Patents by Inventor Murielle Rinaldi-Carmona

Murielle Rinaldi-Carmona has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • 3-Acylindole derivatives, preparation and therapeutic use thereof
    Patent number: 7741363
    Abstract: The invention relates to compounds of formula (I), wherein X, R1, R2, R3, R4 and R5 are as described herein. The invention also includes preparative methods for the preparation of compounds of formula (I). A method for the therapeutic use of the inventive compounds is also disclosed and claimed.
    Type: Grant
    Filed: May 14, 2008
    Date of Patent: June 22, 2010
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Claude Vernhet, Murielle Rinaldi-Carmona, CaroleElisabeth Guillaumont-Legeay
  • 1-BENZYLPYRAZOLE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
    Publication number: 20100144818
    Abstract: The present invention relates to compounds corresponding to formula (I): in which Y, R1, R2, R3, R4, R5 and R6 are as defined herein. The present invention also relates to the methods of preparation and the therapeutic applications of the compounds of formula (I).
    Type: Application
    Filed: December 3, 2009
    Publication date: June 10, 2010
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Laurent BOULU, Joseph MILLAN, Murielle RINALDI-CARMONA
  • N-[(4,5-DIPHENYL-2-THIENYL)METHYL]AMINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
    Publication number: 20100137402
    Abstract: The subject of the present invention is compounds corresponding to formula (I): Wherein X, R1, R2, R3 and R4 are as described herein. The invention also relates to a method for the preparation and application of said compounds as cannabinoid CB1 receptor antagonists.
    Type: Application
    Filed: February 8, 2010
    Publication date: June 3, 2010
    Applicant: SANOFI-AVENTIS
    Inventors: Jean-Philippe DUCOUX, Francis BARTH, Murielle RINALDI-CARMONA, Christian CONGY
  • N-[(4,5-diphenyl-2-thienyl)methyl]amine derivatives, their preparation and their therapeutic application
    Patent number: 7687537
    Abstract: The subject of the present invention is compounds corresponding to formula (I): Wherein X, R1, R2, R3 and R4 are as described herein. The invention also relates to a method for the preparation and application of said compounds as cannabinoid CB1 receptor antagonists.
    Type: Grant
    Filed: August 1, 2007
    Date of Patent: March 30, 2010
    Assignee: Sanofi-Aventis
    Inventors: Jean-Philippe Ducoux, Francis Barth, Murielle Rinaldi-Carmona, Christian Congy
  • N-[(4,5-diphenyl-3-alkyl-2-thienyl)methyl]amine [amide, sulfonamide, carbamate and urea) derivatives as cannabinoid CB1 receptor antagonists
    Patent number: 7674821
    Abstract: The invention concerns compounds of formula (I), wherein X, R1, R2, R3, R4 and R5 are as defined herein. The invention also concerns a method for preparing said compounds and their use as cannabinoid CB1 receptor antagonists.
    Type: Grant
    Filed: June 18, 2007
    Date of Patent: March 9, 2010
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Jean-Phillipe Ducoux, Murielle Rinaldi-Carmona
  • SUBSTITUTED N-(4-CYANO-1H-PYRAZOL-3-YL)METHYLAMINE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
    Publication number: 20100041709
    Abstract: The present invention relates to compounds corresponding to formula (I): Wherein X, R1, R2, R3 and R4 are as defined herein. The invention further relates to preparation and therapeutic use of these compounds.
    Type: Application
    Filed: June 24, 2009
    Publication date: February 18, 2010
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian Congy, Serge Martinez, Murielle Rinaldi-Carmona, Martine Vernhet
  • (1,5-diphenyl-1-pyrazol-3-yl)oxadiazole derivatives, preparation method thereof and use of same in therapeutics
    Patent number: 7632852
    Abstract: The invention relates to compounds having formula (I): Wherein R1, R2, R3 and R4 are as defined herein. The invention also relates to a method of preparing said compounds and to the application thereof in therapeutics.
    Type: Grant
    Filed: August 8, 2007
    Date of Patent: December 15, 2009
    Assignee: Sanofi-aventis
    Inventors: Francis Barth, Christian Congy, Patrick Gueule, Murielle Rinaldi-Carmona, Didier Van Broeck
  • Heterocyclic derivatives, preparation and therapeutic use thereof
    Patent number: 7618991
    Abstract: The invention concerns compounds of formula (I): Wherein X, Y, R1, R2, R3 and R4 are as described herein. The invention also concerns a method for preparing same and the therapeutic use thereof.
    Type: Grant
    Filed: May 23, 2008
    Date of Patent: November 17, 2009
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Murielle Rinaldi-Carmona
  • Derivatives of 4,5-diarylpyrrole, preparation method thereof and use of same in therapeutics
    Patent number: 7618995
    Abstract: The invention relates to compounds having formula (I): Wherein X, R1, R2, R3, R4 and R5 are as defined herein. The invention also relates to the preparation method thereof and the use of same in therapeutics.
    Type: Grant
    Filed: December 7, 2007
    Date of Patent: November 17, 2009
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Laurent Hortala, Murielle Rinaldi-Carmona
  • SUBSTITUTED 2,5-DIHYDRO-3H-PYRAZOLO[4,3-C]PYRIDAZIN-3-ONE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE OF THE SAME
    Publication number: 20090281107
    Abstract: The invention relates to compounds having the formula (I): Wherein R1, R2, R3 and R4 are as described herein. Also disclosed are the method of preparation and their use in therapy.
    Type: Application
    Filed: May 19, 2009
    Publication date: November 12, 2009
    Applicant: SANOFI-AVENTIS
    Inventors: Christian CONGY, Victor DOS SANTOS, Murielle RINALDI-CARMONA, Arnaud ROUQUETTE, Didier VAN BROECK
  • PYRROLE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
    Publication number: 20090281116
    Abstract: The invention relates to compounds having the formula (I): Wherein R1, R2, R3, R4, R5, R6, R7 and R9 and A-R9 are as defined herein. Also disclosed are the preparative methods for the compounds of formula (I) and their use in therapy.
    Type: Application
    Filed: May 14, 2009
    Publication date: November 12, 2009
    Applicant: SANOFI-AVENTIS
    Inventors: Francis Barth, Christian Congy, Laurent Hortala, Murielle Rinaldi-Carmona
  • N-[(4,5-diphenyl-2-thienyl)methyl]sulfonamide derivatives, preparation thereof and their therapeutic application
    Patent number: 7589120
    Abstract: The invention relates to compounds of formula (I): Wherein X, R1, R2, R3 and R4 are as described herein. The invention also relates to a method for preparing the aforementioned compounds and to their therapeutic application.
    Type: Grant
    Filed: July 10, 2007
    Date of Patent: September 15, 2009
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Jean-Philippe Ducoux, Murielle Rinaldi-Carmona
  • N-[4,5-diphenylpyrimidin-2-yl)methyl]amine derivatives, the preparation thereof and their therapeutic use
    Patent number: 7541361
    Abstract: The invention relates to compounds of formula (I): Wherein X, R1, R2, R3, R4 and R5 are as defined herein. The invention also relates to a method for preparing the aforementioned compounds and to their therapeutic use.
    Type: Grant
    Filed: January 3, 2008
    Date of Patent: June 2, 2009
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Patrick Gueule, Murielle Rinaldi-Carmona
  • 1,5-diarylpyrrole derivatives, preparation method thereof and application of same in therapeutics
    Patent number: 7524971
    Abstract: The invention relates to compounds having formula (I): Wherein X, R1, R2, R3, R4, R5 and R6 are as defined herein. The invention also relates to a method of preparing said compounds and to die application thereof in therapeutics.
    Type: Grant
    Filed: August 2, 2007
    Date of Patent: April 28, 2009
    Assignee: Sanofi - Aventis
    Inventors: Francis Barth, Christian Congy, Laurent Hortala, Murielle Rinaldi-Carmona
  • 4-cyanopyrazole-3-carboxamide derivatives, preparation and application thereof
    Patent number: 7521471
    Abstract: The invention relates to 4-cyanopyrazole-3-carboxamide derivatives of formula (I): in which R1, R2, R3, R4, R5, R6, R7, R8 are as described herein. Also disclosed and claimed are the method of preparation and therapeutic application of compound of formula (I).
    Type: Grant
    Filed: August 1, 2007
    Date of Patent: April 21, 2009
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Serge Martinez, Murielle Rinaldi-Carmona
  • Thiophene-2-carboxamide derivatives, preparation and therapeutic application thereof
    Patent number: 7462631
    Abstract: The invention discloses and claims a compound of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7, R8 and R11 are as defined herein. Further embodiments of the invention include a method of preparation of a compound of formula (I), its pharmaceutical composition and a method of treatment of a disease using a compound of formula (I).
    Type: Grant
    Filed: April 7, 2006
    Date of Patent: December 9, 2008
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Jean-Philippe Ducoux, Murielle Rinaldi-Carmona, Christian Congy
  • DIARYLTRIAZOLMETHYLAMINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF
    Publication number: 20080293794
    Abstract: The invention concerns compounds of formula (I): Wherein X, R1, R2, R3 and R4 are as described herein. The invention also concerns a method for preparing same and the therapeutic use thereof.
    Type: Application
    Filed: May 22, 2008
    Publication date: November 27, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Murielle RINALDI-CARMONA
  • 3-ACYLINDOLE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF
    Publication number: 20080275102
    Abstract: The invention relates to compounds of formula (I), wherein X, R1, R2, R3, R4 and R5 are as described herein. The invention also includes preparative methods for the preparation of compounds of formula (I). A method for the therapeutic use of the inventive compounds is also disclosed and claimed.
    Type: Application
    Filed: May 14, 2008
    Publication date: November 6, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Claude VERNHET, Murielle RINALDI-CARMONA, Carole Elisabeth GUILLAUMONT-LEGEAY
  • HETEROCYCLIC DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF
    Publication number: 20080269303
    Abstract: The invention concerns compounds of formula (I): Wherein X, Y, R1, R2, R3 and R4 are as described herein. The invention also concerns a method for preparing same and the therapeutic use thereof.
    Type: Application
    Filed: May 23, 2008
    Publication date: October 30, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Murielle RINALDI-CARMONA
  • PYRROLE DERIVATIVES, INTERMEDIATES THEREFOR, PREPARATION AND THERAPEUTIC USE THEREOF
    Publication number: 20080194581
    Abstract: The invention concerns compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7, R8 and R9 are as defined herein. The invention also concerns the method for preparing said compounds including the intermediates therefor and their therapeutic use.
    Type: Application
    Filed: April 14, 2008
    Publication date: August 14, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Laurent HORTALA, Murielle RINALDI-CARMONA