Additional C=o Bonded Directly To Urea Nitrogen Patents (Class 514/594)
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Publication number: 20070275066Abstract: The present invention relates to a sustained release drug delivery system composed of a water insoluble polymer, and more particularly, to a sustained release drug delivery system comprising: a crystalline core material; an active ingredient layer which is formed on an outer surface of the crystalline core material and comprises a pharmacologically active ingredient and a water insoluble polymer; and a sustained release layer which is formed on an outer surface of the active ingredient layer and comprises a sustained release film forming material. The present invention also relates to a sustained release drug delivery system which releases an effective drug in an aqueous solution or a body fluid for 24 hours by using a sustained release film forming material and a plasticizer together to provide sustained release of a pharmacologically active ingredient.Type: ApplicationFiled: August 23, 2006Publication date: November 29, 2007Applicant: Korea Research Institute of Chemical TechnologyInventors: Sun Hang Cho, Byung Cheol Shin, Soon Hong Yuk, Jin A. Seo, Ji Sun Park
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Publication number: 20070253992Abstract: A poison bait in the form of gel which comprises an active ingredient for controlling wood harmful insect, water and cellulose ether has an excellent efficacy for controlling wood harmful insects, wherein the content ratio of water:the cellulose ether is 4:1 to 3:4.Type: ApplicationFiled: April 5, 2007Publication date: November 1, 2007Applicant: SUMITOMO CHEMICAL COMPANY, LIMITEDInventors: Shun-ichi KUBOTA, Kazuhide Nakada
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Patent number: 7288572Abstract: The present invention relates to novel insecticidally and acaricidally active compound combinations of N2-[1,1-dimethyl-2-(methylsulphonyl)ethyl]-3-iodo-N1-{2-methyl-4-[1,2,2,2-tetrafluoro-1-(trifluoromethyl)ethyl]phenyl}phthalamide of the formula (I) and active compounds identified in the disclosure.Type: GrantFiled: September 15, 2006Date of Patent: October 30, 2007Assignee: Bayer CropScience AGInventors: Jörg Konze, Wolfram Andersch, Dietrich Stübler, Rüdiger Fischer
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Patent number: 7232929Abstract: The invention relates to new 2,2,3,3-tetramethylcyclopropane carboxamide derivative compounds, pharmaceutical compositions thereof and uses thereof for treating psychotic disorders, neurodegenerative diseases, epilepsy and pain.Type: GrantFiled: February 15, 2004Date of Patent: June 19, 2007Assignee: Yissum Research Development Company of the Hebrew University of JerusalemInventors: Meir Bialer, Boris Yagen, Eyal Sobol, Dan Kaufmann
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Patent number: 7195773Abstract: A pesticidal composition comprising a pesticidally effective amount of at least one of a pyridic compound of the formula (I) or it salt and at least one of other pesticides: wherein Y is a haloalkyl group, m is 0 or 1, and Q is or a substituted or unsubstituted heterocyclic group, (wherein X is an oxygen atom or a sulfur atom, R1 and R2 are respectively independently a hydrogen atom, a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkenyl group, a substituted or unsubstituted alkynyl group, a substituted or unsubstituted cycloalkyl group, and the like.Type: GrantFiled: October 22, 2001Date of Patent: March 27, 2007Assignee: Ishihara Sangyo Kaisha, Ltd.Inventors: Masayuki Morita, Mitsugu Iwasa
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Patent number: 7179941Abstract: The invention relates to compounds of the formula I in which the radicals are defined as specified, and also to their physiologically tolerated salts. The compounds are suitable, for example, as medicaments for preventing and treating type 2 diabetes.Type: GrantFiled: January 23, 2004Date of Patent: February 20, 2007Assignee: Sanofi-Aventis Deutschland GmbHInventors: Elisabeth Defossa, Dieter Kadereit, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Karl-Ulrich Wendt, Erich Von Roedern, Karl Schoenafinger, Alfons Enhsen
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Patent number: 6852760Abstract: Compositions and methods of using the same for the treatment of diabetes and other disorders of glucose metabolism are provided. Compositions may include an anti-diabetic agent and one or more of a bioavailable source of chromium and vanadium.Type: GrantFiled: September 17, 1999Date of Patent: February 8, 2005Assignee: Akesis Pharmaceuticals, Inc.Inventors: Stuart A. Fine, Kevin J. Kinsella
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Patent number: 6812250Abstract: The invention relates to carboxamide-substituted phenylurea derivatives and their physiologically tolerated salts and physiologically functional derivatives. Compounds of the formula I in which the radicals have the stated meanings, and the physiologically tolerated salts thereof and process for their preparation are described. The compounds are suitable, for example, for treating type II diabetes.Type: GrantFiled: May 24, 2002Date of Patent: November 2, 2004Assignee: Aventis Pharma Deutschland GmbHInventors: Elisabeth Defossa, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Erich von Roedern, Stefan Peukert, Alfons Enhsen, Armin Bauer, Bernd Neises, Karl Ulrich Wendt
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Publication number: 20040213824Abstract: Termites can be controlled by applying a composition comprising N-(2,6-difluorobenzoyl)-N′-[2 -chloro-3,5-bis(trifluoromethyl)phenyl]urea and dried yeast.Type: ApplicationFiled: April 26, 2004Publication date: October 28, 2004Applicant: SUMITOMO CHEMICAL COMPANY, LIMITEDInventor: Takaaki Itoh
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Publication number: 20040192739Abstract: In one aspect, the present invention provides a method for modulating an Edg-2 receptor mediated biological activity in a cell. A cell expressing the Edg-2 receptor is contacted with an modulator of the Edg-2 receptor, which modulates the Edg-2 receptor mediated biological activity. In another aspect, the present invention provides a method for modulating Edg-2 receptor mediated biological activity in a subject. A therapeutically effective amount of an modulator of the Edg-2 receptor is administered to the subject.Type: ApplicationFiled: January 16, 2004Publication date: September 30, 2004Inventors: David Solow-Cordero, Geetha Shankar, Juliet V. Spencer, Charles Gluchowski
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Publication number: 20040167181Abstract: In one aspect, the present invention provides a method of inhibiting an Edg-3 receptor mediated biological activity in a cell. A cell expressing the Edg-3 receptor is contacted with an amount of an Edg-3 receptor inhibitor sufficient to inhibit the Edg-3 receptor mediated biological activity. Preferably, the inhibitor is not a phospholipid.Type: ApplicationFiled: January 16, 2004Publication date: August 26, 2004Inventors: David Solow-Cordero, Geetha Shankar, Juliet V. Spencer, Charles Gluchowski
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Publication number: 20040152743Abstract: The invention relates to heterocyclically substituted benzoylureas and also to their physiologically tolerated salts and physiologically functional derivatives.Type: ApplicationFiled: July 11, 2003Publication date: August 5, 2004Applicant: Aventis Pharma Deutschland GmbHInventors: Karl Schoenafinger, Elisabeth Defossa, Dieter Kadereit, Erich Von Roedern, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Karl-Ulrich Wendt
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Publication number: 20040102518Abstract: The invention relates to N-benzoylureidocinnamic acid derivatives and to their physiologically tolerated salts and physiologically functional derivatives.Type: ApplicationFiled: June 6, 2003Publication date: May 27, 2004Applicant: Aventis Pharma AGInventors: Karl Schoenafinger, Elisabeth Defossa, Dieter Kadereit, Erich Von Roedern, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Karl-Ulrich Wendt
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Publication number: 20040097593Abstract: Novel acyl urea, thiourea, carbamate, thiocarbamate and related compounds are provided which are effective in inhibiting the cytokine-mediated inflammatory response in cultured cells, in ameliorating bone destruction in an animal model of arthritis and in lowering blood glucose levels in animal models of Type II diabetes mellitus. The compounds are disclosed as useful for a variety of treatments including the treatment of diabetes mellitus, insulin resistance, inflammation, inflammatory diseases, immunological diseases and cancer.Type: ApplicationFiled: May 7, 2003Publication date: May 20, 2004Inventors: Partha Neogi, Debedranath Dey, Joseph C. Fuller, Liang Chen, Ta-Kai Li
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Publication number: 20040087659Abstract: The invention relates to urea- and urethane-substituted acylureas and to their physiologically tolerated salts and physiologically functional derivatives.Type: ApplicationFiled: July 11, 2003Publication date: May 6, 2004Inventors: Elisabeth Defossa, Dieter Kadereit, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Karl-Ulrich Wendt, Erich Von Roedern, Karl Schoenafinger
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Publication number: 20040087491Abstract: A class of compounds is described which can be used for the treatment of viral infections.Type: ApplicationFiled: October 30, 2003Publication date: May 6, 2004Inventors: Daniel L. Flynn, Kenneth Williams, Susan L. Hockerman, Jeffrey Zablocki
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Publication number: 20040067943Abstract: Compounds of the formula (I), in which M is a central building block selected from the group below in which Al, A2, K1 and K2 are as defined in the description, are novel effective tryptase inhibitors.Type: ApplicationFiled: August 18, 2003Publication date: April 8, 2004Inventor: Thomas Martin
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Patent number: 6710085Abstract: The present invention is directed to new compositions of matter comprising the reaction products of a carboxylic acid and a urea having the formula: where R1, R2, R3 and R4 are the same or different and are selected from the group consisting of hydrogen, substituted and unsubstituted alkyl, allyl, vinyl and alkoxyl groups having from 1-6 carbon atoms, substituted and unsubstituted phenyl groups and the halides. Preferably, the reaction product of the present invention is N,N′-diformylurea or N,N′-diacetylurea. These reaction products, e.g., diformylurea, have been found to produce significantly improved growth in a variety of agricultural products when applied to the seed, to the surrounding soil or to the foliage of the emerging plant. Because of the similarity in the carbon, nitrogen, oxygen structure of these reaction products with many biological compounds, it is believed that the reaction products of the present invention may find use in a variety of biological applications.Type: GrantFiled: July 29, 2002Date of Patent: March 23, 2004Assignee: Stoller Enterprises, Inc.Inventor: Frank William Dean
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Publication number: 20030212141Abstract: The present invention is directed to a new class of serotonin 5HT2 antagonists and thier use in the treatment of a variety of diseases.Type: ApplicationFiled: April 9, 2003Publication date: November 13, 2003Inventors: Thaddeus R. Nieduzak, Mark W. Dudley, John H. Kehne
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Patent number: 6632840Abstract: Monoacyl-substituted guanidines of formula III, or a salt or acid thereof, and their use as medicine or diagnostic aid: in which X(2) isType: GrantFiled: March 24, 2000Date of Patent: October 14, 2003Assignee: Hoechst AktiengesellschaftInventors: Heinz-Werner Kleemann, Hans-Jochen Lang, Andreas Weichert, Peter Crause, Wolfgang Scholz, Udo Albus, Jan-Robert Schwark
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Publication number: 20030176497Abstract: The invention relates to carboxamide-substituted phenylurea derivatives and their physiologically tolerated salts and physiologically functional derivatives.Type: ApplicationFiled: May 24, 2002Publication date: September 18, 2003Inventors: Elisabeth Defossa, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Erich von Roedern, Stefan Peukert, Alfons Enhsen, Armin Bauer, Bernd Neises, Karl Ulrich Wendt
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Publication number: 20030175319Abstract: Termites can be controlled by applying an effective amount of N-[2-chloro-3,5-bis(trifluoromethyl)phenyl]-N′-(2,6-difluorobenzoyl)urea supported on cellulose.Type: ApplicationFiled: February 25, 2003Publication date: September 18, 2003Applicant: SUMITOMO CHEMICAL COMPANY, LIMITEDInventors: Seietsu Aki, Hiromi Eguchi
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Publication number: 20030158260Abstract: A method of successfully controlling sea lice in commercial fish farming, in an efficient and environmentally friendly way, with the compounds named in claim 1, preferably by injection, and a method of automating this type of control, are described.Type: ApplicationFiled: January 22, 2003Publication date: August 21, 2003Inventor: Hariolf Schmid
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Publication number: 20030153591Abstract: There is now described a method of controlling pests with pymetrozine, profenofos, a benzoylurea-derivative or a carbamat-derivative; more specifically a method of controlling pests in and on transgenic crops of useful plants, such as, for example, in crops of maize, cereals, soya beans, tomatoes, cotton, potatoes, rice and mustard, with pymetrozine, profenofos, a benzoylurea-derivative, especially lufenuron; or a carbamat-derivative, especially fenoxycarb; characterized in that a pesticidal composition comprising pymetrozine, profenofos, a benzoylurea-derivative or a carbamat-derivative, in free form or in agrochemically useful salt form and at least one auxiliary is applied to the pests or their environment, in particular to the crop plant itself.Type: ApplicationFiled: October 17, 2002Publication date: August 14, 2003Inventor: Bruce Lee
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Publication number: 20030139459Abstract: A veterinary preparation for fleas is described, which consists of an amount that is effective against fleas of a combination of a compound of formula (I), wherein R1 hydrogen, C1-C6-alkyl or C3-C7-cycloalkyl; R2 is hydrogen, C1-C6-alkyl or C3-C7-cycloalkyl; R3 is hydrogen or C1-C6-alkyl; and A is heterocycly which is unsubstituted or substituted once or repeatedly by identical or different halogen atoms; and a compound of formula (II), wherein X is halogen, X1 is hydrogen or halogen; X2 is hydrogen or halogen; Y is partially or completely halogenated C1-C6-alkoxy, or partially or completely halogenated C1-C6-alkoxy which is interrupted by one oxygen atom, or partially or completely halogenated C2-C6-alkenyl; Y1 is hydrogen or halogen; Y2 is hydrogen or halogen; Y3 is hydrogen or halogen; Z1 is hydrogen or C1-C3-alkyl; and Z2 is hydrogen or C1-C3-alkyl; and a physiologically acceptable formulation excipient.Type: ApplicationFiled: December 12, 2002Publication date: July 24, 2003Inventors: Olivier Tinembart, Michel Franc, Jean Steffan
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Patent number: 6566304Abstract: The invention relates to use of (a) compounds of phosphorus containing at least partly lipophilic organic radicals together with (b) urea and/or urea derivatives in selected quantity ratios of (a) to (b) as a soil additive for biologically controlling plant-parasitic soil nematodes by strengthening the correspondingly antagonistic soil potential, more particularly by strengthening the growth of antagonistic and/or nematicidal rhizosphere bacteria and/or corresponding mycorrhiza strains—and at the same time strengthening the growth of cultivated plants in soil. The multicomponent mixtures which strengthen bacterial growth are preferably introduced into the region of the plant roots in the form of an aqueous preparation using plant-compatible emulsifiers before and/or during plant growth. Components (a) and (b) are used in such quantity ratios that the ratio by weight of C to N is no higher than 6:1 and preferably no higher than 5:1.Type: GrantFiled: February 6, 2001Date of Patent: May 20, 2003Assignee: Cognis Deutschland GmbHInventors: Doris Bell, Bettina Kopp-Holtwiesche, Stephan Von Tapavicza
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Patent number: 6528543Abstract: Glucokinase activating compounds of the formula wherein R1 and R2 are independently hydrogen, halo, amino, nitro, cyano, sulfonamido, lower alkyl, perfluoro-lower alkyl, lower alkyl thio, perfluoro-lower alkyl thio, lower alkyl sulfonyl, or perfluoro-lower alkyl sulfonyl; R3 is cycloalkyl having from 3 to 7 carbon atoms or lower alkyl having from 2 to 4 carbon atoms; R4 is hydrogen, lower alkyl, lower alkenyl, hydroxy lower alkyl, halo lower alkyl, R5 and R6 are hydrogen or lower alkyl; and n is 0, 1, 2, 3 or 4; or a pharmaceutically acceptable salt thereofType: GrantFiled: March 21, 2000Date of Patent: March 4, 2003Assignee: Hoffman-La Roche Inc.Inventors: Fred Thomas Bizzarro, Wendy Lea Corbett, Antonio Focella, Joseph Francis Grippo, Nancy-Ellen Haynes, George William Holland, Robert Francis Kester, Paige Erin Mahaney, Ramakanth Sarabu
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Patent number: 6506778Abstract: The invention is directed to acylphenylurea derivatives and their physiologically tolerated salts and physiologically functional derivatives. Compounds of the formula I in which the radicals have the stated meanings, and their physiologically tolerated salts and a process for their preparation are described. The compounds are suitable, for example, for treating type II diabetes.Type: GrantFiled: June 8, 2001Date of Patent: January 14, 2003Assignee: Aventis Pharma Deutschland GmbHInventors: Elisabeth Defossa, Thomas Klabunde, Hans-Joerg Burger, Andreas Herling, Karl-Heinz Baringhaus
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Patent number: 6436999Abstract: Diacyl-substituted guanidines of the formula I are described where X(1) and X(2) are as defined herein. The compounds are suitable for use as antiarrhythmic pharmaceuticals possessing a cardioprotective component for the prophylaxis and treatment of infarction and for the treatment of angina pectoris, in connection with which they also inhibit or strongly reduce, in a preventitive manner the pathophysiological processes associated with the genesis of ischemically induced damage, in particular associated with the elicitation of ischemically induced cardiac arrhythmias.Type: GrantFiled: April 18, 1997Date of Patent: August 20, 2002Assignee: Hoechst AktiengesellschaftInventors: Heinz-Werner Kleemann, Hans-Jochen Lang, Andreas Weichert, Peter Crause, Wolfgang Scholz, Udo Albus, Jan-Robert Schwark
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Patent number: 6416752Abstract: An improved termite bait composition comprises a powdered cellulosic attractant having a particle size in the range of approximately 1 to 100 micrometers and a termite killing agent. Also disclosed are a method for controlling termites by applying the termite bait composition to a termite infested area and a termite bait composition package for use in a termite bait station comprising the termite bait composition contained within a termite attractive package.Type: GrantFiled: January 4, 2001Date of Patent: July 9, 2002Assignee: Whitmire Micro-Gen Research Laboratories, Inc.Inventors: Ronald O. Richardson, Robin L. Kern
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Publication number: 20020058683Abstract: A veterinary preparation for fleas is described, which consists of an amount that is effective against fleas of a combination of a compound of formula (I), wherein R1 hydrogen, C1-C6-alkyl or C3-C7-cycloalkyl; R2 is hydrogen, C1-C6-alkyl or C3-C7-cycloalkyl; R3 is hydrogen or C1-C6-alkyl; and A is heterocycly which is unsubstituted or substituted once or repeatedly by identical or different halogen atoms; and a compound of formula (II), wherein X is halogen, X1 is hydrogen or halogen; X2 is hydrogen or halogen; Y is partially or completely halogenated C1-C6-alkoxy, or partially or completely halogenated C1-C6-alkoxy which is interrupted by one oxygen atom, or partially or completely halogenated C2-C6-alkenyl; Y1 is hydrogen or halogen; Y2 is hydrogen or halogen; Y3 is hydrogen or halogen; Z1 is hydrogen or C1-C3-alkyl; and Z2 is hydrogen or C1-C3-alkyl; and a physiologically acceptable formulation excipient.Type: ApplicationFiled: April 3, 2001Publication date: May 16, 2002Inventors: Olivier Tinembart, Michel Franc, Jean Steffan
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Patent number: 6368588Abstract: The present invention relates to an ant or yellow jacket bait that is particularly effective for controlling carpenter ants. The bait is comprised mostly of sugars in a viscous and fluid form that may be readily dispensed into an ant station at room temperatures, and provides a moist, sweet surface that is attractive to ants.Type: GrantFiled: June 22, 2000Date of Patent: April 9, 2002Assignee: FMC CorporationInventors: Larry G. Faehl, James B. Ballard
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Patent number: 6348493Abstract: The present invention provides new methods for the treatment of viral hepatitis C involving the administration of vitamin E and other compounds with antioxidant properties. Treatment with high doses of vitamin E is effective in treating chronic hepatitis C in patients refractory to interferon. In addition, new methods are described for the treatment of hepatic fibrosis and hepatic conditions manifesting hepatic fibrosis involving the administration of butylated hydroxytoluene and a metabolite of pentoxifylline, 1-[3-carboxypropyl]-3, 7-dimethylxanthine. Furthermore, new methods are described for the treatment and prevention of hepatic disorders involving the use of 2,6-di-tert-butylphenol derivatives.Type: GrantFiled: November 28, 2000Date of Patent: February 19, 2002Assignee: The Regents of the University of CaliforniaInventor: Mario Chojkier
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Patent number: 6337078Abstract: Controlled release compositions of matter are disclosed comprising complexes for treating a population of one or more aquatic organisms in a column of water. The complexes comprise at least one system wherein the system comprises at least one bioactive agent as a component selected for treating a population of aquatic organisms, at least one carrier component, and at least one coating component for regulating the controlled release rate and release profile of the bioactive agent in water or at least one bioactive agent and one joint-function component that can serve as both a carrier and coating to regulate the controlled release rate and release profile of the bioactive agent in water, with or without optional binder components and/or additional formulation materials. The components are selected to sink or float so that the complexes will permeate and/or remain in any planar or volumetric segment of a water column for a period of time that is sufficient to effectively treat a population of aquatic organisms.Type: GrantFiled: December 10, 1999Date of Patent: January 8, 2002Assignee: Lee County Mosquito Control DistrictInventor: Richard Levy
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Patent number: 6333355Abstract: The present invention provides a method to control ecto-parasites of a host animals wherein 1-(2,6-difluorobenzoyl)-3-[2-fluoro-4-(1,1,2,3,3,3-hexafluoropropoxy)phenyl]urea is applied to the said host animals. By the method of the present invention, ecto-parasites of animals can be controlled effectively for a long period of time.Type: GrantFiled: November 17, 1998Date of Patent: December 25, 2001Assignee: Sumitomo Chemical Company, LimitedInventors: Satoshi Sembo, Tatsuya Mori, Noriyasu Sakamoto
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Publication number: 20010044470Abstract: The present invention provides a method to control ecto-parasites of a host animals wherein 1-(2,6-difluorobenzoyl)-3-[2-fluoro-4-(1,1,2,3,3,3-hexafluoropropoxy)phenyl]urea is applied to the said host animals.Type: ApplicationFiled: November 17, 1998Publication date: November 22, 2001Inventors: SATOSHI SEMBO, TATSUYA MORI, NORIYASU SAKAMOTO
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Publication number: 20010031790Abstract: A method of lowering plasma levels of &agr;-dicarbonyl precursors of advanced alycation end products such as methylglyoxal in a patient having type 2 diabetes by administrating metformin in a dosage at least twenty five percent in excess of its antidiabetic therapeutic regimen for the patient is provided. The high dosage of metformin acts to reduce plasma levels of &agr;-dicarbonyl compounds by a mechanism distinct from that whereby it exerts its antidiabetic activity.Type: ApplicationFiled: December 13, 2000Publication date: October 18, 2001Inventors: Paul J. Beisswenger, Benjamin S. Szwergold
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Patent number: 6303657Abstract: Compounds of the formula (I) wherein R1 and R2 are H, methyl, or ethyl, provided that at least one of R1 or R2 is methyl or ethyl, have unexpected activity against ants. Compounds wherein at least one of R1 and R2 is methyl or ethyl are novel.Type: GrantFiled: November 7, 2000Date of Patent: October 16, 2001Assignee: Dow AgroSciences LLCInventors: Ronald J. Spragia, George W. Johnson, Laura L. Karr, Jeff M. Edwards, Brian M. Schneider
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Patent number: 6270784Abstract: The present invention relates to new active compound combinations of pyrethroids with insect development inhibitors, for achieving a long-term effect against animal pests with high effectiveness, fewer environmentally polluting properties and a toxicologically favourable control concept.Type: GrantFiled: February 10, 1998Date of Patent: August 7, 2001Assignee: Bayer AktiengesellschaftInventors: Klaus Mrusek, Manfred-Heinrich Schütte
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Patent number: 6245327Abstract: The present invention relates to an ant or yellow jacket bait that is particularly effective for controlling carpenter ants. The bait is comprised mostly of sugars in a viscous and fluid form that may be readily dispeised into an ant station at room temperatures, and provides a moist, sweet surface that is attractive to ants.Type: GrantFiled: March 25, 1996Date of Patent: June 12, 2001Assignee: FMC CorporationInventors: Larry G. Faehl, James B. Ballard
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Patent number: 6245816Abstract: Compounds of the formula (I) wherein R1 and R2 are H, methyl, or ethyl, have unexpected activity against ants. Compounds wherein at least one of R1 and R2 is methyl or ethyl are novel.Type: GrantFiled: March 24, 2000Date of Patent: June 12, 2001Inventors: Ronald J. Spragia, George W. Johnson, Laura L. Karr, Jeff M. Edwards, Brian M. Schneider
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Patent number: 6221912Abstract: Compounds of the formula (I) wherein R1 and R2 are H, methyl, or ethyl, have unexpected activity against cockroaches. Compounds wherein at least one of R1 and R2 is methyl or ethyl are novel.Type: GrantFiled: November 10, 1998Date of Patent: April 24, 2001Assignee: Dow AgroSciences LLCInventors: Ronald J. Spragia, George W. Johnson, Laura L. Karr, Jeff M. Edwards, Brian M. Schneider
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Patent number: 6114378Abstract: A fungicidal mixture comprisinga) an oxime ether of the formula I ##STR1## where the substituents have the following meaning: X is oxygen or amino (NH);Y is CH or N;Z is oxygen, sulfur, amino (NH) or C.sub.1 -C.sub.4 -alkylamino (N--C.sub.1 -C.sub.4 -alkyl);R' is C.sub.1 -C.sub.6 -alkyl, C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.2 -C.sub.6 -haloalkenyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.3 -C.sub.6 -haloalkynyl, C.sub.3 -C.sub.6 -cycloalkylmethyl, or benzyl which may be partially or fully halogenated and/or may carry one to three of the following radicals: cyano, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -haloalkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -haloalkoxy and C.sub.1 -C.sub.Type: GrantFiled: October 21, 1998Date of Patent: September 5, 2000Assignee: BASF AktiengesellschaftInventors: Ruth Muller, Herbert Bayer, Hubert Sauter, Eberhard Ammermann, Gisela Lorenz, Siegfried Strathmann, Klaus Schelberger, Maria Scherer
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Patent number: 6110971Abstract: The present invention provides a pharmaceutical or veterinary composition comprising, a carrier and an active ingredient being a compound of the following formula I: ##STR1## wherein R.sup.1 and R.sup.2 are each independently hydrogen, halogen or methoxy, as well as salts of the compound of formula I.Further provided by the invention is a method of treatment of fungal infection, comprising administering to a patient in need, an effective amount of the compound of said formula I.Type: GrantFiled: February 4, 1999Date of Patent: August 29, 2000Assignee: Novartis Animal Health US, Inc.Inventors: Yair Ben-Ziony, Boaz Arzi
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Patent number: 6093415Abstract: Combinations of a chitin synthesis inhibitor (e.g. hexaflumuron, flufenoxuron, lufenuron, and dimiin) with a juvenile hormone mimic (e.g. methoprene and pyriproxyfen) afford synergistic activity against termites.Type: GrantFiled: February 11, 1998Date of Patent: July 25, 2000Assignee: Dow AgroSciences LLCInventors: Laura L. Karr, Ronald J. Sbragia
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Patent number: 6057370Abstract: A method for controlling insects of Lepidoptera on a genetically altered cotton plant having incorporated therein a gene derived from Bacillus thuringiensis (Bt) which codes for and expresses a protein having pesticide activity comprising the steps of applying to the foliage of said genetically altered cotton plant a pesticidally active amount of certain substituted benzoyl urea compounds.Type: GrantFiled: May 27, 1997Date of Patent: May 2, 2000Inventors: Robert Timothy Weiland, Paul Thomas McDonald, Kevin Leo Kelley
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Patent number: 6057355Abstract: A pesticidal combination comprising a compound of formula (I) and a 1-arylpyrazole of formula (II).Type: GrantFiled: April 10, 1998Date of Patent: May 2, 2000Assignee: Rhone-Poulenc Inc.Inventors: Charles Lee Haas, Michael Thomas Pilato, Philip Reid Timmons, Tai-Teh Wu, Scot Kevin Huber, Bernard Leroux
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Patent number: 6040345Abstract: Compounds of formula (I): ##STR1## wherein R.sup.1 is H or F and R.sup.2 is CF.sub.3 or CF.sub.2 CF.sub.3, exhibit unexpectedly superior activity against cockroaches and are also useful to control other insects.Type: GrantFiled: October 31, 1997Date of Patent: March 21, 2000Assignee: Dow AgroSciences LLCInventors: Ronald E. Hackler, Kathryn E. Lawrence
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Patent number: 6025397Abstract: Compounds of the formula (I) ##STR1## wherein R.sup.1 and R.sup.2 are H, methyl, or ethyl, have unexpected activity against fleas. Compounds wherein at least one of R.sup.1 and R.sup.2 is methyl or ethyl are novel.Type: GrantFiled: November 10, 1998Date of Patent: February 15, 2000Assignee: Dow AgroSciences LLCInventors: Ronald J. Soragia, George W. Johnson, Laura L. Karr, Brian M. Schneider, Jeff M. Edwards
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Patent number: 6022882Abstract: The present invention relates to a novel benzoyl urea derivative which exhibits potent growth-retarding activity against pests and which is represented by formula (I), ##STR1## in which A represents N or CH, and X.sup.1 and X.sup.2 independently of one another represent hydrogen, fluoro, chloro or bromo.Type: GrantFiled: December 21, 1998Date of Patent: February 8, 2000Assignee: Dongbu Hannong Chemical Co., Ltd.Inventors: Jung Ho Kim, Yong Woo Shin, Jung Nyoung Heo, Eui Deok Kim, Joon Seo Park, Hyun Sam Song