual Property GMBH
    Inventors: Chatan Charan, Sarvajna Dwivedi
  • Process for preparing pyridyl-substituted pyrazoles
    Patent number: 9340526
    Abstract: The present invention relates to a process for preparing 1-pyridyl-substituted pyrazoles, comprising the reaction of acetyleneketones with pyridylhydrazine derivatives to give 1-pyridyl-substituted dihydro-1H-pyrazoles, the further reaction thereof with elimination of water to give 1-pyridyl-substituted trihalomethylpyrazoles, and the further processing thereof.
    Type: Grant
    Filed: March 23, 2015
    Date of Patent: May 17, 2016
    Assignee: Bayer Intellectual Property GmbH
    Inventors: Sergii Pazenok, Norbert Lui, Harry Blaschke