Patents by Inventor Murielle Rinaldi-Carmona

Murielle Rinaldi-Carmona has filed for patents to protect the following inventions. This listing includes patent applications that are pending as well as patents that have already been granted by the United States Patent and Trademark Office (USPTO).

  • DERIVATIVES OF 4,5-DIARYLPYRROLE, PREPARATION METHOD THEREOF AND USE OF SAME IN THERAPEUTICS
    Publication number: 20080176924
    Abstract: The invention relates to compounds having formula (I): Wherein X, R1, R2, R3, R4 and R5 are as defined herein. The invention also relates to the preparation method thereof and the use of same in therapeutics.
    Type: Application
    Filed: December 7, 2007
    Publication date: July 24, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Laurent HORTALA, Murielle RINALDI-CARMONA
  • N-[(4,5-DIPHENYLPYRIMIDIN-2-YL)METHYL]AMINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR THERAPEUTIC USE
    Publication number: 20080176867
    Abstract: The invention relates to compounds of formula (I): Wherein X, R1, R2, R3, R4 and R5 are as defined herein. The invention also relates to a method for preparing the aforementioned compounds and to their therapeutic use.
    Type: Application
    Filed: January 3, 2008
    Publication date: July 24, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Patrick GUEULE, Murielle RINALDI-CARMONA
  • Terphenyl derivatives, preparation thereof, compositions containing same
    Patent number: 7390924
    Abstract: The invention relates to terphenyl derivatives of formula: and to their preparation and to the pharmaceutical compositions comprising them. These compounds exhibit an antagonist activity with respect to CB1 cannabinoid receptors.
    Type: Grant
    Filed: April 10, 2003
    Date of Patent: June 24, 2008
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Serge Martinez, Murielle Rinaldi-Carmona
  • Pyrrole derivatives, their preparation and their therapeutic use
    Patent number: 7381727
    Abstract: The invention concerns compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7, R8 and R9 are as defined herein. The invention also concerns the method for preparing said compounds and their therapeutic use.
    Type: Grant
    Filed: January 22, 2007
    Date of Patent: June 3, 2008
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Laurent Hortala, Murielle Rinaldi-Carmona
  • DERIVATIVES OF N-[(1,5-DIPHENYL-1H-PYRAZOL-3-YL)METHYL] SULFONAMIDE, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS
    Publication number: 20080070962
    Abstract: The present invention relates to compounds corresponding to the formula (I): In which R1, R2, R3, R4 and R5 are as described herein. The invention also relates to the method of preparation of said compounds and their application in therapeutics.
    Type: Application
    Filed: September 21, 2007
    Publication date: March 20, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis Barth, Christian Congy, Serge Martinez, Philippe Pointeau, Murielle Rinaldi-Carmona
  • Diphenylpyridine derivatives, preparation and therapeutic application thereof
    Patent number: 7345059
    Abstract: The invention relates to 5,6-diphenylpyridine-3-carboxamide derivatives of general formula (I): where: R1 represents hydrogen or a (C1-C4)alkyl; R2 represents: a monoazo saturated heterocycle of 5 to 7 atoms, the nitrogen atom being substituted with a (C1-C4)alkanoyl; NR10R11; a nonaromatic (C3-C10) carbocycle more than tri-substituted with (C1-C4)alkyl; a nonaromatic (C11-C12) carbocycle unsubstituted or mono- or polysubstituted with (C1-C4)alkyl; a monooxygenated saturated heterocycle with 5 to 7 atoms, more than tri-substituted with (C1-C4)alkyl; or R1 and R2, together with the nitrogen atom to which the above are bonded, form a 4-disubstituted piperidin-1-yl group; the salts, solvates and hydrates thereof. The invention further relates to a method for production and therapeutic application thereof.
    Type: Grant
    Filed: December 22, 2005
    Date of Patent: March 18, 2008
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Laurent Hortala, Murielle Rinaldi-Carmona
  • (1,5-DIPHENYL-1H-PYRAZOL-3-YL)OXADIAZOLE DERIVATIVES, PREPARATION METHOD THEREOF AND USE OF SAME IN THERAPEUTICS
    Publication number: 20080039510
    Abstract: The invention relates to compounds having formula (I): Wherein R1, R2, R3 and R4 are as defined herein. The invention also relates to a method of preparing said compounds and to the application thereof in therapeutics.
    Type: Application
    Filed: August 8, 2007
    Publication date: February 14, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Patrick GUEULE, Murielle RINALDI-CARMONA, Didier VAN BROECK
  • PYRIDINE DERIVATIVES, PREPARATION AND THERAPEUTIC APPLICATION THEREOF
    Publication number: 20080021070
    Abstract: The invention relates to compounds of formula (I): Wherein Z, R3 to R9 are as described herein. The invention also relates to methods of preparation of compounds of formula (I) and intermediates thereof. The compounds of this invention are active at CB1 cannabinoid receptor site, and are therefore, useful as pharmaceutical agents in treating a variety of diseases caused by the effects of CB1 cannabinoid receptors.
    Type: Application
    Filed: April 3, 2007
    Publication date: January 24, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Lionel Barre, Francis Barth, Christian Congy, Murielle Rinaldi-Carmona, Philippe Pointeau
  • Oxazole derivatives, preparation and therapeutic use thereof
    Patent number: 7320978
    Abstract: This invention relates to compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7 and R8 are as described herein. The invention further relates to a method for prevention and therapeutic use thereof.
    Type: Grant
    Filed: August 1, 2006
    Date of Patent: January 22, 2008
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Joelle Arnaud-Taillades, Christian Congy, Murielle Rinaldi-Carmona
  • 1,5-DIARYLPYRROLE DERIVATIVES, PREPARATION METHOD THEREOF AND APPLICATION OF SAME IN THERAPEUTICS
    Publication number: 20080015245
    Abstract: The invention relates to compounds having formula (I): Wherein X, R1, R2, R3, R4, R5 and R6 are as defined herein. The invention also relates to a method of preparing said compounds and to die application thereof in therapeutics.
    Type: Application
    Filed: August 2, 2007
    Publication date: January 17, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Laurent HORTALA, Murielle RINALDI-CARMONA
  • N-[(4,5-DIPHENYL-2-THIENYL)METHYL]AMINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
    Publication number: 20080009543
    Abstract: The subject of the present invention is compounds corresponding to formula (I): Wherein X, R1, R2, R3 and R4 are as described herein. The invention also relates to a method for the preparation and application of said compounds as cannabinoid CB1 receptor antagonists.
    Type: Application
    Filed: August 1, 2007
    Publication date: January 10, 2008
    Applicant: SANOFI-AVENTIS
    Inventors: Jean-Philippe DUCOUX, Francis Barth, Murielle Rinaldi-Carmona, Christian Congy
  • 4-CYANOPYRAZOLE-3-CARBOXAMIDE DERIVATIVES, PREPARATION AND APPLICATION THEREOF
    Publication number: 20070293541
    Abstract: The invention relates to 4-cyanopyrazole-3-carboxamide derivatives of formula (I): in which R1, R2, R3, R4, R5, R6, R7, R8 are as described herein. Also disclosed and claimed are the method of preparation and therapeutic application of compound of formula (I).
    Type: Application
    Filed: August 1, 2007
    Publication date: December 20, 2007
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Serge MARTINEZ, Murielle RINALDI-CARMONA
  • N-[(4,5-DIPHENYL-2-THIENYL)METHYL]SULFONAMIDE DERIVATIVES, PREPARATION THEREOF AND THEIR THERAPEUTIC APPLICATION
    Publication number: 20070287744
    Abstract: The invention relates to compounds of formula (I): Wherein X, R1, R2, R3 and R4 are as described herein. The invention also relates to a method for preparing the aforementioned compounds and to their therapeutic application.
    Type: Application
    Filed: July 10, 2007
    Publication date: December 13, 2007
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Jean-Philippe DUCOUX, Murielle RINALDI-CARMONA
  • N-[(4,5-DIPHENYL-3-ALKYL-2-THIENYL)METHYL]AMINE [AMIDE, SULFONAMIDE, CARBAMATE AND UREA) DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS
    Publication number: 20070270470
    Abstract: The invention concerns compounds of formula (I), wherein X, R1, R2, R3, R4 and R5 are as defined herein. The invention also concerns a method for preparing said compounds and their use as cannabinoid CB1 receptor antagonists.
    Type: Application
    Filed: June 18, 2007
    Publication date: November 22, 2007
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Christian CONGY, Jean-Phillipe DUCOUX, Murielle RINALDI-CARMONA
  • Derivatives of N-[(1,5-diphenyl-1H-pyrazol-3-yl)methyl]sulfonamide, their preparation and their application in therapeutics
    Patent number: 7297710
    Abstract: The present invention relates to compounds corresponding to the formula (I): In which R1, R2, R3, R4 and R5 are as described herein. The invention also relates to the method of preparation of said compounds and their application in therapeutics.
    Type: Grant
    Filed: July 12, 2006
    Date of Patent: November 20, 2007
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Serge Martinez, Philippe Pointeau, Murielle Rinaldi-Carmona
  • Derivatives of N?-(1,5-diphenyl-1H-pyrazol-3-yl) sulfonamide with CB1 receptor affinity
    Patent number: 7294645
    Abstract: The invention relates to compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7, R8, R9 are as defined herein. The invention also relates to the preparation method thereof and to the use of same in therapeutics.
    Type: Grant
    Filed: July 6, 2006
    Date of Patent: November 13, 2007
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Serge Martinez, Murielle Rinaldi-Carmona, Christian Congy
  • 4-cyanopyrazole-3-carboxamide derivatives, preparation, and application thereof
    Patent number: 7282516
    Abstract: The invention relates to 4-cyanopyrazole-3-carboxamide derivatives of formula (I): in which R1, R2, R3, R4, R5, R6, R7, R8 are as described herein. Also disclosed and claimed are the method of preparation and therapeutic application of compound of formula (I).
    Type: Grant
    Filed: December 22, 2005
    Date of Patent: October 16, 2007
    Assignee: Sanofi-Aventis
    Inventors: Francis Barth, Christian Congy, Serge Martinez, Murielle Rinaldi-Carmona
  • PYRROLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC USE
    Publication number: 20070149596
    Abstract: The invention concerns compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7, R8 and R9 are as defined herein. The invention also concerns the method for preparing said compounds and their therapeutic use.
    Type: Application
    Filed: January 22, 2007
    Publication date: June 28, 2007
    Applicant: SANOFI-AVENTIS
    Inventors: Francis Barth, Christian Congy, Laurent Hortala, Murielle Rinaldi-Carmona
  • OXAZOLE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF
    Publication number: 20070043060
    Abstract: This invention relates to compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7 and R8 are as described herein. The invention further relates to a method for prevention and therapeutic use thereof.
    Type: Application
    Filed: August 1, 2006
    Publication date: February 22, 2007
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Joelle ARNAUD-TAILLADES, Christian CONGY, Murielle RINALDI-CARMONA
  • DERIVATIVES OF N-' (1,5-DIPHENYL-1H-PYRAZOL-3-YL) SULFONAMIDE WITH CB1 RECEPTOR AFFINITY
    Publication number: 20070021486
    Abstract: The invention relates to compounds of formula (I): Wherein R1, R2, R3, R4, R5, R6, R7, R8, R9 are as defined herein. The invention also relates to the preparation method thereof and to the use of same in therapeutics.
    Type: Application
    Filed: July 6, 2006
    Publication date: January 25, 2007
    Applicant: SANOFI-AVENTIS
    Inventors: Francis BARTH, Serge MARTINEZ, Murielle RINALDI-CARMONA, Christian CONGY